sk&f-38393 and spiperone

sk&f-38393 has been researched along with spiperone in 80 studies

Research

Studies (80)

TimeframeStudies, this research(%)All Research%
pre-199026 (32.50)18.7374
1990's40 (50.00)18.2507
2000's9 (11.25)29.6817
2010's5 (6.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH1
Jiang, H; Li, Z; Liu, H; Lu, W; Qian, W; Sun, H; Zhang, L; Zhao, R; Zhen, X; Zhou, S; Zhou, Y; Zhu, L1
Chen, K; Gao, B; Guo, L; Jiang, H; Li, Z; Liu, H; Qian, W; Sun, H; Yang, H; Zhen, X; Zhou, S; Zhou, Y; Zhu, L1
Chen, J; Du, P; Fu, W; Li, W; Xu, L; Yuan, C; Zhang, L; Zhen, X1
Choi, AL; Gallo, F; Martínez de la Escalera, G; Weiner, RI1
Jenner, P; Marsden, CD; Rose, S; Thomas, KL2
Lucki, I; McGonigle, P; Subramaniam, S1
LaHoste, GJ; Marshall, JF1
Katz, JL; Terry, P1
O'Boyle, KM; Waddington, JL5
Gong, L; Kostrzewa, RM1
Michel, AD; Nunes, JL; Sharif, NA; Whiting, RL1
Linseman, MA1
Bédard, PJ; Di Paolo, T; Gagnon, C1
Lucki, I; McGonigle, P; Neisewander, JL1
Murray, AM; Waddington, JL2
Nowak, JZ; Schorderet, M1
Bédard, PJ; Di Paolo, T; Rouillard, C1
Beaulieu, M; Felder, R; Kebabian, JW1
Dreher, JK; Jackson, DM1
Segawa, T; Zhang, X1
Brewster, WK; Lee, RC; Lewis, MH; Lovenberg, TW; Mailman, RB; Mottola, DM; Nichols, DE; Riggs, RM1
Arnt, J; Hyttel, J1
Carlsson, A; Hjorth, S1
Crocker, AD; Faunt, JE1
Bijak, M; Smiałowski, A1
Dall'Olio, R; Gandolfi, O; Montanaro, N; Roncada, P1
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW1
Arnt, J; Hyttel, J; Nowak, G1
Burchill, SA; Thody, AJ1
Bondy, SC; Breese, GR; Duncan, GE; Iorio, LC; Mueller, RA; Napier, TC1
Bédard, PJ; Bouchard, S; Boucher, R; Di Paolo, T; Falardeau, P1
Friedhoff, AJ; Rosengarten, H; Schweitzer, JW2
Brunello, N; Monopoli, A; Ongini, E; Racagni, G; Rovescalli, AC1
Salama, AI; Saller, CF1
Arnt, J1
Briley, M; Langer, SZ; Lehmann, J1
Bass, LS; Clardy, J; Dandridge, PA; Garvey, E; Hahn, RA; Kaiser, C; Sarau, HM; Setler, PE1
Senogles, SE1
Chuang, YC; Huang, WT; Lin, MT; Liu, HS; Won, SJ1
Abarca, J; Bustos, G; Gysling, K; Roth, RH1
del Valle, M; García, AG; López, MG; Maroto, R; Mellström, B; Naranjo, JR1
Katz, JL; Witkin, JM1
Guo, J; Kostrzewa, FP; Kostrzewa, RM1
Dall'Olio, R; Gandolfi, O; Rimondini, R1
Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD1
Atrens, DM; Hunt, GE; Jackson, DM1
Chuang, DM; Kirch, DG; Li, R; Wyatt, RJ1
Burnham, P; Louis, JC; Magal, E; Varon, S1
Dall'Olio, R; Gandolfi, O1
Aloyo, VJ; Chen, JF; Weiss, B1
Matsokis, NA; Panagopoulos, NT; Valcana, T1
Deveney, AM; Waddington, JL1
Furukawa, T; Morishita, H1
Braghiroli, L; De Feo, G; Giacomelli, S; Koppenaal, DW; Ponzianelli, A1
Ball, GF; Balthazart, J; Castagna, C1
Cook, CD; Picker, MJ; Rodefer, JS1
Bradley, RJ; Dwyer, DS; Liu, Y1
Hu, JY; Jin, GZ1
Gu, Q; Kwong, E1
Gao, X; Wu, G; Zhang, Y2
Hu, G; Qin, W1
Chu, J; Wilcox, RE; Wilczynski, W1
Fu, Y; Jin, GZ; Zhu, XZ; Zhu, ZT1
Ebadi, M; Govitrapong, P; Santanavanich, C1
Katz, JL; Kopajtic, TA; Terry, P1
Chen, J; Ma, L; Wang, F; Zhang, H; Zhen, X1
Coffeen, U; del Angel, R; López-Avila, A; López-Muñoz, FJ; Ortega-Legaspi, JM; Pellicer, F1
Pfister, G; Schramm, KW; Ud-Daula, A1
Barnes, S; Brecha, NC; Grove, JC; Hirano, AA; Liu, X1
Baindur, N; Bakthavachalam, V; Madras, BK; Neumeyer, JL1
Booth, RG; Brown, RL; Bucholtz, EC; Tropsha, A; Wyrick, SD1

Reviews

1 review(s) available for sk&f-38393 and spiperone

ArticleYear
Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
    Cellular and molecular neurobiology, 1990, Volume: 10, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates

1990

Other Studies

79 other study(ies) available for sk&f-38393 and spiperone

ArticleYear
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
    Nature, 1991, Apr-18, Volume: 350, Issue:6319

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection

1991
Design, synthesis, and pharmacological evaluation of novel tetrahydroprotoberberine derivatives: selective inhibitors of dopamine D₁ receptor.
    Bioorganic & medicinal chemistry, 2012, Aug-01, Volume: 20, Issue:15

    Topics: Berberine Alkaloids; Dose-Response Relationship, Drug; Drug Design; HEK293 Cells; Humans; Models, Molecular; Molecular Structure; Receptors, Dopamine D1; Structure-Activity Relationship

2012
Asymmetric total synthesis and identification of tetrahydroprotoberberine derivatives as new antipsychotic agents possessing a dopamine D(1), D(2) and serotonin 5-HT(1A) multi-action profile.
    Bioorganic & medicinal chemistry, 2013, Feb-15, Volume: 21, Issue:4

    Topics: Animals; Antipsychotic Agents; Berberine; Berberine Alkaloids; CHO Cells; Cricetinae; Cricetulus; Dopamine D2 Receptor Antagonists; HEK293 Cells; Humans; Microwaves; Motor Activity; Protein Binding; Rats; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D1; Receptors, Dopamine D2; Schizophrenia; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Functional reversal of (-)-Stepholidine analogues by replacement of benzazepine substructure using the ring-expansion strategy.
    Chemical biology & drug design, 2016, Volume: 88, Issue:4

    Topics: Benzazepines; Berberine; Binding Sites; Biological Assay; Dopamine D2 Receptor Antagonists; Humans; Models, Molecular; Receptors, Dopamine D1; Receptors, Dopamine D2

2016
Dopaminergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via D1-receptors positively coupled to adenylate cyclase.
    Endocrinology, 1992, Volume: 131, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Benzazepines; Bromocriptine; Cell Line; Cyclic AMP; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Gonadotropin-Releasing Hormone; Kinetics; Nerve Tissue Proteins; Neurons; Norepinephrine; Phosphoproteins; Receptors, Dopamine D1; RNA, Messenger; Spiperone

1992
Dissociation of the striatal D-2 dopamine receptor from adenylyl cyclase following 6-hydroxydopamine-induced denervation.
    Biochemical pharmacology, 1992, Jul-07, Volume: 44, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Benzazepines; Corpus Striatum; Cyclic AMP; Denervation; Dopamine; Ergolines; Female; Homovanillic Acid; Oxidopamine; Prosencephalon; Quinpirole; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1992
Acute reserpine treatment induces down regulation of D-1 dopamine receptor associated adenylyl cyclase activity in rat striatum.
    Biochemical pharmacology, 1992, Jul-07, Volume: 44, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Corpus Striatum; Cyclic AMP; Dose-Response Relationship, Drug; Down-Regulation; Female; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone

1992
Effects of chronic treatment with selective agonists on the subtypes of dopamine receptors.
    Brain research, 1992, Feb-07, Volume: 571, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Body Temperature Regulation; Brain; Caudate Nucleus; Dopamine Agents; Drug Interactions; Ergolines; Kinetics; Male; Nucleus Accumbens; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reference Values; Spiperone; Substantia Nigra

1992
Dopamine supersensitivity and D1/D2 synergism are unrelated to changes in striatal receptor density.
    Synapse (New York, N.Y.), 1992, Volume: 12, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Oxidopamine; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone; Stereotyped Behavior; Time Factors; Tritium

1992
Differential antagonism of the effects of dopamine D1-receptor agonists on feeding behavior in the rat.
    Psychopharmacology, 1992, Volume: 109, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agonists; Dose-Response Relationship, Drug; Feeding Behavior; Food Deprivation; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone

1992
Agonist and antagonist interactions with D1 dopamine receptors: agonist-induced masking of D1 receptors depends on intrinsic activity.
    Neuropharmacology, 1992, Volume: 31, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics; Animals; Benzazepines; Binding, Competitive; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Indoles; Kinetics; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1992
Supersensitized D1 receptors mediate enhanced oral activity after neonatal 6-OHDA.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Female; Mouth; Movement; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1991
Dopamine D2-receptors mediate hypothermia in mice: ICV and IP effects of agonists and antagonists.
    Neurochemical research, 1991, Volume: 16, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Body Temperature Regulation; Cerebral Ventricles; Domperidone; Dopamine Agents; Dopamine Antagonists; Ergolines; Hypothermia; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1991
Effects of dopaminergic agents on alcohol consumption by rats in a limited access paradigm.
    Psychopharmacology, 1990, Volume: 100, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Amphetamine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drinking Behavior; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1990
Effect of chronic treatment of MPTP monkeys with dopamine D-1 and/or D-2 receptor agonists.
    European journal of pharmacology, 1990, Mar-13, Volume: 178, Issue:1

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Brain; Bromocriptine; Carbidopa; Catecholamines; Dopamine Agents; Female; Levodopa; Macaca fascicularis; Receptors, Dopamine; Spiperone

1990
Behavioral and neurochemical effects of chronic administration of reserpine and SKF-38393 in rats.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Spiperone; Stereotyped Behavior; Tritium

1991
The interaction of clozapine with dopamine D1 versus dopamine D2 receptor-mediated function: behavioural indices.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Clozapine; Dopamine; Grooming; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1990
Effects of chronic treatment of MPTP monkeys with bromocriptine alone or in combination with SKF 38393.
    European journal of pharmacology, 1990, Aug-28, Volume: 185, Issue:2-3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Brain; Brain Chemistry; Bromocriptine; Dopamine; Female; Homovanillic Acid; Kinetics; Levodopa; Macaca fascicularis; Motor Activity; MPTP Poisoning; Parkinson Disease, Secondary; Receptors, Dopamine; Spiperone

1990
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
Role of D1 and D2 dopamine receptors in mediating locomotor activity elicited from the nucleus accumbens of rats.
    Brain research, 1989, May-22, Volume: 487, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Ketanserin; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Septal Nuclei; Spiperone; Time Factors

1989
The induction of grooming and vacuous chewing by a series of selective D-1 dopamine receptor agonists: two directions of D-1:D-2 interaction.
    European journal of pharmacology, 1989, Feb-07, Volume: 160, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine Agents; Dose-Response Relationship, Drug; Grooming; Isoquinolines; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior

1989
Selective blockade of dopamine D-1 receptor by SCH 23390 affects dopamine agonist binding to 3H-spiperone labeled D-2 receptors in rat striatum.
    Japanese journal of pharmacology, 1989, Volume: 50, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Guanosine Triphosphate; In Vitro Techniques; Male; Pertussis Toxin; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Virulence Factors, Bordetella

1989
Dihydrexidine, a novel selective high potency full dopamine D-1 receptor agonist.
    European journal of pharmacology, 1989, Jul-04, Volume: 166, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Binding, Competitive; Corpus Striatum; Dopamine Agents; In Vitro Techniques; Male; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Spiperone

1989
Differential involvement of dopamine D-1 and D-2 receptors in the circling behaviour induced by apomorphine, SK & F 38393, pergolide and LY 171555 in 6-hydroxydopamine-lesioned rats.
    Psychopharmacology, 1985, Volume: 85, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Appetite Depressants; Benzazepines; Electric Stimulation; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sympathectomy, Chemical; Time Factors

1985
Structural determinants of selective affinity for brain D-1 dopamine receptors within a series of 1-phenyl-1H-3-benzazepine analogues of SK&F 38393 and SCH 23390.
    European journal of pharmacology, 1985, Sep-24, Volume: 115, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Appetite Depressants; Benzazepines; Brain; Corpus Striatum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Thioxanthenes

1985
Postsynaptic dopamine (DA) receptor stimulator properties of the putative DA autoreceptor-selective agonist B-HT 920 uncovered by co-treatment with the D-1 agonist SK&F 38393.
    Psychopharmacology, 1987, Volume: 93, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Appetite Depressants; Azepines; Benzazepines; Male; Motor Activity; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Synapses

1987
The effects of selective dopamine receptor agonists and antagonists on body temperature in rats.
    European journal of pharmacology, 1987, Jan-20, Volume: 133, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Body Temperature; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1987
Excitatory and inhibitory action of dopamine on hippocampal neurons in vitro. Involvement of D2 and D1 receptors.
    Neuroscience, 1987, Volume: 23, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Culture Techniques; Dopamine; Dopamine Antagonists; Haloperidol; Hippocampus; Male; Neurons; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1987
Behavioral and biochemical expression of D1-receptor supersensitivity following SCH 23390 repeated administrations.
    Brain research, 1988, Jul-12, Volume: 455, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Benzazepines; Corpus Striatum; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1988
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
    Advances in experimental medicine and biology, 1988, Volume: 235

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1988
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.
    European journal of pharmacology, 1988, Aug-24, Volume: 153, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone

1988
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
    The Journal of endocrinology, 1986, Volume: 111, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride

1986
6-hydroxydopamine treatments enhance behavioral responses to intracerebral microinjection of D1- and D2-dopamine agonists into nucleus accumbens and striatum without changing dopamine antagonist binding.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Corpus Striatum; Dopamine; Dopamine Antagonists; Ergolines; Female; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Microinjections; Motor Activity; Nucleus Accumbens; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Spiperone

1987
Behavioral and biochemical effect of chronic treatment with D-1 and/or D-2 dopamine agonists in MPTP monkeys.
    European journal of pharmacology, 1988, May-20, Volume: 150, Issue:1-2

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Benzazepines; Brain Chemistry; Dopamine; Dyskinesia, Drug-Induced; Female; Homovanillic Acid; Macaca fascicularis; Motor Activity; Parkinson Disease, Secondary; Pyridines; Receptors, Dopamine; Spiperone

1988
New substituted 1-phenyl-3-benzazepine analogues of SK&F 38393 and N-methyl-thienopyridine analogues of dihydroxynomifensine with selective affinity for the D-1 dopamine receptor in human post-mortem brain.
    Neuropharmacology, 1987, Volume: 26, Issue:12

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Benzazepines; Binding, Competitive; Brain Chemistry; Humans; In Vitro Techniques; Kinetics; Ligands; Nomifensine; Putamen; Pyridines; Receptors, Dopamine; Spiperone; Thiophenes

1987
Selective dopamine D2 receptor reduction enhances a D1-mediated oral dyskinesia in rats.
    Life sciences, 1986, Jul-07, Volume: 39, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dopamine Antagonists; Jaw; Rats; Rats, Inbred F344; Rats, Inbred Strains; Receptors, Dopamine; Species Specificity; Spiperone; Stereotyped Behavior; Tetrabenazine

1986
Absence of [3H]SCH 23390 specific binding sites in anterior pituitary: dissociation from effects on prolactin secretion.
    European journal of pharmacology, 1987, Mar-17, Volume: 135, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Corpus Striatum; Cyproheptadine; Ergolines; Kinetics; Male; Metergoline; Pituitary Gland, Anterior; Prolactin; Quinpirole; Rats; Rats, Inbred Strains; Spiperone

1987
Dopamine receptor subtypes: in vivo biochemical evidence for functional interaction.
    European journal of pharmacology, 1985, Feb-26, Volume: 109, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Corpus Striatum; Dopamine; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1985
Hyperactivity induced by stimulation of separate dopamine D-1 and D-2 receptors in rats with bilateral 6-OHDA lesions.
    Life sciences, 1985, Aug-26, Volume: 37, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Benzazepines; Clopenthixol; Dopamine; Dose-Response Relationship, Drug; Ergolines; Flupenthixol; Hydroxydopamines; Hypothalamus; Male; Motor Activity; Oxidopamine; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone

1985
Characterization of dopamine autoreceptor and [3H]spiperone binding sites in vitro with classical and novel dopamine receptor agonists.
    European journal of pharmacology, 1983, Mar-18, Volume: 88, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Apomorphine; Benzazepines; Binding Sites; Bromocriptine; Butyrophenones; Cats; Caudate Nucleus; Dopamine; Electric Stimulation; Female; In Vitro Techniques; Male; Phentolamine; Receptors, Dopamine; Spiperone; Sulpiride; Tritium

1983
Selective and stereospecific interactions of R-SK & F 38393 with [3H]piflutixol but not [3H]spiperone binding to striatal D1 and D2 dopamine receptors: comparisons with SCH 23390.
    European journal of pharmacology, 1984, Mar-02, Volume: 98, Issue:3-4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Appetite Depressants; Benzazepines; Binding, Competitive; Butyrophenones; Corpus Striatum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism; Thioxanthenes

1984
Induction of oral dyskinesias in naive rats by D1 stimulation.
    Life sciences, 1983, Dec-19, Volume: 33, Issue:25

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dyskinesia, Drug-Induced; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride

1983
Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.
    European journal of pharmacology, 1984, Oct-30, Volume: 106, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; In Vitro Techniques; Isoquinolines; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereoisomerism; Thioxanthenes

1984
Absolute stereochemistry and dopaminergic activity of enantiomers of 2,3,4,5-tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Binding, Competitive; Chemical Phenomena; Chemistry; Dogs; In Vitro Techniques; Male; Molecular Conformation; Rats; Receptors, Dopamine; Renal Circulation; Spiperone; Stereoisomerism; Substantia Nigra; Vasodilator Agents

1982
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
    Endocrinology, 1994, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella

1994
Suppression of natural killer cell activity in mouse spleen lymphocytes by several dopamine receptor antagonists.
    Experientia, 1995, Apr-15, Volume: 51, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cytotoxicity, Immunologic; Dopamine Antagonists; Flupenthixol; Fluphenazine; Killer Cells, Natural; Mice; Mice, Inbred C3H; Pimozide; Spiperone; Spleen; Thiothixene; Trifluoperazine

1995
Changes in extracellular levels of glutamate and aspartate in rat substantia nigra induced by dopamine receptor ligands: in vivo microdialysis studies.
    Neurochemical research, 1995, Volume: 20, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aspartic Acid; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Extracellular Space; Glutamic Acid; Kinetics; Ligands; Male; Microdialysis; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Spiperone; Substantia Nigra; Tetrodotoxin; Time Factors

1995
Expression of the bovine striatal D2 receptor, but not the D1 receptor, in bovine adrenal medulla.
    Molecular pharmacology, 1995, Volume: 47, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenal Medulla; Animals; Base Sequence; Benzazepines; Catecholamines; Cattle; Caudate Nucleus; Cell Membrane; Corpus Striatum; Gene Expression; Iodine Radioisotopes; Kinetics; Microsomes; Molecular Sequence Data; Radioligand Assay; Receptors, Dopamine D1; Receptors, Dopamine D2; Sequence Homology, Nucleic Acid; Spiperone; Tritium

1995
Behavioral effects of dopaminergic agonists and antagonists alone and in combination in the squirrel monkey.
    Psychopharmacology, 1993, Volume: 113, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Reinforcement Schedule; Saimiri; Spiperone

1993
Ontogenetic quinpirole treatment induces vertical jumping activity in rats.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Behavior, Animal; Benzazepines; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Injections, Intraperitoneal; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1993
D-cycloserine decreases both D1 and D2 dopamine receptors number and their function in rat brain.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Cell Membrane; Cycloserine; Dizocilpine Maleate; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; In Vitro Techniques; Kinetics; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone

1994
An autoradiographic study of the differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on striatal and extrastriatal D-1 and D-2 dopamine receptors in the rat.
    Neuropharmacology, 1994, Volume: 33, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Densitometry; Dopamine Agonists; Dopamine Antagonists; Ergolines; Male; Neostriatum; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1994
Reward summation and the effects of dopamine D1 and D2 agonists and antagonists on fixed-interval responding for brain stimulation.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Brain; Bromocriptine; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Drug Interactions; Electric Stimulation; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule; Reward; Self Stimulation; Spiperone

1994
Effect of chronic haloperidol treatment on dopamine-induced inositol phosphate formation in rat brain slices.
    Neurochemical research, 1994, Volume: 19, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Brain; Corpus Striatum; Dopamine; Dopamine Antagonists; Frontal Lobe; Haloperidol; Hippocampus; In Vitro Techniques; Inositol; Inositol Phosphates; Male; Organ Specificity; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Reference Values; Spiperone

1994
Convergent regulation by ciliary neurotrophic factor and dopamine of tyrosine hydroxylase expression in cultures of rat substantia nigra.
    Neuroscience, 1993, Volume: 52, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Cells, Cultured; Ciliary Neurotrophic Factor; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Ergolines; Glial Fibrillary Acidic Protein; Haloperidol; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphopyruvate Hydratase; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Proteins; Spiperone; Substantia Nigra; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase

1993
Chronic treatment with MK-801 decreases D2 dopamine receptor function in rat striatum.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Corpus Striatum; Dizocilpine Maleate; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Grooming; In Vitro Techniques; Kinetics; Ligands; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone

1993
Continuous treatment with the D2 dopamine receptor agonist quinpirole decreases D2 dopamine receptors, D2 dopamine receptor messenger RNA and proenkephalin messenger RNA, and increases mu opioid receptors in mouse striatum.
    Neuroscience, 1993, Volume: 54, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Behavior, Animal; Blotting, Northern; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Down-Regulation; Enkephalins; Ergolines; Image Processing, Computer-Assisted; Male; Mice; Nucleic Acid Hybridization; Oligonucleotide Probes; Protein Precursors; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger; Spiperone; Up-Regulation

1993
Cerebellar and striatal dopamine receptors: effects of reeler and weaver murine mutations.
    Journal of neuroscience research, 1993, Aug-01, Volume: 35, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebellum; Corpus Striatum; Dopamine; Kinetics; Mice; Mice, Neurologic Mutants; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Species Specificity; Spiperone

1993
Pharmacological characterization of behavioural responses to SK&F 83959 in relation to 'D1-like' dopamine receptors not linked to adenylyl cyclase.
    British journal of pharmacology, 1995, Volume: 116, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Behavior, Animal; Benzamides; Benzazepines; Binding, Competitive; Chromans; Dopamine Agonists; Dopamine Antagonists; Enzyme Induction; Isoquinolines; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone; Tetrahydroisoquinolines

1995
Existence of dopamine D1 receptor on the sympathetic nerve endings in the guinea-pig vas deferens.
    European journal of pharmacology, 1997, Jun-11, Volume: 328, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Brimonidine Tartrate; Dopamine Agonists; Dopamine Antagonists; Electric Stimulation; Guinea Pigs; Idazoxan; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Presynaptic Terminals; Quinoxalines; Receptors, Dopamine D1; Spiperone; Synaptic Transmission; Vas Deferens

1997
A sensitive assay for studying dopaminergic activity in cultures of rat pituitary cells.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cell Count; Cells, Cultured; Cyproheptadine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Evaluation, Preclinical; Female; Haloperidol; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Spiperone

1997
Differential effects of D1 and D2 dopamine-receptor agonists and antagonists on appetitive and consummatory aspects of male sexual behavior in Japanese quail.
    Physiology & behavior, 1997, Volume: 62, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Coturnix; Dopamine Agonists; Dopamine Antagonists; Male; Sexual Behavior, Animal; Spiperone

1997
Selective attenuation of the antinociceptive effects of mu opioids by the putative dopamine D3 agonist 7-OH-DPAT.
    Psychopharmacology, 1999, Volume: 144, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Opioid; Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cycloparaffins; Dopamine Agonists; Dopamine Antagonists; Drug Antagonism; Male; Morphine; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Spiperone; Tetrahydronaphthalenes

1999
Dopamine receptor antagonists modulate glucose uptake in rat pheochromocytoma (PC12) cells.
    Neuroscience letters, 1999, Oct-29, Volume: 274, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Biological Transport; Chlorpromazine; Clozapine; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fluphenazine; Glucose; Haloperidol; PC12 Cells; Pimozide; Rats; Receptors, Dopamine D2; Spiperone; Sulpiride; Tritium

1999
Supraspinal D2 receptor involved in antinociception induced by l-tetrahydropalmatine.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Non-Narcotic; Animals; Benzazepines; Berberine Alkaloids; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Injections, Spinal; Male; Pain Threshold; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1999
Activity-dependent and use-dependent regulation of dopamine-receptor clustering.
    Neuroreport, 2000, Aug-21, Volume: 11, Issue:12

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Bromocriptine; Dopamine Agonists; Dopamine Antagonists; Microscopy, Confocal; Rats; Rats, Long-Evans; Receptor Aggregation; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

2000
Effects of dopaminergic agents on carrageenan hyperalgesia in rats.
    European journal of pharmacology, 2000, Oct-06, Volume: 406, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Carrageenan; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Hindlimb; Hyperalgesia; Injections; Injections, Intraventricular; Male; Pain; Pain Measurement; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Sodium Chloride; Spiperone; Time Factors

2000
Effects of dopaminergic agents on carrageenan hyperalgesia after intrathecal administration to rats.
    European journal of pharmacology, 2001, Apr-20, Volume: 418, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Carrageenan; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Hindlimb; Hot Temperature; Hyperalgesia; Injections, Spinal; Male; Pain Measurement; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone

2001
[Differential regulation of dopamine receptors on pre- and postsynaptic Na+, K(+)-ATPase in rat striatum].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1997, Volume: 32, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Female; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sodium-Potassium-Exchanging ATPase; Spiperone; Synaptic Membranes

1997
Pharmacological characterization of the D1- and D2-like dopamine receptors from the brain of the leopard frog, Rana pipiens.
    Brain, behavior and evolution, 2001, Volume: 57, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Brain; Radioligand Assay; Rana pipiens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Species Specificity; Spiperone; Sulpiride

2001
Biphasic firing response of nucleus accumbens neurons elicited by THPB-18 and its correlation with DA receptor subtypes.
    Acta pharmacologica Sinica, 2004, Volume: 25, Issue:12

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Berberine Alkaloids; Dopamine D2 Receptor Antagonists; Male; Neurons; Nucleus Accumbens; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Ventral Tegmental Area

2004
Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway.
    Journal of pineal research, 2005, Volume: 38, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acyltransferases; Animals; Benzazepines; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Melatonin; Phosphorylation; Pineal Gland; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Transcription, Genetic

2005
Effects of dopamine D1-like receptor agonists on food-maintained operant behavior in rats.
    Behavioural pharmacology, 2006, Volume: 17, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Synergism; Food; Male; Metergoline; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reinforcement Schedule; Reward; Spiperone

2006
Chronic SKF83959 induced less severe dyskinesia and attenuated L-DOPA-induced dyskinesia in 6-OHDA-lesioned rat model of Parkinson's disease.
    Neuropharmacology, 2007, Volume: 53, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Drug Administration Schedule; Drug Interactions; Dyskinesia, Drug-Induced; Levodopa; Male; Movement; Oxidopamine; Parkinson Disease; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Spiperone; Sympatholytics; Time Factors

2007
Dopamine receptors in the anterior insular cortex modulate long-term nociception in the rat.
    European journal of pain (London, England), 2008, Volume: 12, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Afferent Pathways; Animals; Apomorphine; Benzazepines; Cerebral Cortex; Chronic Disease; Dopamine; Dopamine Agonists; Dopamine Antagonists; Hot Temperature; Male; Microinjections; Models, Neurological; Neuralgia; Nociceptors; Pain; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Sciatic Neuropathy; Self Mutilation; Spiperone

2008
Identification of dopamine receptor in Tetrahymena thermophila by fluorescent ligands.
    Pakistan journal of biological sciences : PJBS, 2012, Dec-01, Volume: 15, Issue:23

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Fluorescent Dyes; Ligands; Microscopy, Confocal; Microscopy, Fluorescence; Protozoan Proteins; Receptors, Dopamine D1; Rhodamines; Spiperone; Tetrahymena thermophila

2012
Dopamine D1 receptor modulation of calcium channel currents in horizontal cells of mouse retina.
    Journal of neurophysiology, 2016, 08-01, Volume: 116, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Biophysical Phenomena; Calcium; Calcium Channel Blockers; Calcium Channels; Connexins; Dopamine; Dopamine Agonists; Dopamine Antagonists; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; omega-Conotoxin GVIA; Plant Lectins; Receptors, Dopamine D1; Retina; Retinal Horizontal Cells; RNA, Untranslated; Spiperone

2016
Fluorescent probes for dopamine receptors: synthesis and characterization of fluorescein and 7-nitrobenz-2-oxa-1,3-diazol-4-yl conjugates of D-1 and D-2 receptor ligands.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:11

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine Antagonists; Fluorescent Dyes; Ligands; Macaca fascicularis; Oxadiazoles; Receptors, Dopamine; Stereoisomerism; Structure-Activity Relationship

1991
Synthesis, evaluation, and comparative molecular field analysis of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for histamine H(1) receptors.
    Journal of medicinal chemistry, 1999, Aug-12, Volume: 42, Issue:16

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ligands; Models, Molecular; Pyrilamine; Radioligand Assay; Structure-Activity Relationship; Tetrahydronaphthalenes

1999