sk&f 77434 has been researched along with sk&f-38393 in 26 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 16 (61.54) | 18.2507 |
2000's | 9 (34.62) | 29.6817 |
2010's | 1 (3.85) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Baindur, N; Baldessarini, RJ; Kula, NS; Neumeyer, JL | 1 |
Cheng, J; McCorvy, JD; Tan, L; Yan, W | 1 |
Chang, JP; Peter, RE; Wong, AO | 1 |
Self, DW; Stein, L | 1 |
Katz, JL; Terry, P | 1 |
Briggs, CA; Frail, DE; Kang, CH; Kebabian, JW; Paxson, CL; Pollock, NJ; Rakowski, RF | 1 |
Murray, AM; Waddington, JL | 1 |
Edwards, MA; Kantak, KM; Spealman, RD | 1 |
Garrett, BE; Holtzman, SG | 1 |
Silverman, PB | 1 |
Meyer, ME; Shults, JM | 1 |
Barthalmus, GT; Temple, JG | 1 |
Kamijo, N; Nagao, T; Ono, H | 1 |
Bergman, J; Grech, DM; Spealman, RD | 1 |
Abrahams, BS; Beninger, RJ; Mallet, PE; Rutherford, JD | 1 |
Bergman, J; Tidey, JW | 1 |
Lalonde, R; Lestienne, F; Thullier, F | 1 |
Platt, DM; Rowlett, JK; Spealman, RD | 1 |
Bergman, J; Caine, SB; Mello, NK; Negus, SS | 1 |
Bergman, J; Mutschler, NH | 1 |
Cauli, O; Morelli, M | 1 |
Desai, RI; Katz, JL; Terry, P | 2 |
Katz, JL; Kopajtic, TA; Terry, P | 1 |
1 review(s) available for sk&f 77434 and sk&f-38393
Article | Year |
---|---|
Biased Ligands of G Protein-Coupled Receptors (GPCRs): Structure-Functional Selectivity Relationships (SFSRs) and Therapeutic Potential.
Topics: Animals; Drug Discovery; Humans; Ligands; Receptors, G-Protein-Coupled; Signal Transduction; Structure-Activity Relationship | 2018 |
25 other study(ies) available for sk&f 77434 and sk&f-38393
Article | Year |
---|---|
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Stereoisomeric probes for the D1 dopamine receptor: synthesis and characterization of R-(+) and S-(-) enantiomers of 3-allyl-7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine and its 6-bromo analogue.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Brain; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 1992 |
Dopamine stimulates growth hormone release from the pituitary of goldfish, Carassius auratus, through the dopamine D1 receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Bromocriptine; Domperidone; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Goldfish; Gonadotropin-Releasing Hormone; Growth Hormone; Pituitary Gland; Quinpirole; Radioimmunoassay; Receptors, Dopamine | 1992 |
The D1 agonists SKF 82958 and SKF 77434 are self-administered by rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reinforcement, Psychology; Self Administration | 1992 |
Differential antagonism of the effects of dopamine D1-receptor agonists on feeding behavior in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agonists; Dose-Response Relationship, Drug; Feeding Behavior; Food Deprivation; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone | 1992 |
Activation of the 5-HT1C receptor expressed in Xenopus oocytes by the benzazepines SCH 23390 and SKF 38393.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Choroid Plexus; Cloning, Molecular; Dopamine Agents; Dopamine Antagonists; In Vitro Techniques; Oocytes; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Serotonin; RNA, Messenger; Serotonin; Signal Transduction; Swine; Xenopus laevis | 1991 |
The interaction of clozapine with dopamine D1 versus dopamine D2 receptor-mediated function: behavioural indices.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Clozapine; Dopamine; Grooming; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1990 |
Effects of N-methyl-D-aspartate antagonists in rats discriminating different doses of cocaine: comparison with direct and indirect dopamine agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cocaine; Discrimination Learning; Dopamine Agonists; Male; N-Methylaspartate; Oxazines; Piperazines; Rats; Rats, Wistar | 1995 |
Caffeine cross-tolerance to selective dopamine D1 and D2 receptor agonists but not to their synergistic interaction.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Administration, Oral; Analysis of Variance; Animals; Apomorphine; Caffeine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Drug Tolerance; Ergolines; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1994 |
On-off effects of dopamine receptor agonists in the hemi-parkinsonian rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cocaine; Dopamine Agents; Dose-Response Relationship, Drug; Female; Injections, Intraperitoneal; Motor Activity; Oxidopamine; Parkinson Disease; Rats; Rats, Sprague-Dawley | 1993 |
Dopamine D1 receptor family agonists, SK&F38393, SK&F77434, and SK&F82958, differentially affect locomotor activities in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drug Synergism; Motor Activity; Physical Stimulation; Rats; Receptors, Dopamine D1; Stereotyped Behavior | 1993 |
Effects of monoamine oxidase inhibitors and dopamine agonists on the behavior of mammal- and frog-eating snakes.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Appetitive Behavior; Clorgyline; Colubridae; Dopamine Agents; Dose-Response Relationship, Drug; Feeding Behavior; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Motor Activity; Receptors, Dopamine; Receptors, Dopamine D1; Selegiline; Snakes; Species Specificity; Stereotyped Behavior | 1994 |
Depression of the monosynaptic reflex by apomorphine or bromocriptine is not mediated by D1/D2 receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Bromocriptine; Decerebrate State; Depression, Chemical; Dopamine Agents; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Monosynaptic; Sulpiride; Synaptic Transmission | 1993 |
Self-administration of D1 receptor agonists by squirrel monkeys.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Receptors, Dopamine D1; Saimiri; Self Administration | 1996 |
Place conditioning with the dopamine D1-like receptor agonist SKF 82958 but not SKF 81297 or SKF 77434.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Motor Activity; Rats; Rats, Wistar; Receptors, Dopamine D1 | 1998 |
Drug discrimination in methamphetamine-trained monkeys: agonist and antagonist effects of dopaminergic drugs.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic Agents; Animals; Benzazepines; Catalepsy; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Ergolines; Male; Methamphetamine; Oxazines; Receptors, Dopamine D1; Receptors, Dopamine D2; Saimiri | 1998 |
Effects of dopaminergic agents and of an NMDA receptor antagonist on motor coordination in Lurcher mutant mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Carbidopa; Dextromethorphan; Dopamine Agonists; Dopamine Antagonists; Female; Levodopa; Male; Mice; Mice, Neurologic Mutants; Olivopontocerebellar Atrophies; Psychomotor Performance; Receptors, N-Methyl-D-Aspartate | 1999 |
Dissociation of cocaine-antagonist properties and motoric effects of the D1 receptor partial agonists SKF 83959 and SKF 77434.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Catalepsy; Cocaine; Discrimination Learning; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Muscle Rigidity; Receptors, Dopamine D1; Saimiri | 2000 |
Effects of dopamine D1-like and D2-like agonists in rats trained to discriminate cocaine from saline: influence of experimental history.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cocaine; Dextroamphetamine; Discrimination Learning; Discrimination, Psychological; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetrahydronaphthalenes | 2000 |
Effects of chronic administration of the D1 receptor partial agonist SKF 77434 on cocaine self-administration in rhesus monkeys.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Eating; Female; Macaca mulatta; Reaction Time; Receptors, Dopamine D1; Self Administration | 2002 |
Subchronic caffeine administration sensitizes rats to the motor-activating effects of dopamine D(1) and D(2) receptor agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Dopamine Agonists; Drug Synergism; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2002 |
Comparison of the discriminative-stimulus effects of SKF 38393 with those of other dopamine receptor agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Cocaine; Discrimination Learning; Discrimination, Psychological; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Humans; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2003 |
A comparison of the locomotor stimulant effects of D1-like receptor agonists in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Cocaine; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Hydrolysis; Male; Mice; Motor Activity; Phosphatidylinositols; Receptors, Dopamine D1; Time Factors | 2005 |
Effects of dopamine D1-like receptor agonists on food-maintained operant behavior in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Synergism; Food; Male; Metergoline; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reinforcement Schedule; Reward; Spiperone | 2006 |