senktide has been researched along with sr 142806 in 4 studies
| Studies (senktide) | Trials (senktide) | Recent Studies (post-2010) (senktide) | Studies (sr 142806) | Trials (sr 142806) | Recent Studies (post-2010) (sr 142806) |
|---|---|---|---|---|---|
| 292 | 1 | 50 | 28 | 0 | 12 |
| Protein | Taxonomy | senktide (IC50) | sr 142806 (IC50) |
|---|---|---|---|
| Cytochrome P450 3A4 | Homo sapiens (human) | 1 | |
| Cytochrome P450 2C19 | Homo sapiens (human) | 7 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (50.00) | 18.2507 |
| 2000's | 1 (25.00) | 29.6817 |
| 2010's | 1 (25.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Chung, FZ; Oxender, DL; Tian, Y; Wu, LH | 1 |
| Brawner, ME; Elshourbagy, NA; Foley, JJ; Giardina, GA; Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Potts, W; Sarau, HM; Schmidt, DB; Webb, EF | 1 |
| Ames, RS; Brawner, ME; Buckley, PT; Elshourbagy, NA; Feild, JA; Foley, JJ; Giardina, GA; Hay, DW; Luttmann, MA; Nuthulaganti, P; Sarau, HM; Schmidt, DB | 1 |
| Batt, F; Blanc, S; Dutheuil, G; El Bousmaqui, M; Fraser, GL; Hoveyda, HR; Korac, J; Lapin, A; Lenoir, F; Noël, S; Roy, MO | 1 |
4 other study(ies) available for senktide and sr 142806
| Article | Year |
|---|---|
The unpredicted high affinities of a large number of naturally occurring tachykinins for chimeric NK1/NK3 receptors suggest a role for an inhibitory domain in determining receptor specificity.
Topics: Amino Acid Sequence; Binding, Competitive; Humans; Ligands; Membrane Proteins; Molecular Sequence Data; Neurokinin A; Neurokinin B; Phosphatidylinositols; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Recombinant Fusion Proteins; Structure-Activity Relationship; Substance P; Tachykinins | 1996 |
Nonpeptide tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor antagonist.
Topics: Animals; Calcium; CHO Cells; Cricetinae; Dogs; Humans; Mice; Piperidines; Quinolines; Rabbits; Radioligand Assay; Rats; Receptors, Neurokinin-3; Receptors, Tachykinin | 1997 |
Molecular and pharmacological characterization of the murine tachykinin NK(3) receptor.
Topics: Amino Acid Sequence; Animals; Calcium; Cloning, Molecular; Humans; Mice; Molecular Sequence Data; Neurokinin A; Quinolines; Receptors, Neurokinin-3 | 2001 |
Discovery and optimization of novel antagonists to the human neurokinin-3 receptor for the treatment of sex-hormone disorders (Part I).
Topics: Androgens; Animals; Brain; Caco-2 Cells; Chemistry Techniques, Synthetic; CHO Cells; Cricetulus; Crystallography, X-Ray; Drug Discovery; Endocrine System Diseases; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; High-Throughput Screening Assays; Humans; Ligands; Luteinizing Hormone; Male; Rats, Sprague-Dawley; Receptors, Neurokinin-3; Structure-Activity Relationship | 2015 |