Page last updated: 2024-09-03

septide and pyrrolidonecarboxylic acid

septide has been researched along with pyrrolidonecarboxylic acid in 81 studies

Compound Research Comparison

Studies
(septide)
Trials
(septide)
Recent Studies (post-2010)
(septide)
Studies
(pyrrolidonecarboxylic acid)
Trials
(pyrrolidonecarboxylic acid)
Recent Studies (post-2010) (pyrrolidonecarboxylic acid)
84023,005101671

Research

Studies (81)

TimeframeStudies, this research(%)All Research%
pre-19906 (7.41)18.7374
1990's59 (72.84)18.2507
2000's14 (17.28)29.6817
2010's2 (2.47)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ferretti, JA; Jernigan, RL; Jiang, SP; Sumner, SC1
Chang, FY; Lee, SD; Wang, PS; Yeh, GH2
Beaujouan, JC; Chassaing, G; Glowinski, J; Lavielle, S; Loeuillet, D; Petitet, F; Saffroy, M; Torrens, Y1
Kisara, K; Ohba, M; Sakurada, S; Sakurada, T; Tan-No, K; Terenius, L; Yamada, T1
Andrews, PV; Boyd, RL; Eglezos, A; Helme, RD1
Eliakim, R; Karmeli, F; Okon, E; Rachmilewitz, D1
Guard, S; Suman-Chauhan, N; Watling, KJ; Williams, BJ1
Gunne, L; Johansson, PE; Liminga, U1
Maggi, CA; Patacchini, R; Quartara, L; Rovero, P; Santicioli, P1
Kisara, K; Manome, Y; Ohba, M; Sakurada, S; Sakurada, T; Tan-no, K; Yamada, T1
Byk, G; Chorev, M; Gilon, C; Halle, D; Selinger, Z1
Chang, FY; Ouyang, A; Sharp, D1
Fardin, V; Garret, C1
Chorev, M; Devor, M; Frey, J; Gilon, C; Laufer, R; Papir-Kricheli, D; Selinger, Z1
Magneney, S; Mayer, M; Michelot, R; Potier, P; Schmitt, P1
Drapeau, G; Maggi, CA; Meli, A; Patacchini, R; Regoli, D; Renzi, D; Rovero, P; Santicioli, P; Surrenti, C1
Chang, KS; Li, XS; Tanz, RD1
Harting, J; Reuss, K; Wienrich, M1
Barbanti, G; Beneforti, P; Maggi, CA; Meli, A; Patacchini, R; Rovero, P; Santicioli, P; Turini, D1
Beaujouan, JC; Glowinski, J; Saffroy, M; Torrens, Y2
Maggi, CA; Patacchini, R1
Bock, MD; Doble, A; Fardin, V; Garret, C; Heuillet, E; Le Guern, J; Mayaux, JF; Ménager, J; Pradier, L1
Fong, TM; Huang, RR; Strader, CD; Yu, H1
Bordey, A; Emonds-Alt, X; Feltz, P; Gauthier, T; Le Fur, G; Lefevre, IA; Oury-Donat, F; Soubrie, P; Thurneyssen, O1
Burcher, E; Lavielle, S; Zeng, XP1
Boni, P; Evangelista, S; Maggi, CA1
Maggi, CA; Meini, S; Patacchini, R1
Giachetti, A; Giuliani, S; Maggi, CA; Meini, S; Patacchini, R; Potier, E; Quartara, L; Sisto, A1
Hill, RG; Longmore, J; Razzaque, Z; Shaw, D1
Goso, C; Manzini, S; Palma, C1
Burcher, E; Stamatakos, C1
Brunissen, A; Carruette, A; Chassaing, G; Garret, C; Lavielle, S1
Hall, JM; Mitchell, D; Morton, IK1
Burcher, E; Zeng, XP1
Chang, DK; Guo, W; Lee, CM; Wong, TC1
Giuliani, S; Maggi, CA; Meini, S; Patacchini, R1
Bock, MD; Clerc, F; Fardin, V; Flamand, O; Foucault, F; Garret, C; Jolly, A1
Brunner, S; John, C; Tanaka, DT1
Ahluwalia, A; Giuliani, S; Maggi, CA1
Glowinski, J1
Betschart, J; Blanchard, JC; Garret, C; Grall, I; Piot, O; Ravard, S1
Chung, FZ; Huang, CC; Pu, Y; Tian, Y; Wu, LH1
Desban, M; Gauchy, C; Glowinski, J; Kemel, ML1
John, C; Kazem, E; Tanaka, DT1
Cavero, I; Floch, A; Thiry, C1
Bertrand, C; Emanueli, C; Figini, M; Geppetti, P; Javdan, P1
Carmody, J; Messlinger, K; Pawlak, M1
Chrétien, L; Gobeil, F; Jukic, D; Nguyen, QT; Nguyen-Le, XK; Regoli, D1
Hastrup, H; Schwartz, TW1
Fox, AJ; Naeem, S; Patel, IA; Urbán, L; Walpole, C1
Bertrand, C; Emanueli, C; Figini, M; Geppetti, P; Regoli, D; Sicuteri, R1
Beaujouan, JC; Chassaing, G; Glowinski, J; Lavielle, S; Saffroy, M; Sagan, S; Torrens, Y1
Bunnett, NW; Moore, BA; Sharkey, KA; Vanner, S1
Baamonde, A; Hidalgo, A; Menéndez, L1
Berthier, A; Dreux, C; Huleux, C; Rossignol, B1
Cody, C; Jones, RS; Maubach, KA1
Evans, RH; Ofner, S; Olpe, HR; Pozza, MF; Schoeffel, C1
Criscuoli, M; Lippi, A; Maggi, CA; Santicioli, P1
Bornstein, JC; Burcher, E; Johnson, PJ1
Bourque, MJ; Robitaille, R1
Ciucci, A; Manzini, S; Palma, C; Werge, TM1
Alvarez-Vega, M; Baamonde, A; Gutiérrez, M; Hidalgo, A; Menéndez, L1
Boquet, D; Couraud, JY; Créminon, C; Frobert, Y; Grassi, J; Sagot, MA; Wijkhuisen, A1
Barbot, L; Cellier, E; Couture, R; Iyengar, S1
Amadesi, S; Bertrand, C; Geppetti, P; Nadel, JA; Ricciardolo, FL; Trevisani, M1
Holzer, P; Shahbazian, A1
Bertrand, PP; Bian, XC; Bornstein, JC; Furness, JB1
Alvarez-Vega, M; Baamonde, A; Hidalgo, A; Menéndez, L1
Allouard, N; Bert, L; Bougault, I; Le-Fur, G; Rodier, D; Soubrié, P; Steinberg, R1
Glowinski, J; Godeheu, G; Kemel, ML; Pérez, S; Soubrié, P1
Baamonde, A; Hidalgo, A; Lastra, A; Menéndez, L; Villanueva, N1
Aggio, A; Ciccocioppo, R; Loreto, MF; Onori, L; Taddei, G; Tonini, M; Vicini, R1
Bolle, P; Severini, C; Tucci, P; Valeri, P1
Furuta, T; Kaneko, T; Koyano, K; Tomioka, R; Yanagawa, Y1
De Man, JG; De Schepper, HU; De Winter, BY; Herman, AG; Pelckmans, PA; Seerden, TC2
Bian, GL; Chen, LW; Wang, YQ; Wei, LC; Yung, KL1
Chan, YS; Chen, LW; Chu, JM; Yung, KK1
Bleeker, D; Heitman, LH; IJzerman, AP; Nederpelt, I; Tuijt, B1

Reviews

1 review(s) available for septide and pyrrolidonecarboxylic acid

ArticleYear
The 'septide-sensitive' tachykinin receptor: still an enigma.
    Trends in pharmacological sciences, 1995, Volume: 16, Issue:11

    Topics: Animals; Cell Line; DNA, Complementary; Guinea Pigs; Ileum; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Receptors, Tachykinin; Substance P; Transfection; Type C Phospholipases; Urinary Bladder

1995

Other Studies

80 other study(ies) available for septide and pyrrolidonecarboxylic acid

ArticleYear
Conformational analysis of receptor selective tachykinin analogs: senktide and septide.
    Journal of biomolecular structure & dynamics, 1992, Volume: 10, Issue:3

    Topics: Amino Acid Sequence; Circular Dichroism; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Peptide Fragments; Protein Conformation; Pyrrolidonecarboxylic Acid; Substance P

1992
The motor actions of natural neurokinins and their specific agonists on the gastrointestinal tract of the rat.
    The Chinese journal of physiology, 1992, Volume: 35, Issue:4

    Topics: Animals; Charcoal; Gastrointestinal Motility; Injections, Intraperitoneal; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Pilot Projects; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins

1992
[A new tachykinin receptor revealed by substance P analogues in the guinea pig ileum].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 1992, Mar-26, Volume: 314, Issue:7

    Topics: Animals; Cell Membrane; Duodenum; Guinea Pigs; Ileum; Muscle Contraction; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P

1992
N-terminal substance P fragments inhibit the spinally induced, NK 1 receptor mediated behavioural responses in mice.
    Life sciences, 1990, Volume: 47, Issue:20

    Topics: Animals; Behavior, Animal; Bombesin; Injections, Spinal; Male; Mice; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Somatostatin; Spinal Cord; Substance P; Tachykinins

1990
Tachykinin-mediated modulation of the primary antibody response in rats: evidence for mediation by an NK-2 receptor.
    Journal of neuroimmunology, 1991, Volume: 32, Issue:1

    Topics: Animals; Animals, Newborn; Antibody Formation; Capsaicin; Denervation; Female; Immune System; Lymph Nodes; Male; Neurokinin A; Peptide Fragments; Peripheral Nerves; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins

1991
Gastric mucosal damage by ethanol is mediated by substance P and prevented by ketotifen, a mast cell stabilizer.
    Gastroenterology, 1991, Volume: 100, Issue:5 Pt 1

    Topics: Animals; Azepines; Cimetidine; Ethanol; Gastric Acid; Gastric Mucosa; Gastrins; Hydroxyzine; In Vitro Techniques; Ketotifen; Leukotriene B4; Male; Mast Cells; Pepsin A; Peptide Fragments; Platelet Activating Factor; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; SRS-A; Substance P; Triazoles

1991
Pharmacological characterization of tachykinin-stimulated inositol phospholipid hydrolysis in peripheral tissues.
    British journal of pharmacology, 1990, Volume: 101, Issue:4

    Topics: Animals; Cricetinae; Guinea Pigs; Hydrolysis; Ileum; In Vitro Techniques; Muscles; Parotid Gland; Peptide Fragments; Peptides, Cyclic; Phosphatidylinositols; Pyrrolidonecarboxylic Acid; Rats; Substance P; Tachykinins; Urinary Bladder

1990
Intranigral tachykinin NK3 receptor agonist elicits oral movements in rats.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 38, Issue:3

    Topics: Animals; Female; Infusions, Parenteral; Mastication; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Substantia Nigra; Tachykinins

1991
Tachykinin receptors in the guinea-pig isolated bronchi.
    European journal of pharmacology, 1991, May-17, Volume: 197, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Bronchi; Guinea Pigs; In Vitro Techniques; Male; Molecular Sequence Data; Neurokinin A; Oligopeptides; Peptide Fragments; Phenoxybenzamine; Protease Inhibitors; Pyrrolidonecarboxylic Acid; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tachykinins

1991
Differential effects of substance P analogs on neurokinin 1 receptor agonists in the mouse spinal cord.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:1

    Topics: Analgesics; Animals; Behavior, Animal; Injections, Spinal; Male; Mice; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Spinal Cord; Substance P

1991
Backbone cyclization: A new method for conferring conformational constraint on peptides.
    Biopolymers, 1991, Volume: 31, Issue:6

    Topics: Amino Acid Sequence; Cyclization; Molecular Sequence Data; Peptide Fragments; Peptides; Protein Conformation; Pyrrolidonecarboxylic Acid; Substance P

1991
Multiple neurokinin receptor subtypes are present in the colon of the cat and rat.
    Annals of the New York Academy of Sciences, 1991, Volume: 632

    Topics: Animals; Atropine; Cats; Colon; In Vitro Techniques; Isometric Contraction; Muscle, Smooth; Neurokinin B; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tetrodotoxin

1991
Species differences between [3H] substance P binding in rat and guinea-pig shown by the use of peptide agonists and antagonists.
    European journal of pharmacology, 1991, Aug-29, Volume: 201, Issue:2-3

    Topics: Animals; Brain Chemistry; Guinea Pigs; Ileum; In Vitro Techniques; Male; Peptide Fragments; Peptides; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Receptors, Tachykinin; Species Specificity; Substance P; Tachykinins

1991
Behavioural effects of receptor-specific substance P agonists.
    Pain, 1987, Volume: 31, Issue:2

    Topics: Animals; Behavior, Animal; Injections, Spinal; Male; Muscle Hypotonia; Pain Measurement; Paralysis; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Sciatic Nerve; Spinal Nerve Roots; Stereotyped Behavior; Substance P

1987
N-acylated pentapeptides antagonists of substance P on guinea-pig ileum.
    Biochemical and biophysical research communications, 1988, Oct-14, Volume: 156, Issue:1

    Topics: Acylation; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Oligopeptides; Peptide Fragments; Pyrrolidonecarboxylic Acid; Structure-Activity Relationship; Substance P

1988
Effect of thiorphan on response of the guinea-pig gallbladder to tachykinins.
    European journal of pharmacology, 1989, Jun-08, Volume: 165, Issue:1

    Topics: Animals; Captopril; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioimmunoassay; Substance P; Tachykinins; Thiorphan

1989
Effect of age and methacholine on the rate and coronary flow of isolated hearts of diabetic rats.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: Aging; Animals; Atropine; Blood Glucose; Body Weight; Coronary Circulation; Diabetes Mellitus, Experimental; Heart; Heart Rate; In Vitro Techniques; Male; Methacholine Compounds; Organ Size; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Substance P; Time Factors

1989
Effects of receptor-selective neurokinin agonists and a neurokinin antagonist on the electrical activity of spinal cord neurones in culture.
    British journal of pharmacology, 1989, Volume: 98, Issue:3

    Topics: Animals; Cells, Cultured; Electrophysiology; Female; Glutamates; Membrane Potentials; Microelectrodes; Neurons; Peptide Fragments; Pregnancy; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Spinal Cord; Substance P; Tetrodotoxin

1989
Further studies on the motor response of the human isolated urinary bladder to tachykinins, capsaicin and electrical field stimulation.
    General pharmacology, 1989, Volume: 20, Issue:5

    Topics: Adult; Aged; Autonomic Nervous System; Calcitonin Gene-Related Peptide; Capsaicin; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Pyrrolidonecarboxylic Acid; Substance P; Tachykinins; Thiorphan; Urinary Bladder

1989
Involvement of septide-sensitive tachykinin receptors in inositol phospholipid hydrolysis in the rat urinary bladder.
    Peptides, 1995, Volume: 16, Issue:4

    Topics: Amino Acid Sequence; Animals; Benzamides; Hydrolysis; Indoles; Isoindoles; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Phosphatidylinositols; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Urinary Bladder

1995
Tachykinin NK1 receptors mediate both vasoconstrictor and vasodilator responses in the rabbit isolated jugular vein.
    European journal of pharmacology, 1995, Sep-05, Volume: 283, Issue:1-3

    Topics: Animals; Dose-Response Relationship, Drug; Endothelium; Jugular Veins; Male; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Tachykinin; Substance P; Tachykinins; Vasoconstriction; Vasodilation

1995
Septide: an agonist for the NK1 receptor acting at a site distinct from substance P.
    Molecular pharmacology, 1994, Volume: 45, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Cell Line; Cell Membrane; Indoles; Inositol Phosphates; Isoindoles; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioligand Assay; Rats; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Transfection

1994
Interaction of substance P with the second and seventh transmembrane domains of the neurokinin-1 receptor.
    Biochemistry, 1994, Mar-15, Volume: 33, Issue:10

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Peptide Fragments; Protein Structure, Secondary; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Transfection

1994
SR 140333, a novel, selective, and potent nonpeptide antagonist of the NK1 tachykinin receptor: characterization on the U373MG cell line.
    Journal of neurochemistry, 1994, Volume: 62, Issue:4

    Topics: Astrocytoma; Binding, Competitive; Calcium; Electric Conductivity; Genes, fos; Humans; Inositol Phosphates; Iodine Radioisotopes; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Potassium; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Stereoisomerism; Substance P; Succinimides; Taurine; Transcription, Genetic; Tumor Cells, Cultured

1994
Evidence for tachykinin NK-2 receptors in guinea-pig airways from binding and functional studies, using [125I]-[Lys5,Tyr(I2)7,MeLeu9,Nle10]-NKA(4-10).
    Neuropeptides, 1994, Volume: 26, Issue:1

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Bronchi; Drug Interactions; Female; Guinea Pigs; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neuropeptides; Peptide Fragments; Protease Inhibitors; Protein Binding; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Substance P; Tachykinins

1994
In vivo evidence for the activation of a septide-sensitive tachykinin receptor in guinea pig bronchoconstriction.
    Life sciences, 1994, Volume: 54, Issue:19

    Topics: Animals; Biphenyl Compounds; Bronchial Spasm; Bronchoconstriction; Dose-Response Relationship, Drug; Guinea Pigs; Hypnotics and Sedatives; Male; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Receptors, Tachykinin; Substance P; Sulfones

1994
Tachykinin NK1 receptor subtypes in the rat urinary bladder.
    British journal of pharmacology, 1994, Volume: 111, Issue:3

    Topics: Animals; Benzamides; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Tachykinin; Substance P; Sulfones; Tachykinins; Urinary Bladder

1994
Comparison of tachykinin NK1 and NK2 receptors in the circular muscle of the guinea-pig ileum and proximal colon.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Colon; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Nifedipine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Sulfones

1994
Differences in the effects of NK1-receptor antagonists, (+/-)-CP 96,345 and CP 99,994, on agonist-induced responses in guinea-pig trachea.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Biphenyl Compounds; Guinea Pigs; In Vitro Techniques; Indoles; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Substance P; Trachea

1994
Different susceptibility to neurokinin 1 receptor antagonists of substance P and septide-induced interleukin-6 release from U373 MG human astrocytoma cell line.
    Neuroscience letters, 1994, Apr-25, Volume: 171, Issue:1-2

    Topics: Astrocytoma; Binding, Competitive; Brain Neoplasms; Humans; Interleukin-6; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Pyrrolidonecarboxylic Acid; Substance P; Tumor Cells, Cultured

1994
Septide but not substance P stimulates inhibitory neurons in guinea-pig ileum.
    European journal of pharmacology, 1994, Jun-13, Volume: 258, Issue:3

    Topics: Animals; Guinea Pigs; Ileum; In Vitro Techniques; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P

1994
Highly potent substance P antagonists substituted with beta-phenyl- or beta-benzyl-proline at position 10.
    European journal of pharmacology, 1994, Jun-13, Volume: 258, Issue:3

    Topics: Amino Acid Sequence; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Rabbits; Rats; Receptors, Neurokinin-1; Structure-Activity Relationship; Substance P

1994
Typical and atypical NK1 tachykinin receptor characteristics in the rabbit isolated iris sphincter.
    British journal of pharmacology, 1994, Volume: 112, Issue:3

    Topics: Animals; In Vitro Techniques; Iris; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phenoxybenzamine; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P

1994
Use of selective antagonists for further characterization of tachykinin NK-2, NK-1 and possible "septide-selective" receptors in guinea pig bronchus.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: Amino Acid Sequence; Animals; Bronchi; Female; Guinea Pigs; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Substance P; Tachykinins

1994
Conformational study of two substance P hexapeptides by two-dimensional NMR.
    International journal of peptide and protein research, 1993, Volume: 41, Issue:2

    Topics: Amino Acid Sequence; Chloroform; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Peptide Fragments; Protein Conformation; Protein Folding; Pyrrolidonecarboxylic Acid; Solvents; Stereoisomerism; Substance P; Trifluoroethanol; Water

1993
Evidence for the presence of a septide-sensitive tachykinin receptor in the circular muscle of the guinea-pig ileum.
    European journal of pharmacology, 1993, Apr-28, Volume: 235, Issue:2-3

    Topics: Animals; Biphenyl Compounds; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscles; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tachykinins

1993
Variations in affinities for the NK1 receptor: differences between the non-peptide substance P antagonists RP 67580 and CP-96,345 and the agonist septide.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Binding, Competitive; Biphenyl Compounds; Brain; Cell Line; Dogs; Guinea Pigs; Humans; Indoles; Isoindoles; Mice; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Receptors, Neurokinin-1; Submandibular Gland; Substance P

1993
Neuromodulation mediated by neurokinin-1 subtype receptors in adult rabbit airways.
    The American journal of physiology, 1993, Volume: 265, Issue:3 Pt 1

    Topics: Acetylcholine; Animals; Electric Stimulation; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nervous System Physiological Phenomena; Parasympathetic Nervous System; Peptide Fragments; Physalaemin; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tetrodotoxin; Trachea

1993
Demonstration of a 'septide-sensitive' inflammatory response in rat skin.
    British journal of pharmacology, 1995, Volume: 116, Issue:4

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Blood Proteins; Capillary Permeability; Dermatitis, Contact; Dose-Response Relationship, Drug; Edema; Indoles; Isoindoles; Male; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Nitric Oxide Synthase; p-Methoxy-N-methylphenethylamine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1995
Comparative behavioural profile of centrally administered tachykinin NK1, NK2 and NK3 receptor agonists in the guinea-pig.
    British journal of pharmacology, 1995, Volume: 116, Issue:5

    Topics: Animals; Behavior, Animal; Guinea Pigs; Injections, Intraventricular; Male; Motor Activity; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

1995
Structural motifs encoded by individual exons of the human neurokinin-1 receptor gene interact differentially with selective agonists and antagonists.
    Journal of neurochemistry, 1996, Volume: 67, Issue:3

    Topics: Amino Acid Sequence; Cloning, Molecular; Exons; Humans; Iodine Radioisotopes; Molecular Sequence Data; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phosphatidylinositols; Piperidines; Protein Binding; Pyrrolidonecarboxylic Acid; Quinuclidines; Radioligand Assay; Receptors, Neurokinin-1; Recombinant Fusion Proteins; Stereoisomerism; Substance P

1996
Distinct regulations by septide and the neurokinin-1 tachykinin receptor agonist [pro9]substance P of the N-methyl-D-aspartate-evoked release of dopamine in striosome- and matrix-enriched areas of the rat striatum.
    Neuroscience, 1996, Volume: 73, Issue:4

    Topics: Animals; Corpus Striatum; Dopamine; Extracellular Matrix; Indoles; Isoindoles; Male; N-Methylaspartate; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P

1996
Neurokinin subtype receptors mediating substance P contraction in immature rabbit airways.
    Pediatric research, 1996, Volume: 39, Issue:1

    Topics: Animals; Atropine; Bronchi; Glycopeptides; Isometric Contraction; Muscle, Smooth; Neostigmine; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea

1996
Pharmacological evidence that NK-2 tachykinin receptors mediate hypotension in the guinea pig but not in the rat.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Animals; Benzamides; Blood Pressure; Guinea Pigs; Hypotension; Indoles; Isoindoles; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1996
Evidence that tachykinins relax the guinea-pig trachea via nitric oxide release and by stimulation of a septide-insensitive NK1 receptor.
    British journal of pharmacology, 1996, Volume: 117, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Neurokinin A; Neurokinin B; Nitric Oxide; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P; Tachykinins; Trachea

1996
Lack of a role for substance P in the control of dural arterial flow.
    Experimental brain research, 1996, Volume: 111, Issue:3

    Topics: Animals; Cerebral Arteries; Dura Mater; Electric Stimulation; Indoles; Isoindoles; Laser-Doppler Flowmetry; Male; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Regional Blood Flow; Substance P

1996
Neurokinin receptors in the guinea pig ileum.
    Pharmacology, 1996, Volume: 52, Issue:1

    Topics: Acetylcholine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Biphenyl Compounds; Guinea Pigs; Ileum; Male; Myenteric Plexus; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stereoisomerism; Structure-Activity Relationship; Substance P

1996
Septide and neurokinin A are high-affinity ligands on the NK-1 receptor: evidence from homologous versus heterologous binding analysis.
    FEBS letters, 1996, Dec-16, Volume: 399, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; COS Cells; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Protein Binding; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P

1996
Receptors mediating tachykinin-evoked depolarisations of neurons in the neonatal rat spinal cord.
    Acta biologica Hungarica, 1996, Volume: 47, Issue:1-4

    Topics: Animals; Animals, Newborn; Biphenyl Compounds; Evoked Potentials; In Vitro Techniques; Indoles; Isoindoles; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spinal Cord; Substance P; Tachykinins

1996
Differential activation of the epithelial and smooth muscle NK1 receptors by synthetic tachykinin agonists in guinea-pig trachea.
    British journal of pharmacology, 1997, Volume: 121, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Epithelium; Guinea Pigs; Male; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Peptide Fragments; Physalaemin; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Substance P; Tachykinins; Trachea

1997
High affinity binding of [3H]propionyl-[Met(O2)11]substance P(7-11), a tritiated septide-like peptide, in Chinese hamster ovary cells expressing human neurokinin-1 receptors and in rat submandibular glands.
    Molecular pharmacology, 1997, Volume: 52, Issue:1

    Topics: Animals; Binding Sites; CHO Cells; Cricetinae; Male; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Submandibular Gland; Substance P

1997
Characterization of neurokinin-1 receptors in the submucosal plexus of guinea pig ileum.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 1

    Topics: Animals; Electric Stimulation; Female; Ganglia, Autonomic; Guinea Pigs; Ileum; Immunohistochemistry; In Vitro Techniques; Intestinal Mucosa; Male; Membrane Potentials; Microscopy, Video; Muscle, Smooth; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rabbits; Rats; Receptors, Neurokinin-1; Submucous Plexus; Substance P; Vasodilation

1997
Spinal calmodulin inhibitors reduce N-methyl-D-aspartate- and septide-induced nociceptive behavior.
    European journal of pharmacology, 1997, Sep-17, Volume: 335, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Enzyme Inhibitors; Imidazoles; Injections, Intraventricular; Male; N-Methylaspartate; Neurokinin A; Pain; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Spinal Cord; Substance P; Sulfonamides

1997
A "septide-sensitive" receptor is not involved in tachykinin-mediated secretory and inositol phosphate responses in rat parotid gland: are several transduction pathways involved after the stimulation of the NK1 receptor?
    Journal of neurochemistry, 1998, Volume: 70, Issue:2

    Topics: Animals; Cells, Cultured; Indoles; Inositol Phosphates; Isoindoles; Kinetics; Male; Neurokinin-1 Receptor Antagonists; Parotid Gland; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Salivary Proteins and Peptides; Signal Transduction; Substance P; Tachykinins

1998
Tachykinins may modify spontaneous epileptiform activity in the rat entorhinal cortex in vitro by activating GABAergic inhibition.
    Neuroscience, 1998, Volume: 83, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Entorhinal Cortex; Epilepsy; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Phosphinic Acids; Propanolamines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Substance P; Synapses; Tachykinins

1998
The potency of the novel tachykinin receptor antagonist CGP49823 at rat and gerbil motoneurones in vitro.
    European journal of pharmacology, 1998, Jan-26, Volume: 342, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Gerbillinae; In Vitro Techniques; Motor Neurons; Neurokinin-1 Receptor Antagonists; Neuromuscular Depolarizing Agents; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinolines; Rats; Rats, Inbred Strains; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P

1998
Depolarization evoked co-release of tachykinins from enteric nerves in the guinea-pig proximal colon.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:3

    Topics: Animals; Calcium; Colon; Enteric Nervous System; Guinea Pigs; Neurokinin A; Peptide Fragments; Piperidines; Potassium Chloride; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Tachykinin; Substance P; Tachykinins

1998
Roles of neuronal NK1 and NK3 receptors in synaptic transmission during motility reflexes in the guinea-pig ileum.
    British journal of pharmacology, 1998, Volume: 124, Issue:7

    Topics: Animals; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Synaptic Transmission

1998
Endogenous peptidergic modulation of perisynaptic Schwann cells at the frog neuromuscular junction.
    The Journal of physiology, 1998, Oct-01, Volume: 512 ( Pt 1)

    Topics: Acetylcholinesterase; Animals; Calcium; GTP-Binding Proteins; Muscarine; Muscle, Skeletal; Neostigmine; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Peptide Fragments; Pertussis Toxin; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rana pipiens; Receptors, Neurokinin-1; Schwann Cells; Substance P; Synapses; Virulence Factors, Bordetella

1998
Point mutation increases a form of the NK1 receptor with high affinity for neurokinin A and B and septide.
    British journal of pharmacology, 1998, Volume: 125, Issue:2

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Neurokinin A; Neurokinin B; Peptide Fragments; Point Mutation; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-1; Recombinant Proteins; Substance P

1998
Comparison of the effects of calmidazolium, morphine and bupivacaine on N-methyl-D-aspartate- and septide-induced nociceptive behaviour.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:6

    Topics: Analgesics; Animals; Bupivacaine; Imidazoles; Male; Morphine; N-Methylaspartate; Pain; Pain Measurement; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Spinal Cord; Substance P

1998
Rat gastrointestinal motor responses mediated via activation of neurokinin receptors.
    Journal of gastroenterology and hepatology, 1999, Volume: 14, Issue:1

    Topics: Animals; Chromates; Chromium Radioisotopes; Gastric Emptying; Gastrointestinal Motility; Intubation, Gastrointestinal; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sodium Compounds; Substance P

1999
Identification in the NK1 tachykinin receptor of a domain involved in recognition of neurokinin A and septide but not of substance P.
    FEBS letters, 1999, Mar-26, Volume: 447, Issue:2-3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Chlorocebus aethiops; COS Cells; DNA, Complementary; Humans; In Vitro Techniques; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Point Mutation; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Tachykinins

1999
Characterization of central and peripheral effects of septide with the use of five tachykinin NK1 receptor antagonists in the rat.
    British journal of pharmacology, 1999, Volume: 127, Issue:3

    Topics: Acetamides; Animals; Behavior, Animal; Blood Pressure; Capillary Permeability; Heart Rate; Indoles; Injections, Intraventricular; Male; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-1; Stereoisomerism; Substance P

1999
Role of nitric oxide and septide-insensitive NK(1) receptors in bronchoconstriction induced by aerosolised neurokinin A in guinea-pigs.
    British journal of pharmacology, 2000, Volume: 129, Issue:5

    Topics: Aerosols; Airway Resistance; Animals; Bronchoconstriction; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P

2000
Further evidence for the presence of "septide-sensitive" tachykinin binding sites in tissues possessing solely NK(1) tachykinin receptors.
    Biochemical and biophysical research communications, 2000, Apr-13, Volume: 270, Issue:2

    Topics: Animals; Binding Sites; CHO Cells; Cricetinae; Humans; Indoles; Iodine Radioisotopes; Isoindoles; Mice; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protein Isoforms; Pyrrolidonecarboxylic Acid; Radioligand Assay; Rats; Receptors, Neurokinin-1; Substance P; Tetrazoles; Tumor Cells, Cultured

2000
Differences in circular muscle contraction and peristaltic motor inhibition caused by tachykinin NK1 receptor agonists in the guinea-pig small intestine.
    Neurogastroenterology and motility, 2000, Volume: 12, Issue:2

    Topics: Adenosine Triphosphate; Animals; Enzyme Inhibitors; Female; Guinea Pigs; Intestine, Small; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Piperidines; Purinergic P2 Receptor Antagonists; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sincalide; Spasm; Substance P; Suramin; Tetrodotoxin

2000
Evidence for functional NK1-tachykinin receptors on motor neurones supplying the circular muscle of guinea-pig small and large intestine.
    Neurogastroenterology and motility, 2000, Volume: 12, Issue:4

    Topics: Animals; Colon; Duodenum; Enzyme Inhibitors; Guinea Pigs; Ileum; Immunohistochemistry; In Vitro Techniques; Indomethacin; Motor Neurons; Muscle, Smooth; Nitric Oxide Synthase; Nitroarginine; Peptide Fragments; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Substance P

2000
Effects of the calcium release inhibitor dantrolene and the Ca2+-ATPase inhibitor thapsigargin on spinal nociception in rats.
    Pharmacology, 2001, Volume: 62, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics; Animals; Behavior, Animal; Calcium; Calcium-Transporting ATPases; Dantrolene; Enzyme Inhibitors; Male; Muscle Relaxants, Central; N-Methylaspartate; Pain; Pain Measurement; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Spinal Cord; Substance P; Thapsigargin

2001
Permissive role of neurokinin NK(3) receptors in NK(1) receptor-mediated activation of the locus coeruleus revealed by SR 142801.
    Synapse (New York, N.Y.), 2002, Volume: 43, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antiemetics; Dose-Response Relationship, Drug; Guinea Pigs; Locus Coeruleus; Male; Neural Pathways; Neurokinin-1 Receptor Antagonists; Neurons; Norepinephrine; Peptide Fragments; Piperidines; Prefrontal Cortex; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tetrazoles

2002
Facilitation by endogenous tachykinins of the NMDA-evoked release of acetylcholine after acute and chronic suppression of dopaminergic transmission in the matrix of the rat striatum.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Mar-01, Volume: 22, Issue:5

    Topics: Acetylcholine; Animals; Benzamides; Corpus Striatum; Dopamine; Dopamine Antagonists; Enzyme Inhibitors; In Vitro Techniques; Male; N-Methylaspartate; Neural Inhibition; Neurons; Oxidopamine; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Synaptic Transmission; Tachykinins; Time Factors

2002
Spinal nociceptin inhibits septide but not N-methyl-D-aspartate-induced nociceptive behavior in rats.
    European journal of pharmacology, 2002, Jun-07, Volume: 445, Issue:1-2

    Topics: Animals; Behavior, Animal; Injections, Spinal; Male; N-Methylaspartate; Naloxone; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Opioid; Spinal Cord; Substance P

2002
Peristalsis regulation by tachykinin NK1 receptors in the rabbit isolated distal colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 285, Issue:2

    Topics: Alanine; Animals; Atropine; Colon; Drug Interactions; Enzyme Inhibitors; Indoles; Kinetics; Male; Neurokinin-1 Receptor Antagonists; Nitric Oxide Synthase; Nitroarginine; Peptide Fragments; Peristalsis; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Rabbits; Receptors, Neurokinin-1; Substance P

2003
Biologic activity of the tachykinins on lamb and sheep gallbladder.
    Peptides, 2003, Volume: 24, Issue:4

    Topics: Animals; Binding Sites; Capsaicin; Dose-Response Relationship, Drug; Female; Gallbladder; Male; Muscles; Neurokinin A; Neurokinin B; Peptide Fragments; Physalaemin; Protein Structure, Tertiary; Pyrrolidonecarboxylic Acid; Receptors, Tachykinin; Sheep; Substance P; Tachykinins

2003
GABAergic basal forebrain neurons that express receptor for neurokinin B and send axons to the cerebral cortex.
    The Journal of comparative neurology, 2004, May-17, Volume: 473, Issue:1

    Topics: Animals; Animals, Newborn; Axons; Calbindin 2; Calbindins; Cell Count; Cerebral Cortex; Cholera Toxin; Choline O-Acetyltransferase; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Immunoenzyme Techniques; Immunohistochemistry; In Situ Hybridization; In Vitro Techniques; Isoenzymes; Male; Membrane Potentials; Neurons; Neuropeptide Y; Parvalbumins; Patch-Clamp Techniques; Peptide Fragments; Polypyrimidine Tract-Binding Protein; Prosencephalon; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-3; S100 Calcium Binding Protein G; Somatostatin; Substance P; Wheat Germ Agglutinin-Horseradish Peroxidase Conjugate

2004
Functional characterisation of tachykinin receptors in the circular muscle layer of the mouse ileum.
    Regulatory peptides, 2005, Sep-15, Volume: 130, Issue:3

    Topics: Action Potentials; Analgesics; Animals; Antipsychotic Agents; Atropine; Electric Stimulation; Ileum; Indoles; Isoindoles; Mice; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Nitroarginine; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

2005
The role of tachykinins in circular muscle contractility of the murine ileum: a functional investigation.
    Autonomic neuroscience : basic & clinical, 2006, Jun-30, Volume: 126-127

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Ilium; In Vitro Techniques; Male; Mice; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nitroarginine; Peptide Fragments; Potassium Chloride; Pyrrolidonecarboxylic Acid; Substance P; Tachykinins; Tetrodotoxin

2006
Neurokinin-3 peptide instead of neurokinin-1 synergistically exacerbates kainic acid-inducing degeneration of neurons in the substantia nigra of mice.
    Journal of neurochemistry, 2008, Volume: 105, Issue:1

    Topics: Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Drug Synergism; Fluoresceins; Kainic Acid; Male; Mice; Mice, Inbred Strains; Nerve Degeneration; Nerve Tissue Proteins; Neurokinin-1 Receptor Antagonists; Neurons; Organic Chemicals; Peptide Fragments; Pyrrolidonecarboxylic Acid; Quinolines; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Substantia Nigra; Tetrazolium Salts; Thiazoles

2008
Neuroprotective effects of neurokinin receptor one in dopaminergic neurons are mediated through Akt/PKB cell signaling pathway.
    Neuropharmacology, 2011, Volume: 61, Issue:8

    Topics: Analysis of Variance; Animals; Apomorphine; bcl-Associated Death Protein; Caspase 3; Cell Death; Cell Line, Tumor; Corpus Striatum; Disease Models, Animal; Dopamine Agonists; Dopaminergic Neurons; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Gene Expression Regulation; L-Lactate Dehydrogenase; Male; Motor Activity; Neuroblastoma; Neurokinin-1 Receptor Antagonists; Neuroprotective Agents; Neurotoxicity Syndromes; Oxidopamine; Peptide Fragments; Proto-Oncogene Proteins c-akt; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Rotarod Performance Test; Signal Transduction; Substance P; Sympatholytics; Time Factors; Tyrosine 3-Monooxygenase

2011
Kinetic binding and activation profiles of endogenous tachykinins targeting the NK1 receptor.
    Biochemical pharmacology, 2016, Oct-15, Volume: 118

    Topics: Algorithms; Animals; Astrocytoma; Binding, Competitive; Cell Line, Tumor; CHO Cells; Cricetulus; Electric Impedance; Humans; Kinetics; Ligands; Nerve Tissue Proteins; Neuroglia; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Radioligand Assay; Receptors, Neurokinin-1; Recombinant Proteins; Substance P; Tachykinins

2016