Page last updated: 2024-09-03

sk&f 86466 and spironolactone

sk&f 86466 has been researched along with spironolactone in 1 studies

Compound Research Comparison

Studies
(sk&f 86466)
Trials
(sk&f 86466)
Recent Studies (post-2010)
(sk&f 86466)
Studies
(spironolactone)
Trials
(spironolactone)
Recent Studies (post-2010) (spironolactone)
73397,2229601,923

Protein Interaction Comparison

ProteinTaxonomysk&f 86466 (IC50)spironolactone (IC50)
Chain A, Mineralocorticoid receptorHomo sapiens (human)0.049
Chain A, Mineralocorticoid receptorHomo sapiens (human)0.049
Estrogen receptorHomo sapiens (human)5.702
Glucocorticoid receptorHomo sapiens (human)4.0745
Progesterone receptorHomo sapiens (human)1.675
Glycine receptor subunit alpha-1Rattus norvegicus (Norway rat)1.9025
Mineralocorticoid receptor Homo sapiens (human)0.0315
Androgen receptorHomo sapiens (human)0.3585
Androgen receptorRattus norvegicus (Norway rat)0.406
Glycine receptor subunit betaRattus norvegicus (Norway rat)1.9025
Glycine receptor subunit alpha-2Rattus norvegicus (Norway rat)1.9025
Glycine receptor subunit alpha-3Rattus norvegicus (Norway rat)1.9025
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)6.92
Cytochrome P450 2C19Homo sapiens (human)3

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1

Other Studies

1 other study(ies) available for sk&f 86466 and spironolactone

ArticleYear
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009