Page last updated: 2024-08-24

sertindole and raclopride

sertindole has been researched along with raclopride in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's1 (20.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Audinot, V; Chaput, C; Conte, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L1
Balle, T; Bang-Andersen, B; Christoffersen, CT; Jensen, M; Kristensen, JL; Püschl, A; Risgaard, R1
Balle, T; Bang-Andersen, B; Christoffersen, CT; Jensen, KG; Jørgensen, M; Jørgensen, PN1
Farde, L; Halldin, C; Mack, RJ; Nyberg, S1
Brennum, LT; Kreilgaard, M; Olsen, CK1

Trials

1 trial(s) available for sertindole and raclopride

ArticleYear
D2 occupancy, extrapyramidal side effects and antipsychotic drug treatment: a pilot study with sertindole in healthy subjects.
    International clinical psychopharmacology, 1997, Volume: 12 Suppl 1

    Topics: Administration, Oral; Adult; Antipsychotic Agents; Basal Ganglia Diseases; Brain; Humans; Imidazoles; Indoles; Injections, Intravenous; Male; Pilot Projects; Raclopride; Receptors, Dopamine D2; Salicylamides; Tomography, Emission-Computed

1997

Other Studies

4 other study(ies) available for sertindole and raclopride

ArticleYear
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study.
    European journal of pharmacology, 1998, Aug-21, Volume: 355, Issue:2-3

    Topics: Animals; Antipsychotic Agents; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Sulfur Radioisotopes

1998
Exploring the neuroleptic substituent in octoclothepin: potential ligands for positron emission tomography with subnanomolar affinity for α(1)-adrenoceptors.
    Journal of medicinal chemistry, 2010, Oct-14, Volume: 53, Issue:19

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Cattle; Cell Line; Cell Membrane Permeability; Cerebral Cortex; Cricetinae; Crystallography, X-Ray; Dibenzothiepins; Humans; Ligands; Models, Molecular; Piperazines; Positron-Emission Tomography; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Stereoisomerism; Structure-Activity Relationship

2010
Discovery of novel α₁-adrenoceptor ligands based on the antipsychotic sertindole suitable for labeling as PET ligands.
    Bioorganic & medicinal chemistry, 2013, Jan-01, Volume: 21, Issue:1

    Topics: Animals; Antipsychotic Agents; Brain; Caco-2 Cells; CHO Cells; Cricetinae; Humans; Imidazoles; Indoles; Ligands; Positron-Emission Tomography; Rats; Receptors, Adrenergic, alpha-1

2013
Using pharmacokinetic-pharmacodynamic modelling as a tool for prediction of therapeutic effective plasma levels of antipsychotics.
    European journal of pharmacology, 2008, Apr-28, Volume: 584, Issue:2-3

    Topics: Administration, Oral; Animals; Antipsychotic Agents; Basal Ganglia; Behavior, Animal; Benzodiazepines; Binding, Competitive; Clozapine; Conditioning, Psychological; Dopamine Antagonists; Haloperidol; Imidazoles; Indoles; Injections, Subcutaneous; Male; Models, Biological; Olanzapine; Protein Binding; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Reproducibility of Results; Risperidone

2008