Page last updated: 2024-09-05

solifenacin succinate and oxybutynin

solifenacin succinate has been researched along with oxybutynin in 54 studies

Compound Research Comparison

Studies
(solifenacin succinate)
Trials
(solifenacin succinate)
Recent Studies (post-2010)
(solifenacin succinate)
Studies
(oxybutynin)
Trials
(oxybutynin)
Recent Studies (post-2010) (oxybutynin)
5221943432,6076191,670

Protein Interaction Comparison

ProteinTaxonomysolifenacin succinate (IC50)oxybutynin (IC50)
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)2.5951
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.027
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.002
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.0032
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.0035
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.0027
Sodium-dependent noradrenaline transporter Homo sapiens (human)2.5951
Cytochrome P450 2C19Homo sapiens (human)0.6
D(3) dopamine receptorHomo sapiens (human)0.4288
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.792
Sodium-dependent dopamine transporter Homo sapiens (human)0.0855
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.0242

Research

Studies (54)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's21 (38.89)29.6817
2010's30 (55.56)24.3611
2020's3 (5.56)2.80

Authors

AuthorsStudies
Honda, K; Ikeda, K; Kobayashi, S; Miyata, K; Suzuki, M; Takeuchi, M; Yamada, T1
Ikeda, K; Kobayashi, S; Miyata, K1
Hatanaka, T; Ikeda, K; Kobayashi, S; Miyata, K; Ohtake, A; Sasamata, M; Sato, S; Ukai, M1
Sand, PK1
Miyata, K; Oki, T; Sato, S; Yamada, S1
Krivoborodov, GG; Mazo, EB1
MacDiarmid, SA; Staskin, DR1
Appell, RA; McCrery, RJ; Smith, PP1
Oki, T; Takeuchi, C; Yamada, S1
Brubaker, L; Chapple, C; Coyne, KS; Kopp, Z1
Hegde, SS; Michel, MC1
Hatanaka, T; Miyata, K; Noguchi, Y; Ohtake, A; Okutsu, H; Saitoh, C; Sasamata, M; Sato, S; Suzuki, M; Ukai, M; Yuyama, H1
Cardozo, L; Cartwright, R; Robinson, D; Vella, M1
Bertozzi, R; Cipriani, S; Colli, E; Meschia, M; Montorsi, F; Olivieri, L; Parazzini, F1
Chugh, A; Gupta, JB; Hegde, LG; Kumar, N; Meru, AV; Naruganahalli, KS; Ray, A; Sinha, S1
Hilas, O; Lam, S1
Duggan, P; Wong, C1
Brenes, FJ; Chapple, CR; Rosenberg, MT1
Fujino, T; Ito, Y; Matsui, M; Noguchi, Y; Ohtake, A; Oyunzul, L; Sasamata, M; Suzuki, M; Yamada, S; Yoshida, A; Yuyama, H1
Bolodeoku, J; Edgar, C; Tretter, RN; Wesnes, KA1
Cardozo, L; Sidhu, M; Thorpe, A; Warner, J1
Wyndaele, JJ1
Barkin, J; Carlson, K; Drutz, H; Egerdie, B; Gajewski, JB; Herschorn, S; Paradiso-Hardy, F; Pommerville, P; Radomski, S; Schulz, J; Stothers, L1
Herschorn, S; Piwko, C; Vicente, C1
Fujino, T; Kageyama, A; Nozawa, Y; Yamada, S; Yoshida, A1
Jakobsen, SM; Kersten, H; Molden, E1
Bungay, PJ; Callegari, E; Fenner, KS; Kay, GG; Kempshall, S; LaPerle, JL; Malhotra, B; Michel, MC; Webster, R1
Schröder, A; Thüroff, JW1
Chess-Williams, R; Moro, C; Uchiyama, J1
Cody, JD; Ellis, G; Hay-Smith, EJ; Herbison, GP; Madhuvrata, P1
Kane, RL; Ramakrishnan, R; Sainfort, F; Shamliyan, T; Wyman, JF1
Alessandri, F; Candiani, M; Ferrero, S; Leone Roberti Maggiore, U; Origoni, M; Remorgida, V; Salvatore, S; Venturini, PL1
Compion, G; Dale, M; Stow, B; Tretter, R; Wagg, A2
Cornu, JN1
Abrams, P; Hart, WM; Munro, V; Nazir, J; Retsa, P1
Akino, H; Fujiuchi, Y; Fuse, H; Kitagawa, Y; Miyazawa, K; Namiki, M; Suzuki, K; Yokoyama, O1
Kosilov, KV; Kosilova, LV; Krasnykh, MA; Loparev, SA1
Blak, B; Hakimi, Z; Johnson, M; Nazir, J; Odeyemi, IA1
Trivedi, D1
Barkin, J; Berner, T; Diles, D; Franks, B1
Hikiyama, E; Ito, Y; Kashiwabara, M; Onoue, S; Yamada, S; Yoshida, A1
Hsiao, SM; Kuo, HC; Lin, HH1
Ahamed, AA; Lim, V; Masten Singh, PK; Naidu, P; Nalliah, S; Wg, P1
Dandolu, V; Lua, LL; Pathak, P1
Aballéa, S; Hakimi, Z; Kelleher, C; Maman, K; Mankowski, C; Nazir, J; Odeyemi, I1
Herbison, P; McKenzie, JE1
Cetinel, B; Dincer, M; Gultekin, MH; Guzelsoy, M; Onal, B; Turegun, FA1
Almeida, FG; Bernardo, WM; Sacomani, CAR; Silvinato, A1
Hansson, F; Kilany, S; Milsom, I; Schiotz, HA; Svensson, M1
Panicker, JN; Richardson, K; Welk, B1
Gomes, T; Herschorn, S; Jarvi, K; Juurlink, D; Matta, R; Nam, RK1
Hiren Prajapati, HP; Krunal Vishavadia, KV; Madhu Sharma, MS; Sandip Solanki, SS1

Reviews

20 review(s) available for solifenacin succinate and oxybutynin

ArticleYear
Elevating our therapeutic expectations in overactive bladder.
    Journal of the American Academy of Nurse Practitioners, 2004, Volume: 16, Issue:10 Suppl

    Topics: Benzhydryl Compounds; Benzilates; Benzofurans; Constipation; Cresols; Delayed-Action Preparations; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Treatment Outcome; Urinary Incontinence; Vision Disorders; Xerostomia

2004
[Neurological aspect of the hyperactive urinary bladder syndrome].
    Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova, 2005, Volume: 105, Issue:7

    Topics: Benzilates; Brain; Brain Diseases; Cerebrovascular Circulation; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Parkinson Disease; Positron-Emission Tomography; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder, Neurogenic

2005
Using anticholinergics to treat overactive bladder: the issue of treatment tolerability.
    The American journal of medicine, 2006, Volume: 119, Issue:3 Suppl 1

    Topics: Benzhydryl Compounds; Benzilates; Benzofurans; Cholinergic Antagonists; Cresols; Humans; Mandelic Acids; Nortropanes; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Incontinence

2006
The emergence of new drugs for overactive bladder.
    Expert opinion on emerging drugs, 2006, Volume: 11, Issue:1

    Topics: Acetylcholine; Amines; Animals; Anticonvulsants; Benzhydryl Compounds; Cresols; Cyclohexanecarboxylic Acids; Drug Evaluation, Preclinical; Gabapentin; gamma-Aminobutyric Acid; Humans; Mandelic Acids; Muscarinic Antagonists; Muscle, Smooth; Phenylpropanolamine; Product Surveillance, Postmarketing; Quinuclidines; Randomized Controlled Trials as Topic; Receptor, Muscarinic M3; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urinary Incontinence

2006
Patient-reported outcomes in overactive bladder: importance for determining clinical effectiveness of treatment.
    Urology, 2006, Volume: 68, Issue:2 Suppl

    Topics: Benzhydryl Compounds; Clinical Trials as Topic; Cresols; Health Status; Humans; Mandelic Acids; Muscarinic Antagonists; Patient Compliance; Patient Satisfaction; Phenylpropanolamine; Quality of Life; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Neurogenic; Urinary Incontinence, Stress

2006
Treatment of the overactive bladder syndrome with muscarinic receptor antagonists: a matter of metabolites?
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 374, Issue:2

    Topics: Benzhydryl Compounds; Benzilates; Benzofurans; Cresols; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Parasympatholytics; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive

2006
New developments in the treatment of urinary incontinence.
    Minerva urologica e nefrologica = The Italian journal of urology and nephrology, 2006, Volume: 58, Issue:4

    Topics: Administration, Cutaneous; Adrenergic Uptake Inhibitors; Benzofurans; Drug Therapy, Combination; Duloxetine Hydrochloride; Humans; Mandelic Acids; Muscarinic Antagonists; Pyrrolidines; Quality of Life; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Thiophenes; Treatment Outcome; Urinary Bladder, Overactive; Urinary Incontinence, Stress

2006
Number of daytime micturitions and volume voided per micturition in the evaluation of efficacy of drugs for overactive bladder: findings from randomized clinical trials.
    European urology, 2007, Volume: 52, Issue:2

    Topics: Benzhydryl Compounds; Cresols; Humans; Mandelic Acids; Muscarinic Antagonists; Phenylpropanolamine; Quinuclidines; Randomized Controlled Trials as Topic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive; Urination

2007
Update on drugs for overactive bladder syndrome.
    Drug and therapeutics bulletin, 2007, Volume: 45, Issue:6

    Topics: Benzhydryl Compounds; Benzilates; Benzofurans; Cholinergic Antagonists; Cresols; Humans; Mandelic Acids; Muscarinic Antagonists; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Randomized Controlled Trials as Topic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive

2007
Pharmacologic management of overactive bladder.
    Clinical interventions in aging, 2007, Volume: 2, Issue:3

    Topics: Benzhydryl Compounds; Benzofurans; Cresols; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Overactive

2007
Listening to the patient: a flexible approach to the use of antimuscarinic agents in overactive bladder syndrome.
    BJU international, 2009, Volume: 104, Issue:7

    Topics: Benzofurans; Drug Administration Schedule; Humans; Mandelic Acids; Multicenter Studies as Topic; Muscarinic Antagonists; Patient Satisfaction; Pyrrolidines; Quinuclidines; Randomized Controlled Trials as Topic; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder, Overactive

2009
New strategies for medical management of overactive bladder in children.
    Current opinion in urology, 2010, Volume: 20, Issue:4

    Topics: Benzhydryl Compounds; Benzilates; Botulinum Toxins; Child; Cresols; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Phenylpropanolamine; Quinuclidines; Receptors, Muscarinic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive; Urination

2010
Which anticholinergic drug for overactive bladder symptoms in adults.
    The Cochrane database of systematic reviews, 2012, Jan-18, Volume: 1

    Topics: Adult; Benzhydryl Compounds; Cholinergic Antagonists; Cresols; Humans; Mandelic Acids; Phenylpropanolamine; Quinuclidines; Randomized Controlled Trials as Topic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive; Urinary Incontinence

2012
Benefits and harms of pharmacologic treatment for urinary incontinence in women: a systematic review.
    Annals of internal medicine, 2012, Jun-19, Volume: 156, Issue:12

    Topics: Benzhydryl Compounds; Benzilates; Benzofurans; Comparative Effectiveness Research; Cresols; Female; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Phenylpropanolamine; Pyrrolidines; Quality of Life; Quinuclidines; Randomized Controlled Trials as Topic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Incontinence

2012
Pharmacokinetics and toxicity of antimuscarinic drugs for overactive bladder treatment in females.
    Expert opinion on drug metabolism & toxicology, 2012, Volume: 8, Issue:11

    Topics: Benzhydryl Compounds; Benzilates; Benzofurans; Chronic Disease; Cresols; Drug Combinations; Female; Humans; Imidazoles; Mandelic Acids; Muscarinic Antagonists; Nocturia; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive; Urinary Incontinence

2012
Cochrane Review Summary: Pelvic floor muscle training added to another active treatment versus the same active treatment alone for urinary incontinence in women.
    Primary health care research & development, 2015, Volume: 16, Issue:6

    Topics: Clenbuterol; Combined Modality Therapy; Duloxetine Hydrochloride; Electric Stimulation; Exercise Therapy; Female; Hot Temperature; Humans; Mandelic Acids; Patient Satisfaction; Pelvic Floor; Solifenacin Succinate; Treatment Outcome; Urinary Incontinence; Urological Agents

2015
Comparison of efficacy and tolerability of pharmacological treatment for the overactive bladder in women: A network meta-analysis.
    Australian family physician, 2017, Volume: 46, Issue:3

    Topics: Dose-Response Relationship, Drug; Female; Humans; Mandelic Acids; Randomized Controlled Trials as Topic; Solifenacin Succinate; Urinary Bladder, Overactive; Urological Agents; Women's Health

2017
Comparative efficacy and tolerability of solifenacin 5 mg/day versus other oral antimuscarinic agents in overactive bladder: A systematic literature review and network meta-analysis.
    Neurourology and urodynamics, 2018, Volume: 37, Issue:3

    Topics: Benzhydryl Compounds; Benzilates; Humans; Mandelic Acids; Muscarinic Antagonists; Network Meta-Analysis; Solifenacin Succinate; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Overactive

2018
Which anticholinergic is best for people with overactive bladders? A network meta-analysis.
    Neurourology and urodynamics, 2019, Volume: 38, Issue:2

    Topics: Benzhydryl Compounds; Benzilates; Benzofurans; Cholinergic Antagonists; Humans; Imidazoles; Mandelic Acids; Network Meta-Analysis; Pyrrolidines; Solifenacin Succinate; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Overactive

2019
The cognitive effect of anticholinergics for patients with overactive bladder.
    Nature reviews. Urology, 2021, Volume: 18, Issue:11

    Topics: Benzhydryl Compounds; Benzofurans; Cholinergic Antagonists; Cognition; Cognitive Dysfunction; Dementia; Humans; Mandelic Acids; Prodromal Symptoms; Pyrrolidines; Risk Assessment; Risk Factors; Solifenacin Succinate; Tolterodine Tartrate; Urinary Bladder, Overactive

2021

Trials

7 trial(s) available for solifenacin succinate and oxybutynin

ArticleYear
Solifenacin for overactive bladder in women unsuccessfully treated with immediate release oxybutynin: a pilot study.
    Journal of obstetrics and gynaecology : the journal of the Institute of Obstetrics and Gynaecology, 2009, Volume: 29, Issue:1

    Topics: Adult; Aged; Cholinergic Antagonists; Female; Humans; Mandelic Acids; Middle Aged; Nocturia; Pilot Projects; Quality of Life; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Treatment Failure; Urinary Bladder, Overactive

2009
Exploratory pilot study assessing the risk of cognitive impairment or sedation in the elderly following single doses of solifenacin 10 mg.
    Expert opinion on drug safety, 2009, Volume: 8, Issue:6

    Topics: Aged; Attention; Cognition; Cognition Disorders; Cross-Over Studies; Executive Function; Female; Humans; Hypnotics and Sedatives; Learning; Male; Mandelic Acids; Memory; Memory, Short-Term; Muscarinic Antagonists; Neuropsychological Tests; Parasympatholytics; Pilot Projects; Quinuclidines; Reaction Time; Risk; Sample Size; Solifenacin Succinate; Tetrahydroisoquinolines

2009
Tolerability of 5 mg solifenacin once daily versus 5 mg oxybutynin immediate release 3 times daily: results of the VECTOR trial.
    The Journal of urology, 2010, Volume: 183, Issue:5

    Topics: Adult; Aged; Aged, 80 and over; Canada; Chi-Square Distribution; Double-Blind Method; Drug Administration Schedule; Female; Humans; Incidence; Male; Mandelic Acids; Middle Aged; Muscarinic Antagonists; Quinuclidines; Severity of Illness Index; Solifenacin Succinate; Surveys and Questionnaires; Tetrahydroisoquinolines; Treatment Outcome; Urinary Bladder, Overactive; Xerostomia

2010
Canadian cost-effectiveness analysis of solifenacin compared to oxybutynin immediate-release in patients with overactive bladder.
    Journal of medical economics, 2010, Volume: 13, Issue:3

    Topics: Canada; Cost-Benefit Analysis; Female; Humans; Male; Mandelic Acids; Markov Chains; Muscarinic Antagonists; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder, Overactive

2010
Randomised, multicentre, placebo-controlled, double-blind crossover study investigating the effect of solifenacin and oxybutynin in elderly people with mild cognitive impairment: the SENIOR study.
    European urology, 2013, Volume: 64, Issue:1

    Topics: Age Factors; Aged; Aged, 80 and over; Aging; Analysis of Variance; Attention; Cognition; Cognitive Dysfunction; Cross-Over Studies; Double-Blind Method; Female; Humans; Least-Squares Analysis; Male; Mandelic Acids; Memory; Muscarinic Antagonists; Quinuclidines; Risk Factors; Solifenacin Succinate; Tetrahydroisoquinolines; Time Factors; Treatment Outcome; United Kingdom; Urinary Bladder, Overactive; Urological Agents

2013
[Treatment of overactive bladder in older women increased doses of antimuscarinic drugs safe and effective alternative to existing methods].
    Advances in gerontology = Uspekhi gerontologii, 2014, Volume: 27, Issue:1

    Topics: Aged; Benzhydryl Compounds; Benzilates; Cresols; Dose-Response Relationship, Drug; Double-Blind Method; Drug Monitoring; Drug Synergism; Drug Therapy, Combination; Female; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Phenylpropanolamine; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Overactive; Urinary Incontinence, Urge; Urodynamics

2014
Which antimuscarinic agents used in the treatment of overactive bladder increase heart rate? a prospective randomized clinical trial.
    International urology and nephrology, 2019, Volume: 51, Issue:3

    Topics: Adult; Aged; Benzhydryl Compounds; Benzilates; Benzofurans; Blood Pressure; Female; Heart Rate; Humans; Male; Mandelic Acids; Middle Aged; Muscarinic Antagonists; Nortropanes; Prospective Studies; Pyrrolidines; Solifenacin Succinate; Tolterodine Tartrate; Urinary Bladder, Overactive

2019

Other Studies

27 other study(ies) available for solifenacin succinate and oxybutynin

ArticleYear
M(3) receptor antagonism by the novel antimuscarinic agent solifenacin in the urinary bladder and salivary gland.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 366, Issue:2

    Topics: Animals; Benzofurans; Bradycardia; Calcium; Carbachol; Cells, Cultured; Cytosol; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; In Vitro Techniques; Isoquinolines; Kinetics; Male; Mandelic Acids; Mice; Mice, Inbred BALB C; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Pyrrolidines; Quinuclidines; Rats; Receptor, Muscarinic M3; Receptors, Muscarinic; Salivary Glands; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder

2002
Comparison of in vitro selectivity profiles of solifenacin succinate (YM905) and current antimuscarinic drugs in bladder and salivary glands: a Ca2+ mobilization study in monkey cells.
    Life sciences, 2004, Jan-02, Volume: 74, Issue:7

    Topics: Animals; Benzhydryl Compounds; Benzofurans; Calcium; Calcium Signaling; Carbachol; Cresols; Dose-Response Relationship, Drug; In Vitro Techniques; Inhibitory Concentration 50; Macaca fascicularis; Male; Mandelic Acids; Muscarinic Antagonists; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Solifenacin Succinate; Submandibular Gland; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder

2004
In vitro and in vivo tissue selectivity profile of solifenacin succinate (YM905) for urinary bladder over salivary gland in rats.
    European journal of pharmacology, 2004, May-25, Volume: 492, Issue:2-3

    Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Calcium; Cresols; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Mandelic Acids; Muscarinic Antagonists; Myocytes, Smooth Muscle; Organ Specificity; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Rats; Rats, Wistar; Solifenacin Succinate; Submandibular Gland; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder

2004
Muscarinic receptor binding, plasma concentration and inhibition of salivation after oral administration of a novel antimuscarinic agent, solifenacin succinate in mice.
    British journal of pharmacology, 2005, Volume: 145, Issue:2

    Topics: Administration, Oral; Animals; Depression, Chemical; In Vitro Techniques; Male; Mandelic Acids; Mice; Muscarinic Antagonists; Quinuclidines; Radioligand Assay; Receptors, Muscarinic; Salivary Glands; Salivation; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder

2005
Comparative evaluation of exocrine muscarinic receptor binding characteristics and inhibition of salivation of solifenacin in mice.
    Biological & pharmaceutical bulletin, 2006, Volume: 29, Issue:7

    Topics: Administration, Oral; Animals; Kinetics; Male; Mandelic Acids; Mice; Mice, Inbred Strains; Parasympatholytics; Quinuclidines; Receptors, Muscarinic; Saliva; Salivation; Solifenacin Succinate; Tetrahydroisoquinolines

2006
Pharmacological characterization of a new antimuscarinic agent, solifenacin succinate, in comparison with other antimuscarinic agents.
    Biological & pharmaceutical bulletin, 2007, Volume: 30, Issue:1

    Topics: Animals; Atropine; Benzhydryl Compounds; Benzilates; Benzofurans; Binding, Competitive; Carbachol; CHO Cells; Cholinergic Agonists; Cresols; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mandelic Acids; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; N-Methylscopolamine; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Muscarinic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Transfection; Urinary Bladder; Urinary Bladder, Overactive; Urination

2007
Comparative in vivo uroselectivity profiles of anticholinergics, tested in a novel anesthetized rabbit model.
    European journal of pharmacology, 2007, Oct-31, Volume: 572, Issue:2-3

    Topics: Anesthesia; Animals; Benzhydryl Compounds; Benzofurans; Carbachol; Cholinergic Antagonists; Cresols; Injections, Intra-Arterial; Male; Mandelic Acids; Phenylpropanolamine; Pressure; Pyrrolidines; Quinuclidines; Rabbits; Salivary Glands; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder

2007
Comparison of muscarinic receptor selectivity of solifenacin and oxybutynin in the bladder and submandibular gland of muscarinic receptor knockout mice.
    European journal of pharmacology, 2009, Aug-01, Volume: 615, Issue:1-3

    Topics: Administration, Oral; Animals; Dose-Response Relationship, Drug; Male; Mandelic Acids; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Muscarinic Antagonists; Protein Binding; Quinuclidines; Radioligand Assay; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Solifenacin Succinate; Submandibular Gland; Tetrahydroisoquinolines; Urinary Bladder

2009
The cost-effectiveness of solifenacin vs fesoterodine, oxybutynin immediate-release, propiverine, tolterodine extended-release and tolterodine immediate-release in the treatment of patients with overactive bladder in the UK National Health Service.
    BJU international, 2010, Volume: 106, Issue:4

    Topics: Benzhydryl Compounds; Benzilates; Cost-Benefit Analysis; Cresols; Decision Trees; Delayed-Action Preparations; Humans; Mandelic Acids; Muscarinic Antagonists; Phenylpropanolamine; Quality of Life; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Overactive

2010
Pediatrics: combining antimuscarinics shows promise for overactive bladder.
    Nature reviews. Urology, 2010, Volume: 7, Issue:2

    Topics: Benzhydryl Compounds; Child; Cresols; Drug Therapy, Combination; Humans; Mandelic Acids; Muscarinic Antagonists; Pediatrics; Phenylpropanolamine; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive

2010
Loss of muscarinic and purinergic receptors in urinary bladder of rats with hydrochloric acid-induced cystitis.
    Urology, 2010, Volume: 76, Issue:4

    Topics: Adenosine Triphosphate; Animals; Benzhydryl Compounds; Benzofurans; Cresols; Cystitis; Disease Models, Animal; Down-Regulation; Female; Hydrochloric Acid; Mandelic Acids; N-Methylscopolamine; Organophosphonates; Phenols; Phenylpropanolamine; Pirenzepine; Polycyclic Compounds; Pyridoxal Phosphate; Pyrrolidines; Quinuclidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Purinergic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urination; Urodynamics

2010
Evaluation of brain anticholinergic activities of urinary spasmolytic drugs using a high-throughput radio receptor bioassay.
    Journal of the American Geriatrics Society, 2011, Volume: 59, Issue:3

    Topics: Benzhydryl Compounds; Benzofurans; Biological Assay; Brain; Cognition Disorders; Cresols; Humans; In Vitro Techniques; Mandelic Acids; Muscarinic Antagonists; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate

2011
A comprehensive non-clinical evaluation of the CNS penetration potential of antimuscarinic agents for the treatment of overactive bladder.
    British journal of clinical pharmacology, 2011, Volume: 72, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; Benzhydryl Compounds; Benzofurans; Blood-Brain Barrier; Brain; Cell Line; Chromatography, High Pressure Liquid; Cresols; Humans; Male; Mandelic Acids; Muscarinic Antagonists; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Randomized Controlled Trials as Topic; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Solifenacin Succinate; Tandem Mass Spectrometry; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder, Overactive

2011
Urothelial/lamina propria spontaneous activity and the role of M3 muscarinic receptors in mediating rate responses to stretch and carbachol.
    Urology, 2011, Volume: 78, Issue:6

    Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Carbachol; Cresols; Diamines; Mandelic Acids; Mucous Membrane; Muscarinic Antagonists; Muscle Contraction; Phenylpropanolamine; Piperidines; Pirenzepine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Stress, Mechanical; Swine; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urothelium

2011
Overactive bladder medical management in the elderly: it is time to go beyond the tip of the iceberg.
    European urology, 2013, Volume: 64, Issue:1

    Topics: Aging; Cognition; Cognitive Dysfunction; Female; Humans; Male; Mandelic Acids; Muscarinic Antagonists; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder, Overactive; Urological Agents

2013
Reply from authors re: Jean-Nicolas Cornu. Overactive bladder medical management in the elderly: it is time to go beyond the tip of the iceberg. Eur Urol 2013;64:82-3.
    European urology, 2013, Volume: 64, Issue:1

    Topics: Aging; Cognition; Cognitive Dysfunction; Female; Humans; Male; Mandelic Acids; Muscarinic Antagonists; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder, Overactive; Urological Agents

2013
Cost-effectiveness analysis of solifenacin versus oxybutynin immediate-release in the treatment of patients with overactive bladder in the United Kingdom.
    Journal of medical economics, 2013, Volume: 16, Issue:10

    Topics: Benzhydryl Compounds; Cohort Studies; Cost-Benefit Analysis; Cresols; Humans; Incontinence Pads; Mandelic Acids; Markov Chains; Medication Adherence; Models, Economic; Muscarinic Antagonists; Patient Dropouts; Phenylpropanolamine; Quality-Adjusted Life Years; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Treatment Outcome; United Kingdom; Urinary Bladder, Overactive; Urinary Incontinence

2013
Factors influencing patient satisfaction with antimuscarinic treatment of overactive bladder syndrome: results of a real-life clinical study.
    International journal of urology : official journal of the Japanese Urological Association, 2014, Volume: 21, Issue:4

    Topics: Aged; Aged, 80 and over; Benzhydryl Compounds; Benzilates; Cresols; Cross-Sectional Studies; Female; Humans; Imidazoles; Japan; Male; Mandelic Acids; Middle Aged; Muscarinic Antagonists; Patient Satisfaction; Phenylpropanolamine; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Overactive

2014
Drug treatment patterns for the management of men with lower urinary tract symptoms associated with benign prostatic hyperplasia who have both storage and voiding symptoms: a study using the health improvement network UK primary care data.
    Current medical research and opinion, 2015, Volume: 31, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Aged; Benzhydryl Compounds; Cresols; Family Practice; Humans; Lower Urinary Tract Symptoms; Male; Mandelic Acids; Middle Aged; Muscarinic Antagonists; Phenylpropanolamine; Primary Health Care; Prostatic Hyperplasia; Quinuclidines; Retrospective Studies; Solifenacin Succinate; Sulfonamides; Tamsulosin; Tetrahydroisoquinolines; Tolterodine Tartrate; United Kingdom

2015
Alpha blocker monotherapy versus combination therapy with antimuscarinics in men with persistent LUTS refractory to alpha-adrenergic treatment: patterns of persistence.
    The Canadian journal of urology, 2015, Volume: 22, Issue:4

    Topics: Administrative Claims, Healthcare; Adrenergic alpha-Antagonists; Aged; Benzofurans; Doxazosin; Drug Therapy, Combination; Humans; Longitudinal Studies; Male; Mandelic Acids; Medication Adherence; Middle Aged; Muscarinic Antagonists; Ontario; Prazosin; Prostatic Hyperplasia; Prostatism; Pyrrolidines; Quinazolines; Retrospective Studies; Solifenacin Succinate; Sulfonamides; Tamsulosin; Tolterodine Tartrate

2015
Muscarinic Receptor Binding in Rat Bladder Urothelium and Detrusor Muscle by Intravesical Solifenacin.
    Biological & pharmaceutical bulletin, 2016, Volume: 39, Issue:7

    Topics: Administration, Intravesical; Animals; Benzilates; Male; Mandelic Acids; Muscarinic Antagonists; Muscle, Smooth; Nortropanes; Rats, Sprague-Dawley; Receptors, Muscarinic; Solifenacin Succinate; Urinary Bladder; Urological Agents; Urothelium

2016
Treatment Outcome of Overactive Bladder Patients Receiving Antimuscarinic Therapy for More than One Year.
    Lower urinary tract symptoms, 2018, Volume: 10, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Constipation; Female; Humans; Male; Mandelic Acids; Middle Aged; Muscarinic Antagonists; Retrospective Studies; Severity of Illness Index; Solifenacin Succinate; Time Factors; Tolterodine Tartrate; Treatment Outcome; Urinary Bladder, Overactive; Urodynamics; Vision Disorders; Xerostomia; Young Adult

2018
Comparing anticholinergic persistence and adherence profiles in overactive bladder patients based on gender, obesity, and major anticholinergic agents.
    Neurourology and urodynamics, 2017, Volume: 36, Issue:8

    Topics: Adolescent; Adult; Cholinergic Antagonists; Female; Humans; Male; Mandelic Acids; Medication Adherence; Middle Aged; Obesity; Quality of Life; Sex Factors; Solifenacin Succinate; Tolterodine Tartrate; Urinary Bladder, Overactive; Young Adult

2017
Overactive bladder - pharmacological treatment.
    Revista da Associacao Medica Brasileira (1992), 2019, May-02, Volume: 65, Issue:4

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Antidepressive Agents; Benzilates; Benzofurans; Brazil; Clinical Decision-Making; Drug Therapy, Combination; Humans; Mandelic Acids; Muscarinic Antagonists; Nortropanes; Pyrrolidines; Solifenacin Succinate; Thiazoles; Tolterodine Tartrate; Urinary Bladder, Overactive

2019
A Nordic registry-based study of drug treatment patterns in overactive bladder patients.
    Scandinavian journal of urology, 2019, Volume: 53, Issue:4

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Aged; Aged, 80 and over; Benzhydryl Compounds; Benzofurans; Denmark; Female; Humans; Male; Mandelic Acids; Middle Aged; Muscarinic Antagonists; Norway; Practice Patterns, Physicians'; Prospective Studies; Pyrrolidines; Registries; Solifenacin Succinate; Sweden; Thiazoles; Tolterodine Tartrate; Urinary Bladder, Overactive

2019
Receipt of Overactive Bladder Drugs and Incident Dementia: A Population-based Case-control Study.
    European urology focus, 2022, Volume: 8, Issue:5

    Topics: Aged; Canada; Case-Control Studies; Dementia; Humans; Muscarinic Antagonists; Solifenacin Succinate; Tolterodine Tartrate; Urinary Bladder, Overactive

2022
[Assessment of prescribing practices in overactive bladder pharmacotherapy across different specialties of India: a prescription trend analysis].
    Urologiia (Moscow, Russia : 1999), 2023, Issue:2

    Topics: Acetanilides; Humans; Muscarinic Antagonists; Prescriptions; Solifenacin Succinate; Tolterodine Tartrate; Urinary Bladder, Overactive; Urological Agents

2023