sk&f 100330-a has been researched along with gamma-aminobutyric acid in 15 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Studies (sk&f 100330-a) | Trials (sk&f 100330-a) | Recent Studies (post-2010) (sk&f 100330-a) | Studies (gamma-aminobutyric acid) | Trials (gamma-aminobutyric acid) | Recent Studies (post-2010) (gamma-aminobutyric acid) |
---|---|---|---|---|---|
20 | 0 | 0 | 40,215 | 1,423 | 9,631 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 9 (60.00) | 18.7374 |
1990's | 5 (33.33) | 18.2507 |
2000's | 1 (6.67) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ali, FE; Bondinell, WE; Dandridge, PA; Frazee, JS; Garvey, E; Girard, GR; Kaiser, C; Ku, TW; Lafferty, JJ; Moonsammy, GI | 1 |
Agmo, A; Gutiérrez, M; Guzmán, M; Pruneda, R | 1 |
Enna, SJ; Ferkany, JW; Karbon, EW | 1 |
Andersen, KE; Braestrup, C; Knutsen, LJ; Nielsen, EB; Sonnewald, U; Suzdak, PD | 1 |
Falch, E; Krogsgaard-Larsen, P | 1 |
Falch, E; Krogsgaard-Larsen, P; Larsson, OM; Schousboe, A | 1 |
Bonanno, G; Raiteri, M | 2 |
Bennett, JP; Cruz, CJ; Ferrari, MB | 1 |
Löscher, W | 1 |
Löscher, W; Schwark, WS | 1 |
Enna, SJ; Zorn, SH | 1 |
Agmo, A; Soria, P | 1 |
Golovanevsky, V; Kanner, BI | 1 |
Bonanno, G; Raiteri, L; Raiteri, M; Stigliani, S; Zedda, L | 1 |
15 other study(ies) available for sk&f 100330-a and gamma-aminobutyric acid
Article | Year |
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Orally active and potent inhibitors of gamma-aminobutyric acid uptake.
Topics: 4-Aminobutyrate Transaminase; Administration, Oral; Alkylation; Amino Acids; Animals; Brain; Carboxylic Acids; gamma-Aminobutyric Acid; Glutamate Decarboxylase; In Vitro Techniques; Male; Neurotransmitter Uptake Inhibitors; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Stereoisomerism; Synaptosomes | 1985 |
GABAergic drugs and conflict behavior in the rat: lack of similarities with the actions of benzodiazepines.
Topics: Alkynes; Aminocaproates; Animals; Baclofen; Behavior, Animal; Benzodiazepines; Bicuculline; Brain; Conflict, Psychological; Drug Interactions; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Nicotinic Acids; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission | 1991 |
Biochemical and behavioral studies following subchronic administration of GABA uptake inhibitors in mice.
Topics: Animals; Anticonvulsants; Catalepsy; Epilepsy, Tonic-Clonic; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; Molecular Structure; Nicotinic Acids; Nipecotic Acids; Pentylenetetrazole; Receptors, Dopamine; Receptors, GABA-A; Time Factors | 1991 |
Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor.
Topics: Animals; Anticonvulsants; Carbolines; Clonazepam; Convulsants; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred DBA; Neurotransmitter Uptake Inhibitors; Nicotinic Acids; Nipecotic Acids; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures; Tiagabine | 1991 |
GABA uptake inhibitors containing mono- and diarylmethoxyalkyl N-substituents.
Topics: Anticonvulsants; gamma-Aminobutyric Acid; Neurotransmitter Uptake Inhibitors; Nicotinic Acids; Nipecotic Acids; Structure-Activity Relationship; Synaptosomes | 1989 |
Kinetic characterization of inhibition of gamma-aminobutyric acid uptake into cultured neurons and astrocytes by 4,4-diphenyl-3-butenyl derivatives of nipecotic acid and guvacine.
Topics: Animals; Anticonvulsants; Astrocytes; Cells, Cultured; Cerebral Cortex; Chemical Phenomena; Chemistry; GABA Antagonists; gamma-Aminobutyric Acid; Mice; Mice, Inbred Strains; Neurons; Nicotinic Acids; Nipecotic Acids; Proline | 1988 |
Coexistence of carriers for dopamine and GABA uptake on a same nerve terminal in the rat brain.
Topics: Aminobutyrates; Animals; Anticonvulsants; Brain Chemistry; Dopamine; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Nerve Endings; Nicotinic Acids; Nipecotic Acids; Norepinephrine; Rats; Rats, Inbred Strains; Serotonin; Synaptosomes | 1987 |
Presence of a gamma-aminobutyric acid (GABA) uptake system on cholinergic terminals of rat hippocampus: evidence for neuronal coexistence of acetylcholine and GABA?
Topics: Acetylcholine; Animals; Choline; Cholinergic Fibers; gamma-Aminobutyric Acid; Hemicholinium 3; Hippocampus; Male; Neurons; Nicotinic Acids; Nipecotic Acids; Rats; Rats, Inbred Strains | 1987 |
GABA-mimetic drugs enhance apomorphine-induced contralateral turning in rats with unilateral nigrostriatal dopamine denervation: implications for the therapy of Parkinson's disease.
Topics: Alkynes; Aminocaproates; Animals; Antiparkinson Agents; Apomorphine; Drug Synergism; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Nicotinic Acids; Parkinson Disease; Rats; Rats, Inbred Strains | 1987 |
Anticonvulsant action in the epileptic gerbil of novel inhibitors of GABA uptake.
Topics: Animals; Anticonvulsants; Depression, Chemical; Epilepsy; Female; gamma-Aminobutyric Acid; Gerbillinae; Male; Nicotinic Acids; Nipecotic Acids | 1985 |
Comparison of the anticonvulsant effects of two novel GABA uptake inhibitors and diazepam in amygdaloid kindled rats.
Topics: Amygdala; Animals; Anticonvulsants; Diazepam; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Kindling, Neurologic; Nicotinic Acids; Nipecotic Acids; Rats; Rats, Inbred Strains; Seizures | 1985 |
GABA uptake inhibitors produce a greater antinociceptive response in the mouse tail-immersion assay than other types of GABAergic drugs.
Topics: Analgesics; Animals; Biological Transport; Brain; Corpus Striatum; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Nicotinic Acids; Nipecotic Acids; Oxotremorine; Pain; Tail | 1985 |
GABAergic drugs and sexual motivation, receptivity and exploratory behaviors in the female rat.
Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Exploratory Behavior; Female; gamma-Aminobutyric Acid; Male; Nicotinic Acids; Rats; Rats, Wistar; Sexual Behavior, Animal | 1997 |
The reactivity of the gamma-aminobutyric acid transporter GAT-1 toward sulfhydryl reagents is conformationally sensitive. Identification of a major target residue.
Topics: Carrier Proteins; Ethyl Methanesulfonate; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; HeLa Cells; Humans; Membrane Proteins; Membrane Transport Proteins; Mutagenesis, Site-Directed; Nicotinic Acids; Organic Anion Transporters; Protein Structure, Secondary; Sulfhydryl Reagents | 1999 |
Multiple mechanisms of transmitter release evoked by "pathologically" elevated extracellular [K+]: involvement of transporter reversal and mitochondrial calcium.
Topics: Animals; Anticonvulsants; Brain Chemistry; Calcium; Carrier Proteins; Cerebral Cortex; Chelating Agents; Clonazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Exocytosis; Extracellular Space; Fluorescent Dyes; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Male; Membrane Proteins; Membrane Transport Proteins; Nicotinic Acids; Organic Anion Transporters; Potassium Chloride; Rats; Rats, Sprague-Dawley; Sodium-Calcium Exchanger; Synaptosomes; Thiazepines; Tritium | 2002 |