Page last updated: 2024-08-24

sertindole and cyclosporine

sertindole has been researched along with cyclosporine in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Broccatelli, F; Carosati, E; Cruciani, G; Frosini, M; Goracci, L; Neri, A; Oprea, TI1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Brincat, JP; Broccatelli, F; Carosati, E; Cruciani, G; Frosini, M; Kaatz, GW; Neri, A; Sabatini, S1
Andersen, K; Andersen, L; Badolo, L; Balle, T; Chou, YW; Farde, L; Gjervig Jensen, K; Halldin, C; Hjorth Alifrangis, L; Perregaard, J1

Other Studies

4 other study(ies) available for sertindole and cyclosporine

ArticleYear
A novel approach for predicting P-glycoprotein (ABCB1) inhibition using molecular interaction fields.
    Journal of medicinal chemistry, 2011, Mar-24, Volume: 54, Issue:6

    Topics: Animals; Aripiprazole; ATP Binding Cassette Transporter, Subfamily B, Member 1; Butyrophenones; Cell Line, Tumor; Cell Membrane Permeability; Drug Design; Humans; Hydrophobic and Hydrophilic Interactions; Ligands; Mice; Models, Molecular; Molecular Structure; Piperazines; Piperidines; Protein Binding; Quantitative Structure-Activity Relationship; Quinolones

2011
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Ligand Promiscuity between the Efflux Pumps Human P-Glycoprotein and S. aureus NorA.
    ACS medicinal chemistry letters, 2012, Mar-08, Volume: 3, Issue:3

    Topics:

2012
New alpha(1)-adrenoceptor antagonists derived from the antipsychotic sertindole - carbon-11 labelling and pet examination of brain uptake in the cynomolgus monkey.
    Nuclear medicine and biology, 2004, Volume: 31, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Antipsychotic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Brain; Caco-2 Cells; Carbon Radioisotopes; Cyclosporine; Drug Evaluation, Preclinical; Humans; Imidazoles; Indoles; Isotope Labeling; Kinetics; Macaca fascicularis; Male; Metabolic Clearance Rate; Mice; Positron-Emission Tomography; Protein Binding; Radiopharmaceuticals; Receptors, Adrenergic, alpha-1

2004