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sertindole and octoclothepine, (s)-isomer

sertindole has been researched along with octoclothepine, (s)-isomer in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andersen, K; Bøgesø, KP; Gundertofte, K; Liljefors, T; Perregaard, J1
Andersen, K; Balle, T; Larsen, AK; Liljefors, T; Perregaard, J; Ramirez, MT; Søby, KK1
Balle, T; Bang-Andersen, B; Christoffersen, CT; Jensen, M; Kristensen, JL; Püschl, A; Risgaard, R1

Other Studies

3 other study(ies) available for sertindole and octoclothepine, (s)-isomer

ArticleYear
Development of a receptor-interaction model for serotonin 5-HT2 receptor antagonists. Predicting selectivity with respect to dopamine D2 receptors.
    Journal of medicinal chemistry, 1994, Apr-01, Volume: 37, Issue:7

    Topics: Indans; Indoles; Models, Chemical; Molecular Conformation; Receptors, Dopamine D2; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1994
Synthesis and structure-affinity relationship investigations of 5-heteroaryl-substituted analogues of the antipsychotic sertindole. A new class of highly selective alpha(1) adrenoceptor antagonists.
    Journal of medicinal chemistry, 2003, Jan-16, Volume: 46, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Azoles; Brain; Cell Line; Cricetinae; Humans; Imidazoles; In Vitro Techniques; Indoles; Pyridines; Pyrimidines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Receptors, Dopamine; Receptors, Serotonin; Structure-Activity Relationship; Triazoles

2003
Exploring the neuroleptic substituent in octoclothepin: potential ligands for positron emission tomography with subnanomolar affinity for α(1)-adrenoceptors.
    Journal of medicinal chemistry, 2010, Oct-14, Volume: 53, Issue:19

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Cattle; Cell Line; Cell Membrane Permeability; Cerebral Cortex; Cricetinae; Crystallography, X-Ray; Dibenzothiepins; Humans; Ligands; Models, Molecular; Piperazines; Positron-Emission Tomography; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Stereoisomerism; Structure-Activity Relationship

2010