Page last updated: 2024-09-03

sk&f 86466 and 1-(5-isoquinolinesulfonyl)-2-methylpiperazine dihydrochloride

sk&f 86466 has been researched along with 1-(5-isoquinolinesulfonyl)-2-methylpiperazine dihydrochloride in 1 studies

Compound Research Comparison

Studies
(sk&f 86466)
Trials
(sk&f 86466)
Recent Studies (post-2010)
(sk&f 86466)
Studies
(1-(5-isoquinolinesulfonyl)-2-methylpiperazine dihydrochloride)
Trials
(1-(5-isoquinolinesulfonyl)-2-methylpiperazine dihydrochloride)
Recent Studies (post-2010) (1-(5-isoquinolinesulfonyl)-2-methylpiperazine dihydrochloride)
7339501

Protein Interaction Comparison

ProteinTaxonomysk&f 86466 (IC50)1-(5-isoquinolinesulfonyl)-2-methylpiperazine dihydrochloride (IC50)
Serine/threonine-protein kinase D3Homo sapiens (human)6
Protein kinase C gamma typeHomo sapiens (human)6
Protein kinase C beta typeHomo sapiens (human)6
Protein kinase C alpha typeHomo sapiens (human)6
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)3.5
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)3.5
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)3.5
Protein kinase C eta typeHomo sapiens (human)6
Protein kinase C iota typeHomo sapiens (human)6
Protein kinase C epsilon typeHomo sapiens (human)6
Protein kinase C theta typeHomo sapiens (human)6
Protein kinase C zeta typeHomo sapiens (human)6
Protein kinase C delta typeHomo sapiens (human)6
Serine/threonine-protein kinase D1Homo sapiens (human)6

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1

Other Studies

1 other study(ies) available for sk&f 86466 and 1-(5-isoquinolinesulfonyl)-2-methylpiperazine dihydrochloride

ArticleYear
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009