sk&f 97541 has been researched along with baclofen in 34 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 9 (26.47) | 18.2507 |
| 2000's | 23 (67.65) | 29.6817 |
| 2010's | 1 (2.94) | 24.3611 |
| 2020's | 1 (2.94) | 2.80 |
| Authors | Studies |
|---|---|
| Baumann, PA; Brugger, F; Froestl, W; Gentsch, C; Hall, RG; Jaekel, J; Mickel, SJ; Olpe, HR; Strub, D; von Sprecher, G | 1 |
| Alstermark, C; Amin, K; Dinn, SR; Elebring, T; Fitzpatrick, K; Fjellström, O; Geiss, WB; Gottfries, J; Guzzo, PR; Harding, JP; Holmén, A; Kothare, M; Lehmann, A; Mattsson, JP; Nilsson, K; Sundén, G; Swanson, M; von Unge, S; Woo, AM; Wyle, MJ; Zheng, X | 1 |
| Benham, CD; Evans, ML; Howson, W; Lacey, MG; Seabrook, GR | 1 |
| Howson, W; Lacey, MG; Seabrook, GR | 2 |
| Cunningham, JR; Neal, MJ | 1 |
| Lipton, SA; Pan, ZH | 1 |
| Bon, C; Galvan, M | 1 |
| Hashimoto, T; Kuriyama, K | 1 |
| Blackshaw, LA; Dent, J; Lehmann, A; Staunton, E | 1 |
| Bexis, S; Froestl, W; Kerr, DI; Marino, V; Ong, J; Parker, DA | 1 |
| Giniatullin, R; Nistri, A; Sokolova, E | 1 |
| Duty, S; Johnston, T | 1 |
| Jackson, GL; Kuehl, D | 1 |
| Carai, MA; Colombo, G; Froestl, W; Gessa, GL; Serra, S; Vacca, G | 1 |
| Besheer, J; Hodge, CW; Lepoutre, V | 1 |
| Farb, DH; Gravielle, MC; Lyons, HR; Martin, SC; Russek, SJ; Steiger, JL | 1 |
| Martinez, V; Piqueras, L | 1 |
| Priest, CA; Puche, AC | 1 |
| Baber, SR; Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD | 1 |
| Carter, LP; Chen, W; Coop, A; France, CP; Koek, W; Lamb, RJ; Wu, H | 1 |
| Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD; Richards, TA | 2 |
| Carter, LP; Coop, A; France, CP; Koek, W; Wu, H | 1 |
| Carter, LP; Chen, W; Coop, A; France, CP; Koek, W | 1 |
| Coop, A; Koek, W; Mercer, SL | 1 |
| Balcar, VJ; Griffin, JL; Nasrallah, FA; Rae, C | 1 |
| Filip, M; Frankowska, M | 1 |
| Filip, M; Frankowska, M; Przegaliński, E | 1 |
| Mares, P | 1 |
| Baumann, O; Blenau, W; Rotte, C; Walz, B; Witte, J | 1 |
| Coop, A; France, CP; Koek, W; Mercer, SL | 1 |
| Dlouhá, K; Kagan, D; Roubalová, L; Svoboda, P | 1 |
| Frankowska, M; Gamberini, S; Gawlińska, K; Gawliński, D; Jastrzębska, J; Pieniążek, R; Suder, A; Wydra, K | 1 |
34 other study(ies) available for sk&f 97541 and baclofen
| Article | Year |
|---|---|
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.
Topics: Animals; Behavior, Animal; Cats; Crystallography, X-Ray; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Organophosphonates; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Stereoisomerism; Structure-Activity Relationship | 1995 |
Synthesis and pharmacological evaluation of novel gamma-aminobutyric acid type B (GABAB) receptor agonists as gastroesophageal reflux inhibitors.
Topics: Animals; Dose-Response Relationship, Drug; GABA Agonists; GABA-B Receptor Agonists; Gastroesophageal Reflux; Humans; Magnetic Resonance Spectroscopy; Spectrometry, Mass, Fast Atom Bombardment | 2008 |
Presynaptic inhibition mediated by GABAB receptors in rat striatal brain slices.
Topics: Action Potentials; Animals; Baclofen; Corpus Striatum; GABA-A Receptor Antagonists; Neurons; Organophosphorus Compounds; Rats; Receptors, GABA-A; Synapses | 1991 |
Subpopulations of GABA-mediated synaptic potentials in slices of rat dorsal striatum are differentially modulated by presynaptic GABAB receptors.
Topics: Animals; Baclofen; Caudate Nucleus; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Organophosphorus Compounds; Putamen; Rats; Receptors, GABA-A; Synaptic Membranes | 1991 |
Electrophysiological characterization of potent agonists and antagonists at pre- and postsynaptic GABAB receptors on neurones in rat brain slices.
Topics: Animals; Baclofen; Bicuculline; Brain; Corpus Striatum; Electrophysiology; GABA-A Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Neurons; Organophosphorus Compounds; Rats; Receptors, GABA-A; Substantia Nigra; Synapses | 1990 |
Baclofen enhancement of acetylcholine release from amacrine cells in the rabbit retina by reduction of glycinergic inhibition.
Topics: Acetylcholine; Animals; Baclofen; Bicuculline; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Muscarine; Organophosphorus Compounds; Rabbits; Retina; Strychnine | 1995 |
Multiple GABA receptor subtypes mediate inhibition of calcium influx at rat retinal bipolar cell terminals.
Topics: Animals; Axons; Baclofen; Bicuculline; Calcium; Cells, Cultured; gamma-Aminobutyric Acid; Nerve Endings; Organophosphorus Compounds; Picrotoxin; Potassium; Propylamines; Rats; Receptors, GABA; Receptors, GABA-A; Retina | 1995 |
Electrophysiological actions of GABAB agonists and antagonists in rat dorso-lateral septal neurones in vitro.
Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Dose-Response Relationship, Drug; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Membrane Potentials; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-B; Septal Nuclei | 1996 |
In vivo evidence that GABA(B) receptors are negatively coupled to adenylate cyclase in rat striatum.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Isoproterenol; Locomotion; Male; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Signal Transduction | 1997 |
Inhibition of transient LES relaxations and reflux in ferrets by GABA receptor agonists.
Topics: Animals; Baclofen; Behavior, Animal; Deglutition; Esophagogastric Junction; Female; Ferrets; GABA Agonists; gamma-Aminobutyric Acid; Gastroesophageal Reflux; Hydrogen-Ion Concentration; Manometry; Muscle Relaxation; Organophosphonates; Organophosphorus Compounds; Phosphinic Acids; Pressure; Time Factors | 1999 |
CGP 36216 is a selective antagonist at GABA(B) presynaptic receptors in rat brain.
Topics: Animals; Autoreceptors; Baclofen; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Neocortex; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B | 2001 |
The ATP-mediated fast current of rat dorsal root ganglion neurons is a novel effector for GABA(B) receptor activation.
Topics: Adenosine Triphosphate; Animals; Baclofen; Benzylamines; Cells, Cultured; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ganglia, Spinal; Membrane Potentials; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Phosphinic Acids; Picrotoxin; Rats; Receptors, GABA-A; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X3 | 2003 |
GABA(B) receptor agonists reverse akinesia following intranigral or intracerebroventricular injection in the reserpine-treated rat.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Globus Pallidus; Hypokinesia; Injections, Intraventricular; Male; Motor Activity; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Reserpine; Substantia Nigra | 2003 |
Effects of applying gamma-aminobutyric acid(B) drugs into the medial basal hypothalamus on basal luteinizing hormone concentrations and on luteinizing hormone surges in the female sheep.
Topics: Animals; Baclofen; Benzylamines; Breeding; Estrogens; Female; GABA Agonists; GABA-B Receptor Agonists; Hypothalamus, Middle; Luteinizing Hormone; Organophosphorus Compounds; Ovariectomy; Phosphinic Acids; Pituitary Gland, Anterior; Seasons; Sheep | 2004 |
Suppression of GABA(B) receptor function in vivo by disulfide reducing agent, DL-dithiothreitol (DTT).
Topics: Animals; Baclofen; Conditioning, Operant; Discrimination Learning; Dithiothreitol; Drug Interactions; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Hydroxybutyrates; Male; Mice; Mice, Inbred DBA; Organophosphonates; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Long-Evans; Reflex | 2004 |
GABA(B) receptor agonists reduce operant ethanol self-administration and enhance ethanol sedation in C57BL/6J mice.
Topics: Analysis of Variance; Animals; Baclofen; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; GABA Agonists; GABA-B Receptor Agonists; Hypnotics and Sedatives; Male; Mice; Mice, Inbred C57BL; Motor Activity; Organophosphorus Compounds; Receptors, GABA-B; Reflex; Self Administration | 2004 |
Differential expression of gamma-aminobutyric acid type B receptor subunit mRNAs in the developing nervous system and receptor coupling to adenylyl cyclase in embryonic neurons.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Binding Sites; Blotting, Western; Chlorocebus aethiops; COS Cells; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; GABA Agonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; In Situ Hybridization; Inhibitory Concentration 50; Male; Nervous System; Neurons; Organophosphorus Compounds; Phosphodiesterase Inhibitors; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; Tritium | 2004 |
Peripheral GABAB agonists stimulate gastric acid secretion in mice.
Topics: Animals; Antibodies, Monoclonal; Atropine; Baclofen; Deoxyglucose; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gastric Acid; Gastrins; Imidazoles; Injections, Intravenous; Male; Mice; Mice, Knockout; Muscimol; Organophosphorus Compounds; Pentagastrin; Peptides, Cyclic; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Somatostatin; Somatostatin; Time Factors; Vagotomy | 2004 |
GABAB receptor expression and function in olfactory receptor neuron axon growth.
Topics: Analysis of Variance; Animals; Animals, Newborn; Axons; Baclofen; Cells, Cultured; Drug Interactions; Embryo, Mammalian; Female; GABA Agonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gene Expression Regulation; Glutamate Decarboxylase; Growth Cones; Immunohistochemistry; In Vitro Techniques; Male; Mice; Olfactory Bulb; Olfactory Mucosa; Olfactory Receptor Neurons; Organophosphorus Compounds; Pregnancy; Receptors, GABA-B; Time Factors | 2004 |
Analysis of gamma-aminobutyric acid-mediated responses in the pulmonary vascular bed of the cat.
Topics: Animals; Baclofen; Blood Vessels; Cats; Dose-Response Relationship, Drug; Female; Glyburide; Lung; Male; Meclofenamic Acid; Organophosphorus Compounds; Receptors, GABA-A; Receptors, GABA-B | 2004 |
Discriminative stimulus effects of gamma-hydroxybutyrate (GHB) in rats discriminating GHB from baclofen and diazepam.
Topics: 4-Butyrolactone; Anesthetics, Intravenous; Animals; Baclofen; Benzocycloheptenes; Benzylamines; Butylene Glycols; Diazepam; Discrimination, Psychological; Dithiothreitol; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Sodium Oxybate | 2005 |
Analysis of responses to St. John's Wort in the feline pulmonary vascular bed.
Topics: Acetylcholine; Animals; Arachidonic Acid; Baclofen; Bicuculline; Bradykinin; Calcium Channel Agonists; Cats; Dose-Response Relationship, Drug; Female; GABA Antagonists; Hypericum; Male; Meclofenamic Acid; Muscimol; Nicardipine; Nitric Oxide Donors; Organophosphorus Compounds; Ornithine; Pinacidil; Plant Extracts; Prospective Studies; Pulmonary Artery; Pulmonary Circulation; Vasodilator Agents | 2004 |
Discriminative stimulus effects of flumazenil: perceptual masking by baclofen, and lack of substitution with gamma-hydroxybutyrate and its precursors 1,4-butanediol and gamma-butyrolactone.
Topics: 4-Butyrolactone; Animals; Baclofen; Benzocycloheptenes; Butylene Glycols; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Organophosphorus Compounds; Sodium Oxybate | 2006 |
Analysis of responses to kava kava in the feline pulmonary vascular bed.
Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Bradykinin; Calcium Channel Blockers; Calcium Channels; Cats; Cyclooxygenase Inhibitors; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; Kava; Lung; Meclofenamic Acid; Muscimol; Nicardipine; Nitric Oxide Synthase; Organophosphorus Compounds; Ornithine; Pinacidil; Plant Extracts; Receptors, GABA; Vasodilator Agents | 2006 |
Discriminative stimulus effects of GHB and GABA(B) agonists are differentially attenuated by CGP35348.
Topics: Analysis of Variance; Animals; Baclofen; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Sodium Oxybate | 2006 |
Cataleptic effects of gamma-hydroxybutyrate (GHB), its precursor gamma-butyrolactone (GBL), and GABAB receptor agonists in mice: differential antagonism by the GABAB receptor antagonist CGP35348.
Topics: 4-Butyrolactone; Animals; Baclofen; Catalepsy; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Male; Mice; Mice, Inbred C57BL; Narcolepsy; Organophosphorus Compounds; Receptors, GABA-B; Sodium Oxybate; Substance-Related Disorders | 2007 |
Understanding your inhibitions: modulation of brain cortical metabolism by GABA(B) receptors.
Topics: Animals; Baclofen; Benzylamines; Carbon Isotopes; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Guinea Pigs; Molecular Structure; Morpholines; Nuclear Magnetic Resonance, Biomolecular; Organophosphorus Compounds; Phosphinic Acids; Principal Component Analysis; Receptors, GABA-B | 2007 |
Effects of GABA(B) receptor agents on cocaine priming, discrete contextual cue and food induced relapses.
Topics: Animals; Baclofen; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Cues; Disease Models, Animal; Dose-Response Relationship, Drug; Extinction, Psychological; Feeding Behavior; GABA Agonists; GABA Antagonists; Injections, Intravenous; Male; Morpholines; Organophosphorus Compounds; Phenols; Rats; Rats, Wistar; Receptors, GABA-B; Reinforcement, Psychology; Secondary Prevention; Self Administration | 2007 |
Effects of GABA(B) receptor antagonist, agonists and allosteric positive modulator on the cocaine-induced self-administration and drug discrimination.
Topics: Animals; Baclofen; Cocaine; Discrimination Learning; GABA Modulators; Male; Morpholines; Motor Activity; Organophosphorus Compounds; Phenols; Rats; Rats, Wistar; Receptors, GABA-B; Self Administration | 2007 |
Anticonvulsant action of GABA-B receptor agonist SKF97541 differs from that of baclofen.
Topics: Age Factors; Animals; Anticonvulsants; Baclofen; Disease Models, Animal; Dose-Response Relationship, Drug; GABA Agonists; GABA-B Receptor Agonists; Male; Organophosphorus Compounds; Pentylenetetrazole; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-B; Seizures | 2008 |
Source, topography and excitatory effects of GABAergic innervation in cockroach salivary glands.
Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Electrophysiology; Fluorescent Antibody Technique; GABA Agonists; gamma-Aminobutyric Acid; Neurons; Organophosphorus Compounds; Periplaneta; Phosphinic Acids; Salivary Glands | 2009 |
Behavioral effects of gamma-hydroxybutyrate, its precursor gamma-butyrolactone, and GABA(B) receptor agonists: time course and differential antagonism by the GABA(B) receptor antagonist 3-aminopropyl(diethoxymethyl)phosphinic acid (CGP35348).
Topics: 4-Butyrolactone; Anesthetics, Intravenous; Animals; Baclofen; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Injections, Intramuscular; Kinetics; Organophosphorus Compounds; Sodium Oxybate | 2009 |
Ontogenetic development of GABA(B)-receptor signaling cascade in plasma membranes isolated from rat brain cortex; the number of GABA(B)-receptors is high already shortly after the birth.
Topics: Animals; Animals, Newborn; Baclofen; Binding Sites; Cell Membrane; Cerebral Cortex; GABA-B Receptor Agonists; Organophosphorus Compounds; Rats; Receptors, GABA-B; Signal Transduction; Time Factors | 2012 |
The impact of GABA
Topics: Animals; Baclofen; Behavior, Addictive; Behavior, Animal; Brain; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Depression; Disease Models, Animal; Drug-Seeking Behavior; GABA-B Receptor Agonists; Male; Organophosphorus Compounds; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Reinforcement, Psychology; Reward | 2020 |