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sk&f 97541 and gamma-aminobutyric acid

sk&f 97541 has been researched along with gamma-aminobutyric acid in 22 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (40.91)18.2507
2000's13 (59.09)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baumann, PA; Brugger, F; Froestl, W; Gentsch, C; Hall, RG; Jaekel, J; Mickel, SJ; Olpe, HR; Strub, D; von Sprecher, G1
Chebib, M; Hanrahan, JR; Hibbs, DE; Johnston, GA; Kim, HL; Kumar, RJ; Salam, NK1
Howson, W; Lacey, MG; Seabrook, GR1
Cunningham, JR; Neal, MJ1
Lipton, SA; Pan, ZH1
Lipton, SA; Pan, ZH; Zhang, D; Zhang, X1
Chang, Y; Weiss, DS1
Euler, T; Wässle, H1
Fukunaga, A; Hasegawa, H; Imamura, K; Matsuno, A; Ogawa, C; Ozoe, Y1
Blackshaw, LA; Dent, J; Lehmann, A; Staunton, E1
Greka, A; Lipton, SA; Zhang, D1
Mezler, M; Müller, T; Raming, K1
Herzig, KH; Hoepfner, M; Jansen, A; Riecken, EO; Scherübl, H1
Bexis, S; Froestl, W; Kerr, DI; Marino, V; Ong, J; Parker, DA1
Giniatullin, R; Nistri, A; Sokolova, E1
Lasater, EM; Vigh, J1
Carai, MA; Colombo, G; Froestl, W; Gessa, GL; Serra, S; Vacca, G1
Farb, DH; Gravielle, MC; Lyons, HR; Martin, SC; Russek, SJ; Steiger, JL1
Martinez, V; Piqueras, L1
Hamasaka, Y; Nässel, DR; Wegener, C1
Chebib, M; Hanrahan, JR; Johnston, GA; Kumar, RJ; Mewett, KN; Morriss, G; Wooller, S1
Baumann, O; Blenau, W; Rotte, C; Walz, B; Witte, J1

Other Studies

22 other study(ies) available for sk&f 97541 and gamma-aminobutyric acid

ArticleYear
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.
    Journal of medicinal chemistry, 1995, Aug-18, Volume: 38, Issue:17

    Topics: Animals; Behavior, Animal; Cats; Crystallography, X-Ray; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Organophosphonates; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Stereoisomerism; Structure-Activity Relationship

1995
Novel gamma-aminobutyric acid rho1 receptor antagonists; synthesis, pharmacological activity and structure-activity relationships.
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Female; GABA Antagonists; Ligands; Models, Molecular; Molecular Structure; Oocytes; Structure-Activity Relationship; Xenopus laevis

2008
Subpopulations of GABA-mediated synaptic potentials in slices of rat dorsal striatum are differentially modulated by presynaptic GABAB receptors.
    Brain research, 1991, Oct-25, Volume: 562, Issue:2

    Topics: Animals; Baclofen; Caudate Nucleus; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Organophosphorus Compounds; Putamen; Rats; Receptors, GABA-A; Synaptic Membranes

1991
Baclofen enhancement of acetylcholine release from amacrine cells in the rabbit retina by reduction of glycinergic inhibition.
    The Journal of physiology, 1995, Jan-15, Volume: 482 ( Pt 2)

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Muscarine; Organophosphorus Compounds; Rabbits; Retina; Strychnine

1995
Multiple GABA receptor subtypes mediate inhibition of calcium influx at rat retinal bipolar cell terminals.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:4

    Topics: Animals; Axons; Baclofen; Bicuculline; Calcium; Cells, Cultured; gamma-Aminobutyric Acid; Nerve Endings; Organophosphorus Compounds; Picrotoxin; Potassium; Propylamines; Rats; Receptors, GABA; Receptors, GABA-A; Retina

1995
Agonist-induced closure of constitutively open gamma-aminobutyric acid channels with mutated M2 domains.
    Proceedings of the National Academy of Sciences of the United States of America, 1997, Jun-10, Volume: 94, Issue:12

    Topics: Amino Acid Sequence; Animals; Cloning, Molecular; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Ion Channels; Macromolecular Substances; Membrane Potentials; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Organophosphorus Compounds; Point Mutation; Rats; Receptors, GABA; Receptors, Glycine; Receptors, Nicotinic; Recombinant Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Virulence Factors, Bordetella; Xenopus laevis

1997
Substitutions of the highly conserved M2 leucine create spontaneously opening rho1 gamma-aminobutyric acid receptors.
    Molecular pharmacology, 1998, Volume: 53, Issue:3

    Topics: Animals; Chlorides; Female; gamma-Aminobutyric Acid; Humans; Leucine; Mutagenesis, Site-Directed; Oocytes; Organophosphorus Compounds; Picrotoxin; Receptors, GABA; Xenopus laevis

1998
Different contributions of GABAA and GABAC receptors to rod and cone bipolar cells in a rat retinal slice preparation.
    Journal of neurophysiology, 1998, Volume: 79, Issue:3

    Topics: Animals; Azetidinecarboxylic Acid; Bicuculline; Chloride Channels; Excitatory Amino Acid Agonists; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Organophosphorus Compounds; Patch-Clamp Techniques; Quisqualic Acid; Rats; Receptors, GABA; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Retinal Cone Photoreceptor Cells; Retinal Rod Photoreceptor Cells

1998
Insecticidal properties of 3-aminopropyl(methyl)phosphinic acid and its effect on K(+)-evoked release of acetylcholine from cockroach synaptosomes.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1999, Volume: 122, Issue:2

    Topics: Acetylcholine; Animals; Female; GABA Antagonists; gamma-Aminobutyric Acid; Houseflies; Insecticides; Male; Organophosphorus Compounds; Periplaneta; Potassium; Synaptosomes

1999
Inhibition of transient LES relaxations and reflux in ferrets by GABA receptor agonists.
    The American journal of physiology, 1999, Volume: 277, Issue:4

    Topics: Animals; Baclofen; Behavior, Animal; Deglutition; Esophagogastric Junction; Female; Ferrets; GABA Agonists; gamma-Aminobutyric Acid; Gastroesophageal Reflux; Hydrogen-Ion Concentration; Manometry; Muscle Relaxation; Organophosphonates; Organophosphorus Compounds; Phosphinic Acids; Pressure; Time Factors

1999
Expression of GABA(C) receptor rho1 and rho2 subunits during development of the mouse retina.
    The European journal of neuroscience, 2000, Volume: 12, Issue:10

    Topics: Age Factors; Animals; Animals, Newborn; Bicuculline; Fetus; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; Mice; Mice, Inbred C57BL; Neurons, Afferent; Organophosphorus Compounds; Picrotoxin; Receptors, GABA; Retina; RNA, Messenger

2000
Cloning and functional expression of GABA(B) receptors from Drosophila.
    The European journal of neuroscience, 2001, Volume: 13, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Line; Central Nervous System; Cloning, Molecular; Cyclic AMP; Drosophila melanogaster; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Invertebrate; Gene Expression Regulation, Developmental; GTP-Binding Proteins; Humans; Insect Proteins; Kidney; Molecular Sequence Data; Oocytes; Organophosphorus Compounds; Phosphinic Acids; Phylogeny; Potassium Channels; Potassium Channels, Inwardly Rectifying; Propanolamines; Receptors, GABA-B; Sequence Homology, Amino Acid; Xenopus

2001
GABA(C) receptors in neuroendocrine gut cells: a new GABA-binding site in the gut.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 441, Issue:2-3

    Topics: Acrylates; Animals; Bicuculline; Calcium; Cholecystokinin; Cytarabine; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Immunohistochemistry; Intestinal Neoplasms; Kinetics; Mice; Mice, Transgenic; Neuroendocrine Tumors; Organophosphorus Compounds; Pyridazines; Receptors, GABA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured

2000
CGP 36216 is a selective antagonist at GABA(B) presynaptic receptors in rat brain.
    European journal of pharmacology, 2001, Volume: 415, Issue:2-3

    Topics: Animals; Autoreceptors; Baclofen; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Neocortex; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B

2001
The ATP-mediated fast current of rat dorsal root ganglion neurons is a novel effector for GABA(B) receptor activation.
    Neuroscience letters, 2003, Mar-06, Volume: 338, Issue:3

    Topics: Adenosine Triphosphate; Animals; Baclofen; Benzylamines; Cells, Cultured; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Membrane Potentials; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Rats; Receptors, GABA-A; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X3

2003
Intracellular calcium release resulting from mGluR1 receptor activation modulates GABAA currents in wide-field retinal amacrine cells: a study with caffeine.
    The European journal of neuroscience, 2003, Volume: 17, Issue:11

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amacrine Cells; Animals; Anticoagulants; Bicuculline; Caffeine; Calcium; Calcium Channels; Carps; Cells, Cultured; Central Nervous System Stimulants; Chelating Agents; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electric Conductivity; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Heparin; Immunohistochemistry; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Kainic Acid; Membrane Potentials; Methoxyhydroxyphenylglycol; Organophosphorus Compounds; Patch-Clamp Techniques; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Retina; Ryanodine

2003
Suppression of GABA(B) receptor function in vivo by disulfide reducing agent, DL-dithiothreitol (DTT).
    Psychopharmacology, 2004, Volume: 174, Issue:2

    Topics: Animals; Baclofen; Conditioning, Operant; Discrimination Learning; Dithiothreitol; Drug Interactions; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Hydroxybutyrates; Male; Mice; Mice, Inbred DBA; Organophosphonates; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Long-Evans; Reflex

2004
Differential expression of gamma-aminobutyric acid type B receptor subunit mRNAs in the developing nervous system and receptor coupling to adenylyl cyclase in embryonic neurons.
    The Journal of comparative neurology, 2004, May-17, Volume: 473, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Binding Sites; Blotting, Western; Chlorocebus aethiops; COS Cells; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; GABA Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; In Situ Hybridization; Inhibitory Concentration 50; Male; Nervous System; Neurons; Organophosphorus Compounds; Phosphodiesterase Inhibitors; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; Tritium

2004
Peripheral GABAB agonists stimulate gastric acid secretion in mice.
    British journal of pharmacology, 2004, Volume: 142, Issue:6

    Topics: Animals; Antibodies, Monoclonal; Atropine; Baclofen; Deoxyglucose; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gastric Acid; Gastrins; Imidazoles; Injections, Intravenous; Male; Mice; Mice, Knockout; Muscimol; Organophosphorus Compounds; Pentagastrin; Peptides, Cyclic; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Somatostatin; Somatostatin; Time Factors; Vagotomy

2004
GABA modulates Drosophila circadian clock neurons via GABAB receptors and decreases in calcium.
    Journal of neurobiology, 2005, Volume: 65, Issue:3

    Topics: Animals; Animals, Genetically Modified; Blotting, Western; Calcium; Cell Count; Cells, Cultured; Circadian Rhythm; Diagnostic Imaging; Dose-Response Relationship, Drug; Drosophila; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Green Fluorescent Proteins; Immunohistochemistry; Isoenzymes; Larva; Neurons; Organophosphorus Compounds; Picrotoxin; Receptors, GABA-A; Serotonin

2005
(3-Aminocyclopentyl)methylphosphinic acids: novel GABA(C) receptor antagonists.
    Neuropharmacology, 2007, Volume: 52, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Oocytes; Organophosphorus Compounds; Patch-Clamp Techniques; Receptors, GABA; Xenopus laevis

2007
Source, topography and excitatory effects of GABAergic innervation in cockroach salivary glands.
    The Journal of experimental biology, 2009, Volume: 212, Issue:Pt 1

    Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Electrophysiology; Fluorescent Antibody Technique; GABA Agonists; gamma-Aminobutyric Acid; Neurons; Organophosphorus Compounds; Periplaneta; Phosphinic Acids; Salivary Glands

2009