Page last updated: 2024-09-03

sk&f 104078 and 8-hydroxy-2-(di-n-propylamino)tetralin

sk&f 104078 has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 1 studies

Compound Research Comparison

Studies
(sk&f 104078)
Trials
(sk&f 104078)
Recent Studies (post-2010)
(sk&f 104078)
Studies
(8-hydroxy-2-(di-n-propylamino)tetralin)
Trials
(8-hydroxy-2-(di-n-propylamino)tetralin)
Recent Studies (post-2010) (8-hydroxy-2-(di-n-propylamino)tetralin)
29003,5307389

Protein Interaction Comparison

ProteinTaxonomysk&f 104078 (IC50)8-hydroxy-2-(di-n-propylamino)tetralin (IC50)
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.0012
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0032
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.81
D(2) dopamine receptorBos taurus (cattle)0.8
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.81
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.81
D(2) dopamine receptorRattus norvegicus (Norway rat)2.8959
Lysosomal alpha-glucosidaseBos taurus (cattle)0.0021

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19901 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brown, CM; Kilpatrick, AT; MacKinnon, AC; Spedding, M1

Other Studies

1 other study(ies) available for sk&f 104078 and 8-hydroxy-2-(di-n-propylamino)tetralin

ArticleYear
The alpha 2-adrenoceptor antagonist SK&F 104078 has high affinity for 5-HT1A and 5-HT2 receptors.
    European journal of pharmacology, 1989, Jul-18, Volume: 166, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Benzazepines; Binding, Competitive; Cerebral Cortex; In Vitro Techniques; Ketanserin; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Tetrahydronaphthalenes

1989