Page last updated: 2024-09-03

serotonin-o-carboxymethyl-gly-tyr and cp 93129

serotonin-o-carboxymethyl-gly-tyr has been researched along with cp 93129 in 3 studies

Compound Research Comparison

Studies
(serotonin-o-carboxymethyl-gly-tyr)
Trials
(serotonin-o-carboxymethyl-gly-tyr)
Recent Studies (post-2010)
(serotonin-o-carboxymethyl-gly-tyr)
Studies
(cp 93129)
Trials
(cp 93129)
Recent Studies (post-2010) (cp 93129)
2000109011

Protein Interaction Comparison

ProteinTaxonomyserotonin-o-carboxymethyl-gly-tyr (IC50)cp 93129 (IC50)
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)3
5-hydroxytryptamine receptor 1DHomo sapiens (human)2.2
5-hydroxytryptamine receptor 2CHomo sapiens (human)6.4
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.015

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bruinvels, AT; Hoyer, D; Landwehrmeyer, B; Palacios, JM; Probst, A1
Castanon, N; Chauveau, J; Chaveau, J; Hen, R; Macor, JE; Moskowitz, MA; Scearce, K; Waeber, C; Yu, XJ1
Castro, ME; Mostany, R; Pazos, A1

Other Studies

3 other study(ies) available for serotonin-o-carboxymethyl-gly-tyr and cp 93129

ArticleYear
A comparative autoradiographic study of 5-HT1D binding sites in human and guinea-pig brain using different radioligands.
    Brain research. Molecular brain research, 1994, Volume: 21, Issue:1-2

    Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Dipeptides; Female; Guinea Pigs; Humans; Iodine Radioisotopes; Kinetics; Ligands; Male; Organ Specificity; Pyridines; Pyrroles; Receptors, Serotonin; Serotonin; Species Specificity; Sumatriptan; Tritium; Yohimbine

1994
5-Carboxamido-tryptamine, CP-122,288 and dihydroergotamine but not sumatriptan, CP-93,129, and serotonin-5-O-carboxymethyl-glycyl -tyrosinamide block dural plasma protein extravasation in knockout mice that lack 5-hydroxytryptamine1B receptors.
    Molecular pharmacology, 1996, Volume: 49, Issue:5

    Topics: Animals; Capillary Permeability; Dihydroergotamine; Dipeptides; Mice; Mice, Knockout; Pyridines; Pyrroles; Pyrrolidines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion

1996
Autoradiographic characterisation of [35S]GTPgammaS binding stimulation mediated by 5-HT1B receptor in postmortem human brain.
    Neuropharmacology, 2005, Volume: 48, Issue:1

    Topics: Aged; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain; Dipeptides; Drug Interactions; Female; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidones; Postmortem Changes; Protein Binding; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfur Isotopes

2005