Page last updated: 2024-09-03

sk&f 86466 and buspirone hydrochloride

sk&f 86466 has been researched along with buspirone hydrochloride in 2 studies

Compound Research Comparison

Studies
(sk&f 86466)
Trials
(sk&f 86466)
Recent Studies (post-2010)
(sk&f 86466)
Studies
(buspirone hydrochloride)
Trials
(buspirone hydrochloride)
Recent Studies (post-2010) (buspirone hydrochloride)
73391705

Protein Interaction Comparison

ProteinTaxonomysk&f 86466 (IC50)buspirone hydrochloride (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.74
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.74
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.74

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berger, J; Brown, CM; Clark, RD; Fisher, LE; Kilpatrick, AT; MacKinnon, AC; Spedding, M; Weinhardt, KK1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1

Other Studies

2 other study(ies) available for sk&f 86466 and buspirone hydrochloride

ArticleYear
1,9-Alkano-bridged 2,3,4,5-tetrahydro-1H-3-benzazepines with affinity for the alpha 2-adrenoceptor and the 5-HT1A receptor.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:2

    Topics: Animals; Benzazepines; Cerebral Cortex; Chemical Phenomena; Chemistry; Chemistry, Physical; In Vitro Techniques; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Structure-Activity Relationship; Thermodynamics

1990
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009