Page last updated: 2024-08-25

siguazodan and rolipram

siguazodan has been researched along with rolipram in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's16 (72.73)18.2507
2000's6 (27.27)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Hassall, GA; Parrott, DP; Souness, JE1
Conanan, ND; Ellis, JL1
Chen, J; Meeker, SN; Undem, BJ1
Lamb, J; Murray, KJ; Turner, NC; Worby, A1
Coates, WJ; Dolan, JS; Grimsditch, D; Lamb, J; Murray, KJ; Turner, NC; Warrington, BH; Worby, A1
Bochnowicz, S; Hay, DW; Kotzer, CJ; Luttmann, MA; Osborn, RR; Torphy, TJ; Underwood, DC1
Advenier, C; Girard, V; Martin, CA; Molimard, M; Qian, Y1
Advenier, C; Karlsson, JA; Naline, E; Qian, Y; Raeburn, D1
Karlsson, JA; Raeburn, D; Tomkinson, A1
Furman, BL; Pyne, NJ; Shafiee-Nick, R1
Banner, KH; Bertin, B; Moodley, I; Page, CP1
Dahl, SG; Lagente, V; Payne, AN; Planquois, JM; Ruffin-Morin, Y2
Essayan, DM; Huang, SK; Kagey-Sobotka, A; Lichtenstein, LM1
Dahl, R; Nielsen-Kudsk, F; Thirstrup, S1
Braun, U; Kaasik, A; Minajeva, A; Ohisalo, JJ; Paju, K; Seppet, EK; Vetter, R1
Landells, LJ; O'Connor, BJ; Page, CP; Souness, JE; Spina, D1
De Witt, BJ; Kadowitz, PJ; Marrone, JR1
Cunningham, FM; Lees, P; Page, CP; Rickards, KJ1
Delgado, M; Fernandez-Alfonso, MS; Fuentes, JA1
Kam, MF; Lau, HY1

Other Studies

22 other study(ies) available for siguazodan and rolipram

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Inhibition of pig aortic smooth muscle cell DNA synthesis by selective type III and type IV cyclic AMP phosphodiesterase inhibitors.
    Biochemical pharmacology, 1992, Sep-01, Volume: 44, Issue:5

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Aorta; Cell Division; Colforsin; Cyclic AMP; DNA Replication; Guanidines; Isoenzymes; Isoquinolines; Muscle, Smooth, Vascular; Pyridazines; Pyrrolidinones; Rolipram; Swine; Tetrahydroisoquinolines; Thymidine

1992
Modulation of relaxant responses evoked by a nitric oxide donor and by nonadrenergic, noncholinergic stimulation by isozyme-selective phosphodiesterase inhibitors in guinea pig trachea.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 272, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Atropine; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Electric Stimulation; Guanidines; Guinea Pigs; Indomethacin; Isoenzymes; Muscle Relaxation; Nitric Oxide; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Propranolol; Purinones; Pyridazines; Pyrrolidinones; Receptors, Adrenergic; Receptors, Cholinergic; Rolipram; Trachea; Vasoactive Intestinal Peptide; Xanthines

1995
Inhibition of neurally mediated nonadrenergic, noncholinergic contractions of guinea pig bronchus by isozyme-selective phosphodiesterase inhibitors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:2

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Bronchi; Bronchoconstriction; Electric Stimulation; Guanidines; Guinea Pigs; Isoenzymes; Male; Phosphodiesterase Inhibitors; Purinones; Pyridazines; Pyrrolidinones; Rolipram; Vagus Nerve

1994
Relaxation of guinea-pig trachea by cyclic AMP phosphodiesterase inhibitors and their enhancement by sodium nitroprusside.
    British journal of pharmacology, 1994, Volume: 111, Issue:4

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Nitroprusside; Phosphodiesterase Inhibitors; Pyridazines; Pyrrolidinones; Rolipram; Trachea

1994
Pulmonary effects of type V cyclic GMP specific phosphodiesterase inhibition in the anaesthetized guinea-pig.
    British journal of pharmacology, 1994, Volume: 111, Issue:4

    Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Anesthesia; Animals; Bronchoconstriction; Cyclic GMP; Guanidines; Guinea Pigs; Male; Nitroprusside; Parasympatholytics; Phosphodiesterase Inhibitors; Purinones; Pyridazines; Pyrrolidinones; Rolipram; Trachea

1994
Comparison of phosphodiesterase III, IV and dual III/IV inhibitors on bronchospasm and pulmonary eosinophil influx in guinea pigs.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:1

    Topics: Animals; Antigens; Bronchial Spasm; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Drug Synergism; Eosinophils; Guanidines; Guinea Pigs; Histamine Antagonists; In Vitro Techniques; Isoenzymes; Leukotriene D4; Male; Phosphodiesterase Inhibitors; Plethysmography, Whole Body; Pulmonary Eosinophilia; Pyridazines; Pyrrolidinones; Rolipram; Trachea

1994
Rolipram, but not siguazodan or zaprinast, inhibits the excitatory noncholinergic neurotransmission in guinea-pig bronchi.
    The European respiratory journal, 1994, Volume: 7, Issue:2

    Topics: Animals; Bronchi; Electric Stimulation; Female; Guanidines; Guinea Pigs; In Vitro Techniques; Male; Nerve Fibers; Phosphodiesterase Inhibitors; Purinones; Pyridazines; Pyrrolidinones; Rolipram; Synaptic Transmission

1994
Effects of rolipram and siguazodan on the human isolated bronchus and their interaction with isoprenaline and sodium nitroprusside.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: Albuterol; Bronchi; Guanidines; Humans; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Nitroprusside; Phosphodiesterase Inhibitors; Pyridazines; Pyrrolidinones; Rolipram

1993
Comparison of the effects of selective inhibitors of phosphodiesterase types III and IV in airway smooth muscle with differing beta-adrenoceptor subtypes.
    British journal of pharmacology, 1993, Volume: 108, Issue:1

    Topics: Albuterol; Animals; Bronchi; Cattle; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Methacholine Chloride; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phosphodiesterase Inhibitors; Pyridazines; Pyrrolidinones; Rolipram; Trachea

1993
Effects of type-selective phosphodiesterase inhibitors on glucose-induced insulin secretion and islet phosphodiesterase activity.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Analysis of Variance; Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Glucose; Guanidines; Insulin; Insulin Secretion; Islets of Langerhans; Isoenzymes; Male; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Purinones; Pyrazines; Pyridazines; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Rolipram; Thiophenes

1995
Effect of isoenzyme selective phosphodiesterase inhibitors on the proliferation of murine thymus and spleen cells.
    Pulmonary pharmacology, 1996, Volume: 9, Issue:1

    Topics: Animals; Cell Division; Female; Guanidines; Lymphocyte Activation; Mice; Phosphodiesterase Inhibitors; Pyridazines; Pyrrolidinones; Rolipram; Spleen; Thymus Gland

1996
Salbutamol potentiates the relaxant effects of selective phosphodiesterase inhibitors on guinea pig isolated trachea.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adrenergic beta-Agonists; Albuterol; Animals; Drug Synergism; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Male; Milrinone; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Osmolar Concentration; Phosphodiesterase Inhibitors; Purinones; Pyridazines; Pyridones; Pyrrolidinones; Rolipram; Theophylline; Trachea

1996
Differential inhibition by selective phosphodiesterase inhibitors of antigen, LTC4 and histamine-induced contraction of guinea-pig isolated trachea.
    Pulmonary pharmacology, 1996, Volume: 9, Issue:4

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Bronchoconstrictor Agents; Bronchodilator Agents; Guanidines; Guinea Pigs; Histamine Antagonists; In Vitro Techniques; Leukotriene C4; Male; Milrinone; Muscle Tonus; Ovalbumin; Phosphodiesterase Inhibitors; Purinones; Pyridazines; Pyridones; Pyrrolidinones; Rolipram; Theophylline; Trachea

1996
Regulation of interleukin-13 by type 4 cyclic nucleotide phosphodiesterase (PDE) inhibitors in allergen-specific human T lymphocyte clones.
    Biochemical pharmacology, 1997, Apr-04, Volume: 53, Issue:7

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Allergens; Clone Cells; Gene Expression; Glycoproteins; Guanidines; Humans; Interleukin-13; Lymphocyte Activation; Lymphocytes; Phosphodiesterase Inhibitors; Pyridazines; Pyrrolidinones; Rolipram

1997
Interaction between prostaglandins and selective phosphodiesterase inhibitors in isolated guinea-pig trachea in vitro.
    European journal of pharmacology, 1997, Aug-27, Volume: 333, Issue:2-3

    Topics: Animals; Cyclooxygenase Inhibitors; Dinoprost; Dinoprostone; Drug Interactions; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxytocics; Phosphodiesterase Inhibitors; Purinones; Pyridazines; Pyrrolidinones; Rolipram; Trachea

1997
Mechanisms of thyroid hormone control over sensitivity and maximal contractile responsiveness to beta-adrenergic agonists in atria.
    Molecular and cellular biochemistry, 1998, Volume: 184, Issue:1-2

    Topics: Adrenergic beta-Agonists; Animals; Atrial Function; Calcium-Binding Proteins; Calcium-Transporting ATPases; Cyclic AMP; GTP-Binding Proteins; Guanidines; Isoproterenol; Myocardial Contraction; Phenylisopropyladenosine; Phosphorylation; Pyridazines; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Rolipram; Thyroid Hormones

1998
A biochemical and functional assessment of monocyte phosphodiesterase activity in healthy and asthmatic subjects.
    Pulmonary pharmacology & therapeutics, 2000, Volume: 13, Issue:5

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adult; Aged; Asthma; Case-Control Studies; Guanidines; Humans; Middle Aged; Monocytes; Phosphodiesterase Inhibitors; Pyridazines; Rolipram; Theophylline; Tumor Necrosis Factor-alpha

2000
Comparison of responses to siguazodan, rolipram, and zaprinast in the feline pulmonary vascular bed.
    European journal of pharmacology, 2000, Oct-13, Volume: 406, Issue:2

    Topics: Animals; Blood Pressure; Cats; Dose-Response Relationship, Drug; Female; Guanidines; Male; Phosphodiesterase Inhibitors; Pulmonary Circulation; Purinones; Pyridazines; Rolipram

2000
Phosphodiesterase activity in neutrophils from horses with chronic obstructive pulmonary disease.
    Veterinary immunology and immunopathology, 2000, Oct-31, Volume: 76, Issue:3-4

    Topics: Animals; Dose-Response Relationship, Immunologic; Guanidines; Horse Diseases; Horses; Isoenzymes; Neutrophils; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Pulmonary Disease, Chronic Obstructive; Pyridazines; Pyridines; Rolipram

2000
Histamine up-regulates phosphodiesterase IV activity in U-937 cells through H2 receptor stimulation and cAMP increase.
    Medical science monitor : international medical journal of experimental and clinical research, 2003, Volume: 9, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Diphenhydramine; Guanidines; Histamine; Humans; Kinetics; Purinones; Pyridazines; Ranitidine; Receptors, Histamine H2; Rolipram; U937 Cells

2003
Inhibition of mast cell histamine release by specific phosphodiesterase inhibitors.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2005, Volume: 54 Suppl 1

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Guanidines; Histamine; Mast Cells; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Protein Isoforms; Pyridazines; Rats; Rats, Sprague-Dawley; Rolipram

2005