sk&f 77434 and sk&f-38393

sk&f 77434 has been researched along with sk&f-38393 in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's16 (61.54)18.2507
2000's9 (34.62)29.6817
2010's1 (3.85)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Baindur, N; Baldessarini, RJ; Kula, NS; Neumeyer, JL1
Cheng, J; McCorvy, JD; Tan, L; Yan, W1
Chang, JP; Peter, RE; Wong, AO1
Self, DW; Stein, L1
Katz, JL; Terry, P1
Briggs, CA; Frail, DE; Kang, CH; Kebabian, JW; Paxson, CL; Pollock, NJ; Rakowski, RF1
Murray, AM; Waddington, JL1
Edwards, MA; Kantak, KM; Spealman, RD1
Garrett, BE; Holtzman, SG1
Silverman, PB1
Meyer, ME; Shults, JM1
Barthalmus, GT; Temple, JG1
Kamijo, N; Nagao, T; Ono, H1
Bergman, J; Grech, DM; Spealman, RD1
Abrahams, BS; Beninger, RJ; Mallet, PE; Rutherford, JD1
Bergman, J; Tidey, JW1
Lalonde, R; Lestienne, F; Thullier, F1
Platt, DM; Rowlett, JK; Spealman, RD1
Bergman, J; Caine, SB; Mello, NK; Negus, SS1
Bergman, J; Mutschler, NH1
Cauli, O; Morelli, M1
Desai, RI; Katz, JL; Terry, P2
Katz, JL; Kopajtic, TA; Terry, P1

Reviews

1 review(s) available for sk&f 77434 and sk&f-38393

ArticleYear
Biased Ligands of G Protein-Coupled Receptors (GPCRs): Structure-Functional Selectivity Relationships (SFSRs) and Therapeutic Potential.
    Journal of medicinal chemistry, 2018, 11-21, Volume: 61, Issue:22

    Topics: Animals; Drug Discovery; Humans; Ligands; Receptors, G-Protein-Coupled; Signal Transduction; Structure-Activity Relationship

2018

Other Studies

25 other study(ies) available for sk&f 77434 and sk&f-38393

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Stereoisomeric probes for the D1 dopamine receptor: synthesis and characterization of R-(+) and S-(-) enantiomers of 3-allyl-7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine and its 6-bromo analogue.
    Journal of medicinal chemistry, 1992, Apr-17, Volume: 35, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Brain; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship

1992
Dopamine stimulates growth hormone release from the pituitary of goldfish, Carassius auratus, through the dopamine D1 receptors.
    Endocrinology, 1992, Volume: 130, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Bromocriptine; Domperidone; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Goldfish; Gonadotropin-Releasing Hormone; Growth Hormone; Pituitary Gland; Quinpirole; Radioimmunoassay; Receptors, Dopamine

1992
The D1 agonists SKF 82958 and SKF 77434 are self-administered by rats.
    Brain research, 1992, Jun-12, Volume: 582, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reinforcement, Psychology; Self Administration

1992
Differential antagonism of the effects of dopamine D1-receptor agonists on feeding behavior in the rat.
    Psychopharmacology, 1992, Volume: 109, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agonists; Dose-Response Relationship, Drug; Feeding Behavior; Food Deprivation; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone

1992
Activation of the 5-HT1C receptor expressed in Xenopus oocytes by the benzazepines SCH 23390 and SKF 38393.
    British journal of pharmacology, 1991, Volume: 104, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Choroid Plexus; Cloning, Molecular; Dopamine Agents; Dopamine Antagonists; In Vitro Techniques; Oocytes; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Serotonin; RNA, Messenger; Serotonin; Signal Transduction; Swine; Xenopus laevis

1991
The interaction of clozapine with dopamine D1 versus dopamine D2 receptor-mediated function: behavioural indices.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Clozapine; Dopamine; Grooming; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1990
Effects of N-methyl-D-aspartate antagonists in rats discriminating different doses of cocaine: comparison with direct and indirect dopamine agonists.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cocaine; Discrimination Learning; Dopamine Agonists; Male; N-Methylaspartate; Oxazines; Piperazines; Rats; Rats, Wistar

1995
Caffeine cross-tolerance to selective dopamine D1 and D2 receptor agonists but not to their synergistic interaction.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Administration, Oral; Analysis of Variance; Animals; Apomorphine; Caffeine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Drug Tolerance; Ergolines; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2

1994
On-off effects of dopamine receptor agonists in the hemi-parkinsonian rat.
    European journal of pharmacology, 1993, Sep-21, Volume: 242, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cocaine; Dopamine Agents; Dose-Response Relationship, Drug; Female; Injections, Intraperitoneal; Motor Activity; Oxidopamine; Parkinson Disease; Rats; Rats, Sprague-Dawley

1993
Dopamine D1 receptor family agonists, SK&F38393, SK&F77434, and SK&F82958, differentially affect locomotor activities in rats.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 46, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drug Synergism; Motor Activity; Physical Stimulation; Rats; Receptors, Dopamine D1; Stereotyped Behavior

1993
Effects of monoamine oxidase inhibitors and dopamine agonists on the behavior of mammal- and frog-eating snakes.
    Physiology & behavior, 1994, Volume: 55, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Appetitive Behavior; Clorgyline; Colubridae; Dopamine Agents; Dose-Response Relationship, Drug; Feeding Behavior; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Motor Activity; Receptors, Dopamine; Receptors, Dopamine D1; Selegiline; Snakes; Species Specificity; Stereotyped Behavior

1994
Depression of the monosynaptic reflex by apomorphine or bromocriptine is not mediated by D1/D2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Bromocriptine; Decerebrate State; Depression, Chemical; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Monosynaptic; Sulpiride; Synaptic Transmission

1993
Self-administration of D1 receptor agonists by squirrel monkeys.
    Psychopharmacology, 1996, Volume: 125, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Receptors, Dopamine D1; Saimiri; Self Administration

1996
Place conditioning with the dopamine D1-like receptor agonist SKF 82958 but not SKF 81297 or SKF 77434.
    European journal of pharmacology, 1998, Feb-19, Volume: 343, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Motor Activity; Rats; Rats, Wistar; Receptors, Dopamine D1

1998
Drug discrimination in methamphetamine-trained monkeys: agonist and antagonist effects of dopaminergic drugs.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic Agents; Animals; Benzazepines; Catalepsy; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Ergolines; Male; Methamphetamine; Oxazines; Receptors, Dopamine D1; Receptors, Dopamine D2; Saimiri

1998
Effects of dopaminergic agents and of an NMDA receptor antagonist on motor coordination in Lurcher mutant mice.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 63, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Carbidopa; Dextromethorphan; Dopamine Agonists; Dopamine Antagonists; Female; Levodopa; Male; Mice; Mice, Neurologic Mutants; Olivopontocerebellar Atrophies; Psychomotor Performance; Receptors, N-Methyl-D-Aspartate

1999
Dissociation of cocaine-antagonist properties and motoric effects of the D1 receptor partial agonists SKF 83959 and SKF 77434.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Catalepsy; Cocaine; Discrimination Learning; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Muscle Rigidity; Receptors, Dopamine D1; Saimiri

2000
Effects of dopamine D1-like and D2-like agonists in rats trained to discriminate cocaine from saline: influence of experimental history.
    Experimental and clinical psychopharmacology, 2000, Volume: 8, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cocaine; Dextroamphetamine; Discrimination Learning; Discrimination, Psychological; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetrahydronaphthalenes

2000
Effects of chronic administration of the D1 receptor partial agonist SKF 77434 on cocaine self-administration in rhesus monkeys.
    Psychopharmacology, 2002, Volume: 160, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Eating; Female; Macaca mulatta; Reaction Time; Receptors, Dopamine D1; Self Administration

2002
Subchronic caffeine administration sensitizes rats to the motor-activating effects of dopamine D(1) and D(2) receptor agonists.
    Psychopharmacology, 2002, Volume: 162, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Dopamine Agonists; Drug Synergism; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2

2002
Comparison of the discriminative-stimulus effects of SKF 38393 with those of other dopamine receptor agonists.
    Behavioural pharmacology, 2003, Volume: 14, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Cocaine; Discrimination Learning; Discrimination, Psychological; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Humans; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2

2003
A comparison of the locomotor stimulant effects of D1-like receptor agonists in mice.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Cocaine; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Hydrolysis; Male; Mice; Motor Activity; Phosphatidylinositols; Receptors, Dopamine D1; Time Factors

2005
Effects of dopamine D1-like receptor agonists on food-maintained operant behavior in rats.
    Behavioural pharmacology, 2006, Volume: 17, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Synergism; Food; Male; Metergoline; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reinforcement Schedule; Reward; Spiperone

2006