sk&f 100330-a has been researched along with tiagabine in 2 studies
| Studies (sk&f 100330-a) | Trials (sk&f 100330-a) | Recent Studies (post-2010) (sk&f 100330-a) | Studies (tiagabine) | Trials (tiagabine) | Recent Studies (post-2010) (tiagabine) |
|---|---|---|---|---|---|
| 20 | 0 | 0 | 571 | 102 | 111 |
| Protein | Taxonomy | sk&f 100330-a (IC50) | tiagabine (IC50) |
|---|---|---|---|
| Sodium- and chloride-dependent GABA transporter 1 | Rattus norvegicus (Norway rat) | 2.2107 | |
| Sodium- and chloride-dependent GABA transporter 1 | Homo sapiens (human) | 0.2213 | |
| Sodium- and chloride-dependent GABA transporter 1 | Mus musculus (house mouse) | 0.1968 | |
| Sodium- and chloride-dependent betaine transporter | Mus musculus (house mouse) | 0.27 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 1 (50.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 1 (50.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Faust, MR; Höfner, G; Pabel, J; Wanner, KT | 1 |
| Andersen, KE; Braestrup, C; Knutsen, LJ; Nielsen, EB; Sonnewald, U; Suzdak, PD | 1 |
2 other study(ies) available for sk&f 100330-a and tiagabine
| Article | Year |
|---|---|
Azetidine derivatives as novel gamma-aminobutyric acid uptake inhibitors: synthesis, biological evaluation, and structure-activity relationship.
Topics: Animals; Azetidines; Biological Transport; Cattle; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; Inhibitory Concentration 50; Structure-Activity Relationship | 2010 |
Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor.
Topics: Animals; Anticonvulsants; Carbolines; Clonazepam; Convulsants; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred DBA; Neurotransmitter Uptake Inhibitors; Nicotinic Acids; Nipecotic Acids; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures; Tiagabine | 1991 |