serine and quinazolines

serine has been researched along with quinazolines in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19901 (4.55)18.7374
1990's2 (9.09)18.2507
2000's7 (31.82)29.6817
2010's12 (54.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hutchison, DJ; Rader, JI1
Dreslin, JA; Grizzuti, K; Gros, P; Kajiji, S1
Eguchi, K; Eguchi, S; Frank, GD; Hirata, Y; Inagami, T; Iwasaki, H; Marumo, F; Motley, ED; Ueno, H1
Choi, JI; Jeong, SW; Yoon, MH1
Bassères, DS; Bohlander, SK; Davis, RJ; Dayaram, T; Delmotte, MH; Giese, NA; Gilliland, DG; Hiddemann, W; Lokker, N; Radomska, HS; Schnittger, S; Small, D; Sternberg, DW; Tenen, DG; Yamamoto, Y; Zhang, P; Zheng, R1
Asahina, H; Dosaka-Akita, H; Kinoshita, I; Nishimura, M; Yamazaki, K; Yokouchi, H1
Anderson, KS; Atreya, CE; Doan, LT; Martucci, WE; Vargo, MA1
Kawanishi, M; Koizumi, K; Nishimura, M; Saiki, I; Sakurai, H; Shin, MS; Singhirunnusorn, P; Suzuki, S1
Angelillo-Scherrer, A; Hirt, L; Price, M; Thevenet, J1
Aung, HH; Barnholt, KE; Kota, RS; Rutledge, JC1
Arellano-Plancarte, A; Catt, KJ; Hernandez-Aranda, J; Olivares-Reyes, JA1
Cho, S; Jeong, YS; Kang, YK; Ko, Y; Park, JS1
Akar, U; Arun, BK; Hortobagyi, GN; LaFortune, TA; Nieves-Alicea, R; Tari, AM; Ueno, NT; Zhang, D1
Borsuk, E; Kubiak, JZ; Meglicki, M; Pasternak, M; Teperek-Tkacz, M1
Lenihan, DJ; Subbiah, IM; Tsimberidou, AM1
Assiddiq, BF; Chan, SP; Chong, PK; Lim, YP; Tan, KY; Toy, W1
Hellman, U; Kazi, JU; Lundby, A; Mohlin, S; Olsen, JV; Påhlman, S; Rönnstrand, L; Sun, J1
Asara, JM; Choi, JH; Cui, H; Ding, HF; Ding, J; Dong, Z; Huang, S; Li, T; Wang, X; Yang, L; Zha, Y; Zhao, E1
Kontani, Y; Kusudo, T; Mori, N; Okamatsu, Y; Saito, M; Takeuchi, T; Wang, T; Yamashita, H; Yamashita, Y1
Altiok, S; Doshi, P; Fulp, W; Haura, EB; Sasser, K; Smith, MA; Song, L1
Katayama, K; Noguchi, K; Sugimoto, Y; Takami, M1
Cao, LL; Guan, PP; Huang, XS; Liang, YY; Wang, P1

Other Studies

22 other study(ies) available for serine and quinazolines

ArticleYear
Selection and characterization of mutant strains of Streptococcus faecium var. durans resistant to methasquin and amethopterin.
    Cancer research, 1972, Volume: 32, Issue:4

    Topics: Culture Media; Depression, Chemical; Drug Antagonism; Drug Resistance, Microbial; Drug Synergism; Folic Acid; Folic Acid Antagonists; Genetics, Microbial; Methotrexate; Mutation; Purines; Quinazolines; Serine; Streptococcus; Tetrahydrofolates; Thymine Nucleotides

1972
Structurally distinct MDR modulators show specific patterns of reversal against P-glycoproteins bearing unique mutations at serine939/941.
    Biochemistry, 1994, May-03, Volume: 33, Issue:17

    Topics: Amino Acid Sequence; Animals; Cell Survival; CHO Cells; Clone Cells; Cricetinae; Cyclosporine; Dibenzocycloheptenes; Drug Resistance; Glycoproteins; Isoquinolines; Mice; Phenylalanine; Point Mutation; Quinazolines; Quinolines; Recombinant Proteins; Serine; Transfection; Vinblastine

1994
Intracellular signaling of angiotensin II-induced p70 S6 kinase phosphorylation at Ser(411) in vascular smooth muscle cells. Possible requirement of epidermal growth factor receptor, Ras, extracellular signal-regulated kinase, and Akt.
    The Journal of biological chemistry, 1999, Dec-24, Volume: 274, Issue:52

    Topics: Angiotensin II; Animals; Calcium; CHO Cells; Cricetinae; ErbB Receptors; Muscle, Smooth, Vascular; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Quinazolines; ras Proteins; Rats; Rats, Sprague-Dawley; Ribosomal Protein S6 Kinases; Serine; Transcriptional Activation; Tyrphostins

1999
Spinal gabapentin and antinociception: mechanisms of action.
    Journal of Korean medical science, 2003, Volume: 18, Issue:2

    Topics: Acetates; Adrenergic alpha-Antagonists; Adrenergic Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amines; Analgesics; Animals; Atropine; Cyclohexanecarboxylic Acids; Dihydroergocristine; Enzyme Inhibitors; Excitatory Amino Acid Agonists; GABA Antagonists; Gabapentin; gamma-Aminobutyric Acid; Injections, Spinal; Leucine; Male; Mecamylamine; Muscarinic Antagonists; N-Methylaspartate; Naloxone; Narcotic Antagonists; Nicotinic Antagonists; Pain Measurement; Quinazolines; Rats; Rats, Sprague-Dawley; Serine; Spinal Cord; Thapsigargin; Triazoles

2003
Block of C/EBP alpha function by phosphorylation in acute myeloid leukemia with FLT3 activating mutations.
    The Journal of experimental medicine, 2006, Feb-20, Volume: 203, Issue:2

    Topics: Aged; CCAAT-Enhancer-Binding Protein-alpha; Cell Differentiation; Cell Line; Enzyme Activation; Female; fms-Like Tyrosine Kinase 3; Granulocytes; Humans; K562 Cells; Leukemia, Myeloid, Acute; Male; MAP Kinase Kinase 1; Myeloid Cells; Phosphorylation; Piperazines; Point Mutation; Quinazolines; Serine; Tumor Cells, Cultured; U937 Cells

2006
Non-responsiveness to gefitinib in a patient with lung adenocarcinoma having rare EGFR mutations S768I and V769L.
    Lung cancer (Amsterdam, Netherlands), 2006, Volume: 54, Issue:3

    Topics: Adenocarcinoma; DNA, Neoplasm; Drug Resistance, Neoplasm; ErbB Receptors; Gefitinib; Humans; Isoleucine; Leucine; Lung Neoplasms; Male; Middle Aged; Mutation; Quinazolines; Serine; Valine

2006
Nonconserved residues Ala287 and Ser290 of the Cryptosporidium hominis thymidylate synthase domain facilitate its rapid rate of catalysis.
    Biochemistry, 2007, Jul-17, Volume: 46, Issue:28

    Topics: Alanine; Amino Acid Sequence; Animals; Binding Sites; Catalysis; Chromatography, High Pressure Liquid; Cryptosporidium; Crystallography, X-Ray; Folic Acid; Kinetics; Models, Molecular; Molecular Sequence Data; Multienzyme Complexes; Mutagenesis, Site-Directed; Protein Structure, Tertiary; Protozoan Proteins; Quinazolines; Serine; Tetrahydrofolate Dehydrogenase; Tetrahydrofolates; Thymidine Monophosphate; Thymidylate Synthase

2007
TAK1-mediated serine/threonine phosphorylation of epidermal growth factor receptor via p38/extracellular signal-regulated kinase: NF-{kappa}B-independent survival pathways in tumor necrosis factor alpha signaling.
    Molecular and cellular biology, 2009, Volume: 29, Issue:20

    Topics: Anthracenes; Butadienes; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; HeLa Cells; Humans; Imidazoles; Lactones; MAP Kinase Kinase Kinases; NF-kappa B; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Quinazolines; Resorcinols; RNA, Small Interfering; Serine; Signal Transduction; Threonine; Tumor Necrosis Factor-alpha

2009
Coagulation factor Xa activates thrombin in ischemic neural tissue.
    Journal of neurochemistry, 2009, Volume: 111, Issue:3

    Topics: Animals; Animals, Newborn; Anticoagulants; Cell Death; Factor Xa; Fondaparinux; Gene Expression Regulation; Glucose; Hippocampus; Hypoxia; Ischemia; JNK Mitogen-Activated Protein Kinases; Organ Culture Techniques; Polysaccharides; Pyrroles; Quinazolines; Rats; Receptor, PAR-1; Serine; Signal Transduction; Thrombin

2009
Adenosine blocks IFN-gamma-induced phosphorylation of STAT1 on serine 727 to reduce macrophage activation.
    Journal of immunology (Baltimore, Md. : 1950), 2009, Nov-15, Volume: 183, Issue:10

    Topics: Adenosine; Adenosine A3 Receptor Antagonists; Analgesics; Animals; Cell Line; Dihydropyridines; Gene Expression; Humans; Interferon-gamma; Janus Kinases; Macrophage Activation; Macrophages; Mice; Microarray Analysis; Phosphorylation; Quinazolines; Receptor, Adenosine A3; Serine; Signal Transduction; STAT1 Transcription Factor; Transcriptional Activation; Triazoles; Tyrosine

2009
Angiotensin-induced EGF receptor transactivation inhibits insulin signaling in C9 hepatic cells.
    Biochemical pharmacology, 2010, Mar-01, Volume: 79, Issue:5

    Topics: Angiotensin II; Animals; Cell Line; Enzyme Inhibitors; ErbB Receptors; Hepatocytes; Insulin; Insulin Resistance; Phosphorylation; Proto-Oncogene Proteins c-akt; Quinazolines; Rats; Receptor, Insulin; Serine; Signal Transduction; Threonine; Transcriptional Activation; Tyrphostins; Vasoconstrictor Agents

2010
Phosphorylation of serine-10 of histone H3 shields modified lysine-9 selectively during mitosis.
    Genes to cells : devoted to molecular & cellular mechanisms, 2010, Volume: 15, Issue:3

    Topics: Animals; Aurora Kinase B; Benzamides; Cell Cycle; Chromobox Protein Homolog 5; Chromosomal Proteins, Non-Histone; Female; Histones; Lysine; Male; Methylation; Mice; Mitosis; NIH 3T3 Cells; Phosphorylation; Protein Kinase Inhibitors; Quinazolines; Serine

2010
Silencing kinase-interacting stathmin gene enhances erlotinib sensitivity by inhibiting Ser¹⁰ p27 phosphorylation in epidermal growth factor receptor-expressing breast cancer.
    Molecular cancer therapeutics, 2010, Volume: 9, Issue:11

    Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Carcinoma; Cell Line, Tumor; Cyclin-Dependent Kinase Inhibitor p27; Drug Resistance, Neoplasm; Drug Synergism; Erlotinib Hydrochloride; Female; Gene Silencing; Genes, erbB-1; Humans; Mice; Mice, Nude; Phosphorylation; Protein Binding; Protein Kinases; Quinazolines; RNA, Small Interfering; Serine; Stathmin; Xenograft Model Antitumor Assays

2010
Phosphorylation of histone H3 serine 10 in early mouse embryos: active phosphorylation at late S phase and differential effects of ZM447439 on first two embryonic mitoses.
    Cell cycle (Georgetown, Tex.), 2010, Dec-01, Volume: 9, Issue:23

    Topics: Anaphase; Animals; Aurora Kinase A; Aurora Kinase B; Aurora Kinases; Benzamides; Cell Cycle Proteins; Embryo, Mammalian; Female; G1 Phase; Histones; Kinetochores; Mad2 Proteins; Male; Mice; Mitosis; Phosphorylation; Protein Serine-Threonine Kinases; Quinazolines; S Phase; Serine; Spindle Apparatus; Telophase

2010
Cardiovascular toxicity profiles of vascular-disrupting agents.
    The oncologist, 2011, Volume: 16, Issue:8

    Topics: Angiogenesis Inhibitors; Bibenzyls; Cardiovascular System; Clinical Trials as Topic; Humans; Neoplasms; Neovascularization, Pathologic; Organophosphorus Compounds; Quinazolines; Serine; Xanthones

2011
EGFR S1166 phosphorylation induced by a combination of EGF and gefitinib has a potentially negative impact on lung cancer cell growth.
    Journal of proteome research, 2012, Aug-03, Volume: 11, Issue:8

    Topics: Amino Acid Motifs; Amino Acid Sequence; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Epidermal Growth Factor; ErbB Receptors; Gefitinib; Humans; Lung Neoplasms; Molecular Sequence Data; Peptide Fragments; Phosphorylation; Protein Processing, Post-Translational; Quinazolines; Serine; Tandem Mass Spectrometry; Tyrosine

2012
The PI3-kinase isoform p110δ is essential for cell transformation induced by the D816V mutant of c-Kit in a lipid-kinase-independent manner.
    Oncogene, 2014, Nov-13, Volume: 33, Issue:46

    Topics: Adenine; Animals; Binding Sites; Blotting, Western; Cell Line; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cell Transformation, Neoplastic; Chlorocebus aethiops; Chromones; Class Ia Phosphatidylinositol 3-Kinase; COS Cells; Female; Mice, Inbred Strains; Mice, Nude; Morpholines; Mutation, Missense; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Binding; Proto-Oncogene Proteins c-kit; Quinazolines; RNA Interference; Serine; Tyrosine

2014
The histone H3 methyltransferase G9A epigenetically activates the serine-glycine synthesis pathway to sustain cancer cell survival and proliferation.
    Cell metabolism, 2013, Dec-03, Volume: 18, Issue:6

    Topics: Animals; Autophagy; Azepines; Bone Neoplasms; Cell Line, Tumor; Cell Proliferation; Cell Survival; Epigenomics; Glycine; HeLa Cells; Histocompatibility Antigens; Histone-Lysine N-Methyltransferase; Histones; Humans; Methylation; Mice; Microtubule-Associated Proteins; Quinazolines; Ribosomes; Serine; Transcription, Genetic

2013
Evodiamine inhibits insulin-stimulated mTOR-S6K activation and IRS1 serine phosphorylation in adipocytes and improves glucose tolerance in obese/diabetic mice.
    PloS one, 2013, Volume: 8, Issue:12

    Topics: 3T3-L1 Cells; Adipocytes; Adipose Tissue, White; AMP-Activated Protein Kinases; Animals; Diabetes Mellitus, Experimental; Evodia; Female; Glucose; Glucose Tolerance Test; Hypoglycemic Agents; Insulin Receptor Substrate Proteins; Insulin Resistance; Mice; Mice, Obese; Phosphorylation; Quinazolines; Ribosomal Protein S6 Kinases; Serine; Signal Transduction; TOR Serine-Threonine Kinases

2013
Antitumor efficacy of the anti-interleukin-6 (IL-6) antibody siltuximab in mouse xenograft models of lung cancer.
    Journal of thoracic oncology : official publication of the International Association for the Study of Lung Cancer, 2014, Volume: 9, Issue:7

    Topics: Adenocarcinoma; Animals; Antibodies, Monoclonal; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cell Line, Tumor; Disease Models, Animal; Erlotinib Hydrochloride; Female; Fibroblasts; Humans; Interleukin-6; Lung Neoplasms; Mice; Phosphorylation; Proto-Oncogene Proteins; Proto-Oncogene Proteins p21(ras); Quinazolines; ras Proteins; Serine; STAT3 Transcription Factor; Tyrosine

2014
Protein kinase C alpha-mediated phosphorylation of PIM-1L promotes the survival and proliferation of acute myeloid leukemia cells.
    Biochemical and biophysical research communications, 2018, 09-10, Volume: 503, Issue:3

    Topics: Apoptosis; Cell Line, Tumor; Cell Proliferation; Humans; Leukemia, Myeloid, Acute; Phosphorylation; Protein Isoforms; Protein Kinase C-alpha; Proto-Oncogene Proteins c-pim-1; Pyrroles; Quinazolines; Serine

2018
Cyclooxygenase-2 is Essential for Mediating the Effects of Calcium Ions on Stimulating Phosphorylation of Tau at the Sites of Ser 396 and Ser 404.
    Journal of Alzheimer's disease : JAD, 2019, Volume: 68, Issue:3

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Animals; Blotting, Western; Calcium; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Humans; Lactones; Male; Maze Learning; Mice; Mice, Transgenic; Phosphorylation; Prostaglandin-E Synthases; Quinazolines; Real-Time Polymerase Chain Reaction; Serine; Sulfones; tau Proteins

2019