Page last updated: 2024-09-03

sk&f 86466 and 4-iodoclonidine

sk&f 86466 has been researched along with 4-iodoclonidine in 2 studies

Compound Research Comparison

Studies
(sk&f 86466)
Trials
(sk&f 86466)
Recent Studies (post-2010)
(sk&f 86466)
Studies
(4-iodoclonidine)
Trials
(4-iodoclonidine)
Recent Studies (post-2010) (4-iodoclonidine)
733943210
7339801

Protein Interaction Comparison

ProteinTaxonomysk&f 86466 (IC50)4-iodoclonidine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.0015
Alpha-2B adrenergic receptorHomo sapiens (human)0.0015
Alpha-2C adrenergic receptorHomo sapiens (human)0.0015
high affinity choline transporter 1 isoform aHomo sapiens (human)0.979

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dreshaj, I; Ernsberger, P; Haxhiu, MA; Schäfer, SG1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1

Other Studies

2 other study(ies) available for sk&f 86466 and 4-iodoclonidine

ArticleYear
Selective antihypertensive action of moxonidine is mediated mainly by I1-imidazoline receptors in the rostral ventrolateral medulla.
    Journal of cardiovascular pharmacology, 1994, Volume: 24 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Affinity Labels; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Binding, Competitive; Blood Gas Analysis; Blood Pressure; Blood Pressure Determination; Cattle; Clonidine; Disease Models, Animal; Heart Rate; Hypertension; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Medulla Oblongata; Microinjections; Radioligand Assay; Rats; Rats, Inbred SHR; Receptors, Drug

1994
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009