Page last updated: 2024-09-05

sorafenib and fr 148083

sorafenib has been researched along with fr 148083 in 3 studies

Compound Research Comparison

Studies
(sorafenib)
Trials
(sorafenib)
Recent Studies (post-2010)
(sorafenib)
Studies
(fr 148083)
Trials
(fr 148083)
Recent Studies (post-2010) (fr 148083)
6,5207305,25123021

Protein Interaction Comparison

ProteinTaxonomysorafenib (IC50)fr 148083 (IC50)
Dual specificity mitogen-activated protein kinase kinase 7Homo sapiens (human)0.8
Mitogen-activated protein kinase kinase kinase 7Homo sapiens (human)0.017
Mitogen-activated protein kinase 1Homo sapiens (human)2.5393
Nuclear receptor subfamily 2 group C member 2Homo sapiens (human)0.009
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)0.0296
Transcription factor p65Homo sapiens (human)0.25
TGF-beta-activated kinase 1 and MAP3K7-binding protein 1Homo sapiens (human)0.0087
Phospholipase A-2-activating proteinHomo sapiens (human)0.011

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Ide, M; Kamikawa, T; Kashiwagi, H; Matsuo, A; Miura, T; Morikami, K; Muraoka, T; Nishihara, M1
Caballero, E; García-Cárceles, J; Gil, C; Martínez, A1

Reviews

1 review(s) available for sorafenib and fr 148083

ArticleYear
Kinase Inhibitors as Underexplored Antiviral Agents.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Animals; Antiviral Agents; Drug Repositioning; Humans; Protein Kinase Inhibitors; Virus Diseases; Viruses

2022

Other Studies

2 other study(ies) available for sorafenib and fr 148083

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Identification of a selective inhibitor of transforming growth factor β-activated kinase 1 by biosensor-based screening of focused libraries.
    Bioorganic & medicinal chemistry letters, 2017, 02-15, Volume: 27, Issue:4

    Topics: Biosensing Techniques; Humans; Kinetics; MAP Kinase Kinase Kinases; Protein Kinase Inhibitors; Surface Plasmon Resonance

2017