septide has been researched along with pyrrolidonecarboxylic acid in 81 studies
Studies (septide) | Trials (septide) | Recent Studies (post-2010) (septide) | Studies (pyrrolidonecarboxylic acid) | Trials (pyrrolidonecarboxylic acid) | Recent Studies (post-2010) (pyrrolidonecarboxylic acid) |
---|---|---|---|---|---|
84 | 0 | 2 | 3,005 | 101 | 671 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 6 (7.41) | 18.7374 |
1990's | 59 (72.84) | 18.2507 |
2000's | 14 (17.28) | 29.6817 |
2010's | 2 (2.47) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ferretti, JA; Jernigan, RL; Jiang, SP; Sumner, SC | 1 |
Chang, FY; Lee, SD; Wang, PS; Yeh, GH | 2 |
Beaujouan, JC; Chassaing, G; Glowinski, J; Lavielle, S; Loeuillet, D; Petitet, F; Saffroy, M; Torrens, Y | 1 |
Kisara, K; Ohba, M; Sakurada, S; Sakurada, T; Tan-No, K; Terenius, L; Yamada, T | 1 |
Andrews, PV; Boyd, RL; Eglezos, A; Helme, RD | 1 |
Eliakim, R; Karmeli, F; Okon, E; Rachmilewitz, D | 1 |
Guard, S; Suman-Chauhan, N; Watling, KJ; Williams, BJ | 1 |
Gunne, L; Johansson, PE; Liminga, U | 1 |
Maggi, CA; Patacchini, R; Quartara, L; Rovero, P; Santicioli, P | 1 |
Kisara, K; Manome, Y; Ohba, M; Sakurada, S; Sakurada, T; Tan-no, K; Yamada, T | 1 |
Byk, G; Chorev, M; Gilon, C; Halle, D; Selinger, Z | 1 |
Chang, FY; Ouyang, A; Sharp, D | 1 |
Fardin, V; Garret, C | 1 |
Chorev, M; Devor, M; Frey, J; Gilon, C; Laufer, R; Papir-Kricheli, D; Selinger, Z | 1 |
Magneney, S; Mayer, M; Michelot, R; Potier, P; Schmitt, P | 1 |
Drapeau, G; Maggi, CA; Meli, A; Patacchini, R; Regoli, D; Renzi, D; Rovero, P; Santicioli, P; Surrenti, C | 1 |
Chang, KS; Li, XS; Tanz, RD | 1 |
Harting, J; Reuss, K; Wienrich, M | 1 |
Barbanti, G; Beneforti, P; Maggi, CA; Meli, A; Patacchini, R; Rovero, P; Santicioli, P; Turini, D | 1 |
Beaujouan, JC; Glowinski, J; Saffroy, M; Torrens, Y | 2 |
Maggi, CA; Patacchini, R | 1 |
Bock, MD; Doble, A; Fardin, V; Garret, C; Heuillet, E; Le Guern, J; Mayaux, JF; Ménager, J; Pradier, L | 1 |
Fong, TM; Huang, RR; Strader, CD; Yu, H | 1 |
Bordey, A; Emonds-Alt, X; Feltz, P; Gauthier, T; Le Fur, G; Lefevre, IA; Oury-Donat, F; Soubrie, P; Thurneyssen, O | 1 |
Burcher, E; Lavielle, S; Zeng, XP | 1 |
Boni, P; Evangelista, S; Maggi, CA | 1 |
Maggi, CA; Meini, S; Patacchini, R | 1 |
Giachetti, A; Giuliani, S; Maggi, CA; Meini, S; Patacchini, R; Potier, E; Quartara, L; Sisto, A | 1 |
Hill, RG; Longmore, J; Razzaque, Z; Shaw, D | 1 |
Goso, C; Manzini, S; Palma, C | 1 |
Burcher, E; Stamatakos, C | 1 |
Brunissen, A; Carruette, A; Chassaing, G; Garret, C; Lavielle, S | 1 |
Hall, JM; Mitchell, D; Morton, IK | 1 |
Burcher, E; Zeng, XP | 1 |
Chang, DK; Guo, W; Lee, CM; Wong, TC | 1 |
Giuliani, S; Maggi, CA; Meini, S; Patacchini, R | 1 |
Bock, MD; Clerc, F; Fardin, V; Flamand, O; Foucault, F; Garret, C; Jolly, A | 1 |
Brunner, S; John, C; Tanaka, DT | 1 |
Ahluwalia, A; Giuliani, S; Maggi, CA | 1 |
Glowinski, J | 1 |
Betschart, J; Blanchard, JC; Garret, C; Grall, I; Piot, O; Ravard, S | 1 |
Chung, FZ; Huang, CC; Pu, Y; Tian, Y; Wu, LH | 1 |
Desban, M; Gauchy, C; Glowinski, J; Kemel, ML | 1 |
John, C; Kazem, E; Tanaka, DT | 1 |
Cavero, I; Floch, A; Thiry, C | 1 |
Bertrand, C; Emanueli, C; Figini, M; Geppetti, P; Javdan, P | 1 |
Carmody, J; Messlinger, K; Pawlak, M | 1 |
Chrétien, L; Gobeil, F; Jukic, D; Nguyen, QT; Nguyen-Le, XK; Regoli, D | 1 |
Hastrup, H; Schwartz, TW | 1 |
Fox, AJ; Naeem, S; Patel, IA; Urbán, L; Walpole, C | 1 |
Bertrand, C; Emanueli, C; Figini, M; Geppetti, P; Regoli, D; Sicuteri, R | 1 |
Beaujouan, JC; Chassaing, G; Glowinski, J; Lavielle, S; Saffroy, M; Sagan, S; Torrens, Y | 1 |
Bunnett, NW; Moore, BA; Sharkey, KA; Vanner, S | 1 |
Baamonde, A; Hidalgo, A; Menéndez, L | 1 |
Berthier, A; Dreux, C; Huleux, C; Rossignol, B | 1 |
Cody, C; Jones, RS; Maubach, KA | 1 |
Evans, RH; Ofner, S; Olpe, HR; Pozza, MF; Schoeffel, C | 1 |
Criscuoli, M; Lippi, A; Maggi, CA; Santicioli, P | 1 |
Bornstein, JC; Burcher, E; Johnson, PJ | 1 |
Bourque, MJ; Robitaille, R | 1 |
Ciucci, A; Manzini, S; Palma, C; Werge, TM | 1 |
Alvarez-Vega, M; Baamonde, A; Gutiérrez, M; Hidalgo, A; Menéndez, L | 1 |
Boquet, D; Couraud, JY; Créminon, C; Frobert, Y; Grassi, J; Sagot, MA; Wijkhuisen, A | 1 |
Barbot, L; Cellier, E; Couture, R; Iyengar, S | 1 |
Amadesi, S; Bertrand, C; Geppetti, P; Nadel, JA; Ricciardolo, FL; Trevisani, M | 1 |
Holzer, P; Shahbazian, A | 1 |
Bertrand, PP; Bian, XC; Bornstein, JC; Furness, JB | 1 |
Alvarez-Vega, M; Baamonde, A; Hidalgo, A; Menéndez, L | 1 |
Allouard, N; Bert, L; Bougault, I; Le-Fur, G; Rodier, D; Soubrié, P; Steinberg, R | 1 |
Glowinski, J; Godeheu, G; Kemel, ML; Pérez, S; Soubrié, P | 1 |
Baamonde, A; Hidalgo, A; Lastra, A; Menéndez, L; Villanueva, N | 1 |
Aggio, A; Ciccocioppo, R; Loreto, MF; Onori, L; Taddei, G; Tonini, M; Vicini, R | 1 |
Bolle, P; Severini, C; Tucci, P; Valeri, P | 1 |
Furuta, T; Kaneko, T; Koyano, K; Tomioka, R; Yanagawa, Y | 1 |
De Man, JG; De Schepper, HU; De Winter, BY; Herman, AG; Pelckmans, PA; Seerden, TC | 2 |
Bian, GL; Chen, LW; Wang, YQ; Wei, LC; Yung, KL | 1 |
Chan, YS; Chen, LW; Chu, JM; Yung, KK | 1 |
Bleeker, D; Heitman, LH; IJzerman, AP; Nederpelt, I; Tuijt, B | 1 |
1 review(s) available for septide and pyrrolidonecarboxylic acid
Article | Year |
---|---|
The 'septide-sensitive' tachykinin receptor: still an enigma.
Topics: Animals; Cell Line; DNA, Complementary; Guinea Pigs; Ileum; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Receptors, Tachykinin; Substance P; Transfection; Type C Phospholipases; Urinary Bladder | 1995 |
80 other study(ies) available for septide and pyrrolidonecarboxylic acid
Article | Year |
---|---|
Conformational analysis of receptor selective tachykinin analogs: senktide and septide.
Topics: Amino Acid Sequence; Circular Dichroism; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Peptide Fragments; Protein Conformation; Pyrrolidonecarboxylic Acid; Substance P | 1992 |
The motor actions of natural neurokinins and their specific agonists on the gastrointestinal tract of the rat.
Topics: Animals; Charcoal; Gastrointestinal Motility; Injections, Intraperitoneal; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Pilot Projects; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins | 1992 |
[A new tachykinin receptor revealed by substance P analogues in the guinea pig ileum].
Topics: Animals; Cell Membrane; Duodenum; Guinea Pigs; Ileum; Muscle Contraction; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P | 1992 |
N-terminal substance P fragments inhibit the spinally induced, NK 1 receptor mediated behavioural responses in mice.
Topics: Animals; Behavior, Animal; Bombesin; Injections, Spinal; Male; Mice; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Somatostatin; Spinal Cord; Substance P; Tachykinins | 1990 |
Tachykinin-mediated modulation of the primary antibody response in rats: evidence for mediation by an NK-2 receptor.
Topics: Animals; Animals, Newborn; Antibody Formation; Capsaicin; Denervation; Female; Immune System; Lymph Nodes; Male; Neurokinin A; Peptide Fragments; Peripheral Nerves; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins | 1991 |
Gastric mucosal damage by ethanol is mediated by substance P and prevented by ketotifen, a mast cell stabilizer.
Topics: Animals; Azepines; Cimetidine; Ethanol; Gastric Acid; Gastric Mucosa; Gastrins; Hydroxyzine; In Vitro Techniques; Ketotifen; Leukotriene B4; Male; Mast Cells; Pepsin A; Peptide Fragments; Platelet Activating Factor; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; SRS-A; Substance P; Triazoles | 1991 |
Pharmacological characterization of tachykinin-stimulated inositol phospholipid hydrolysis in peripheral tissues.
Topics: Animals; Cricetinae; Guinea Pigs; Hydrolysis; Ileum; In Vitro Techniques; Muscles; Parotid Gland; Peptide Fragments; Peptides, Cyclic; Phosphatidylinositols; Pyrrolidonecarboxylic Acid; Rats; Substance P; Tachykinins; Urinary Bladder | 1990 |
Intranigral tachykinin NK3 receptor agonist elicits oral movements in rats.
Topics: Animals; Female; Infusions, Parenteral; Mastication; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Substantia Nigra; Tachykinins | 1991 |
Tachykinin receptors in the guinea-pig isolated bronchi.
Topics: Amino Acid Sequence; Animals; Bronchi; Guinea Pigs; In Vitro Techniques; Male; Molecular Sequence Data; Neurokinin A; Oligopeptides; Peptide Fragments; Phenoxybenzamine; Protease Inhibitors; Pyrrolidonecarboxylic Acid; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tachykinins | 1991 |
Differential effects of substance P analogs on neurokinin 1 receptor agonists in the mouse spinal cord.
Topics: Analgesics; Animals; Behavior, Animal; Injections, Spinal; Male; Mice; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Spinal Cord; Substance P | 1991 |
Backbone cyclization: A new method for conferring conformational constraint on peptides.
Topics: Amino Acid Sequence; Cyclization; Molecular Sequence Data; Peptide Fragments; Peptides; Protein Conformation; Pyrrolidonecarboxylic Acid; Substance P | 1991 |
Multiple neurokinin receptor subtypes are present in the colon of the cat and rat.
Topics: Animals; Atropine; Cats; Colon; In Vitro Techniques; Isometric Contraction; Muscle, Smooth; Neurokinin B; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tetrodotoxin | 1991 |
Species differences between [3H] substance P binding in rat and guinea-pig shown by the use of peptide agonists and antagonists.
Topics: Animals; Brain Chemistry; Guinea Pigs; Ileum; In Vitro Techniques; Male; Peptide Fragments; Peptides; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Receptors, Tachykinin; Species Specificity; Substance P; Tachykinins | 1991 |
Behavioural effects of receptor-specific substance P agonists.
Topics: Animals; Behavior, Animal; Injections, Spinal; Male; Muscle Hypotonia; Pain Measurement; Paralysis; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Sciatic Nerve; Spinal Nerve Roots; Stereotyped Behavior; Substance P | 1987 |
N-acylated pentapeptides antagonists of substance P on guinea-pig ileum.
Topics: Acylation; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Oligopeptides; Peptide Fragments; Pyrrolidonecarboxylic Acid; Structure-Activity Relationship; Substance P | 1988 |
Effect of thiorphan on response of the guinea-pig gallbladder to tachykinins.
Topics: Animals; Captopril; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioimmunoassay; Substance P; Tachykinins; Thiorphan | 1989 |
Effect of age and methacholine on the rate and coronary flow of isolated hearts of diabetic rats.
Topics: Aging; Animals; Atropine; Blood Glucose; Body Weight; Coronary Circulation; Diabetes Mellitus, Experimental; Heart; Heart Rate; In Vitro Techniques; Male; Methacholine Compounds; Organ Size; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Substance P; Time Factors | 1989 |
Effects of receptor-selective neurokinin agonists and a neurokinin antagonist on the electrical activity of spinal cord neurones in culture.
Topics: Animals; Cells, Cultured; Electrophysiology; Female; Glutamates; Membrane Potentials; Microelectrodes; Neurons; Peptide Fragments; Pregnancy; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Spinal Cord; Substance P; Tetrodotoxin | 1989 |
Further studies on the motor response of the human isolated urinary bladder to tachykinins, capsaicin and electrical field stimulation.
Topics: Adult; Aged; Autonomic Nervous System; Calcitonin Gene-Related Peptide; Capsaicin; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Pyrrolidonecarboxylic Acid; Substance P; Tachykinins; Thiorphan; Urinary Bladder | 1989 |
Involvement of septide-sensitive tachykinin receptors in inositol phospholipid hydrolysis in the rat urinary bladder.
Topics: Amino Acid Sequence; Animals; Benzamides; Hydrolysis; Indoles; Isoindoles; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Phosphatidylinositols; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Urinary Bladder | 1995 |
Tachykinin NK1 receptors mediate both vasoconstrictor and vasodilator responses in the rabbit isolated jugular vein.
Topics: Animals; Dose-Response Relationship, Drug; Endothelium; Jugular Veins; Male; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Tachykinin; Substance P; Tachykinins; Vasoconstriction; Vasodilation | 1995 |
Septide: an agonist for the NK1 receptor acting at a site distinct from substance P.
Topics: Animals; Binding Sites; Binding, Competitive; Cell Line; Cell Membrane; Indoles; Inositol Phosphates; Isoindoles; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioligand Assay; Rats; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Transfection | 1994 |
Interaction of substance P with the second and seventh transmembrane domains of the neurokinin-1 receptor.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Peptide Fragments; Protein Structure, Secondary; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Transfection | 1994 |
SR 140333, a novel, selective, and potent nonpeptide antagonist of the NK1 tachykinin receptor: characterization on the U373MG cell line.
Topics: Astrocytoma; Binding, Competitive; Calcium; Electric Conductivity; Genes, fos; Humans; Inositol Phosphates; Iodine Radioisotopes; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Potassium; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Stereoisomerism; Substance P; Succinimides; Taurine; Transcription, Genetic; Tumor Cells, Cultured | 1994 |
Evidence for tachykinin NK-2 receptors in guinea-pig airways from binding and functional studies, using [125I]-[Lys5,Tyr(I2)7,MeLeu9,Nle10]-NKA(4-10).
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Bronchi; Drug Interactions; Female; Guinea Pigs; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neuropeptides; Peptide Fragments; Protease Inhibitors; Protein Binding; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Substance P; Tachykinins | 1994 |
In vivo evidence for the activation of a septide-sensitive tachykinin receptor in guinea pig bronchoconstriction.
Topics: Animals; Biphenyl Compounds; Bronchial Spasm; Bronchoconstriction; Dose-Response Relationship, Drug; Guinea Pigs; Hypnotics and Sedatives; Male; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Receptors, Tachykinin; Substance P; Sulfones | 1994 |
Tachykinin NK1 receptor subtypes in the rat urinary bladder.
Topics: Animals; Benzamides; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Tachykinin; Substance P; Sulfones; Tachykinins; Urinary Bladder | 1994 |
Comparison of tachykinin NK1 and NK2 receptors in the circular muscle of the guinea-pig ileum and proximal colon.
Topics: Animals; Colon; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Nifedipine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones | 1994 |
Differences in the effects of NK1-receptor antagonists, (+/-)-CP 96,345 and CP 99,994, on agonist-induced responses in guinea-pig trachea.
Topics: Animals; Biphenyl Compounds; Guinea Pigs; In Vitro Techniques; Indoles; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Substance P; Trachea | 1994 |
Different susceptibility to neurokinin 1 receptor antagonists of substance P and septide-induced interleukin-6 release from U373 MG human astrocytoma cell line.
Topics: Astrocytoma; Binding, Competitive; Brain Neoplasms; Humans; Interleukin-6; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Pyrrolidonecarboxylic Acid; Substance P; Tumor Cells, Cultured | 1994 |
Septide but not substance P stimulates inhibitory neurons in guinea-pig ileum.
Topics: Animals; Guinea Pigs; Ileum; In Vitro Techniques; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P | 1994 |
Highly potent substance P antagonists substituted with beta-phenyl- or beta-benzyl-proline at position 10.
Topics: Amino Acid Sequence; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Rabbits; Rats; Receptors, Neurokinin-1; Structure-Activity Relationship; Substance P | 1994 |
Typical and atypical NK1 tachykinin receptor characteristics in the rabbit isolated iris sphincter.
Topics: Animals; In Vitro Techniques; Iris; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phenoxybenzamine; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P | 1994 |
Use of selective antagonists for further characterization of tachykinin NK-2, NK-1 and possible "septide-selective" receptors in guinea pig bronchus.
Topics: Amino Acid Sequence; Animals; Bronchi; Female; Guinea Pigs; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Substance P; Tachykinins | 1994 |
Conformational study of two substance P hexapeptides by two-dimensional NMR.
Topics: Amino Acid Sequence; Chloroform; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Peptide Fragments; Protein Conformation; Protein Folding; Pyrrolidonecarboxylic Acid; Solvents; Stereoisomerism; Substance P; Trifluoroethanol; Water | 1993 |
Evidence for the presence of a septide-sensitive tachykinin receptor in the circular muscle of the guinea-pig ileum.
Topics: Animals; Biphenyl Compounds; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscles; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tachykinins | 1993 |
Variations in affinities for the NK1 receptor: differences between the non-peptide substance P antagonists RP 67580 and CP-96,345 and the agonist septide.
Topics: Animals; Binding, Competitive; Biphenyl Compounds; Brain; Cell Line; Dogs; Guinea Pigs; Humans; Indoles; Isoindoles; Mice; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Receptors, Neurokinin-1; Submandibular Gland; Substance P | 1993 |
Neuromodulation mediated by neurokinin-1 subtype receptors in adult rabbit airways.
Topics: Acetylcholine; Animals; Electric Stimulation; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nervous System Physiological Phenomena; Parasympathetic Nervous System; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tetrodotoxin; Trachea | 1993 |
Demonstration of a 'septide-sensitive' inflammatory response in rat skin.
Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Blood Proteins; Capillary Permeability; Dermatitis, Contact; Dose-Response Relationship, Drug; Edema; Indoles; Isoindoles; Male; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Nitric Oxide Synthase; p-Methoxy-N-methylphenethylamine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P | 1995 |
Comparative behavioural profile of centrally administered tachykinin NK1, NK2 and NK3 receptor agonists in the guinea-pig.
Topics: Animals; Behavior, Animal; Guinea Pigs; Injections, Intraventricular; Male; Motor Activity; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P | 1995 |
Structural motifs encoded by individual exons of the human neurokinin-1 receptor gene interact differentially with selective agonists and antagonists.
Topics: Amino Acid Sequence; Cloning, Molecular; Exons; Humans; Iodine Radioisotopes; Molecular Sequence Data; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phosphatidylinositols; Piperidines; Protein Binding; Pyrrolidonecarboxylic Acid; Quinuclidines; Radioligand Assay; Receptors, Neurokinin-1; Recombinant Fusion Proteins; Stereoisomerism; Substance P | 1996 |
Distinct regulations by septide and the neurokinin-1 tachykinin receptor agonist [pro9]substance P of the N-methyl-D-aspartate-evoked release of dopamine in striosome- and matrix-enriched areas of the rat striatum.
Topics: Animals; Corpus Striatum; Dopamine; Extracellular Matrix; Indoles; Isoindoles; Male; N-Methylaspartate; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P | 1996 |
Neurokinin subtype receptors mediating substance P contraction in immature rabbit airways.
Topics: Animals; Atropine; Bronchi; Glycopeptides; Isometric Contraction; Muscle, Smooth; Neostigmine; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea | 1996 |
Pharmacological evidence that NK-2 tachykinin receptors mediate hypotension in the guinea pig but not in the rat.
Topics: Animals; Benzamides; Blood Pressure; Guinea Pigs; Hypotension; Indoles; Isoindoles; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P | 1996 |
Evidence that tachykinins relax the guinea-pig trachea via nitric oxide release and by stimulation of a septide-insensitive NK1 receptor.
Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Neurokinin A; Neurokinin B; Nitric Oxide; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P; Tachykinins; Trachea | 1996 |
Lack of a role for substance P in the control of dural arterial flow.
Topics: Animals; Cerebral Arteries; Dura Mater; Electric Stimulation; Indoles; Isoindoles; Laser-Doppler Flowmetry; Male; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Regional Blood Flow; Substance P | 1996 |
Neurokinin receptors in the guinea pig ileum.
Topics: Acetylcholine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Guinea Pigs; Ileum; Male; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stereoisomerism; Structure-Activity Relationship; Substance P | 1996 |
Septide and neurokinin A are high-affinity ligands on the NK-1 receptor: evidence from homologous versus heterologous binding analysis.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; COS Cells; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Protein Binding; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P | 1996 |
Receptors mediating tachykinin-evoked depolarisations of neurons in the neonatal rat spinal cord.
Topics: Animals; Animals, Newborn; Biphenyl Compounds; Evoked Potentials; In Vitro Techniques; Indoles; Isoindoles; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spinal Cord; Substance P; Tachykinins | 1996 |
Differential activation of the epithelial and smooth muscle NK1 receptors by synthetic tachykinin agonists in guinea-pig trachea.
Topics: Animals; Dose-Response Relationship, Drug; Epithelium; Guinea Pigs; Male; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Peptide Fragments; Physalaemin; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Substance P; Tachykinins; Trachea | 1997 |
High affinity binding of [3H]propionyl-[Met(O2)11]substance P(7-11), a tritiated septide-like peptide, in Chinese hamster ovary cells expressing human neurokinin-1 receptors and in rat submandibular glands.
Topics: Animals; Binding Sites; CHO Cells; Cricetinae; Male; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Submandibular Gland; Substance P | 1997 |
Characterization of neurokinin-1 receptors in the submucosal plexus of guinea pig ileum.
Topics: Animals; Electric Stimulation; Female; Ganglia, Autonomic; Guinea Pigs; Ileum; Immunohistochemistry; In Vitro Techniques; Intestinal Mucosa; Male; Membrane Potentials; Microscopy, Video; Muscle, Smooth; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rabbits; Rats; Receptors, Neurokinin-1; Submucous Plexus; Substance P; Vasodilation | 1997 |
Spinal calmodulin inhibitors reduce N-methyl-D-aspartate- and septide-induced nociceptive behavior.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Enzyme Inhibitors; Imidazoles; Injections, Intraventricular; Male; N-Methylaspartate; Neurokinin A; Pain; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Spinal Cord; Substance P; Sulfonamides | 1997 |
A "septide-sensitive" receptor is not involved in tachykinin-mediated secretory and inositol phosphate responses in rat parotid gland: are several transduction pathways involved after the stimulation of the NK1 receptor?
Topics: Animals; Cells, Cultured; Indoles; Inositol Phosphates; Isoindoles; Kinetics; Male; Neurokinin-1 Receptor Antagonists; Parotid Gland; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Salivary Proteins and Peptides; Signal Transduction; Substance P; Tachykinins | 1998 |
Tachykinins may modify spontaneous epileptiform activity in the rat entorhinal cortex in vitro by activating GABAergic inhibition.
Topics: Animals; Baclofen; Bicuculline; Entorhinal Cortex; Epilepsy; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Phosphinic Acids; Propanolamines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Substance P; Synapses; Tachykinins | 1998 |
The potency of the novel tachykinin receptor antagonist CGP49823 at rat and gerbil motoneurones in vitro.
Topics: Animals; Anti-Anxiety Agents; Gerbillinae; In Vitro Techniques; Motor Neurons; Neurokinin-1 Receptor Antagonists; Neuromuscular Depolarizing Agents; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinolines; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P | 1998 |
Depolarization evoked co-release of tachykinins from enteric nerves in the guinea-pig proximal colon.
Topics: Animals; Calcium; Colon; Enteric Nervous System; Guinea Pigs; Neurokinin A; Peptide Fragments; Piperidines; Potassium Chloride; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Tachykinin; Substance P; Tachykinins | 1998 |
Roles of neuronal NK1 and NK3 receptors in synaptic transmission during motility reflexes in the guinea-pig ileum.
Topics: Animals; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Synaptic Transmission | 1998 |
Endogenous peptidergic modulation of perisynaptic Schwann cells at the frog neuromuscular junction.
Topics: Acetylcholinesterase; Animals; Calcium; GTP-Binding Proteins; Muscarine; Muscle, Skeletal; Neostigmine; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Peptide Fragments; Pertussis Toxin; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rana pipiens; Receptors, Neurokinin-1; Schwann Cells; Substance P; Synapses; Virulence Factors, Bordetella | 1998 |
Point mutation increases a form of the NK1 receptor with high affinity for neurokinin A and B and septide.
Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Neurokinin A; Neurokinin B; Peptide Fragments; Point Mutation; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-1; Recombinant Proteins; Substance P | 1998 |
Comparison of the effects of calmidazolium, morphine and bupivacaine on N-methyl-D-aspartate- and septide-induced nociceptive behaviour.
Topics: Analgesics; Animals; Bupivacaine; Imidazoles; Male; Morphine; N-Methylaspartate; Pain; Pain Measurement; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Spinal Cord; Substance P | 1998 |
Rat gastrointestinal motor responses mediated via activation of neurokinin receptors.
Topics: Animals; Chromates; Chromium Radioisotopes; Gastric Emptying; Gastrointestinal Motility; Intubation, Gastrointestinal; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sodium Compounds; Substance P | 1999 |
Identification in the NK1 tachykinin receptor of a domain involved in recognition of neurokinin A and septide but not of substance P.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Chlorocebus aethiops; COS Cells; DNA, Complementary; Humans; In Vitro Techniques; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Point Mutation; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Tachykinins | 1999 |
Characterization of central and peripheral effects of septide with the use of five tachykinin NK1 receptor antagonists in the rat.
Topics: Acetamides; Animals; Behavior, Animal; Blood Pressure; Capillary Permeability; Heart Rate; Indoles; Injections, Intraventricular; Male; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-1; Stereoisomerism; Substance P | 1999 |
Role of nitric oxide and septide-insensitive NK(1) receptors in bronchoconstriction induced by aerosolised neurokinin A in guinea-pigs.
Topics: Aerosols; Airway Resistance; Animals; Bronchoconstriction; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P | 2000 |
Further evidence for the presence of "septide-sensitive" tachykinin binding sites in tissues possessing solely NK(1) tachykinin receptors.
Topics: Animals; Binding Sites; CHO Cells; Cricetinae; Humans; Indoles; Iodine Radioisotopes; Isoindoles; Mice; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protein Isoforms; Pyrrolidonecarboxylic Acid; Radioligand Assay; Rats; Receptors, Neurokinin-1; Substance P; Tetrazoles; Tumor Cells, Cultured | 2000 |
Differences in circular muscle contraction and peristaltic motor inhibition caused by tachykinin NK1 receptor agonists in the guinea-pig small intestine.
Topics: Adenosine Triphosphate; Animals; Enzyme Inhibitors; Female; Guinea Pigs; Intestine, Small; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Piperidines; Purinergic P2 Receptor Antagonists; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sincalide; Spasm; Substance P; Suramin; Tetrodotoxin | 2000 |
Evidence for functional NK1-tachykinin receptors on motor neurones supplying the circular muscle of guinea-pig small and large intestine.
Topics: Animals; Colon; Duodenum; Enzyme Inhibitors; Guinea Pigs; Ileum; Immunohistochemistry; In Vitro Techniques; Indomethacin; Motor Neurons; Muscle, Smooth; Nitric Oxide Synthase; Nitroarginine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P | 2000 |
Effects of the calcium release inhibitor dantrolene and the Ca2+-ATPase inhibitor thapsigargin on spinal nociception in rats.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics; Animals; Behavior, Animal; Calcium; Calcium-Transporting ATPases; Dantrolene; Enzyme Inhibitors; Male; Muscle Relaxants, Central; N-Methylaspartate; Pain; Pain Measurement; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Spinal Cord; Substance P; Thapsigargin | 2001 |
Permissive role of neurokinin NK(3) receptors in NK(1) receptor-mediated activation of the locus coeruleus revealed by SR 142801.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiemetics; Dose-Response Relationship, Drug; Guinea Pigs; Locus Coeruleus; Male; Neural Pathways; Neurokinin-1 Receptor Antagonists; Neurons; Norepinephrine; Peptide Fragments; Piperidines; Prefrontal Cortex; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tetrazoles | 2002 |
Facilitation by endogenous tachykinins of the NMDA-evoked release of acetylcholine after acute and chronic suppression of dopaminergic transmission in the matrix of the rat striatum.
Topics: Acetylcholine; Animals; Benzamides; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Inhibitors; In Vitro Techniques; Male; N-Methylaspartate; Neural Inhibition; Neurons; Oxidopamine; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Synaptic Transmission; Tachykinins; Time Factors | 2002 |
Spinal nociceptin inhibits septide but not N-methyl-D-aspartate-induced nociceptive behavior in rats.
Topics: Animals; Behavior, Animal; Injections, Spinal; Male; N-Methylaspartate; Naloxone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Opioid; Spinal Cord; Substance P | 2002 |
Peristalsis regulation by tachykinin NK1 receptors in the rabbit isolated distal colon.
Topics: Alanine; Animals; Atropine; Colon; Drug Interactions; Enzyme Inhibitors; Indoles; Kinetics; Male; Neurokinin-1 Receptor Antagonists; Nitric Oxide Synthase; Nitroarginine; Peptide Fragments; Peristalsis; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rabbits; Receptors, Neurokinin-1; Substance P | 2003 |
Biologic activity of the tachykinins on lamb and sheep gallbladder.
Topics: Animals; Binding Sites; Capsaicin; Dose-Response Relationship, Drug; Female; Gallbladder; Male; Muscles; Neurokinin A; Neurokinin B; Peptide Fragments; Physalaemin; Protein Structure, Tertiary; Pyrrolidonecarboxylic Acid; Receptors, Tachykinin; Sheep; Substance P; Tachykinins | 2003 |
GABAergic basal forebrain neurons that express receptor for neurokinin B and send axons to the cerebral cortex.
Topics: Animals; Animals, Newborn; Axons; Calbindin 2; Calbindins; Cell Count; Cerebral Cortex; Cholera Toxin; Choline O-Acetyltransferase; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Immunoenzyme Techniques; Immunohistochemistry; In Situ Hybridization; In Vitro Techniques; Isoenzymes; Male; Membrane Potentials; Neurons; Neuropeptide Y; Parvalbumins; Patch-Clamp Techniques; Peptide Fragments; Polypyrimidine Tract-Binding Protein; Prosencephalon; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-3; S100 Calcium Binding Protein G; Somatostatin; Substance P; Wheat Germ Agglutinin-Horseradish Peroxidase Conjugate | 2004 |
Functional characterisation of tachykinin receptors in the circular muscle layer of the mouse ileum.
Topics: Action Potentials; Analgesics; Animals; Antipsychotic Agents; Atropine; Electric Stimulation; Ileum; Indoles; Isoindoles; Mice; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Nitroarginine; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P | 2005 |
The role of tachykinins in circular muscle contractility of the murine ileum: a functional investigation.
Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Ilium; In Vitro Techniques; Male; Mice; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nitroarginine; Peptide Fragments; Potassium Chloride; Pyrrolidonecarboxylic Acid; Substance P; Tachykinins; Tetrodotoxin | 2006 |
Neurokinin-3 peptide instead of neurokinin-1 synergistically exacerbates kainic acid-inducing degeneration of neurons in the substantia nigra of mice.
Topics: Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Drug Synergism; Fluoresceins; Kainic Acid; Male; Mice; Mice, Inbred Strains; Nerve Degeneration; Nerve Tissue Proteins; Neurokinin-1 Receptor Antagonists; Neurons; Organic Chemicals; Peptide Fragments; Pyrrolidonecarboxylic Acid; Quinolines; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Substantia Nigra; Tetrazolium Salts; Thiazoles | 2008 |
Neuroprotective effects of neurokinin receptor one in dopaminergic neurons are mediated through Akt/PKB cell signaling pathway.
Topics: Analysis of Variance; Animals; Apomorphine; bcl-Associated Death Protein; Caspase 3; Cell Death; Cell Line, Tumor; Corpus Striatum; Disease Models, Animal; Dopamine Agonists; Dopaminergic Neurons; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Gene Expression Regulation; L-Lactate Dehydrogenase; Male; Motor Activity; Neuroblastoma; Neurokinin-1 Receptor Antagonists; Neuroprotective Agents; Neurotoxicity Syndromes; Oxidopamine; Peptide Fragments; Proto-Oncogene Proteins c-akt; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Rotarod Performance Test; Signal Transduction; Substance P; Sympatholytics; Time Factors; Tyrosine 3-Monooxygenase | 2011 |
Kinetic binding and activation profiles of endogenous tachykinins targeting the NK1 receptor.
Topics: Algorithms; Animals; Astrocytoma; Binding, Competitive; Cell Line, Tumor; CHO Cells; Cricetulus; Electric Impedance; Humans; Kinetics; Ligands; Nerve Tissue Proteins; Neuroglia; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Tachykinins | 2016 |