Page last updated: 2024-09-05

sorafenib and gw 3965

sorafenib has been researched along with gw 3965 in 3 studies

Compound Research Comparison

Studies
(sorafenib)
Trials
(sorafenib)
Recent Studies (post-2010)
(sorafenib)
Studies
(gw 3965)
Trials
(gw 3965)
Recent Studies (post-2010) (gw 3965)
6,5207305,2512350164

Protein Interaction Comparison

ProteinTaxonomysorafenib (IC50)gw 3965 (IC50)
Alpha-glucosidase MAL32Saccharomyces cerevisiae S288C4.8
Oxysterols receptor LXR-betaHomo sapiens (human)0.47
Oxysterols receptor LXR-alphaHomo sapiens (human)0.5691

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's2 (66.67)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Chen, Y; Dai, F; Gu, T; Jiang, H; Li, K; Liang, Z; Liu, Y; She, J; Tang, L; Zhan, Z; Zhou, X1
Cai, X; Chen, J; Ji, L; Jiang, S; Liang, X; Liang, Y; Lin, C; Lin, Z; Pan, Y; Tao, L; Wan, Z; Xia, S; Xu, J1

Other Studies

3 other study(ies) available for sorafenib and gw 3965

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
LXR-Mediated Regulation of Marine-Derived Piericidins Aggravates High-Cholesterol Diet-Induced Cholesterol Metabolism Disorder in Mice.
    Journal of medicinal chemistry, 2021, 07-22, Volume: 64, Issue:14

    Topics: Animals; Cholesterol; Cholesterol, Dietary; Diet, High-Fat; Dose-Response Relationship, Drug; Hep G2 Cells; Humans; Liver X Receptors; Male; Mice; Mice, Inbred C57BL; Molecular Structure; Pericarditis; Structure-Activity Relationship; Tumor Cells, Cultured

2021
LXR activation potentiates sorafenib sensitivity in HCC by activating microRNA-378a transcription.
    Theranostics, 2020, Volume: 10, Issue:19

    Topics: Animals; Benzoates; Benzylamines; Carcinoma, Hepatocellular; Cell Line, Tumor; Cell Proliferation; Cell Survival; Down-Regulation; Drug Resistance, Neoplasm; Drug Synergism; Gene Expression Regulation, Neoplastic; Humans; Karyopherins; Liver Neoplasms; Liver X Receptors; Male; Mice; MicroRNAs; Middle Aged; Neoplasm Transplantation; Receptor, IGF Type 1; Sorafenib; Survival Analysis

2020