sk&f 97541 has been researched along with gamma-aminobutyric acid in 22 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 9 (40.91) | 18.2507 |
2000's | 13 (59.09) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Baumann, PA; Brugger, F; Froestl, W; Gentsch, C; Hall, RG; Jaekel, J; Mickel, SJ; Olpe, HR; Strub, D; von Sprecher, G | 1 |
Chebib, M; Hanrahan, JR; Hibbs, DE; Johnston, GA; Kim, HL; Kumar, RJ; Salam, NK | 1 |
Howson, W; Lacey, MG; Seabrook, GR | 1 |
Cunningham, JR; Neal, MJ | 1 |
Lipton, SA; Pan, ZH | 1 |
Lipton, SA; Pan, ZH; Zhang, D; Zhang, X | 1 |
Chang, Y; Weiss, DS | 1 |
Euler, T; Wässle, H | 1 |
Fukunaga, A; Hasegawa, H; Imamura, K; Matsuno, A; Ogawa, C; Ozoe, Y | 1 |
Blackshaw, LA; Dent, J; Lehmann, A; Staunton, E | 1 |
Greka, A; Lipton, SA; Zhang, D | 1 |
Mezler, M; Müller, T; Raming, K | 1 |
Herzig, KH; Hoepfner, M; Jansen, A; Riecken, EO; Scherübl, H | 1 |
Bexis, S; Froestl, W; Kerr, DI; Marino, V; Ong, J; Parker, DA | 1 |
Giniatullin, R; Nistri, A; Sokolova, E | 1 |
Lasater, EM; Vigh, J | 1 |
Carai, MA; Colombo, G; Froestl, W; Gessa, GL; Serra, S; Vacca, G | 1 |
Farb, DH; Gravielle, MC; Lyons, HR; Martin, SC; Russek, SJ; Steiger, JL | 1 |
Martinez, V; Piqueras, L | 1 |
Hamasaka, Y; Nässel, DR; Wegener, C | 1 |
Chebib, M; Hanrahan, JR; Johnston, GA; Kumar, RJ; Mewett, KN; Morriss, G; Wooller, S | 1 |
Baumann, O; Blenau, W; Rotte, C; Walz, B; Witte, J | 1 |
22 other study(ies) available for sk&f 97541 and gamma-aminobutyric acid
Article | Year |
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Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.
Topics: Animals; Behavior, Animal; Cats; Crystallography, X-Ray; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Organophosphonates; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Stereoisomerism; Structure-Activity Relationship | 1995 |
Novel gamma-aminobutyric acid rho1 receptor antagonists; synthesis, pharmacological activity and structure-activity relationships.
Topics: Animals; Female; GABA Antagonists; Ligands; Models, Molecular; Molecular Structure; Oocytes; Structure-Activity Relationship; Xenopus laevis | 2008 |
Subpopulations of GABA-mediated synaptic potentials in slices of rat dorsal striatum are differentially modulated by presynaptic GABAB receptors.
Topics: Animals; Baclofen; Caudate Nucleus; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Organophosphorus Compounds; Putamen; Rats; Receptors, GABA-A; Synaptic Membranes | 1991 |
Baclofen enhancement of acetylcholine release from amacrine cells in the rabbit retina by reduction of glycinergic inhibition.
Topics: Acetylcholine; Animals; Baclofen; Bicuculline; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Muscarine; Organophosphorus Compounds; Rabbits; Retina; Strychnine | 1995 |
Multiple GABA receptor subtypes mediate inhibition of calcium influx at rat retinal bipolar cell terminals.
Topics: Animals; Axons; Baclofen; Bicuculline; Calcium; Cells, Cultured; gamma-Aminobutyric Acid; Nerve Endings; Organophosphorus Compounds; Picrotoxin; Potassium; Propylamines; Rats; Receptors, GABA; Receptors, GABA-A; Retina | 1995 |
Agonist-induced closure of constitutively open gamma-aminobutyric acid channels with mutated M2 domains.
Topics: Amino Acid Sequence; Animals; Cloning, Molecular; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Ion Channels; Macromolecular Substances; Membrane Potentials; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Organophosphorus Compounds; Point Mutation; Rats; Receptors, GABA; Receptors, Glycine; Receptors, Nicotinic; Recombinant Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Virulence Factors, Bordetella; Xenopus laevis | 1997 |
Substitutions of the highly conserved M2 leucine create spontaneously opening rho1 gamma-aminobutyric acid receptors.
Topics: Animals; Chlorides; Female; gamma-Aminobutyric Acid; Humans; Leucine; Mutagenesis, Site-Directed; Oocytes; Organophosphorus Compounds; Picrotoxin; Receptors, GABA; Xenopus laevis | 1998 |
Different contributions of GABAA and GABAC receptors to rod and cone bipolar cells in a rat retinal slice preparation.
Topics: Animals; Azetidinecarboxylic Acid; Bicuculline; Chloride Channels; Excitatory Amino Acid Agonists; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Organophosphorus Compounds; Patch-Clamp Techniques; Quisqualic Acid; Rats; Receptors, GABA; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Retinal Cone Photoreceptor Cells; Retinal Rod Photoreceptor Cells | 1998 |
Insecticidal properties of 3-aminopropyl(methyl)phosphinic acid and its effect on K(+)-evoked release of acetylcholine from cockroach synaptosomes.
Topics: Acetylcholine; Animals; Female; GABA Antagonists; gamma-Aminobutyric Acid; Houseflies; Insecticides; Male; Organophosphorus Compounds; Periplaneta; Potassium; Synaptosomes | 1999 |
Inhibition of transient LES relaxations and reflux in ferrets by GABA receptor agonists.
Topics: Animals; Baclofen; Behavior, Animal; Deglutition; Esophagogastric Junction; Female; Ferrets; GABA Agonists; gamma-Aminobutyric Acid; Gastroesophageal Reflux; Hydrogen-Ion Concentration; Manometry; Muscle Relaxation; Organophosphonates; Organophosphorus Compounds; Phosphinic Acids; Pressure; Time Factors | 1999 |
Expression of GABA(C) receptor rho1 and rho2 subunits during development of the mouse retina.
Topics: Age Factors; Animals; Animals, Newborn; Bicuculline; Fetus; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; Mice; Mice, Inbred C57BL; Neurons, Afferent; Organophosphorus Compounds; Picrotoxin; Receptors, GABA; Retina; RNA, Messenger | 2000 |
Cloning and functional expression of GABA(B) receptors from Drosophila.
Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Line; Central Nervous System; Cloning, Molecular; Cyclic AMP; Drosophila melanogaster; GABA Antagonists; gamma-Aminobutyric Acid; Ganglia, Invertebrate; Gene Expression Regulation, Developmental; GTP-Binding Proteins; Humans; Insect Proteins; Kidney; Molecular Sequence Data; Oocytes; Organophosphorus Compounds; Phosphinic Acids; Phylogeny; Potassium Channels; Potassium Channels, Inwardly Rectifying; Propanolamines; Receptors, GABA-B; Sequence Homology, Amino Acid; Xenopus | 2001 |
GABA(C) receptors in neuroendocrine gut cells: a new GABA-binding site in the gut.
Topics: Acrylates; Animals; Bicuculline; Calcium; Cholecystokinin; Cytarabine; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Immunohistochemistry; Intestinal Neoplasms; Kinetics; Mice; Mice, Transgenic; Neuroendocrine Tumors; Organophosphorus Compounds; Pyridazines; Receptors, GABA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured | 2000 |
CGP 36216 is a selective antagonist at GABA(B) presynaptic receptors in rat brain.
Topics: Animals; Autoreceptors; Baclofen; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Neocortex; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B | 2001 |
The ATP-mediated fast current of rat dorsal root ganglion neurons is a novel effector for GABA(B) receptor activation.
Topics: Adenosine Triphosphate; Animals; Baclofen; Benzylamines; Cells, Cultured; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Membrane Potentials; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Rats; Receptors, GABA-A; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X3 | 2003 |
Intracellular calcium release resulting from mGluR1 receptor activation modulates GABAA currents in wide-field retinal amacrine cells: a study with caffeine.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amacrine Cells; Animals; Anticoagulants; Bicuculline; Caffeine; Calcium; Calcium Channels; Carps; Cells, Cultured; Central Nervous System Stimulants; Chelating Agents; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electric Conductivity; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Heparin; Immunohistochemistry; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Kainic Acid; Membrane Potentials; Methoxyhydroxyphenylglycol; Organophosphorus Compounds; Patch-Clamp Techniques; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Retina; Ryanodine | 2003 |
Suppression of GABA(B) receptor function in vivo by disulfide reducing agent, DL-dithiothreitol (DTT).
Topics: Animals; Baclofen; Conditioning, Operant; Discrimination Learning; Dithiothreitol; Drug Interactions; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Hydroxybutyrates; Male; Mice; Mice, Inbred DBA; Organophosphonates; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Long-Evans; Reflex | 2004 |
Differential expression of gamma-aminobutyric acid type B receptor subunit mRNAs in the developing nervous system and receptor coupling to adenylyl cyclase in embryonic neurons.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Binding Sites; Blotting, Western; Chlorocebus aethiops; COS Cells; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; GABA Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; In Situ Hybridization; Inhibitory Concentration 50; Male; Nervous System; Neurons; Organophosphorus Compounds; Phosphodiesterase Inhibitors; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; Tritium | 2004 |
Peripheral GABAB agonists stimulate gastric acid secretion in mice.
Topics: Animals; Antibodies, Monoclonal; Atropine; Baclofen; Deoxyglucose; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gastric Acid; Gastrins; Imidazoles; Injections, Intravenous; Male; Mice; Mice, Knockout; Muscimol; Organophosphorus Compounds; Pentagastrin; Peptides, Cyclic; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Somatostatin; Somatostatin; Time Factors; Vagotomy | 2004 |
GABA modulates Drosophila circadian clock neurons via GABAB receptors and decreases in calcium.
Topics: Animals; Animals, Genetically Modified; Blotting, Western; Calcium; Cell Count; Cells, Cultured; Circadian Rhythm; Diagnostic Imaging; Dose-Response Relationship, Drug; Drosophila; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Green Fluorescent Proteins; Immunohistochemistry; Isoenzymes; Larva; Neurons; Organophosphorus Compounds; Picrotoxin; Receptors, GABA-A; Serotonin | 2005 |
(3-Aminocyclopentyl)methylphosphinic acids: novel GABA(C) receptor antagonists.
Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Oocytes; Organophosphorus Compounds; Patch-Clamp Techniques; Receptors, GABA; Xenopus laevis | 2007 |
Source, topography and excitatory effects of GABAergic innervation in cockroach salivary glands.
Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Electrophysiology; Fluorescent Antibody Technique; GABA Agonists; gamma-Aminobutyric Acid; Neurons; Organophosphorus Compounds; Periplaneta; Phosphinic Acids; Salivary Glands | 2009 |