sk&f-38393 and clozapine

sk&f-38393 has been researched along with clozapine in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19906 (24.00)18.7374
1990's13 (52.00)18.2507
2000's4 (16.00)29.6817
2010's2 (8.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
George, SR; Guan, HC; Laurier, LG; Ng, G; Niznik, HB; O'Dowd, BF; Seeman, P; Sunahara, RK; Torchia, J; Van Tol, HH1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Artz, MT; Cools, AR; Ellenbroek, BA1
Bakhtiar, R; Bull, DR; Sheehan, MJ1
Altar, CA; Jiang, LH; Kasser, RJ; Wang, RY1
Murray, AM; Waddington, JL1
Breese, GA; Criswell, HE; Mueller, RA1
Adamovage, LA; Kreamer, LD; Salama, AI; Saller, CF1
Ashby, CR; Hitzemann, R; Rubinstein, JE; Wang, RY1
Matsubara, S; Meltzer, HY1
Hu, XT; Wang, RY1
Fenton, HM; Gerhardt, S; Leszczak, E; Liebman, JM1
Bengtsson, A; Jackson, DM; Malmberg, A; Mohell, N1
Chen, JF; Weiss, B1
Fici, GJ; Sethy, VH; VonVoigtlander, PF; Wu, H1
Wirtshafter, D1
Kulkarni, SK; Ninan, I1
Jackson, DM; Liao, Y; Wikström, H1
Bradley, RJ; Dwyer, DS; Liu, Y1
Adachi, K; Cools, AR; Hasegawa, M; Hirose, N; Ikeda, H; Koshikawa, N; Sato, M1
Cory-Slechta, DA; Zuch, CL1
Kaur, G; Kulkarni, SK1
Bekker, A; Chen, X; Fan, Q; Fu, R; Li, J; Mei, Q; Shiwalkar, N; Ye, JH; Zuo, W1
Bandyopadhyaya, A; Rajagopalan, DR; Rajagopalan, P; Rajagopalan, R1

Other Studies

25 other study(ies) available for sk&f-38393 and clozapine

ArticleYear
Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1.
    Nature, 1991, Apr-18, Volume: 350, Issue:6319

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain; Cell Line; Cell Membrane; Cloning, Molecular; Dopamine; Humans; Kinetics; Molecular Sequence Data; Molecular Weight; Oligonucleotide Probes; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D5; RNA, Messenger; Sequence Homology, Nucleic Acid; Transfection

1991
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
The involvement of dopamine D1 and D2 receptors in the effects of the classical neuroleptic haloperidol and the atypical neuroleptic clozapine.
    European journal of pharmacology, 1991, Apr-10, Volume: 196, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Clozapine; Dopamine Agents; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine

1991
Characterization of dopamine autoreceptors in the amygdala: a fast cyclic voltammetric study in vitro.
    Neuroscience letters, 1991, Dec-16, Volume: 134, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; Amygdala; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Dopamine; Electric Stimulation; Ergolines; Male; Metoclopramide; Neurotransmitter Uptake Inhibitors; Nialamide; Piperazines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Secretory Rate; Sulpiride

1991
One year of continuous treatment with haloperidol or clozapine fails to induce a hypersensitive response of caudate putamen neurons to dopamine D1 and D2 receptor agonists.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Administration, Oral; Animals; Clozapine; Dibenzazepines; Dopamine Agents; Drug Interactions; Ergolines; Haloperidol; Male; Neurons; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine

1990
The interaction of clozapine with dopamine D1 versus dopamine D2 receptor-mediated function: behavioural indices.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Benzazepines; Clozapine; Dopamine; Grooming; Male; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1990
Clozapine antagonism of D-1 and D-2 dopamine receptor-mediated behaviors.
    European journal of pharmacology, 1989, Jan-10, Volume: 159, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Appetite Depressants; Behavior, Animal; Benzazepines; Clozapine; Dibenzazepines; Ergolines; Female; Hydroxydopamines; Motor Activity; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Serotonin

1989
Dopamine receptor occupancy in vivo: measurement using N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ).
    Life sciences, 1989, Volume: 45, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Clozapine; Corpus Striatum; Ergolines; Haloperidol; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1989
One year treatment with haloperidol or clozapine fails to alter neostriatal D1- and D2-dopamine receptor sensitivity in the rat.
    Brain research, 1989, Jul-24, Volume: 493, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Colforsin; Corpus Striatum; Cyclic AMP; Dibenzazepines; Drug Synergism; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1989
Effect of typical and atypical antipsychotic drugs on 5-HT2 receptor density in rat cerebral cortex.
    Life sciences, 1989, Volume: 45, Issue:15

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Butyrophenones; Cerebral Cortex; Chlorpromazine; Clozapine; Dibenzazepines; Dibenzothiazepines; Down-Regulation; Flupenthixol; Kinetics; Loxapine; Male; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiro Compounds; Time Factors

1989
Haloperidol and clozapine: differential effects on the sensitivity of caudate-putamen neurons to dopamine agonists and cholecystokinin following one month continuous treatment.
    Brain research, 1989, May-08, Volume: 486, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Benzazepines; Cholecystokinin; Clozapine; Corpus Striatum; Dibenzazepines; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sincalide

1989
Evidence for heterogeneous rotational responsiveness to apomorphine, 3-PPP and SKF 38393 in 6-hydroxydopamine-denervated rats.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Clozapine; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Piperidines; Postural Balance; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sympathectomy, Chemical

1984
Why does clozapine stimulate the motor activity of reserpine-pretreated rats when combined with a dopamine D1 receptor agonist?
    European journal of pharmacology, 1995, Aug-25, Volume: 282, Issue:1-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Antipsychotic Agents; Clozapine; Dopamine Antagonists; Drug Therapy, Combination; Enzyme Inhibitors; Ergolines; Male; Methyltyrosines; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reserpine; Stimulation, Chemical; Tyrosine 3-Monooxygenase

1995
Irreversible blockade of D2 dopamine receptors by fluphenazine-N-mustard increases glutamic acid decarboxylase mRNA in rat striatum.
    Neuroscience letters, 1993, Feb-19, Volume: 150, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Base Sequence; Blotting, Northern; Clozapine; Corpus Striatum; Depression, Chemical; Dopamine D2 Receptor Antagonists; Fluphenazine; Glutamate Decarboxylase; Haloperidol; In Vitro Techniques; Male; Molecular Sequence Data; Oligodeoxyribonucleotides; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; RNA Probes; RNA, Messenger

1993
D1 dopamine receptor activity of anti-parkinsonian drugs.
    Life sciences, 1997, Volume: 60, Issue:18

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antiparkinson Agents; Apomorphine; Benzazepines; Benzothiazoles; Bromocriptine; Cells, Cultured; Cerebellum; Clozapine; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Pergolide; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Tetrahydronaphthalenes; Thiazoles

1997
D1 dopamine receptors mediate neuroleptic-induced Fos expression in the islands of Calleja.
    Synapse (New York, N.Y.), 1998, Volume: 28, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adamantane; Animals; Antiparkinson Agents; Antipsychotic Agents; Benzazepines; Benzopyrans; Clozapine; Dopamine Agonists; Male; Olfactory Pathways; Proto-Oncogene Proteins c-fos; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Salicylamides

1998
Partial agonistic action of clozapine at dopamine D2 receptors in dopamine depleted animals.
    Psychopharmacology, 1998, Volume: 135, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Antipsychotic Agents; Central Nervous System Depressants; Clozapine; Dopamine; Dopamine Agonists; Enzyme Inhibitors; Mice; Motor Activity; Receptors, Dopamine D2; Reserpine; Stereotyped Behavior; Tyrosine 3-Monooxygenase

1998
Is clozapine an (partial) agonist at both dopamine D1 and D2 receptors?
    Psychopharmacology, 1998, Volume: 138, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Body Temperature; Clozapine; Dopamine Agonists; Muscarinic Antagonists; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2

1998
Dopamine receptor antagonists modulate glucose uptake in rat pheochromocytoma (PC12) cells.
    Neuroscience letters, 1999, Oct-29, Volume: 274, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Biological Transport; Chlorpromazine; Clozapine; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Antagonists; Fluphenazine; Glucose; Haloperidol; PC12 Cells; Pimozide; Rats; Receptors, Dopamine D2; Spiperone; Sulpiride; Tritium

1999
Effects of chronic haloperidol and clozapine on vacuous chewing and dopamine-mediated jaw movements in rats: evaluation of a revised animal model of tardive dyskinesia.
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:11-12

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Clozapine; Disease Models, Animal; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dyskinesia, Drug-Induced; Haloperidol; Jaw; Male; Mastication; Quinpirole; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Serotonin Antagonists

1999
Stimulus properties of 7-OH-DPAT versus auto- and postsynaptic receptor-specific doses of quinpirole.
    Pharmacology, biochemistry, and behavior, 2001, Volume: 68, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Clozapine; Dopamine Antagonists; Female; Haloperidol; Maternal Behavior; Motivation; Motor Activity; Pimozide; Rats

2001
Studies on modulation of feeding behavior by atypical antipsychotics in female mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2002, Volume: 26, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adipose Tissue; Animals; Antipsychotic Agents; Body Weight; Clozapine; Eating; Feeding Behavior; Female; Fluoxetine; Hyperphagia; Mice; Mice, Inbred Strains; Organ Size; Quinpirole; Quipazine; Selective Serotonin Reuptake Inhibitors; Weight Gain

2002
Alcohol withdrawal drives depressive behaviors by activating neurons in the rostromedial tegmental nucleus.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2019, Volume: 44, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Clozapine; Dopaminergic Neurons; Ethanol; gamma-Aminobutyric Acid; Male; Microinjections; Neural Inhibition; Neural Pathways; Nucleus Accumbens; Proto-Oncogene Proteins c-fos; Quinoxalines; Quinpirole; Rats; Substance Withdrawal Syndrome; Tegmentum Mesencephali; Ventral Tegmental Area

2019
The synthesis and comparative receptor binding affinities of novel, isomeric pyridoindolobenzazepine scaffolds.
    Bioorganic & medicinal chemistry letters, 2014, Jan-15, Volume: 24, Issue:2

    Topics: Benzodiazepinones; Isomerism; Protein Binding; Protein Structure, Tertiary; Receptors, Cell Surface

2014