Page last updated: 2024-09-04

sk&f 100330-a and clonazepam

sk&f 100330-a has been researched along with clonazepam in 2 studies

Compound Research Comparison

Studies
(sk&f 100330-a)
Trials
(sk&f 100330-a)
Recent Studies (post-2010)
(sk&f 100330-a)
Studies
(clonazepam)
Trials
(clonazepam)
Recent Studies (post-2010) (clonazepam)
20002,719239519

Protein Interaction Comparison

ProteinTaxonomysk&f 100330-a (IC50)clonazepam (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0017
GABA theta subunitRattus norvegicus (Norway rat)0.0017
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0017

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andersen, KE; Braestrup, C; Knutsen, LJ; Nielsen, EB; Sonnewald, U; Suzdak, PD1
Bonanno, G; Raiteri, L; Raiteri, M; Stigliani, S; Zedda, L1

Other Studies

2 other study(ies) available for sk&f 100330-a and clonazepam

ArticleYear
Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor.
    European journal of pharmacology, 1991, Apr-24, Volume: 196, Issue:3

    Topics: Animals; Anticonvulsants; Carbolines; Clonazepam; Convulsants; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred DBA; Neurotransmitter Uptake Inhibitors; Nicotinic Acids; Nipecotic Acids; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures; Tiagabine

1991
Multiple mechanisms of transmitter release evoked by "pathologically" elevated extracellular [K+]: involvement of transporter reversal and mitochondrial calcium.
    Journal of neurochemistry, 2002, Volume: 80, Issue:4

    Topics: Animals; Anticonvulsants; Brain Chemistry; Calcium; Carrier Proteins; Cerebral Cortex; Chelating Agents; Clonazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Exocytosis; Extracellular Space; Fluorescent Dyes; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Male; Membrane Proteins; Membrane Transport Proteins; Nicotinic Acids; Organic Anion Transporters; Potassium Chloride; Rats; Rats, Sprague-Dawley; Sodium-Calcium Exchanger; Synaptosomes; Thiazepines; Tritium

2002