Page last updated: 2024-09-03

sk&f 104856 and bmy 7378

sk&f 104856 has been researched along with bmy 7378 in 3 studies

Compound Research Comparison

Studies
(sk&f 104856)
Trials
(sk&f 104856)
Recent Studies (post-2010)
(sk&f 104856)
Studies
(bmy 7378)
Trials
(bmy 7378)
Recent Studies (post-2010) (bmy 7378)
140039013
1400225025

Protein Interaction Comparison

ProteinTaxonomysk&f 104856 (IC50)bmy 7378 (IC50)
DRattus norvegicus (Norway rat)0.091
D(3) dopamine receptorRattus norvegicus (Norway rat)0.091
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.091
D(4) dopamine receptorRattus norvegicus (Norway rat)0.091
D(2) dopamine receptorRattus norvegicus (Norway rat)0.091

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Botta, M; Cagnotto, A; Manetti, F; Materia, L; Mennini, T; Minneman, KP; Nicoletti, F; Romeo, G; Russo, F1
Pedretti, A; Testa, B; Villa, L; Vistoli, G1
Ballard, S; Blagg, J; Fox, D; Kenny, B1

Reviews

1 review(s) available for sk&f 104856 and bmy 7378

ArticleYear
Pharmacological options in the treatment of benign prostatic hyperplasia.
    Journal of medicinal chemistry, 1997, Apr-25, Volume: 40, Issue:9

    Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Controlled Clinical Trials as Topic; Endothelins; Enzyme Inhibitors; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Adrenergic, alpha; Structure-Activity Relationship

1997

Other Studies

2 other study(ies) available for sk&f 104856 and bmy 7378

ArticleYear
New pyrimido[5,4-b]indoles as ligands for alpha(1)-adrenoceptor subtypes.
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Adrenergic alpha-Antagonists; Animals; Cell Line; Computer Simulation; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quantitative Structure-Activity Relationship; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Structure-Activity Relationship

2003
Range and sensitivity as descriptors of molecular property spaces in dynamic QSAR analyses.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Chemical Phenomena; Chemistry, Physical; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Receptors, Adrenergic, alpha-1; Solvents

2005