Page last updated: 2024-08-26

sk&f 95282 and thiazoles

sk&f 95282 has been researched along with thiazoles in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-19906 (16.67)18.7374
1990's28 (77.78)18.2507
2000's2 (5.56)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bodnar, RJ; Hough, LB; Koch, JE1
Hough, LB; Nalwalk, JW2
Chakravarty, AK; Puri, S; Ray, A; Sen, P1
Maeyama, K; Onodera, K; Sakai, N; Watanabe, T; Yanai, K1
Boussard, M; Jantos, H; Monti, JM; Olivera, S; Orellana, C1
Battles, AH; Hough, LB; Nalwalk, JW1
Eberle, NB; Glick, SD; Gogas, KR; Hough, LB; Lyon, RA; Parsons, ME; Ward, SJ; Young, RC1
Gogas, KR; Hough, LB3
Calcutt, CR; Ganellin, CR; Griffiths, R; Leigh, BK; Maguire, JP; Mitchell, RC; Mylek, ME; Parsons, ME; Smith, IR; Young, RC1
Camarota, NA; Cue, D; Eberle, N; Gogas, KR; Hough, LB; Jackowski, S1
Imaizumi, M; Miyazaki, S; Onodera, K2
Fleckenstein, AE; Lookingland, KJ; Moore, KE2
Wong, CL1
Barke, KE; Bodnar, RJ; Hough, LB; Koch, JE; Nalwalk, JW1
Misawa, M; Onodera, K; Suzuki, T; Takamori, K1
Adami, M; Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C1
Schilling, L; Wahl, M1
Adachi, N; Hirakawa, M; Itano, Y; Oishi, R; Saeki, K; Yamada, T1
D'Souza, T; Dryer, SE; Nowak, JZ; Sek, B1
Eaton, SJ; Eoh, S; Harrington, ME; Hoque, S; Meyer, J1
Ito, C; Onodera, K; Sato, M; Watanabe, T1
Hayashi, Y; Kagawa, K; Mammoto, T; Mashimo, T; Yamamoto, Y; Yamatodani, A; Yoshiya, I1
Imaizumi, M; Miyazaki, S; Onodera, K; Timmerman, H1
Itoh, C; Onodera, K; Sato, M; Watanabe, T1
Misawa, M; Mori, T; Onodera, K; Suzuki, T; Tsuji, M1
Bertaccini, G; Coppelli, G; Coruzzi, G; Poli, E; Pozzoli, C1
Inokuchi, A; Komiyama, S; Liu, F; Ureshino, M; Yokomitsu, S1
Meade, HM; Seeley, NA; Sturman, G1
Chen, Z; Fujii, Y; Kamei, C; Sugimoto, Y; Suzuki, G1
Affricano, D; Angelucci, L; Lombardo, K; Nicolai, R; Scaccianoce, S1
Hough, LB; Lu, Q; Montero, MJ; Nalwalk, JW; Shan, Z; Svokos, K; Wentland, MP1

Other Studies

36 other study(ies) available for sk&f 95282 and thiazoles

ArticleYear
Potentiation of 2-deoxy-D-glucose antinociception, but not hyperphagia by zolantidine, a histamine (H2) receptor antagonist.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:2

    Topics: Animals; Benzothiazoles; Deoxyglucose; Histamine H2 Antagonists; Hot Temperature; Hyperphagia; Male; Nociceptors; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Thiazoles

1992
Inhibition of morphine antinociception by centrally administered histamine H2 receptor antagonists.
    European journal of pharmacology, 1992, Apr-29, Volume: 215, Issue:1

    Topics: Animals; Benzothiazoles; Brain; Cimetidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Morphine; Nociceptors; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles

1992
Central histaminergic involvement during stress in rats.
    Indian journal of experimental biology, 1992, Volume: 30, Issue:8

    Topics: Animals; Antibody Formation; Benzothiazoles; Brain; Corticosterone; Histamine; Histamine H2 Antagonists; Histidine Decarboxylase; Male; Methylhistidines; Peptic Ulcer; Pheniramine; Phenoxypropanolamines; Piperidines; Rats; Rats, Wistar; Stress, Physiological; Thiazoles

1992
Effects of thioperamide, a histamine H3 receptor antagonist, on locomotor activity and brain histamine content in mast cell-deficient W/Wv mice.
    Life sciences, 1991, Volume: 48, Issue:25

    Topics: Animals; Benzothiazoles; Brain Chemistry; Dopamine; Histamine; Histamine Antagonists; Histamine H2 Antagonists; Mast Cells; Methylhistamines; Mice; Mice, Mutant Strains; Motor Activity; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles

1991
Sleep variables are unaltered by zolantidine in rats: are histamine H2-receptors not involved in sleep regulation?
    Brain research bulletin, 1990, Volume: 25, Issue:2

    Topics: Animals; Benzothiazoles; Diphenhydramine; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Male; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Reference Values; Sleep; Thiazoles; Time Factors; Wakefulness

1990
Zolantidine-induced attenuation of morphine antinociception in rhesus monkeys.
    Brain research, 1990, Aug-27, Volume: 526, Issue:1

    Topics: Animals; Benzothiazoles; Dose-Response Relationship, Drug; Double-Blind Method; Female; Histamine H2 Antagonists; Macaca mulatta; Morphine; Pain; Phenoxypropanolamines; Piperidines; Thiazoles

1990
A role for histamine and H2-receptors in opioid antinociception.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:2

    Topics: Analgesia; Animals; Benzothiazoles; Cimetidine; Histamine; Male; Morphine; Phenoxypropanolamines; Piperidines; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Receptors, Opioid; Thiazoles

1989
Inhibition of naloxone-resistant antinociception by centrally administered H2-antagonists.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Analgesia; Animals; Benzothiazoles; Brain; Dose-Response Relationship, Drug; Drug Resistance; Histamine; Histamine H2 Antagonists; Male; Naloxone; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Thiazoles

1989
Zolantidine (SK&F 95282) is a potent selective brain-penetrating histamine H2-receptor antagonist.
    British journal of pharmacology, 1988, Volume: 93, Issue:1

    Topics: Animals; Benzothiazoles; Binding, Competitive; Brain Chemistry; Cimetidine; Cyclic AMP; Female; Guinea Pigs; Hippocampus; Histamine H2 Antagonists; In Vitro Techniques; Male; Phenoxypropanolamines; Piperidines; Rats; Thiazoles; Uterus

1988
Effects of zolantidine a brain-penetrating H2-receptor antagonist, on naloxone-sensitive and naloxone-resistant analgesia.
    Neuropharmacology, 1988, Volume: 27, Issue:4

    Topics: Analgesia; Animals; Benzothiazoles; Brain; Drug Interactions; Drug Resistance; Histamine H2 Antagonists; Male; Naloxone; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Thiazoles

1988
H2-receptor-mediated stress-induced analgesia is dependent on neither pituitary nor adrenal activation.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:3

    Topics: Adrenalectomy; Analgesia; Animals; Benzothiazoles; Electroshock; Histamine H2 Antagonists; Hypophysectomy; Male; Naloxone; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Reference Values; Thiazoles

1988
Actions of the brain-penetrating H2-antagonist zolantidine on histamine dynamics and metabolism in rat brain.
    Biochemical pharmacology, 1988, Dec-15, Volume: 37, Issue:24

    Topics: Animals; Benzothiazoles; Brain; Brain Chemistry; Dose-Response Relationship, Drug; Histamine; Histamine N-Methyltransferase; In Vitro Techniques; Kidney; Kinetics; Methylhistamines; Methyltransferases; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Thiazoles

1988
Effects of thioperamide, a histamine H3-receptor antagonist, on a scopolamine-induced learning deficit using an elevated plus-maze test in mice.
    Life sciences, 1995, Volume: 57, Issue:23

    Topics: Animals; Benzothiazoles; Histamine; Histamine Antagonists; Male; Maze Learning; Mice; Mice, Inbred ICR; Phenoxypropanolamines; Piperidines; Scopolamine; Thiazoles

1995
Histaminergic neurons mediate restraint stress-induced activation of central 5-hydroxytryptaminergic neurons in the rat.
    European journal of pharmacology, 1994, Oct-24, Volume: 264, Issue:2

    Topics: Animals; Benzothiazoles; Histamine; Histamine H2 Antagonists; Histidine Decarboxylase; Hydroxyindoleacetic Acid; Male; Methylhistidines; Neurons; Nucleus Accumbens; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Receptors, Histamine H1; Restraint, Physical; Serotonin; Suprachiasmatic Nucleus; Thiazoles

1994
Effects of a histamine H2 receptor agonist and antagonist on restraint-induced antinociception in female mice.
    European journal of pharmacology, 1995, Jun-12, Volume: 279, Issue:2-3

    Topics: Animals; Benzothiazoles; Cimetidine; Dimaprit; Female; Histamine Agonists; Histamine H2 Antagonists; Mice; Mice, Inbred Strains; Pain Measurement; Phenoxypropanolamines; Piperidines; Reaction Time; Restraint, Physical; Stress, Psychological; Thiazoles

1995
Modulation of morphine antinociception by the brain-penetrating H2 antagonist zolantidine: detailed characterization in five nociceptive test systems.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 50, Issue:3

    Topics: Animals; Benzothiazoles; Blood-Brain Barrier; Histamine H2 Antagonists; Hot Temperature; Male; Morphine; Pain; Pain Measurement; Phenoxypropanolamines; Piperidines; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Thiazoles

1995
Importance of histamine H2 receptors in restraint-morphine interactions.
    Life sciences, 1995, Volume: 57, Issue:13

    Topics: Analysis of Variance; Animals; Benzothiazoles; Histamine; Histamine H2 Antagonists; Male; Morphine; Pain; Phenoxypropanolamines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; Restraint, Physical; Thiazoles; Time Factors

1995
Effects of the histaminergic system on the morphine-induced conditioned place preference in mice.
    Brain research, 1995, Mar-27, Volume: 675, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Benzothiazoles; Conditioning, Operant; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Histamine; Histamine H2 Antagonists; Histidine; Histidine Decarboxylase; Homovanillic Acid; Limbic System; Male; Methylhistidines; Mice; Mice, Inbred Strains; Morphine; Phenoxypropanolamines; Piperidines; Prosencephalon; Thiazoles

1995
Activity of the new histamine H2-receptor antagonist zolantidine at cardiac and gastric H2-receptors.
    Pharmacology, 1994, Volume: 48, Issue:2

    Topics: Animals; Benzothiazoles; Cats; Female; Gastric Fistula; Gastric Mucosa; Guinea Pigs; Heart Rate; Histamine H2 Antagonists; Male; Myocardial Contraction; Phenoxypropanolamines; Piperidines; Ranitidine; Rats; Rats, Wistar; Thiazoles

1994
Activation of noradrenergic neurons projecting to the diencephalon following central administration of histamine is mediated by H1 receptors.
    Brain research, 1994, Feb-28, Volume: 638, Issue:1-2

    Topics: Animals; Benzothiazoles; Cerebral Ventricles; Diencephalon; Histamine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methoxyhydroxyphenylglycol; Neurons; Norepinephrine; Paraventricular Hypothalamic Nucleus; Phenoxypropanolamines; Piperidines; Preoptic Area; Pyrilamine; Rats; Receptors, Histamine H1; Thiazoles

1994
Effects of antihistaminics on experimental brain edema.
    Acta neurochirurgica. Supplementum, 1994, Volume: 60

    Topics: Animals; Antioxidants; Benzothiazoles; Blood-Brain Barrier; Brain Edema; Dexamethasone; Freezing; Histamine; Histamine Antagonists; Histamine H2 Antagonists; Lipid Peroxidation; Male; Parietal Lobe; Phenoxypropanolamines; Piperidines; Pregnatrienes; Pyrilamine; Rats; Rats, Sprague-Dawley; Thiazoles; Water-Electrolyte Balance

1994
Aggravation of ischemic neuronal damage in the rat hippocampus by impairment of histaminergic neurotransmission.
    Brain research, 1993, Jan-29, Volume: 602, Issue:1

    Topics: Animals; Benzothiazoles; Brain Ischemia; Cell Death; Hippocampus; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Methylhistidines; Neurons; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Synaptic Transmission; Thiazoles

1993
Does histamine stimulate cyclic AMP formation in the avian pineal gland via a novel (non-H1, non-H2, non-H3) histamine receptor subtype.
    Neurochemistry international, 1995, Volume: 27, Issue:6

    Topics: Animals; Benzothiazoles; Chickens; Cyclic AMP; Ducks; Histamine; Histamine Agonists; Histamine H2 Antagonists; Ion Channels; Male; Methylation; Phenoxypropanolamines; Pineal Gland; Piperidines; Receptors, Histamine; Stimulation, Chemical; Thiazoles

1995
Circadian rhythm photic phase shifts are not altered by histamine receptor antagonists.
    Brain research bulletin, 1996, Volume: 41, Issue:4

    Topics: Animals; Benzothiazoles; Cimetidine; Circadian Rhythm; Cricetinae; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mesocricetus; Phenoxypropanolamines; Photoperiod; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles

1996
Effects of histamine agents on methamphetamine-induced stereotyped behavior and behavioral sensitization in rats.
    Psychopharmacology, 1997, Volume: 130, Issue:4

    Topics: Animals; Benzothiazoles; Brain; Central Nervous System Stimulants; Histamine Agents; Histidine; Male; Methamphetamine; Methylhistidines; Motor Activity; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Stereotyped Behavior; Thiazoles

1997
Interactions between neuronal histamine and halothane anesthesia in rats.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Anesthetics, Inhalation; Animals; Benzothiazoles; Drug Interactions; Enzyme Inhibitors; Halothane; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Male; Methylhistidines; Microdialysis; Neurons; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Thiazoles

1997
Effects of clobenpropit (VUF-9153), a histamine H3-receptor antagonist, on learning and memory, and on cholinergic and monoaminergic systems in mice.
    Life sciences, 1997, Volume: 61, Issue:4

    Topics: Acetylcholine; Animals; Avoidance Learning; Benzothiazoles; Biogenic Monoamines; Brain; Drug Interactions; Histamine Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Memory; Methylhistamines; Mice; Mice, Inbred ICR; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H3; Scopolamine; Thiazoles; Thiourea

1997
Motor behavioural function for histamine-dopamine interaction in brain.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1998, Volume: 47 Suppl 1

    Topics: Animals; Benzazepines; Benzothiazoles; Brain; Brain Chemistry; Central Nervous System Stimulants; Dopamine Agents; Dopamine Antagonists; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Methamphetamine; Motor Activity; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Stereotyped Behavior; Thiazoles

1998
Cognitive involvement by negative modulation of histamine H2 receptors in passive avoidance task in mice.
    Methods and findings in experimental and clinical pharmacology, 1998, Volume: 20, Issue:4

    Topics: Animals; Avoidance Learning; Benzothiazoles; Cognition; Drug Interactions; Histamine Agonists; Histamine H2 Antagonists; Injections, Intraventricular; Male; Memory; Methylhistamines; Mice; Mice, Inbred ICR; Phenoxypropanolamines; Piperidines; Receptors, Histamine H2; Thiazoles

1998
Generalization of D-, L- and DL-chlorpheniramine and zolantidine to the discriminative stimulus effects of cocaine and methamphetamine.
    Behavioural pharmacology, 1997, Volume: 8, Issue:8

    Topics: Animals; Antidepressive Agents, Tricyclic; Benzothiazoles; Chlorpheniramine; Clomipramine; Cocaine; Desipramine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Stimulus; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Methamphetamine; Middle Aged; Phenoxypropanolamines; Piperazines; Piperidines; Rats; Rats, Inbred F344; Thiazoles

1997
Effects of histamine H2 receptor agonists and antagonists on the isolated guinea pig gallbladder.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:1

    Topics: Animals; Benzothiazoles; Dopamine Agents; Famotidine; Gallbladder; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Phenoxypropanolamines; Piperidines; Pyridines; Receptors, Histamine H2; Sincalide; Thiazoles; Triazoles

1999
Effects of the antihistaminergic drugs diphenhydramine and zolantidine on vestibular-induced hypothalamic neuronal activity in the guinea pig.
    European archives of oto-rhino-laryngology : official journal of the European Federation of Oto-Rhino-Laryngological Societies (EUFOS) : affiliated with the German Society for Oto-Rhino-Laryngology - Head and Neck Surgery, 1999, Volume: 256 Suppl 1

    Topics: Animals; Benzothiazoles; Caloric Tests; Diphenhydramine; Guinea Pigs; Histamine H1 Antagonists; Hypothalamus; Injections, Intravenous; Male; Neurons; Phenoxypropanolamines; Piperidines; Thiazoles; Vestibule, Labyrinth

1999
Histamine H2-receptor modulation in two mouse models of seizure susceptibility.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1999, Volume: 48 Suppl 1

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzothiazoles; Convulsants; Dimaprit; Female; Histamine Agonists; Histamine Antagonists; Male; Mice; Mice, Inbred DBA; Pentylenetetrazole; Phenoxypropanolamines; Piperidines; Receptors, Histamine H2; Seizures; Thiazoles

1999
Effects of histamine and related compounds on regional cerebral blood flow in rats.
    Methods and findings in experimental and clinical pharmacology, 1999, Volume: 21, Issue:9

    Topics: Animals; Benzothiazoles; Blood Pressure; Brain Chemistry; Dimaprit; Diphenhydramine; Drug Interactions; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Thiazoles; Time Factors

1999
Studies on the involvement of histamine in the hypothalamic-pituitary-adrenal axis activation induced by nerve growth factor.
    Life sciences, 2000, Nov-17, Volume: 67, Issue:26

    Topics: Adrenal Glands; Animals; Benzothiazoles; Catheterization; Corticosterone; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypothalamo-Hypophyseal System; Male; Metiamide; Mice; Nerve Growth Factor; Phenoxypropanolamines; Piperidines; Pituitary-Adrenal System; Promethazine; Rats; Rats, Wistar; Thiazoles

2000
Antinociceptive, brain-penetrating derivatives related to improgan, a non-opioid analgesic.
    European journal of pharmacology, 2005, Oct-17, Volume: 522, Issue:1-3

    Topics: Algorithms; Analgesics; Animals; Behavior, Animal; Benzothiazoles; Brain; Cimetidine; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Injections, Intraventricular; Male; Mice; Molecular Structure; Pain; Pain Measurement; Phenoxypropanolamines; Piperidines; Quinazolines; Quinazolinones; Rats; Rats, Sprague-Dawley; Thiazoles; Time Factors; Triazoles

2005