sk&f 89124 has been researched along with ropinirole in 5 studies
Studies (sk&f 89124) | Trials (sk&f 89124) | Recent Studies (post-2010) (sk&f 89124) | Studies (ropinirole) | Trials (ropinirole) | Recent Studies (post-2010) (ropinirole) |
---|---|---|---|---|---|
14 | 0 | 0 | 637 | 129 | 243 |
Protein | Taxonomy | sk&f 89124 (IC50) | ropinirole (IC50) |
---|---|---|---|
D(2) dopamine receptor | Bos taurus (cattle) | 6.81 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 5 (100.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Flaim, KE; Franz, RG; Gaitanopoulos, DE; Gessner, G; Hieble, JP; Kinter, LB; Mann, WA; Stringer, OD; Weinstock, J | 1 |
DeMarinis, RM; Franz, RG; Gallagher, G; Hall, RF; Huffman, WF; Kaiser, C; Ross, ST; Schwartz, MS; Webster, C; Wilson, JW | 1 |
DeMarinis, RM; Gallagher, G; Hieble, JP; Lavanchy, PG; Webster, CA; Wilson, JW | 1 |
DeMarinis, RM; Mico, BA; Swagzdis, JE; Wittendorf, RW | 1 |
Federowicz, DA; Mico, BA; Straub, K; Swagzdis, JE | 1 |
5 other study(ies) available for sk&f 89124 and ropinirole
Article | Year |
---|---|
Synthesis and evaluation of non-catechol D-1 and D-2 dopamine receptor agonists: benzimidazol-2-one, benzoxazol-2-one, and the highly potent benzothiazol-2-one 7-ethylamines.
Topics: Animals; Benzimidazoles; Benzoxazoles; Blood Pressure; Dogs; Female; In Vitro Techniques; Male; Rabbits; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Structure-Activity Relationship; Thiazoles; Vascular Resistance | 1987 |
Syntheses and in vitro evaluation of 4-(2-aminoethyl)-2(3H)-indolones and related compounds as peripheral prejunctional dopamine receptor agonists.
Topics: Animals; Arteries; Ear; Hydralazine; In Vitro Techniques; Indoles; Pyridazines; Rabbits; Rats; Receptors, Dopamine; Structure-Activity Relationship | 1986 |
4-[2-(Di-n-propylamino)ethyl]-2(3H)-indolone: a prejunctional dopamine receptor agonist.
Topics: Animals; Chemical Phenomena; Chemistry; Indoles; Rabbits; Receptors, Dopamine; Vasomotor System | 1985 |
Pharmacokinetics of dopamine-2 agonists in rats and dogs.
Topics: Animals; Biotransformation; Blood Proteins; Dogs; Indoles; Intestinal Absorption; Kinetics; Magnetic Resonance Spectroscopy; Male; Protein Binding; Rats; Rats, Inbred Strains; Receptors, Dopamine; Species Specificity; Sulfonamides | 1986 |
Functional group metabolism of dopamine-2 agonists: conversion of 4-(2-di-n-propylaminoethyl)-2-(3H)-indolone to 4-(2-di-n-propylaminoethyl)-7-hydroxy-2-(3H)-indolone.
Topics: Animals; Biotransformation; Chromatography, High Pressure Liquid; Dogs; Dopamine; Glucuronates; Indoles; Kinetics; Macaca fascicularis; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Rats; Rats, Inbred Strains | 1986 |