Page last updated: 2024-08-16

sibutramine and sr141716

sibutramine has been researched along with sr141716 in 59 studies

Research

Studies (59)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's44 (74.58)29.6817
2010's15 (25.42)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Dourish, CT; Kennett, GA; Vickers, SP; Webster, LJ; Wyatt, A1
Vastag, B1
Halford, JC1
Bérubé-Parent, S; Chaput, JP; Tremblay, A1
Kennedy, RL; Khoo, EY1
Yanovski, SZ1
Astrup, AV; Breum, L; Bruun, JM; Svendsen, OL; Toubro, S1
Cheskin, LJ; Sidhaye, A1
Letonturier, P1
Blackburn, GL; Waltman, BA1
Hamann, A2
Behn, A; Ur, E1
Halpern, A; Mancini, MC1
Caterson, ID; Finer, N1
Cannon, E; Lundquist, LM; Sirimaturos, M1
Boss, O; Hofbauer, KG; Nicholson, JR1
Hofbauer, KG; Nicholson, JR1
Fujioka, K1
Majumdar, SR; Padwal, RS1
Rotthoff, T; Scherbaum, WA1
Formiguera, X; Sierra, A1
Bray, GA; Ryan, DH1
Gargallo, M; Isabel Millán, A; Moreno, B; Rubio, MA1
Zieba, R1
Käser, L; Kolyvanos, NU; Suter, PM; Vetter, W1
Bodary, PF; Eitzman, DT; Iglay, HB1
Kaila, B; Raman, M1
Nau, JY1
Al-Zaman, Y; Aylwin, S1
Davis, RJ; Nomikos, GG1
Aronne, LJ; Neff, LM1
Barnett, A; Rahim, A; Samat, A1
Pagotto, U; Pasquali, R; Vanuzzo, D; Vicennati, V1
Dunbar, AR; Fiksdal, BL; Filtz, CR; Hahn, TW; Jewett, DC; Levine, AS; Novinska, NL; Smith, TR; Wiebelhaus, JM1
Narbro, K; Neovius, M1
Aronne, LJ; Davis, SN; Foster, GD; Pagotto, U1
Idelevich, E; Kirch, W; Schindler, C1
Höcht, C; Mayer, MA; Puyó, A; Taira, CA1
Faludi, G; Halmy, L; Purebl, G; Rihmer, Z1
Choussein, S; Daskalopoulou, SS; Frangos, CC; Makri, AA; Petridou, ET1
Ciccocioppo, R; Cifani, C; Di Francesco, C; Massi, M; Melotto, S; Righetti, C; Tessari, M; Zanoncelli, A1
DeSantis, SM; Johansson, K; Neovius, K; Neovius, M; Rössner, S1
Berghold, A; Horvath, K; Jeitler, K; Matyas, E; Pignitter, N; Siebenhofer, A; Siering, U; Stich, AK1
Amundsen, MO; Berg, C; Engdahl, B; Nordeng, H1
Blundell, JE; Rodgers, RJ; Tallett, AJ1
Axel, AM; Hansen, G; Hansen, HH; Larsen, PJ; Mikkelsen, JD; Raben, A; Tang-Christensen, M1
de Kaste, D; Fijałek, Z; Kaun, N; Maurin, JK; Venhuis, BJ; Vredenbregt, MV1
Madsbad, S1
Bornstein, SR; Chavakis, T; Lamounier-Zepter, V; Schindler, C1
Abrams, K; Ara, R; Cooper, N; Davies, MJ; Dunkley, A; Gray, LJ; Khunti, K; Sutton, A; Warren, FC1
Abrams, K; Ara, R; Blake, L; Cooper, N; Crowther, M; Davies, M; Dunkley, A; Gray, L; Hernández, M; Jackson, R; Khunti, K; Rees, A; Stevenson, M; Sutton, A; Warren, F1
Bedros, JR; Medvegy, M; Pados, G; Simonyi, G1
Colman, E1
Kautzky-Willer, A; Lemmens-Gruber, R1
Berghold, A; Horvath, K; Jeitler, K; Semlitsch, T; Siebenhofer, A; Siering, U1
Baretić, M1
Berghold, A; Horvath, K; Jeitler, K; Meschik, J; Posch, N; Semlitsch, T; Siebenhofer, A1

Reviews

41 review(s) available for sibutramine and sr141716

ArticleYear
Clinical pharmacotherapy for obesity: current drugs and those in advanced development.
    Current drug targets, 2004, Volume: 5, Issue:7

    Topics: Anti-Obesity Agents; Appetite Depressants; Cyclobutanes; Energy Metabolism; Feeding Behavior; Fructose; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Topiramate

2004
Obesity and cardiovascular physiology: impact of some pharmacological agents.
    Current vascular pharmacology, 2005, Volume: 3, Issue:2

    Topics: Animals; Anti-Obesity Agents; Appetite Depressants; Cardiovascular Diseases; Cardiovascular Physiological Phenomena; Clinical Trials as Topic; Cyclobutanes; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Risk Factors

2005
[Drug treatment of obesity].
    Ugeskrift for laeger, 2006, Jan-09, Volume: 168, Issue:2

    Topics: Anti-Obesity Agents; Appetite Depressants; Cyclobutanes; Diethylpropion; Enzyme Inhibitors; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Time Factors; Weight Loss

2006
Pharmacologic treatment of obesity.
    Advances in psychosomatic medicine, 2006, Volume: 27

    Topics: Anti-Obesity Agents; Appetite Depressants; Cyclobutanes; Fructose; Humans; Isoxazoles; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Selective Serotonin Reuptake Inhibitors; Topiramate; Zonisamide

2006
Pharmacotherapy to reduce visceral fat.
    Clinical cornerstone, 2005, Volume: 7, Issue:2-3

    Topics: Anti-Obesity Agents; Coronary Disease; Cyclobutanes; Exercise; Feeding Behavior; Humans; Intra-Abdominal Fat; Lactones; Metabolic Syndrome; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant

2005
[Pharmacotherapy in the treatment of obesity].
    MMW Fortschritte der Medizin, 2006, Mar-02, Volume: 148, Issue:9

    Topics: Anti-Obesity Agents; Appetite Depressants; Cannabinoid Receptor Antagonists; Clinical Trials as Topic; Cyclobutanes; Enzyme Inhibitors; Exercise; Humans; Lactones; Lipase; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Time Factors; Weight Loss

2006
The obesity epidemic and its cardiovascular consequences.
    Current opinion in cardiology, 2006, Volume: 21, Issue:4

    Topics: Appetite Depressants; Body Fat Distribution; Body Mass Index; Cardiovascular Diseases; Cyclobutanes; Humans; Inflammation; Insulin Resistance; Intra-Abdominal Fat; Lactones; Life Style; Lipid Metabolism; Metabolic Syndrome; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Thiazolidinediones; Waist-Hip Ratio

2006
Pharmacological treatment of obesity.
    Arquivos brasileiros de endocrinologia e metabologia, 2006, Volume: 50, Issue:2

    Topics: Amphetamines; Anti-Obesity Agents; Appetite Depressants; Clinical Trials as Topic; Cyclobutanes; Energy Metabolism; Homeostasis; Humans; Lactones; Mazindol; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Weight Loss

2006
Emerging pharmacotherapy for treating obesity and associated cardiometabolic risk.
    Asia Pacific journal of clinical nutrition, 2006, Volume: 15 Suppl

    Topics: Anti-Obesity Agents; Cardiovascular Diseases; Cyclobutanes; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Risk Factors; Safety; Treatment Outcome

2006
Pharmacologic treatment for obesity. Options for today...and tomorrow.
    Advance for nurse practitioners, 2006, Volume: 14, Issue:8

    Topics: Anti-Obesity Agents; Clinical Trials as Topic; Cyclobutanes; Drug Therapy, Combination; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Weight Loss

2006
The obesity epidemic: current and future pharmacological treatments.
    Annual review of pharmacology and toxicology, 2007, Volume: 47

    Topics: Anti-Obesity Agents; Cyclobutanes; Disease Outbreaks; Drug Design; Drugs, Investigational; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant

2007
Pharmacotherapy of obesity.
    Experimental and clinical endocrinology & diabetes : official journal, German Society of Endocrinology [and] German Diabetes Association, 2006, Volume: 114, Issue:9

    Topics: Anti-Obesity Agents; Clinical Trials as Topic; Cyclobutanes; Drug Design; Energy Metabolism; Homeostasis; Humans; Lactones; Life Style; Models, Biological; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Technology, Pharmaceutical

2006
Metabolic syndrome treatment strategies.
    Pharmacotherapy, 2006, Volume: 26, Issue:12 Pt 2

    Topics: Appetite Depressants; Cardiovascular Diseases; Cyclobutanes; Exercise; Humans; Metabolic Syndrome; Obesity; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Risk Factors; Weight Loss

2006
Drug treatments for obesity: orlistat, sibutramine, and rimonabant.
    Lancet (London, England), 2007, Jan-06, Volume: 369, Issue:9555

    Topics: Anti-Obesity Agents; Blood Pressure; Cholesterol, HDL; Cyclobutanes; Half-Life; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Weight Loss

2007
[Pharmacotherapy of obesity].
    Medizinische Monatsschrift fur Pharmazeuten, 2006, Volume: 29, Issue:12

    Topics: Anti-Obesity Agents; Anticonvulsants; Cyclobutanes; Fructose; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Topiramate

2006
[New therapeutic aspects for the control of risk factors in obesity].
    Medicina clinica, 2007, Apr-07, Volume: 128, Issue:13

    Topics: Anti-Obesity Agents; Cyclobutanes; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant

2007
Drug treatment of the overweight patient.
    Gastroenterology, 2007, Volume: 132, Issue:6

    Topics: Animals; Anti-Obesity Agents; Clinical Trials, Phase II as Topic; Cyclobutanes; Humans; Lactones; Obesity; Orlistat; Overweight; Piperidines; Pyrazoles; Rimonabant; Treatment Outcome

2007
Drugs in the treatment of obesity: sibutramine, orlistat and rimonabant.
    Public health nutrition, 2007, Volume: 10, Issue:10A

    Topics: Anti-Obesity Agents; Cyclobutanes; Humans; Lactones; Life Style; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Safety; Treatment Outcome; Weight Loss

2007
[Obesity: a review of currently used antiobesity drugs and new compounds in clinical development].
    Postepy higieny i medycyny doswiadczalnej (Online), 2007, Oct-19, Volume: 61

    Topics: Anti-Obesity Agents; Clinical Trials as Topic; Cyclobutanes; Humans; Lactones; Neurotransmitter Agents; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Treatment Outcome

2007
[Obesity in adults].
    Praxis, 2007, Oct-17, Volume: 96, Issue:42

    Topics: Adult; Aged; Anti-Obesity Agents; Appetite Depressants; Bariatric Surgery; Body Mass Index; Cyclobutanes; Diagnosis, Differential; Enzyme Inhibitors; Humans; Lactones; Male; Middle Aged; Obesity; Obesity, Morbid; Orlistat; Overweight; Piperidines; Prognosis; Pyrazoles; Rimonabant; Time Factors; Weight Loss

2007
Strategies to reduce vascular risk associated with obesity.
    Current vascular pharmacology, 2007, Volume: 5, Issue:4

    Topics: Adiponectin; Anti-Obesity Agents; Cardiovascular Diseases; Cyclobutanes; Diabetes Mellitus, Type 2; Humans; Hyperlipidemias; Hypertension; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Risk Factors

2007
[Pharmacotherapy of obesity].
    Der Internist, 2008, Volume: 49, Issue:1

    Topics: Anti-Obesity Agents; Appetite Depressants; Cyclobutanes; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Treatment Outcome

2008
Obesity: a review of pathogenesis and management strategies.
    Canadian journal of gastroenterology = Journal canadien de gastroenterologie, 2008, Volume: 22, Issue:1

    Topics: Anti-Obesity Agents; Bariatric Surgery; Behavior Therapy; Caloric Restriction; Cyclobutanes; Dietary Carbohydrates; Dietary Fats; Exercise; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Weight Loss

2008
Emerging concepts in the medical and surgical treatment of obesity.
    Frontiers of hormone research, 2008, Volume: 36

    Topics: Adipose Tissue; Amyloid; Anticonvulsants; Antidepressive Agents; Anxiety; Appetite Regulation; Bariatric Surgery; Body Mass Index; Bupropion; Cholecystokinin; Ciliary Neurotrophic Factor; Clinical Trials as Topic; Cyclobutanes; Depression; Diabetes Mellitus, Type 2; Female; Fluoxetine; Fructose; Ghrelin; Humans; Intra-Abdominal Fat; Islet Amyloid Polypeptide; Isoxazoles; Lactones; Leptin; Metabolic Syndrome; Metformin; Obesity; Obesity, Morbid; Orlistat; Oxyntomodulin; Peptide YY; Piperidines; Polycystic Ovary Syndrome; Pyrazoles; Rimonabant; Sertraline; Sleep Apnea, Obstructive; Surgical Procedures, Operative; Topiramate; Zonisamide

2008
Pharmacotherapy for obesity.
    Current atherosclerosis reports, 2007, Volume: 9, Issue:6

    Topics: Amyloid; Anti-Obesity Agents; Appetite Depressants; Body Weight; Chronic Disease; Comorbidity; Cyclobutanes; Exenatide; Gastrointestinal Hormones; Humans; Islet Amyloid Polypeptide; Lactones; Leptin; Metformin; Obesity; Orlistat; Peptides; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Venoms

2007
Pharmacotherapy for obesity in menopausal women.
    Menopause international, 2008, Volume: 14, Issue:2

    Topics: Anti-Obesity Agents; Bariatric Surgery; Cyclobutanes; Diabetes Mellitus, Type 2; Exenatide; Female; Humans; Hypoglycemic Agents; Lactones; Menopause; Metformin; Obesity; Orlistat; Peptides; Piperidines; Pyrazoles; Rimonabant; Risk Factors; Venoms

2008
Cost-effectiveness of pharmacological anti-obesity treatments: a systematic review.
    International journal of obesity (2005), 2008, Volume: 32, Issue:12

    Topics: Anti-Obesity Agents; Appetite Depressants; Body Mass Index; Cost-Benefit Analysis; Cyclobutanes; Europe; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Quality-Adjusted Life Years; Rimonabant; Treatment Outcome; United States

2008
Current pharmacotherapeutic concepts for the treatment of obesity in adults.
    Therapeutic advances in cardiovascular disease, 2009, Volume: 3, Issue:1

    Topics: Adult; Anti-Obesity Agents; Appetite Depressants; Combined Modality Therapy; Cyclobutanes; Enzyme Inhibitors; Humans; Lactones; Lipase; Obesity; Orlistat; Piperidines; Prevalence; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Risk Reduction Behavior; Treatment Outcome; Weight Loss

2009
Recent advances in obesity pharmacotherapy.
    Current clinical pharmacology, 2009, Volume: 4, Issue:1

    Topics: Animals; Anti-Obesity Agents; Cardiovascular Diseases; Cyclobutanes; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant

2009
[Association of obesity and depression].
    Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology, 2008, Volume: 10, Issue:4

    Topics: Anti-Obesity Agents; Antidepressive Agents; Appetite Depressants; Appetite Regulation; Bipolar Disorder; Circadian Rhythm; Cyclobutanes; Depression; Depressive Disorder, Major; Dietary Carbohydrates; Energy Intake; Ghrelin; Humans; Hypothalamo-Hypophyseal System; Insulin Resistance; Leptin; Obesity; Piperidines; Pituitary-Adrenal System; Pyrazoles; Rimonabant; Seasonal Affective Disorder; Sleep Wake Disorders; Surveys and Questionnaires; Weight Gain; Weight Loss

2008
Effect of antiobesity medications in patients with type 2 diabetes mellitus.
    Diabetes, obesity & metabolism, 2009, Volume: 11, Issue:7

    Topics: Adolescent; Adult; Aged; Anti-Obesity Agents; Appetite Depressants; Body Weight; Cyclobutanes; Diabetes Mellitus, Type 2; Female; Humans; Lactones; Male; Middle Aged; Obesity; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Receptor, Cannabinoid, CB1; Rimonabant; Treatment Outcome; Weight Loss; Young Adult

2009
Discontinuation due to adverse events in randomized trials of orlistat, sibutramine and rimonabant: a meta-analysis.
    Obesity reviews : an official journal of the International Association for the Study of Obesity, 2009, Volume: 10, Issue:5

    Topics: Anti-Obesity Agents; Appetite Depressants; Cyclobutanes; Humans; Lactones; Medication Adherence; Odds Ratio; Orlistat; Overweight; Patient Dropouts; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant

2009
Long-term effects of weight-reducing drugs in hypertensive patients.
    The Cochrane database of systematic reviews, 2009, Jul-08, Issue:3

    Topics: Adult; Anti-Obesity Agents; Blood Pressure; Cyclobutanes; Female; Humans; Hypertension; Lactones; Male; Middle Aged; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Time; Weight Loss

2009
[Pharmacological concepts for the treatment of obesity - a therapeutic meander?].
    Deutsche medizinische Wochenschrift (1946), 2011, Volume: 136, Issue:31-32

    Topics: Adverse Drug Reaction Reporting Systems; Appetite Depressants; Body Weight; Brain; Combined Modality Therapy; Cyclobutanes; Diet, Reducing; Drug Approval; Drug Combinations; Drug Recalls; Drugs, Investigational; Forecasting; Humans; Obesity; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant

2011
A systematic review and mixed treatment comparison of pharmacological interventions for the treatment of obesity.
    Obesity reviews : an official journal of the International Association for the Study of Obesity, 2012, Volume: 13, Issue:6

    Topics: Anti-Obesity Agents; Body Mass Index; Cyclobutanes; Humans; Lactones; Life Style; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Treatment Outcome; Weight Loss

2012
What is the clinical effectiveness and cost-effectiveness of using drugs in treating obese patients in primary care? A systematic review.
    Health technology assessment (Winchester, England), 2012, Volume: 16, Issue:5

    Topics: Anti-Obesity Agents; Cost-Benefit Analysis; Cyclobutanes; Drug Costs; Exercise; Female; Humans; Lactones; Male; Middle Aged; Obesity; Orlistat; Piperidines; Primary Health Care; Pyrazoles; Rimonabant; Risk Reduction Behavior; Treatment Outcome

2012
[The pharmacological treatment of obesity: past, present and future].
    Orvosi hetilap, 2012, Mar-11, Volume: 153, Issue:10

    Topics: Amides; Anti-Obesity Agents; Anticonvulsants; Antidepressive Agents; Basal Metabolism; Benzazepines; Benzoxazines; Body Mass Index; Bridged Bicyclo Compounds, Heterocyclic; Ciliary Neurotrophic Factor; Clinical Trials as Topic; Combined Modality Therapy; Cyclobutanes; Dexfenfluramine; Fatty Acids; Female; Fenfluramine; Glucagon-Like Peptide 1; Human Growth Hormone; Humans; Intestinal Absorption; Lactones; Leptin; Life Style; Liraglutide; Male; Norepinephrine; Obesity; Obesity, Morbid; Orlistat; Piperidines; Pyrazoles; Pyridines; Receptor, Melanocortin, Type 4; Rimonabant; Satiation; Serotonin; Sodium-Glucose Transport Proteins; Sucrose; Thyroid Hormones

2012
Obesity and diabetes.
    Handbook of experimental pharmacology, 2012, Issue:214

    Topics: Animals; Cyclobutanes; Diabetes Mellitus; Female; Humans; Incretins; Insulin; Lactones; Male; Metformin; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant; Sex Characteristics; Sulfonylurea Compounds

2012
Long-term effects of weight-reducing drugs in hypertensive patients.
    The Cochrane database of systematic reviews, 2013, Mar-28, Issue:3

    Topics: Adult; Anti-Obesity Agents; Blood Pressure; Cyclobutanes; Diet, Reducing; Female; Humans; Hypertension; Lactones; Male; Middle Aged; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Safety-Based Drug Withdrawals; Time; Weight Loss

2013
Obesity drug therapy.
    Minerva endocrinologica, 2013, Volume: 38, Issue:3

    Topics: Anti-Obesity Agents; Appetite; Combined Modality Therapy; Comorbidity; Cost-Benefit Analysis; Cyclobutanes; Diabetes Mellitus, Type 2; Diet, Diabetic; Drug Combinations; Exercise Therapy; Fructose; Gastrointestinal Hormones; Humans; Incretins; Insulin; Insulin Secretion; Intestines; Lactones; Leptin; Life Style; Models, Biological; Neuropeptides; Obesity; Orlistat; Phentermine; Phytotherapy; Piperidines; Plant Preparations; Pyrazoles; Rimonabant; Topiramate

2013
Long-term effects of weight-reducing drugs in people with hypertension.
    The Cochrane database of systematic reviews, 2016, Mar-02, Volume: 3

    Topics: Adult; Anti-Obesity Agents; Appetite Depressants; Blood Pressure; Cyclobutanes; Diet, Reducing; Female; Fructose; Humans; Hypertension; Lactones; Male; Middle Aged; Orlistat; Phentermine; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Safety-Based Drug Withdrawals; Time; Topiramate; Weight Loss

2016

Other Studies

18 other study(ies) available for sibutramine and sr141716

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Preferential effects of the cannabinoid CB1 receptor antagonist, SR 141716, on food intake and body weight gain of obese (fa/fa) compared to lean Zucker rats.
    Psychopharmacology, 2003, Volume: 167, Issue:1

    Topics: Animals; Appetite Depressants; Cannabinoids; Cyclobutanes; Dose-Response Relationship, Drug; Eating; Energy Metabolism; Male; Motor Activity; Piperidines; Pyrazoles; Rats; Rats, Zucker; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Time Factors; Weight Gain

2003
Experimental drugs take aim at obesity.
    JAMA, 2003, Apr-09, Volume: 289, Issue:14

    Topics: Animals; Anti-Obesity Agents; Ciliary Neurotrophic Factor; Cyclobutanes; Drug Evaluation; Drugs, Investigational; Humans; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Recombinant Proteins; Rimonabant; United States; United States Food and Drug Administration

2003
New options for drug treatment of obesity in patients with Type 2 diabetes.
    Diabetic medicine : a journal of the British Diabetic Association, 2005, Volume: 22 Suppl 4

    Topics: Anti-Obesity Agents; Appetite Depressants; Cannabinoids; Cyclobutanes; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Lactones; Male; Middle Aged; Obesity; Orlistat; Piperidines; Pyrazoles; Rimonabant

2005
Pharmacotherapy for obesity--promise and uncertainty.
    The New England journal of medicine, 2005, Nov-17, Volume: 353, Issue:20

    Topics: Anti-Obesity Agents; Appetite Depressants; Cannabinoid Receptor Antagonists; Cyclobutanes; Dyslipidemias; Humans; Obesity; Piperidines; Pyrazoles; Rimonabant; Weight Loss

2005
[Reducing obesity].
    Presse medicale (Paris, France : 1983), 2006, Volume: 35, Issue:1 Pt 1

    Topics: Adolescent; Adult; Appetite Depressants; Body Mass Index; Cardiovascular Diseases; Child; Cyclobutanes; Female; Humans; Life Style; Male; Middle Aged; Obesity; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Risk Factors; Surveys and Questionnaires; Weight Loss

2006
[Antiobesity drugs--new limitations].
    Revue medicale suisse, 2007, Nov-28, Volume: 3, Issue:135

    Topics: Anti-Obesity Agents; Appetite Depressants; Cyclobutanes; Depression; Drug Therapy, Combination; Evidence-Based Medicine; Humans; Lactones; Obesity, Morbid; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Suicide; Weight Loss

2007
Oral administration of the antiobesity drugs, sibutramine and rimonabant, increases acetylcholine efflux selectively in the medial prefrontal cortex of the rat.
    Molecular psychiatry, 2008, Volume: 13, Issue:3

    Topics: Acetylcholine; Administration, Oral; Analysis of Variance; Animals; Appetite Depressants; Cyclobutanes; Dose-Response Relationship, Drug; Male; Microdialysis; Nucleus Accumbens; Piperidines; Prefrontal Cortex; Pyrazoles; Rats; Rats, Wistar; Rimonabant

2008
[Pharmacological therapy of obesity].
    Giornale italiano di cardiologia (2006), 2008, Volume: 9, Issue:4 Suppl 1

    Topics: Anti-Obesity Agents; Appetite Depressants; Body Mass Index; Bradykinin; Cannabinoid Receptor Antagonists; Cannabinoids; Cyclobutanes; Diabetes Mellitus, Type 2; Double-Blind Method; Economics, Pharmaceutical; Humans; Lactones; Lipase; Meta-Analysis as Topic; Obesity; Orlistat; Piperidines; Practice Guidelines as Topic; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Risk Factors; Time Factors; Weight Loss

2008
Effects of sibutramine and rimonabant in rats trained to discriminate between 22- and 2-h food deprivation.
    Psychopharmacology, 2009, Volume: 203, Issue:2

    Topics: Animals; Appetite Depressants; Cyclobutanes; Discrimination Learning; Discrimination, Psychological; Eating; Food Deprivation; Male; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Time Factors

2009
The endocannabinoid system as a target for obesity treatment.
    Clinical cornerstone, 2008, Volume: 9, Issue:1

    Topics: Amides; Anti-Obesity Agents; Cannabinoid Receptor Modulators; Cyclobutanes; Depression; Endocannabinoids; Humans; Lactones; Life Style; Metabolic Syndrome; Obesity; Orlistat; Piperidines; Pyrazoles; Pyridines; Rimonabant; Risk

2008
Pre-exposure to environmental cues predictive of food availability elicits hypothalamic-pituitary-adrenal axis activation and increases operant responding for food in female rats.
    Addiction biology, 2009, Volume: 14, Issue:4

    Topics: Adrenocorticotropic Hormone; Animals; Anti-Obesity Agents; Appetite Depressants; Cannabinoids; Conditioning, Operant; Corticosterone; Cues; Cyclobutanes; Environment; Feeding Behavior; Female; Fluoxetine; Fructose; Humans; Hypothalamo-Hypophyseal System; Motivation; Piperidines; Pituitary-Adrenal System; Pyrazoles; Rats; Reproducibility of Results; Rimonabant; Selective Serotonin Reuptake Inhibitors; Topiramate

2009
Use of psychotropic drugs and analgesics among users of antiobesity drugs--a population based study.
    Pharmacoepidemiology and drug safety, 2010, Volume: 19, Issue:3

    Topics: Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Analgesics; Anti-Obesity Agents; Child; Cyclobutanes; Databases, Factual; Drug Interactions; Female; Humans; Lactones; Male; Middle Aged; Norway; Orlistat; Piperidines; Practice Patterns, Physicians'; Psychotropic Drugs; Pyrazoles; Rimonabant; Sex Factors; Young Adult

2010
Effects of acute low-dose combined treatment with rimonabant and sibutramine on appetite and weight gain in rats.
    Pharmacology, biochemistry, and behavior, 2010, Volume: 97, Issue:1

    Topics: Animals; Appetite; Cyclobutanes; Drug Administration Schedule; Drug Therapy, Combination; Male; Piperidines; Pyrazoles; Rats; Reaction Time; Rimonabant; Satiety Response; Weight Gain

2010
The novel triple monoamine reuptake inhibitor tesofensine induces sustained weight loss and improves glycemic control in the diet-induced obese rat: comparison to sibutramine and rimonabant.
    European journal of pharmacology, 2010, Jun-25, Volume: 636, Issue:1-3

    Topics: Adipose Tissue; Animals; Appetite; Biogenic Monoamines; Blood Glucose; Bridged Bicyclo Compounds, Heterocyclic; Cyclobutanes; Diet; Eating; Glucose Tolerance Test; Lipids; Male; Neurotransmitter Uptake Inhibitors; Obesity; Piperidines; Pyrazoles; Rats; Rimonabant; Time Factors; Weight Loss

2010
The identification of rimonabant polymorphs, sibutramine and analogues of both in counterfeit Acomplia bought on the internet.
    Journal of pharmaceutical and biomedical analysis, 2011, Jan-05, Volume: 54, Issue:1

    Topics: Chemistry, Pharmaceutical; Chromatography, Liquid; Cyclobutanes; Drug Contamination; Fraud; Internet; Models, Chemical; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Spectroscopy, Near-Infrared; Spectrum Analysis, Raman; X-Ray Diffraction

2011
[Long-term effects of weight-reducing drugs in hypertensive patients--a survey of a Cochrane review].
    Ugeskrift for laeger, 2011, Feb-21, Volume: 173, Issue:8

    Topics: Adult; Anti-Obesity Agents; Appetite Depressants; Blood Pressure; Cardiovascular Diseases; Cyclobutanes; Evidence-Based Medicine; Humans; Hypertension; Lactones; Obesity; Orlistat; Piperidines; Pyrazoles; Randomized Controlled Trials as Topic; Rimonabant; Time Factors; Treatment Outcome; Weight Loss

2011
Food and Drug Administration's Obesity Drug Guidance Document: a short history.
    Circulation, 2012, May-01, Volume: 125, Issue:17

    Topics: Adolescent; Adult; Advisory Committees; Aged; Anti-Obesity Agents; Bariatric Medicine; Body Mass Index; Child; Congresses as Topic; Cyclobutanes; Diabetes Mellitus, Type 2; Drug Approval; Drug Discovery; Female; History, 20th Century; History, 21st Century; Humans; Male; Middle Aged; Multicenter Studies as Topic; Obesity; Outcome Assessment, Health Care; Piperidines; Practice Guidelines as Topic; Pyrazoles; Randomized Controlled Trials as Topic; Reference Standards; Rimonabant; Safety-Based Drug Withdrawals; United States; United States Food and Drug Administration

2012