Page last updated: 2024-09-03

sk&f 104078 and doxazosin

sk&f 104078 has been researched along with doxazosin in 3 studies

Compound Research Comparison

Studies
(sk&f 104078)
Trials
(sk&f 104078)
Recent Studies (post-2010)
(sk&f 104078)
Studies
(doxazosin)
Trials
(doxazosin)
Recent Studies (post-2010) (doxazosin)
29001,372439283

Protein Interaction Comparison

ProteinTaxonomysk&f 104078 (IC50)doxazosin (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.544
Interstitial collagenaseHomo sapiens (human)5.749
Beta-2 adrenergic receptorHomo sapiens (human)2.748
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)2.2155
Alpha-1D adrenergic receptorHomo sapiens (human)0.0034
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.544
Sodium-dependent serotonin transporterHomo sapiens (human)2.688
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.368
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0007
Sodium-dependent dopamine transporter Homo sapiens (human)0.188
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.4022
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)2.2155

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bondinell, WE; Hieble, JP; Ruffolo, RR1
Birkeland, S; Grong, K; Lekven, J; Westby, J1
Grong, K; Hexeberg, E; Lekven, J; Myking, OL; Olweus, J; Westby, J1

Reviews

1 review(s) available for sk&f 104078 and doxazosin

ArticleYear
Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Animals; Humans; Molecular Biology; Molecular Structure; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1995

Other Studies

2 other study(ies) available for sk&f 104078 and doxazosin

ArticleYear
Transmural heterogeneity of postjunctional alpha 2 adrenergic coronary vasoconstriction in hypoperfused cat left ventricle.
    Cardiovascular research, 1992, Volume: 26, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Cats; Coronary Disease; Coronary Vessels; Doxazosin; Male; Regional Blood Flow; Vascular Resistance; Vasoconstriction

1992
Blood flow regulation during acute regional ischemia in feline hearts: importance of postjunctional alpha 1- and alpha 2-adrenoceptors.
    Journal of cardiovascular pharmacology, 1991, Volume: 18, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Catecholamines; Cats; Coronary Circulation; Coronary Disease; Doxazosin; Heart; Male; Myocardium; Oxygen Consumption; Perfusion; Prazosin; Receptors, Adrenergic, alpha; Vascular Resistance

1991