Page last updated: 2024-08-26

sk&f 95282 and pyrilamine

sk&f 95282 has been researched along with pyrilamine in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.88)18.7374
1990's12 (70.59)18.2507
2000's2 (11.76)29.6817
2010's2 (11.76)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brown, TH; Ganellin, CR; Griffiths, R; Jones, M; Mitchell, RC; Rana, KK; Saunders, D; Smith, IR; Sore, NE; Young, RC1
Blake, JF; Curatolo, WJ; Lombardo, F1
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Maeyama, K; Onodera, K; Sakai, N; Watanabe, T; Yanai, K1
Fleckenstein, AE; Lookingland, KJ; Moore, KE2
Schilling, L; Wahl, M1
Adachi, N; Hirakawa, M; Itano, Y; Oishi, R; Saeki, K; Yamada, T1
Eaton, SJ; Eoh, S; Harrington, ME; Hoque, S; Meyer, J1
Ito, C; Onodera, K; Sato, M; Watanabe, T1
Hayashi, Y; Kagawa, K; Mammoto, T; Mashimo, T; Yamamoto, Y; Yamatodani, A; Yoshiya, I1
Imaizumi, M; Miyazaki, S; Onodera, K; Timmerman, H1
Itoh, C; Onodera, K; Sato, M; Watanabe, T1
Chen, Z; Fujii, Y; Kamei, C; Sugimoto, Y; Suzuki, G1
Krishna, DR; Kumar, KV; Palit, G1
Darras, FH; Decker, M; Khan, N; Nurulain, SM; Saad, A; Sadek, B1
Alachkar, A; Gryboś, A; Handzlik, J; Honkisz, E; Kiec-Kononowicz, K; Latacz, G; Lubelska, A; Sadek, B; Siwek, A; Stark, H; Łażewska, D1

Other Studies

17 other study(ies) available for sk&f 95282 and pyrilamine

ArticleYear
Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:3

    Topics: Algorithms; Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry, Physical; Clonidine; Guinea Pigs; Histamine H2 Antagonists; Imipramine; Pyrilamine; Structure-Activity Relationship

1988
Computation of brain-blood partitioning of organic solutes via free energy calculations.
    Journal of medicinal chemistry, 1996, Nov-22, Volume: 39, Issue:24

    Topics: Animals; Blood-Brain Barrier; Brain; Cattle; Cells, Cultured; Endothelium, Vascular; Membrane Lipids; Microcirculation; Molecular Conformation; Molecular Structure; Monte Carlo Method; Permeability; Pharmaceutical Preparations; Software; Solubility; Thermodynamics

1996
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Effects of thioperamide, a histamine H3 receptor antagonist, on locomotor activity and brain histamine content in mast cell-deficient W/Wv mice.
    Life sciences, 1991, Volume: 48, Issue:25

    Topics: Animals; Benzothiazoles; Brain Chemistry; Dopamine; Histamine; Histamine Antagonists; Histamine H2 Antagonists; Mast Cells; Methylhistamines; Mice; Mice, Mutant Strains; Motor Activity; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles

1991
Histaminergic neurons mediate restraint stress-induced activation of central 5-hydroxytryptaminergic neurons in the rat.
    European journal of pharmacology, 1994, Oct-24, Volume: 264, Issue:2

    Topics: Animals; Benzothiazoles; Histamine; Histamine H2 Antagonists; Histidine Decarboxylase; Hydroxyindoleacetic Acid; Male; Methylhistidines; Neurons; Nucleus Accumbens; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Receptors, Histamine H1; Restraint, Physical; Serotonin; Suprachiasmatic Nucleus; Thiazoles

1994
Activation of noradrenergic neurons projecting to the diencephalon following central administration of histamine is mediated by H1 receptors.
    Brain research, 1994, Feb-28, Volume: 638, Issue:1-2

    Topics: Animals; Benzothiazoles; Cerebral Ventricles; Diencephalon; Histamine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methoxyhydroxyphenylglycol; Neurons; Norepinephrine; Paraventricular Hypothalamic Nucleus; Phenoxypropanolamines; Piperidines; Preoptic Area; Pyrilamine; Rats; Receptors, Histamine H1; Thiazoles

1994
Effects of antihistaminics on experimental brain edema.
    Acta neurochirurgica. Supplementum, 1994, Volume: 60

    Topics: Animals; Antioxidants; Benzothiazoles; Blood-Brain Barrier; Brain Edema; Dexamethasone; Freezing; Histamine; Histamine Antagonists; Histamine H2 Antagonists; Lipid Peroxidation; Male; Parietal Lobe; Phenoxypropanolamines; Piperidines; Pregnatrienes; Pyrilamine; Rats; Rats, Sprague-Dawley; Thiazoles; Water-Electrolyte Balance

1994
Aggravation of ischemic neuronal damage in the rat hippocampus by impairment of histaminergic neurotransmission.
    Brain research, 1993, Jan-29, Volume: 602, Issue:1

    Topics: Animals; Benzothiazoles; Brain Ischemia; Cell Death; Hippocampus; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Methylhistidines; Neurons; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Synaptic Transmission; Thiazoles

1993
Circadian rhythm photic phase shifts are not altered by histamine receptor antagonists.
    Brain research bulletin, 1996, Volume: 41, Issue:4

    Topics: Animals; Benzothiazoles; Cimetidine; Circadian Rhythm; Cricetinae; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mesocricetus; Phenoxypropanolamines; Photoperiod; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles

1996
Effects of histamine agents on methamphetamine-induced stereotyped behavior and behavioral sensitization in rats.
    Psychopharmacology, 1997, Volume: 130, Issue:4

    Topics: Animals; Benzothiazoles; Brain; Central Nervous System Stimulants; Histamine Agents; Histidine; Male; Methamphetamine; Methylhistidines; Motor Activity; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Stereotyped Behavior; Thiazoles

1997
Interactions between neuronal histamine and halothane anesthesia in rats.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Anesthetics, Inhalation; Animals; Benzothiazoles; Drug Interactions; Enzyme Inhibitors; Halothane; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Male; Methylhistidines; Microdialysis; Neurons; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Thiazoles

1997
Effects of clobenpropit (VUF-9153), a histamine H3-receptor antagonist, on learning and memory, and on cholinergic and monoaminergic systems in mice.
    Life sciences, 1997, Volume: 61, Issue:4

    Topics: Acetylcholine; Animals; Avoidance Learning; Benzothiazoles; Biogenic Monoamines; Brain; Drug Interactions; Histamine Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Memory; Methylhistamines; Mice; Mice, Inbred ICR; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H3; Scopolamine; Thiazoles; Thiourea

1997
Motor behavioural function for histamine-dopamine interaction in brain.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1998, Volume: 47 Suppl 1

    Topics: Animals; Benzazepines; Benzothiazoles; Brain; Brain Chemistry; Central Nervous System Stimulants; Dopamine Agents; Dopamine Antagonists; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Methamphetamine; Motor Activity; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Stereotyped Behavior; Thiazoles

1998
Effects of histamine and related compounds on regional cerebral blood flow in rats.
    Methods and findings in experimental and clinical pharmacology, 1999, Volume: 21, Issue:9

    Topics: Animals; Benzothiazoles; Blood Pressure; Brain Chemistry; Dimaprit; Diphenhydramine; Drug Interactions; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Thiazoles; Time Factors

1999
Histaminergic H1 receptors mediate L-histidine-induced anxiety in elevated plus-maze test in mice.
    Behavioural pharmacology, 2007, Volume: 18, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzothiazoles; Diazepam; Dose-Response Relationship, Drug; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Mice; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H3

2007
The dual-acting H3 receptor antagonist and AChE inhibitor UW-MD-71 dose-dependently enhances memory retrieval and reverses dizocilpine-induced memory impairment in rats.
    Behavioural brain research, 2016, Jan-15, Volume: 297

    Topics: Animals; Avoidance Learning; Benzothiazoles; Cholinesterase Inhibitors; Disease Models, Animal; Dizocilpine Maleate; Donepezil; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Histamine H3 Antagonists; Indans; Male; Memory; Memory Disorders; Nootropic Agents; Phenoxypropanolamines; Piperidines; Pyrilamine; Pyrroles; Quinazolines; Random Allocation; Rats, Wistar; Receptors, Histamine H3

2016
Anticonvulsant evaluation of novel non-imidazole histamine H3R antagonists in different convulsion models in rats.
    Pharmacology, biochemistry, and behavior, 2018, Volume: 170

    Topics: Animals; Anticonvulsants; Benzothiazoles; Disease Models, Animal; Dose-Response Relationship, Drug; Histamine H3 Antagonists; Humans; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Reaction Time; Seizures; Strychnine

2018