Page last updated: 2024-09-03

sgb 1534 and phentolamine

sgb 1534 has been researched along with phentolamine in 2 studies

Compound Research Comparison

Studies
(sgb 1534)
Trials
(sgb 1534)
Recent Studies (post-2010)
(sgb 1534)
Studies
(phentolamine)
Trials
(phentolamine)
Recent Studies (post-2010) (phentolamine)
20009,141270265

Protein Interaction Comparison

ProteinTaxonomysgb 1534 (IC50)phentolamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.396
Alpha-2A adrenergic receptorHomo sapiens (human)0.006
Cytochrome P450 2D6Homo sapiens (human)10
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0316
Alpha-2B adrenergic receptorHomo sapiens (human)0.018
Alpha-2C adrenergic receptorHomo sapiens (human)0.11
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0316
Alpha-1D adrenergic receptorHomo sapiens (human)0.0173
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.359
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.396
Alpha-1A adrenergic receptorHomo sapiens (human)0.0011
Alpha-1B adrenergic receptorHomo sapiens (human)0.0108
5-hydroxytryptamine receptor 2BHomo sapiens (human)3.807
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0316
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.5495

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Koga, T; Sakai, K; Shiraki, Y1
Aono, J; Ishizuka, N; Nabata, H; Sakai, K1

Other Studies

2 other study(ies) available for sgb 1534 and phentolamine

ArticleYear
Characterization of a novel alpha 1-adrenoceptor antagonist, SGB-1534, in contractile response of isolated canine arterial and venous smooth muscle to exogenous noradrenaline: comparison with prazosin, phentolamine and yohimbine.
    Japanese journal of pharmacology, 1989, Volume: 50, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Prazosin; Quinazolines; Yohimbine

1989
Antihypertensive effects of a novel phenylpiperazine derivative, SGB-1534, on several hypertensive models of rats.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 277, Issue:1

    Topics: Animals; Antihypertensive Agents; Desoxycorticosterone; Hypertension; Hypertension, Renal; Lethal Dose 50; Male; Phentolamine; Posture; Prazosin; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Renin

1985