sk&f-38393 has been researched along with spiperone in 80 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 26 (32.50) | 18.7374 |
1990's | 40 (50.00) | 18.2507 |
2000's | 9 (11.25) | 29.6817 |
2010's | 5 (6.25) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH | 1 |
Jiang, H; Li, Z; Liu, H; Lu, W; Qian, W; Sun, H; Zhang, L; Zhao, R; Zhen, X; Zhou, S; Zhou, Y; Zhu, L | 1 |
Chen, K; Gao, B; Guo, L; Jiang, H; Li, Z; Liu, H; Qian, W; Sun, H; Yang, H; Zhen, X; Zhou, S; Zhou, Y; Zhu, L | 1 |
Chen, J; Du, P; Fu, W; Li, W; Xu, L; Yuan, C; Zhang, L; Zhen, X | 1 |
Choi, AL; Gallo, F; Martínez de la Escalera, G; Weiner, RI | 1 |
Jenner, P; Marsden, CD; Rose, S; Thomas, KL | 2 |
Lucki, I; McGonigle, P; Subramaniam, S | 1 |
LaHoste, GJ; Marshall, JF | 1 |
Katz, JL; Terry, P | 1 |
O'Boyle, KM; Waddington, JL | 5 |
Gong, L; Kostrzewa, RM | 1 |
Michel, AD; Nunes, JL; Sharif, NA; Whiting, RL | 1 |
Linseman, MA | 1 |
Bédard, PJ; Di Paolo, T; Gagnon, C | 1 |
Lucki, I; McGonigle, P; Neisewander, JL | 1 |
Murray, AM; Waddington, JL | 2 |
Nowak, JZ; Schorderet, M | 1 |
Bédard, PJ; Di Paolo, T; Rouillard, C | 1 |
Beaulieu, M; Felder, R; Kebabian, JW | 1 |
Dreher, JK; Jackson, DM | 1 |
Segawa, T; Zhang, X | 1 |
Brewster, WK; Lee, RC; Lewis, MH; Lovenberg, TW; Mailman, RB; Mottola, DM; Nichols, DE; Riggs, RM | 1 |
Arnt, J; Hyttel, J | 1 |
Carlsson, A; Hjorth, S | 1 |
Crocker, AD; Faunt, JE | 1 |
Bijak, M; Smiałowski, A | 1 |
Dall'Olio, R; Gandolfi, O; Montanaro, N; Roncada, P | 1 |
Egawa, M; Friedhoff, AJ; Rosengarten, H; Schweitzer, JW | 1 |
Arnt, J; Hyttel, J; Nowak, G | 1 |
Burchill, SA; Thody, AJ | 1 |
Bondy, SC; Breese, GR; Duncan, GE; Iorio, LC; Mueller, RA; Napier, TC | 1 |
Bédard, PJ; Bouchard, S; Boucher, R; Di Paolo, T; Falardeau, P | 1 |
Friedhoff, AJ; Rosengarten, H; Schweitzer, JW | 2 |
Brunello, N; Monopoli, A; Ongini, E; Racagni, G; Rovescalli, AC | 1 |
Salama, AI; Saller, CF | 1 |
Arnt, J | 1 |
Briley, M; Langer, SZ; Lehmann, J | 1 |
Bass, LS; Clardy, J; Dandridge, PA; Garvey, E; Hahn, RA; Kaiser, C; Sarau, HM; Setler, PE | 1 |
Senogles, SE | 1 |
Chuang, YC; Huang, WT; Lin, MT; Liu, HS; Won, SJ | 1 |
Abarca, J; Bustos, G; Gysling, K; Roth, RH | 1 |
del Valle, M; García, AG; López, MG; Maroto, R; Mellström, B; Naranjo, JR | 1 |
Katz, JL; Witkin, JM | 1 |
Guo, J; Kostrzewa, FP; Kostrzewa, RM | 1 |
Dall'Olio, R; Gandolfi, O; Rimondini, R | 1 |
Gnanalingham, KK; Hunter, AJ; Jenner, P; Marsden, CD | 1 |
Atrens, DM; Hunt, GE; Jackson, DM | 1 |
Chuang, DM; Kirch, DG; Li, R; Wyatt, RJ | 1 |
Burnham, P; Louis, JC; Magal, E; Varon, S | 1 |
Dall'Olio, R; Gandolfi, O | 1 |
Aloyo, VJ; Chen, JF; Weiss, B | 1 |
Matsokis, NA; Panagopoulos, NT; Valcana, T | 1 |
Deveney, AM; Waddington, JL | 1 |
Furukawa, T; Morishita, H | 1 |
Braghiroli, L; De Feo, G; Giacomelli, S; Koppenaal, DW; Ponzianelli, A | 1 |
Ball, GF; Balthazart, J; Castagna, C | 1 |
Cook, CD; Picker, MJ; Rodefer, JS | 1 |
Bradley, RJ; Dwyer, DS; Liu, Y | 1 |
Hu, JY; Jin, GZ | 1 |
Gu, Q; Kwong, E | 1 |
Gao, X; Wu, G; Zhang, Y | 2 |
Hu, G; Qin, W | 1 |
Chu, J; Wilcox, RE; Wilczynski, W | 1 |
Fu, Y; Jin, GZ; Zhu, XZ; Zhu, ZT | 1 |
Ebadi, M; Govitrapong, P; Santanavanich, C | 1 |
Katz, JL; Kopajtic, TA; Terry, P | 1 |
Chen, J; Ma, L; Wang, F; Zhang, H; Zhen, X | 1 |
Coffeen, U; del Angel, R; López-Avila, A; López-Muñoz, FJ; Ortega-Legaspi, JM; Pellicer, F | 1 |
Pfister, G; Schramm, KW; Ud-Daula, A | 1 |
Barnes, S; Brecha, NC; Grove, JC; Hirano, AA; Liu, X | 1 |
Baindur, N; Bakthavachalam, V; Madras, BK; Neumeyer, JL | 1 |
Booth, RG; Brown, RL; Bucholtz, EC; Tropsha, A; Wyrick, SD | 1 |
1 review(s) available for sk&f-38393 and spiperone
Article | Year |
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Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates | 1990 |
79 other study(ies) available for sk&f-38393 and spiperone
Article | Year |
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Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection | 1991 |
Design, synthesis, and pharmacological evaluation of novel tetrahydroprotoberberine derivatives: selective inhibitors of dopamine D₁ receptor.
Topics: Berberine Alkaloids; Dose-Response Relationship, Drug; Drug Design; HEK293 Cells; Humans; Models, Molecular; Molecular Structure; Receptors, Dopamine D1; Structure-Activity Relationship | 2012 |
Asymmetric total synthesis and identification of tetrahydroprotoberberine derivatives as new antipsychotic agents possessing a dopamine D(1), D(2) and serotonin 5-HT(1A) multi-action profile.
Topics: Animals; Antipsychotic Agents; Berberine; Berberine Alkaloids; CHO Cells; Cricetinae; Cricetulus; Dopamine D2 Receptor Antagonists; HEK293 Cells; Humans; Microwaves; Motor Activity; Protein Binding; Rats; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D1; Receptors, Dopamine D2; Schizophrenia; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship | 2013 |
Functional reversal of (-)-Stepholidine analogues by replacement of benzazepine substructure using the ring-expansion strategy.
Topics: Benzazepines; Berberine; Binding Sites; Biological Assay; Dopamine D2 Receptor Antagonists; Humans; Models, Molecular; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2016 |
Dopaminergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via D1-receptors positively coupled to adenylate cyclase.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Benzazepines; Bromocriptine; Cell Line; Cyclic AMP; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Gonadotropin-Releasing Hormone; Kinetics; Nerve Tissue Proteins; Neurons; Norepinephrine; Phosphoproteins; Receptors, Dopamine D1; RNA, Messenger; Spiperone | 1992 |
Dissociation of the striatal D-2 dopamine receptor from adenylyl cyclase following 6-hydroxydopamine-induced denervation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Animals; Benzazepines; Corpus Striatum; Cyclic AMP; Denervation; Dopamine; Ergolines; Female; Homovanillic Acid; Oxidopamine; Prosencephalon; Quinpirole; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1992 |
Acute reserpine treatment induces down regulation of D-1 dopamine receptor associated adenylyl cyclase activity in rat striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Corpus Striatum; Cyclic AMP; Dose-Response Relationship, Drug; Down-Regulation; Female; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone | 1992 |
Effects of chronic treatment with selective agonists on the subtypes of dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Body Temperature Regulation; Brain; Caudate Nucleus; Dopamine Agents; Drug Interactions; Ergolines; Kinetics; Male; Nucleus Accumbens; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reference Values; Spiperone; Substantia Nigra | 1992 |
Dopamine supersensitivity and D1/D2 synergism are unrelated to changes in striatal receptor density.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Oxidopamine; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Spiperone; Stereotyped Behavior; Time Factors; Tritium | 1992 |
Differential antagonism of the effects of dopamine D1-receptor agonists on feeding behavior in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Dopamine Agonists; Dose-Response Relationship, Drug; Feeding Behavior; Food Deprivation; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone | 1992 |
Agonist and antagonist interactions with D1 dopamine receptors: agonist-induced masking of D1 receptors depends on intrinsic activity.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics; Animals; Benzazepines; Binding, Competitive; Cell Membrane; Corpus Striatum; Guanylyl Imidodiphosphate; Indoles; Kinetics; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1992 |
Supersensitized D1 receptors mediate enhanced oral activity after neonatal 6-OHDA.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Dopamine Agents; Dopamine Antagonists; Dose-Response Relationship, Drug; Ergolines; Female; Mouth; Movement; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1991 |
Dopamine D2-receptors mediate hypothermia in mice: ICV and IP effects of agonists and antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Body Temperature Regulation; Cerebral Ventricles; Domperidone; Dopamine Agents; Dopamine Antagonists; Ergolines; Hypothermia; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1991 |
Effects of dopaminergic agents on alcohol consumption by rats in a limited access paradigm.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Amphetamine; Animals; Benzazepines; Dopamine Agents; Dose-Response Relationship, Drug; Drinking Behavior; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Spiperone | 1990 |
Effect of chronic treatment of MPTP monkeys with dopamine D-1 and/or D-2 receptor agonists.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Brain; Bromocriptine; Carbidopa; Catecholamines; Dopamine Agents; Female; Levodopa; Macaca fascicularis; Receptors, Dopamine; Spiperone | 1990 |
Behavioral and neurochemical effects of chronic administration of reserpine and SKF-38393 in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Spiperone; Stereotyped Behavior; Tritium | 1991 |
The interaction of clozapine with dopamine D1 versus dopamine D2 receptor-mediated function: behavioural indices.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Clozapine; Dopamine; Grooming; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1990 |
Effects of chronic treatment of MPTP monkeys with bromocriptine alone or in combination with SKF 38393.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Antiparkinson Agents; Brain; Brain Chemistry; Bromocriptine; Dopamine; Female; Homovanillic Acid; Kinetics; Levodopa; Macaca fascicularis; Motor Activity; MPTP Poisoning; Parkinson Disease, Secondary; Receptors, Dopamine; Spiperone | 1990 |
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone | 1986 |
Role of D1 and D2 dopamine receptors in mediating locomotor activity elicited from the nucleus accumbens of rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Ketanserin; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Septal Nuclei; Spiperone; Time Factors | 1989 |
The induction of grooming and vacuous chewing by a series of selective D-1 dopamine receptor agonists: two directions of D-1:D-2 interaction.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine Agents; Dose-Response Relationship, Drug; Grooming; Isoquinolines; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior | 1989 |
Selective blockade of dopamine D-1 receptor by SCH 23390 affects dopamine agonist binding to 3H-spiperone labeled D-2 receptors in rat striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; Dopamine; Dopamine Agents; Ergolines; Guanosine Triphosphate; In Vitro Techniques; Male; Pertussis Toxin; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sodium; Spiperone; Virulence Factors, Bordetella | 1989 |
Dihydrexidine, a novel selective high potency full dopamine D-1 receptor agonist.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Binding, Competitive; Corpus Striatum; Dopamine Agents; In Vitro Techniques; Male; Phenanthridines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Spiperone | 1989 |
Differential involvement of dopamine D-1 and D-2 receptors in the circling behaviour induced by apomorphine, SK & F 38393, pergolide and LY 171555 in 6-hydroxydopamine-lesioned rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antiparkinson Agents; Antipsychotic Agents; Apomorphine; Appetite Depressants; Benzazepines; Electric Stimulation; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Sympathectomy, Chemical; Time Factors | 1985 |
Structural determinants of selective affinity for brain D-1 dopamine receptors within a series of 1-phenyl-1H-3-benzazepine analogues of SK&F 38393 and SCH 23390.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Appetite Depressants; Benzazepines; Brain; Corpus Striatum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Thioxanthenes | 1985 |
Postsynaptic dopamine (DA) receptor stimulator properties of the putative DA autoreceptor-selective agonist B-HT 920 uncovered by co-treatment with the D-1 agonist SK&F 38393.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Appetite Depressants; Azepines; Benzazepines; Male; Motor Activity; Rats; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Synapses | 1987 |
The effects of selective dopamine receptor agonists and antagonists on body temperature in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Body Temperature; Ergolines; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1987 |
Excitatory and inhibitory action of dopamine on hippocampal neurons in vitro. Involvement of D2 and D1 receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Culture Techniques; Dopamine; Dopamine Antagonists; Haloperidol; Hippocampus; Male; Neurons; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1987 |
Behavioral and biochemical expression of D1-receptor supersensitivity following SCH 23390 repeated administrations.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Benzazepines; Corpus Striatum; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior | 1988 |
Diminished D2 dopamine receptor function and the emergence of repetitive jaw movements.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Disease Models, Animal; Dopamine Antagonists; Dyskinesia, Drug-Induced; Ergolines; Fluphenazine; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior | 1988 |
EEDQ, a tool for ex vivo measurement of occupancy of D-1 and D-2 dopamine receptors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Salicylamides; Spiperone | 1988 |
Dopaminergic inhibition of tyrosinase activity in hair follicular melanocytes of the mouse.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Benzazepines; Bromocriptine; Catechol Oxidase; Depression, Chemical; Dopamine; Ergolines; Female; Hair; Haloperidol; Male; Melanocytes; Mice; Mice, Inbred C3H; Monophenol Monooxygenase; Quinpirole; Skin; Spiperone; Sulpiride | 1986 |
6-hydroxydopamine treatments enhance behavioral responses to intracerebral microinjection of D1- and D2-dopamine agonists into nucleus accumbens and striatum without changing dopamine antagonist binding.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Corpus Striatum; Dopamine; Dopamine Antagonists; Ergolines; Female; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Microinjections; Motor Activity; Nucleus Accumbens; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Spiperone | 1987 |
Behavioral and biochemical effect of chronic treatment with D-1 and/or D-2 dopamine agonists in MPTP monkeys.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Benzazepines; Brain Chemistry; Dopamine; Dyskinesia, Drug-Induced; Female; Homovanillic Acid; Macaca fascicularis; Motor Activity; Parkinson Disease, Secondary; Pyridines; Receptors, Dopamine; Spiperone | 1988 |
New substituted 1-phenyl-3-benzazepine analogues of SK&F 38393 and N-methyl-thienopyridine analogues of dihydroxynomifensine with selective affinity for the D-1 dopamine receptor in human post-mortem brain.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Benzazepines; Binding, Competitive; Brain Chemistry; Humans; In Vitro Techniques; Kinetics; Ligands; Nomifensine; Putamen; Pyridines; Receptors, Dopamine; Spiperone; Thiophenes | 1987 |
Selective dopamine D2 receptor reduction enhances a D1-mediated oral dyskinesia in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dopamine Antagonists; Jaw; Rats; Rats, Inbred F344; Rats, Inbred Strains; Receptors, Dopamine; Species Specificity; Spiperone; Stereotyped Behavior; Tetrabenazine | 1986 |
Absence of [3H]SCH 23390 specific binding sites in anterior pituitary: dissociation from effects on prolactin secretion.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Corpus Striatum; Cyproheptadine; Ergolines; Kinetics; Male; Metergoline; Pituitary Gland, Anterior; Prolactin; Quinpirole; Rats; Rats, Inbred Strains; Spiperone | 1987 |
Dopamine receptor subtypes: in vivo biochemical evidence for functional interaction.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Corpus Striatum; Dopamine; Homovanillic Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1985 |
Hyperactivity induced by stimulation of separate dopamine D-1 and D-2 receptors in rats with bilateral 6-OHDA lesions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzamides; Benzazepines; Clopenthixol; Dopamine; Dose-Response Relationship, Drug; Ergolines; Flupenthixol; Hydroxydopamines; Hypothalamus; Male; Motor Activity; Oxidopamine; Pergolide; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone | 1985 |
Characterization of dopamine autoreceptor and [3H]spiperone binding sites in vitro with classical and novel dopamine receptor agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Apomorphine; Benzazepines; Binding Sites; Bromocriptine; Butyrophenones; Cats; Caudate Nucleus; Dopamine; Electric Stimulation; Female; In Vitro Techniques; Male; Phentolamine; Receptors, Dopamine; Spiperone; Sulpiride; Tritium | 1983 |
Selective and stereospecific interactions of R-SK & F 38393 with [3H]piflutixol but not [3H]spiperone binding to striatal D1 and D2 dopamine receptors: comparisons with SCH 23390.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Appetite Depressants; Benzazepines; Binding, Competitive; Butyrophenones; Corpus Striatum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism; Thioxanthenes | 1984 |
Induction of oral dyskinesias in naive rats by D1 stimulation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Dyskinesia, Drug-Induced; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1983 |
Identification of the enantiomers of SK&F 83566 as specific and stereoselective antagonists at the striatal D-1 dopamine receptor: comparisons with the D-2 enantioselectivity of Ro 22-1319.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Corpus Striatum; In Vitro Techniques; Isoquinolines; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereoisomerism; Thioxanthenes | 1984 |
Absolute stereochemistry and dopaminergic activity of enantiomers of 2,3,4,5-tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Binding, Competitive; Chemical Phenomena; Chemistry; Dogs; In Vitro Techniques; Male; Molecular Conformation; Rats; Receptors, Dopamine; Renal Circulation; Spiperone; Stereoisomerism; Substantia Nigra; Vasodilator Agents | 1982 |
The D2 dopamine receptor mediates inhibition of growth in GH4ZR7 cells: involvement of protein kinase-C epsilon.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alprenolol; Animals; Apomorphine; Benzazepines; Butaclamol; Carcinogens; Cell Division; Cell Line; DNA; Dopamine; Ergolines; Humans; Isoenzymes; Kinetics; Norepinephrine; Pertussis Toxin; Phorbol Esters; Pituitary Neoplasms; Protein Kinase C; Quinpirole; Receptors, Dopamine D2; Salicylamides; Spiperone; Thymidine; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1994 |
Suppression of natural killer cell activity in mouse spleen lymphocytes by several dopamine receptor antagonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cytotoxicity, Immunologic; Dopamine Antagonists; Flupenthixol; Fluphenazine; Killer Cells, Natural; Mice; Mice, Inbred C3H; Pimozide; Spiperone; Spleen; Thiothixene; Trifluoperazine | 1995 |
Changes in extracellular levels of glutamate and aspartate in rat substantia nigra induced by dopamine receptor ligands: in vivo microdialysis studies.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aspartic Acid; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Extracellular Space; Glutamic Acid; Kinetics; Ligands; Male; Microdialysis; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Spiperone; Substantia Nigra; Tetrodotoxin; Time Factors | 1995 |
Expression of the bovine striatal D2 receptor, but not the D1 receptor, in bovine adrenal medulla.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenal Medulla; Animals; Base Sequence; Benzazepines; Catecholamines; Cattle; Caudate Nucleus; Cell Membrane; Corpus Striatum; Gene Expression; Iodine Radioisotopes; Kinetics; Microsomes; Molecular Sequence Data; Radioligand Assay; Receptors, Dopamine D1; Receptors, Dopamine D2; Sequence Homology, Nucleic Acid; Spiperone; Tritium | 1995 |
Behavioral effects of dopaminergic agonists and antagonists alone and in combination in the squirrel monkey.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Reinforcement Schedule; Saimiri; Spiperone | 1993 |
Ontogenetic quinpirole treatment induces vertical jumping activity in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aging; Animals; Behavior, Animal; Benzazepines; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Injections, Intraperitoneal; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1993 |
D-cycloserine decreases both D1 and D2 dopamine receptors number and their function in rat brain.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Cell Membrane; Cycloserine; Dizocilpine Maleate; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; In Vitro Techniques; Kinetics; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone | 1994 |
An autoradiographic study of the differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on striatal and extrastriatal D-1 and D-2 dopamine receptors in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Densitometry; Dopamine Agonists; Dopamine Antagonists; Ergolines; Male; Neostriatum; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1994 |
Reward summation and the effects of dopamine D1 and D2 agonists and antagonists on fixed-interval responding for brain stimulation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Brain; Bromocriptine; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Drug Interactions; Electric Stimulation; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement Schedule; Reward; Self Stimulation; Spiperone | 1994 |
Effect of chronic haloperidol treatment on dopamine-induced inositol phosphate formation in rat brain slices.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Brain; Corpus Striatum; Dopamine; Dopamine Antagonists; Frontal Lobe; Haloperidol; Hippocampus; In Vitro Techniques; Inositol; Inositol Phosphates; Male; Organ Specificity; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Reference Values; Spiperone | 1994 |
Convergent regulation by ciliary neurotrophic factor and dopamine of tyrosine hydroxylase expression in cultures of rat substantia nigra.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Cells, Cultured; Ciliary Neurotrophic Factor; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Ergolines; Glial Fibrillary Acidic Protein; Haloperidol; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Phosphopyruvate Hydratase; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Proteins; Spiperone; Substantia Nigra; Sulpiride; Time Factors; Tyrosine 3-Monooxygenase | 1993 |
Chronic treatment with MK-801 decreases D2 dopamine receptor function in rat striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Corpus Striatum; Dizocilpine Maleate; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Grooming; In Vitro Techniques; Kinetics; Ligands; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Spiperone | 1993 |
Continuous treatment with the D2 dopamine receptor agonist quinpirole decreases D2 dopamine receptors, D2 dopamine receptor messenger RNA and proenkephalin messenger RNA, and increases mu opioid receptors in mouse striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Behavior, Animal; Blotting, Northern; Corpus Striatum; Dopamine Agents; Dopamine D2 Receptor Antagonists; Down-Regulation; Enkephalins; Ergolines; Image Processing, Computer-Assisted; Male; Mice; Nucleic Acid Hybridization; Oligonucleotide Probes; Protein Precursors; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger; Spiperone; Up-Regulation | 1993 |
Cerebellar and striatal dopamine receptors: effects of reeler and weaver murine mutations.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebellum; Corpus Striatum; Dopamine; Kinetics; Mice; Mice, Neurologic Mutants; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Species Specificity; Spiperone | 1993 |
Pharmacological characterization of behavioural responses to SK&F 83959 in relation to 'D1-like' dopamine receptors not linked to adenylyl cyclase.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Behavior, Animal; Benzamides; Benzazepines; Binding, Competitive; Chromans; Dopamine Agonists; Dopamine Antagonists; Enzyme Induction; Isoquinolines; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Spiperone; Tetrahydroisoquinolines | 1995 |
Existence of dopamine D1 receptor on the sympathetic nerve endings in the guinea-pig vas deferens.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Brimonidine Tartrate; Dopamine Agonists; Dopamine Antagonists; Electric Stimulation; Guinea Pigs; Idazoxan; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Presynaptic Terminals; Quinoxalines; Receptors, Dopamine D1; Spiperone; Synaptic Transmission; Vas Deferens | 1997 |
A sensitive assay for studying dopaminergic activity in cultures of rat pituitary cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Bromocriptine; Cell Count; Cells, Cultured; Cyproheptadine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Evaluation, Preclinical; Female; Haloperidol; Pituitary Gland; Prolactin; Rats; Rats, Wistar; Spiperone | 1997 |
Differential effects of D1 and D2 dopamine-receptor agonists and antagonists on appetitive and consummatory aspects of male sexual behavior in Japanese quail.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Coturnix; Dopamine Agonists; Dopamine Antagonists; Male; Sexual Behavior, Animal; Spiperone | 1997 |
Selective attenuation of the antinociceptive effects of mu opioids by the putative dopamine D3 agonist 7-OH-DPAT.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Opioid; Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cycloparaffins; Dopamine Agonists; Dopamine Antagonists; Drug Antagonism; Male; Morphine; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Spiperone; Tetrahydronaphthalenes | 1999 |
Dopamine receptor antagonists modulate glucose uptake in rat pheochromocytoma (PC12) cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Biological Transport; Chlorpromazine; Clozapine; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fluphenazine; Glucose; Haloperidol; PC12 Cells; Pimozide; Rats; Receptors, Dopamine D2; Spiperone; Sulpiride; Tritium | 1999 |
Supraspinal D2 receptor involved in antinociception induced by l-tetrahydropalmatine.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Non-Narcotic; Animals; Benzazepines; Berberine Alkaloids; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Injections, Spinal; Male; Pain Threshold; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 1999 |
Activity-dependent and use-dependent regulation of dopamine-receptor clustering.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding Sites; Bromocriptine; Dopamine Agonists; Dopamine Antagonists; Microscopy, Confocal; Rats; Rats, Long-Evans; Receptor Aggregation; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone | 2000 |
Effects of dopaminergic agents on carrageenan hyperalgesia in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Carrageenan; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Hindlimb; Hyperalgesia; Injections; Injections, Intraventricular; Male; Pain; Pain Measurement; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Sodium Chloride; Spiperone; Time Factors | 2000 |
Effects of dopaminergic agents on carrageenan hyperalgesia after intrathecal administration to rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Carrageenan; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Hindlimb; Hot Temperature; Hyperalgesia; Injections, Spinal; Male; Pain Measurement; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone | 2001 |
[Differential regulation of dopamine receptors on pre- and postsynaptic Na+, K(+)-ATPase in rat striatum].
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Female; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sodium-Potassium-Exchanging ATPase; Spiperone; Synaptic Membranes | 1997 |
Pharmacological characterization of the D1- and D2-like dopamine receptors from the brain of the leopard frog, Rana pipiens.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Binding, Competitive; Brain; Radioligand Assay; Rana pipiens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Species Specificity; Spiperone; Sulpiride | 2001 |
Biphasic firing response of nucleus accumbens neurons elicited by THPB-18 and its correlation with DA receptor subtypes.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Berberine Alkaloids; Dopamine D2 Receptor Antagonists; Male; Neurons; Nucleus Accumbens; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Ventral Tegmental Area | 2004 |
Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acyltransferases; Animals; Benzazepines; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Melatonin; Phosphorylation; Pineal Gland; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Transcription, Genetic | 2005 |
Effects of dopamine D1-like receptor agonists on food-maintained operant behavior in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Drug Synergism; Food; Male; Metergoline; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reinforcement Schedule; Reward; Spiperone | 2006 |
Chronic SKF83959 induced less severe dyskinesia and attenuated L-DOPA-induced dyskinesia in 6-OHDA-lesioned rat model of Parkinson's disease.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Drug Administration Schedule; Drug Interactions; Dyskinesia, Drug-Induced; Levodopa; Male; Movement; Oxidopamine; Parkinson Disease; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Spiperone; Sympatholytics; Time Factors | 2007 |
Dopamine receptors in the anterior insular cortex modulate long-term nociception in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Afferent Pathways; Animals; Apomorphine; Benzazepines; Cerebral Cortex; Chronic Disease; Dopamine; Dopamine Agonists; Dopamine Antagonists; Hot Temperature; Male; Microinjections; Models, Neurological; Neuralgia; Nociceptors; Pain; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Sciatic Neuropathy; Self Mutilation; Spiperone | 2008 |
Identification of dopamine receptor in Tetrahymena thermophila by fluorescent ligands.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Fluorescent Dyes; Ligands; Microscopy, Confocal; Microscopy, Fluorescence; Protozoan Proteins; Receptors, Dopamine D1; Rhodamines; Spiperone; Tetrahymena thermophila | 2012 |
Dopamine D1 receptor modulation of calcium channel currents in horizontal cells of mouse retina.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Biophysical Phenomena; Calcium; Calcium Channel Blockers; Calcium Channels; Connexins; Dopamine; Dopamine Agonists; Dopamine Antagonists; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; omega-Conotoxin GVIA; Plant Lectins; Receptors, Dopamine D1; Retina; Retinal Horizontal Cells; RNA, Untranslated; Spiperone | 2016 |
Fluorescent probes for dopamine receptors: synthesis and characterization of fluorescein and 7-nitrobenz-2-oxa-1,3-diazol-4-yl conjugates of D-1 and D-2 receptor ligands.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Dopamine Antagonists; Fluorescent Dyes; Ligands; Macaca fascicularis; Oxadiazoles; Receptors, Dopamine; Stereoisomerism; Structure-Activity Relationship | 1991 |
Synthesis, evaluation, and comparative molecular field analysis of 1-phenyl-3-amino-1,2,3,4-tetrahydronaphthalenes as ligands for histamine H(1) receptors.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ligands; Models, Molecular; Pyrilamine; Radioligand Assay; Structure-Activity Relationship; Tetrahydronaphthalenes | 1999 |