senktide has been researched along with neurokinin a in 85 studies
Studies (senktide) | Trials (senktide) | Recent Studies (post-2010) (senktide) | Studies (neurokinin a) | Trials (neurokinin a) | Recent Studies (post-2010) (neurokinin a) |
---|---|---|---|---|---|
292 | 1 | 50 | 1,765 | 34 | 91 |
Protein | Taxonomy | senktide (IC50) | neurokinin a (IC50) |
---|---|---|---|
Substance-K receptor | Homo sapiens (human) | 0.0017 | |
Neuromedin-K receptor | Homo sapiens (human) | 0.045 | |
Substance-K receptor | Mesocricetus auratus (golden hamster) | 0.001 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (4.71) | 18.7374 |
1990's | 58 (68.24) | 18.2507 |
2000's | 21 (24.71) | 29.6817 |
2010's | 2 (2.35) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Adami, N; Arkinstall, SJ; Buell, G; Kawashima, E; Maury, K; Missotten, M; Schulz, MF; Talabot, F | 1 |
Brawner, ME; Elshourbagy, NA; Foley, JJ; Giardina, GA; Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Potts, W; Sarau, HM; Schmidt, DB; Webb, EF | 1 |
Cascieri, MA; Harrison, T; Korsgaard, MP; Sadowski, S; Seabrook, GR; Swain, CJ | 1 |
Ames, RS; Brawner, ME; Buckley, PT; Elshourbagy, NA; Feild, JA; Foley, JJ; Giardina, GA; Hay, DW; Luttmann, MA; Nuthulaganti, P; Sarau, HM; Schmidt, DB | 1 |
Chang, FY; Lee, SD; Wang, PS; Yeh, GH | 2 |
Clark, D; Elliott, PJ; Hagan, RM; Overton, P | 1 |
Albus, K; Chao, HH; Hicks, TP | 1 |
Elliott, PJ; Mason, GS | 1 |
Culman, J; Itoi, K; Jost, N; Lebrun, C; Stauss, B; Tschöpe, C; Unger, T | 1 |
Shinkai, M; Takayanagi, I | 1 |
Ballati, L; Giachetti, A; Giuliani, S; Lecci, A; Maggi, CA; Manzini, S; Patacchini, R; Quartara, L; Renzetti, AR; Rovero, P | 1 |
Hall, JM; Mitchell, D; Morton, IK | 1 |
Elliott, PJ; Hagan, RM; Mason, GS; Stephens-Smith, M | 1 |
Beresford, IJ; Deal, MJ; Hagan, RM; Ireland, SJ; Jordan, CC; Ward, P | 1 |
Hall, JM; Morton, IK | 1 |
Kawashima, K; Kobayashi, N; Onishi, Y; Otsuka, M; Sakuma, M; Yanagisawa, M; Yoshioka, K | 1 |
Constantine, JW; Lebel, WS; Woody, HA | 1 |
Barr, AJ; Bernal, AL; Nimmo, AJ; Watson, SP | 1 |
Lorens, SA; Mitsushio, H; Paris, JM | 1 |
Hamaoka, T; Kamiya, H; Matsuoka, Y; Nagashima, A; Takano, Y; Tateishi, K | 1 |
Hicks, CR; Mizoguchi, H | 1 |
Brodin, E; Franck, J; Fried, G | 1 |
Ciccocioppo, R; De Caro, G; Massi, M; Panocka, I; Pompei, P | 1 |
Beaujouan, JC; Glowinski, J; Petitet, F; Saffroy, M; Torrens, Y | 2 |
Guo, JZ; Konishi, S; Murakoshi, T; Otsuka, M; Saito, K; Yoshioka, K; Zhao, FY | 2 |
Itoi, K; Lebrun, CJ; Steckelings, U; Unger, T; Wende, P | 1 |
Giuliani, S; Maggi, CA; Meini, S; Patacchini, R | 1 |
Baranauskas, G; Fisher, ND; Nistri, A | 1 |
Chung, FZ; Hill, DR; Madden, Z; Pinnock, RD; Suman-Chauhan, N; Webdale, L; Woodruff, GN | 1 |
Lefebvre, RA; Smits, GJ | 1 |
Bowery, BJ; Hill, RG; Seabrook, GR | 1 |
Grider, JR; Jin, JG; Makhlouf, GM; Misra, S | 1 |
Boden, PR; Norris, SK; Woodruff, GN | 1 |
Dalforno, G; Gaviraghi, G; Hagan, RM; Palea, S; Pietra, C; Trist, DG | 1 |
Humpel, C; Saria, A | 1 |
Imai, Y; Inoki, R; Takiuchi, S; Tang, FD; Yonehara, N | 1 |
Funayama, N; Shinkai, M; Takayanagi, I | 1 |
Kamiya, HO; Matsumoto, T; Nakayama, Y; Saito, R; Takano, Y | 1 |
Chahl, LA; Johnston, PA | 1 |
De Giorgio, R; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Tramontana, M | 1 |
Marchionni, D; Nisato, D; Roccon, A | 1 |
John, C; Kazem, E; Tanaka, DT | 1 |
Kameyama, T; Shinkai, N; Ukai, M | 3 |
Costa, C; Cozzolino, A; Esposito, C; Falciani, M; Filippelli, A; Porta, R; Rossi, F | 1 |
Fox, AJ; Naeem, S; Patel, IA; Urbán, L; Walpole, C | 1 |
Kawamata, T; Maeda, K; Maeda, S; Nakai, M; Tanaka, C; Yamaguchi, T | 1 |
Hargreaves, RJ; Hill, RG; Shepheard, SL; Williamson, DJ | 1 |
Brelière, JC; Emonds-Alt, X; Le Fur, G; Vilain, P | 1 |
Fisher, L; Pennefather, JN | 1 |
MacNaughton, W; Moore, B; Vanner, S | 1 |
Barnhart, DC; Kimball, BC; Mulholland, MW; Sarosi, GA; Zhang, W | 1 |
Cody, C; Jones, RS; Maubach, KA | 1 |
Bordin, G; Brunelleschi, S; Colangelo, D; Viano, I | 1 |
Ardell, JL; Armour, JA; Hoover, DB; Thompson, GW | 1 |
Petersen, M; Schaible, HG; Segond von Banchet, G | 1 |
Broccardo, M; Improta, G; Tabacco, A | 1 |
Buljubasich, S; Lau, WA; Pennefather, JN; Ventura, S | 1 |
Buckner, CK; Meeker, SN; Pedersen, KE; Undem, BJ | 1 |
Calixto, JB; De Lima, TC; Ribeiro, SJ; Teixeira, RM | 1 |
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ; Widdowson, L | 1 |
Geraghty, DP; Mazzone, SB | 2 |
Crane, LH; Hamlin, GP; Nimmo, AJ; Williams, MJ | 2 |
Holzer, P; Shahbazian, A | 1 |
Coupar, IM; Kerr, KP; Thai, B | 1 |
Baird, AW; Goldhill, J; Moriarty, D; Selve, N | 1 |
Barahona, MV; Bustamante, S; García-Sacristán, A; Hernández, M; Orensanz, LM | 1 |
Burcher, E; Liu, L | 1 |
Barone, FC; Bush, B; Foley, JJ; Giardina, GA; Griswold, DE; Grugni, M; Hay, DW; Kilian, D; Kotzer, CJ; Legos, JJ; Lundberg, D; Luttmann, MA; Martin, LD; Potts, W; Raveglia, LF; Sandhu, P; Sarau, HM; Schmidt, DB; Underwood, DC | 1 |
Jones, RS; Stacey, AE; Woodhall, GL | 1 |
Ogier, R; Raggenbass, M | 1 |
Cunha-Vaz, JG; Gaspar, MN; Macedo, TR; Ribeiro, CA | 1 |
Greenwood-Van Meerveld, B; Venkova, K | 1 |
Couture, R; Deschamps, K | 1 |
Adolfsson, R; Ahlstedt, I; de Verdier, J; Drmota, T; Engberg, S; Johansson, A; Jussila, R; Kristensson, E; Leffler, A; Lindström, E; Novén, A; Påhlman, I; Sigfridsson, K; Sundqvist, M; von Mentzer, B | 1 |
Emala, CW; Gallos, G; Goubaeva, F; Mizuta, F; Mizuta, K; Panettieri, RA; Xu, D; Yang, J; Zhu, D | 1 |
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T | 1 |
Culman, J; Hunt, SP; Tauer, U; Zhao, Y | 1 |
Navarro, VM; Ohkura, S; Okamura, H; Wakabayashi, Y; Yamamura, T | 1 |
85 other study(ies) available for senktide and neurokinin a
Article | Year |
---|---|
Molecular characterisation, expression and localisation of human neurokinin-3 receptor.
Topics: Adult; Amino Acid Sequence; Animals; Base Sequence; Brain; DNA; Gene Expression; Humans; Molecular Sequence Data; Neurokinin A; Polymerase Chain Reaction; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Restriction Mapping; Sequence Homology, Nucleic Acid; Xenopus laevis | 1992 |
Nonpeptide tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor antagonist.
Topics: Animals; Calcium; CHO Cells; Cricetinae; Dogs; Humans; Mice; Piperidines; Quinolines; Rabbits; Radioligand Assay; Rats; Receptors, Neurokinin-3; Receptors, Tachykinin | 1997 |
High affinity, selective neurokinin 2 and neurokinin 3 receptor antagonists from a common structural template.
Topics: Animals; Calcium; CHO Cells; Cricetinae; Fluorescent Dyes; Fura-2; Humans; Lactams; Molecular Conformation; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Spectrometry, Fluorescence; Structure-Activity Relationship | 1998 |
Molecular and pharmacological characterization of the murine tachykinin NK(3) receptor.
Topics: Amino Acid Sequence; Animals; Calcium; Cloning, Molecular; Humans; Mice; Molecular Sequence Data; Neurokinin A; Quinolines; Receptors, Neurokinin-3 | 2001 |
The motor actions of natural neurokinins and their specific agonists on the gastrointestinal tract of the rat.
Topics: Animals; Charcoal; Gastrointestinal Motility; Injections, Intraperitoneal; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Pilot Projects; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins | 1992 |
Neurokinin agonists differentially affect A9 and A10 dopamine cells in the rat.
Topics: Animals; Dopamine; Neurokinin A; Neurons; Peptide Fragments; Rats; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Substantia Nigra; Tegmentum Mesencephali | 1992 |
Tachykinins preferentially excite certain complex cells in the infragranular layers of feline striate cortex.
Topics: Animals; Cats; Evoked Potentials, Visual; Female; Iontophoresis; Male; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Substance P; Tachykinins; Visual Cortex | 1992 |
Behavioural consequences following infusion of selective neurokinin agonists into the median raphe nucleus of the rat.
Topics: Amino Acid Sequence; Animals; Dose-Response Relationship, Drug; Injections; Molecular Sequence Data; Motor Activity; Neurokinin A; Peptide Fragments; Raphe Nuclei; Rats; Substance P | 1992 |
Identification of the central tachykinin receptor subclass involved in substance P-induced cardiovascular and behavioral responses in conscious rats.
Topics: Animals; Behavior, Animal; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Injections, Intraventricular; Male; Neurokinin A; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Tachykinins | 1992 |
Characterization of tachykinin receptors in urinary bladder from guinea pig.
Topics: Animals; Dose-Response Relationship, Drug; Female; Guinea Pigs; Muscle Contraction; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Urinary Bladder | 1990 |
In vivo evidence for tachykininergic transmission using a new NK-2 receptor-selective antagonist, MEN 10,376.
Topics: Animals; Bronchi; Bronchoconstriction; Cerebral Cortex; Cricetinae; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Mesocricetus; Muscle Contraction; Neurokinin A; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Urinary Bladder; Vagus Nerve | 1991 |
Neurokinin receptors in the rabbit iris sphincter characterised by novel agonist ligands.
Topics: Animals; In Vitro Techniques; Iris; Kinetics; Ligands; Male; Neurokinin A; Peptide Fragments; Rabbits; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P | 1991 |
Behavioural and biochemical responses following activation of midbrain dopamine pathways by receptor selective neurokinin agonists.
Topics: Amino Acid Sequence; Animals; Chromatography, High Pressure Liquid; Dopamine; Haloperidol; Limbic System; Male; Mesencephalon; Molecular Sequence Data; Motor Activity; Neural Pathways; Neurokinin A; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Substantia Nigra; Tegmentum Mesencephali | 1991 |
Receptor-selective, peptidase-resistant agonists at neurokinin NK-1 and NK-2 receptors: new tools for investigating neurokinin function.
Topics: Administration, Cutaneous; Amino Acid Sequence; Animals; Bronchoconstriction; Capillary Permeability; Chromatography, High Pressure Liquid; Guinea Pigs; Male; Molecular Sequence Data; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Trachea | 1991 |
Novel ligands confirm NK-1 receptor-mediated modulation of neurotransmission in the guinea pig vas deferens preparation.
Topics: Animals; Electric Stimulation; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Synaptic Transmission; Vas Deferens | 1991 |
Substance P-evoked release of acetylcholine from isolated spinal cord of the newborn rat.
Topics: Acetylcholine; Animals; Animals, Newborn; Calcium; Dihydro-beta-Erythroidine; Edrophonium; Neurokinin A; Neurokinin B; Peptide Fragments; Physostigmine; Potassium; Rats; Rats, Inbred Strains; Secretory Rate; Spinal Cord; Stimulation, Chemical; Substance P; Tetrodotoxin; Veratridine | 1991 |
Inhibition of tachykinin-induced hypotension in dogs by CP-96,345, a selective blocker of NK-1 receptors.
Topics: Animals; Biphenyl Compounds; Blood Pressure; Decerebrate State; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Neurokinin A; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Stereoisomerism; Substance P; Tachykinins | 1991 |
The presence of NK3 tachykinin receptors on rat uterus.
Topics: Animals; Binding, Competitive; Eledoisin; Female; Humans; In Vitro Techniques; Neurokinin A; Peptide Fragments; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Succinimides; Tachykinins; Uterine Contraction; Uterus | 1991 |
Intra-raphe neurokinin-induced hyperactivity: effects of 5,7-dihydroxytryptamine lesions.
Topics: 5,7-Dihydroxytryptamine; Action Potentials; Animals; Catecholamines; Dihydroxytryptamines; Male; Medial Forebrain Bundle; Motor Activity; Neural Pathways; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Substance P | 1989 |
Cardiovascular roles of tachykinin peptides in the nucleus tractus solitarii of rats.
Topics: Animals; Blood Pressure; Cardiovascular System; Dose-Response Relationship, Drug; Heart Rate; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Rats, Inbred Strains; Substance P | 1989 |
Effects of neurokinins on ion transport and sulfated macromolecule release in the isolated ferret trachea.
Topics: Amiloride; Animals; Biological Transport; Bumetanide; Chlorides; Electrodes; Ferrets; In Vitro Techniques; Macromolecular Substances; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Sodium; Substance P; Sulfates; Trachea | 1989 |
Substance P enhances the release of endogenous serotonin from rat ventral spinal cord.
Topics: Animals; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Potassium; Rats; Rats, Inbred Strains; Serotonin; Spinal Cord; Substance P | 1989 |
Selective agonists at NK3 tachykinin receptors inhibit alcohol intake in Sardinian alcohol-preferring rats.
Topics: Alcohol Drinking; Amino Acid Sequence; Animals; Drinking Behavior; Eating; Injections, Intraventricular; Male; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurokinin-3; Substance P; Water Deprivation | 1994 |
A new selective bioassay for tachykinin NK3 receptors based on inositol monophosphate accumulation in the guinea pig ileum.
Topics: Animals; Biphenyl Compounds; Guinea Pigs; Hypnotics and Sedatives; Ileum; In Vitro Techniques; Inositol Phosphates; Male; Muscle, Smooth; Neurokinin A; Peptide Fragments; Phosphatidylinositols; Phospholipids; Receptors, Neurokinin-3; Stimulation, Chemical; Substance P; Tachykinins | 1993 |
Involvement of NK1 receptors in synaptic transmission in the guinea pig coeliac ganglion.
Topics: Animals; Electric Stimulation; Evoked Potentials; Female; Ganglia, Sympathetic; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Receptors, Neurokinin-1; Substance P; Synapses; Synaptic Transmission; Tachykinins | 1993 |
Effects of tachykinins on phosphoinositide metabolism in the hypothalamus: is the NK1 receptor involved?
Topics: Animals; Carbachol; Dose-Response Relationship, Drug; Hypothalamus; In Vitro Techniques; Inositol; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Phosphatidylinositols; Rats; Rats, Wistar; Receptors, Neurokinin-1; Substance P; Tachykinins | 1993 |
Effect of longitudinal muscle-myenteric plexus removal and indomethacin on the response to tachykinin NK-2 and NK-3 receptor agonists in the circular muscle of the guinea-pig ileum.
Topics: Animals; Atropine; Calcium Channel Blockers; Guinea Pigs; Ileum; In Vitro Techniques; Indomethacin; Male; Muscle, Smooth; Myenteric Plexus; Neurokinin A; omega-Conotoxin GVIA; Peptide Fragments; Peptides; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tetrodotoxin | 1994 |
Multiple types of tachykinin receptor mediate a slow excitation of rat spinal motoneurones in vitro.
Topics: Animals; Animals, Newborn; Female; In Vitro Techniques; Male; Membrane Potentials; Motor Neurons; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spinal Cord; Substance P; Tetrodotoxin | 1994 |
Characterization of tachykinin mediated increases in [Ca2+]i in Chinese hamster ovary cells expressing human tachykinin NK3 receptors.
Topics: Animals; Benzamides; Calcium; Calcium-Transporting ATPases; CHO Cells; Cricetinae; Cricetulus; Estrenes; Fura-2; Humans; Inositol Phosphates; Manganese; Neurokinin A; Peptide Fragments; Piperidines; Pyrrolidinones; Receptors, Neurokinin-3; Ryanodine; Second Messenger Systems; Structure-Activity Relationship; Substance P; Tachykinins; Terpenes; Thapsigargin; Type C Phospholipases | 1994 |
Tachykinin receptors involved in the contractile effect of the natural tachykinins in the rat gastric fundus.
Topics: Animals; Biphenyl Compounds; Dose-Response Relationship, Drug; Female; Gastric Fundus; Indoles; Isoindoles; Male; Methacholine Chloride; Muscle Contraction; Neurokinin A; Neurokinin B; Peptide Fragments; Peptides, Cyclic; Rats; Receptors, Tachykinin; Substance P; Tachykinins | 1994 |
Pharmacology of tachykinin receptors on neurones in the ventral tegmental area of rat brain slices.
Topics: Action Potentials; Animals; Electrophysiology; In Vitro Techniques; Microelectrodes; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Rats; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Ventral Tegmental Area | 1995 |
Subtypes of tachykinin receptors on tonic and phasic neurones in coeliac ganglion of the guinea-pig.
Topics: Animals; Female; Ganglia, Sympathetic; Guinea Pigs; In Vitro Techniques; Male; Neurokinin A; Neurons; Peptide Fragments; Receptors, Tachykinin; Substance P | 1995 |
The nonpeptide NK-2 antagonist SR 48968 is also a NK-3 antagonist in the guinea but not in the rat.
Topics: Animals; Benzamides; Binding, Competitive; Cell Membrane; Cerebral Cortex; Enzyme Activation; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Muscle, Smooth; Neurokinin A; Peptide Fragments; Phosphatidylinositols; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Synaptosomes; Tachykinins; Type C Phospholipases | 1993 |
Functional difference between SP and NKA: relaxation of gastric muscle by SP is mediated by VIP and NO.
Topics: Animals; Arginine; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Neurokinin A; Nitric Oxide; Nitroarginine; Peptide Fragments; Stomach; Substance P; Tachykinins; Tetrodotoxin; Vasoactive Intestinal Peptide | 1993 |
Agonists selective for tachykinin NK1 and NK3 receptors excite subpopulations of neurons in the rat medial habenula nucleus in vitro.
Topics: Animals; Electrophysiology; Extracellular Space; In Vitro Techniques; Male; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Tachykinins; Thalamic Nuclei | 1993 |
Further studies on the effects of selective neurokinin agonists upon the activation of micturition reflex in rats. Evidence for a dual NK-1 receptor mediated excitatory and inhibitory activity.
Topics: Animals; Dose-Response Relationship, Drug; Injections, Intra-Arterial; Injections, Intraventricular; Male; Neurokinin A; Peptide Fragments; Physalaemin; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Reflex; Substance P; Urinary Bladder; Urination | 1993 |
Characterization of neurokinin binding sites in rat brain membranes using highly selective ligands.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Brain Chemistry; Eledoisin; Female; Ligands; Membrane Proteins; Molecular Sequence Data; Neurokinin A; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Tachykinins | 1993 |
Involvement of substance P present in small-diameter afferent fibers in microcirculatory hemodynamics of the rat hind instep.
Topics: Afferent Pathways; Animals; Bradykinin; Dose-Response Relationship, Drug; Hindlimb; Male; Microcirculation; Muscle, Smooth, Vascular; Neurokinin A; Peptide Fragments; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Sciatic Nerve; Skin; Substance P | 1993 |
Regional differences in contractile responses to tachykinin agonists and to electrical field stimulation are dependent on distribution of proteinase activity.
Topics: Animals; Bronchi; Electric Stimulation; Endopeptidases; Glycopeptides; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Protease Inhibitors; Rabbits; Substance P; Trachea | 1993 |
The mechanism of central pressor actions of tachykinin NK-3 receptor in the paraventricular nucleus of the hypothalamus in rats.
Topics: Animals; Blood Pressure; Models, Biological; Neurokinin A; Paraventricular Hypothalamic Nucleus; Peptide Fragments; Rats; Receptors, Neurokinin-3; Substance P | 1993 |
Neurokinin-1, -2 and -3 receptors are candidates for a role in the opiate withdrawal response in guinea-pigs.
Topics: Animals; Cerebral Ventricles; Guinea Pigs; Injections, Intraventricular; Motor Activity; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Substance Withdrawal Syndrome | 1993 |
In vivo evidence for the involvement of tachykinin NK3 receptors in the hexamethonium-resistant inhibitory transmission in the rat colon.
Topics: Adrenergic Agents; Animals; Colon; Dose-Response Relationship, Drug; Guanethidine; Hexamethonium; Male; Muscle Contraction; Neurokinin A; NG-Nitroarginine Methyl Ester; Nicotinic Antagonists; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P | 1996 |
Study of SR 142801, a new potent non-peptide NK3 receptor antagonist on cardiovascular responses in conscious guinea-pig.
Topics: Analysis of Variance; Animals; Blood Pressure; Dose-Response Relationship, Drug; Guinea Pigs; Heart Rate; Injections, Intravenous; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Substance P | 1996 |
Neurokinin subtype receptors mediating substance P contraction in immature rabbit airways.
Topics: Animals; Atropine; Bronchi; Glycopeptides; Isometric Contraction; Muscle, Smooth; Neostigmine; Neurokinin A; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Trachea | 1996 |
Neurokinin A and senktide attenuate scopolamine-induced impairment of spontaneous alternation performance in mice.
Topics: Amnesia; Animals; Male; Maze Learning; Mice; Neurokinin A; Peptide Fragments; Psychomotor Performance; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Scopolamine; Substance P | 1996 |
Transglutaminase-synthesized spermine derivative of substance P recognizes rat portal vein neurokinin-3 receptors.
Topics: Androstanes; Animals; Benzimidazoles; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Physalaemin; Piperidines; Portal Vein; Rats; Rats, Wistar; Receptors, Neurokinin-3; Substance P; Thiorphan; Transglutaminases; Vasoconstriction | 1997 |
Receptors mediating tachykinin-evoked depolarisations of neurons in the neonatal rat spinal cord.
Topics: Animals; Animals, Newborn; Biphenyl Compounds; Evoked Potentials; In Vitro Techniques; Indoles; Isoindoles; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Spinal Cord; Substance P; Tachykinins | 1996 |
Possible different mechanism between amyloid-beta (25-35)-and substance P-induced chemotaxis of murine microglia.
Topics: Amyloid beta-Peptides; Animals; Brain; Cells, Cultured; Chemotaxis; Dose-Response Relationship, Drug; Microglia; Neurofibrillary Tangles; Neurokinin A; Peptide Fragments; Rats; Rats, Wistar; Substance P | 1997 |
Intravital microscope studies on the effects of neurokinin agonists and calcitonin gene-related peptide on dural vessel diameter in the anaesthetized rat.
Topics: Anesthetics; Animals; Benzamides; Blood Pressure; Calcitonin Gene-Related Peptide; Dura Mater; Indoles; Isoindoles; Male; Microscopy, Video; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P; Vasodilator Agents | 1997 |
Tachykinin-induced contractions of the guinea pig ileum longitudinal smooth muscle: tonic and phasic muscular activities.
Topics: Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Substance P; Tachykinins | 1997 |
Potencies of agonists acting at tachykinin receptors in the oestrogen-primed rat uterus: effects of peptidase inhibitors.
Topics: Animals; Dipeptides; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Estradiol; Female; Muscle, Smooth; Neurokinin A; Peptide Fragments; Piperidines; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Tachykinins; Uterine Contraction; Uterus | 1997 |
Cellular pathways mediating tachykinin-evoked secretomotor responses in guinea pig ileum.
Topics: Animals; Capsaicin; Electric Stimulation; Evoked Potentials; Guinea Pigs; Ileum; In Vitro Techniques; Intestinal Mucosa; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tachykinins | 1997 |
Tachykinin neuropeptide-evoked intracellular calcium transients in cultured guinea pig myenteric neurons.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Diltiazem; Dipeptides; Fluorometry; Guinea Pigs; Indoles; Lanthanum; Myenteric Plexus; Neurokinin A; Nickel; Nifedipine; Peptide Fragments; Peptides, Cyclic; Receptors, Tachykinin; Substance P; Tachykinins; Virulence Factors, Bordetella | 1998 |
Tachykinins may modify spontaneous epileptiform activity in the rat entorhinal cortex in vitro by activating GABAergic inhibition.
Topics: Animals; Baclofen; Bicuculline; Entorhinal Cortex; Epilepsy; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Phosphinic Acids; Propanolamines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Substance P; Synapses; Tachykinins | 1998 |
Tachykinin receptors are present on human monocytes and play a role in rheumatoid arthritis.
Topics: Aged; Arthritis, Rheumatoid; Cell Separation; Female; Humans; Male; Middle Aged; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Superoxides; Tetradecanoylphorbol Acetate | 1998 |
Involvement of dopamine receptors in beneficial effects of tachykinins on scopolamine-induced impairment of alternation performance in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amnesia; Animals; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Male; Memory; Mice; Neurokinin A; Peptide Fragments; Phenethylamines; Receptors, Cholinergic; Receptors, Dopamine D1; Receptors, Dopamine D2; Scopolamine; Substance P; Sulpiride; Tachykinins | 1998 |
Canine intrinsic cardiac neurons involved in cardiac regulation possess NK1, NK2, and NK3 receptors.
Topics: Animals; Dogs; Heart; Myocardial Contraction; Neurokinin A; Neurons, Afferent; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P | 1998 |
Ameliorative effects of tachykinins on scopolamine-induced impairment of spontaneous alternation performance in mice.
Topics: Animals; Male; Mice; Muscarinic Antagonists; Naloxone; Naltrexone; Narcotic Antagonists; Neurokinin A; Peptide Fragments; Psychomotor Performance; Scopolamine; Substance P; Tachykinins | 1998 |
Rat gastrointestinal motor responses mediated via activation of neurokinin receptors.
Topics: Animals; Chromates; Chromium Radioisotopes; Gastric Emptying; Gastrointestinal Motility; Intubation, Gastrointestinal; Male; Neurokinin A; Neurokinin B; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sodium Compounds; Substance P | 1999 |
Expression of neurokinin-1 receptors on cultured dorsal root ganglion neurons from the adult rat.
Topics: Animals; Cells, Cultured; Ganglia, Spinal; Kinetics; Male; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Time Factors | 1999 |
Central tachykinin NK3 receptors in the inhibitory action on the rat colonic propulsion of a new tachykinin, PG-KII.
Topics: Animals; Colon; Gastrointestinal Transit; Injections, Intraventricular; Male; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins | 1999 |
An immunohistochemical and pharmacological study of tachykinins in the rat and guinea-pig prostate glands.
Topics: Animals; Atropine; Benzamides; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Peptide Fragments; Piperidines; Prostate; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Substance P; Tachykinins | 1999 |
Pharmacological examination of the neurokinin-1 receptor mediating relaxation of human intralobar pulmonary artery.
Topics: Adolescent; Adult; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; Epoprostenol; Female; Humans; In Vitro Techniques; Lung; Male; Middle Aged; Neurokinin A; Nitric Oxide; Peptide Fragments; Phenylephrine; Pulmonary Artery; Receptors, Neurokinin-1; Receptors, Tachykinin; Substance P; Vasoconstriction; Vasodilation | 2000 |
Tachykinin NK(3)receptor involvement in anxiety.
Topics: Animals; Anxiety; Cerebral Ventricles; Injections, Intraventricular; Male; Maze Learning; Mice; Neurokinin A; Neurokinin B; Peptide Fragments; Piperidines; Receptors, Neurokinin-3; Substance P; Tachykinins | 1999 |
Tachykinins increase [3H]acetylcholine release in mouse striatum through multiple receptor subtypes.
Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Choline O-Acetyltransferase; Corpus Striatum; Electrophysiology; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; In Situ Hybridization; Indoles; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurokinin A; Oligopeptides; omega-N-Methylarginine; Peptide Fragments; Phenanthridines; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; RNA, Messenger; Signal Transduction; Substance P; Tachykinins; Tetrodotoxin; Tritium | 2000 |
Respiratory actions of tachykinins in the nucleus of the solitary tract: effect of neonatal capsaicin pretreatment.
Topics: Animals; Animals, Newborn; Capsaicin; Male; Microinjections; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Rats, Wistar; Respiratory Mechanics; Solitary Nucleus; Substance P; Tachykinins | 2000 |
Hormonal variation of rat uterine contractile responsiveness to selective neurokinin receptor agonists.
Topics: Animals; Diestrus; Estrogens; Estrus; Female; Metestrus; Neurokinin A; Ovariectomy; Peptide Fragments; Piperidines; Proestrus; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Uterine Contraction | 2000 |
Differences in circular muscle contraction and peristaltic motor inhibition caused by tachykinin NK1 receptor agonists in the guinea-pig small intestine.
Topics: Adenosine Triphosphate; Animals; Enzyme Inhibitors; Female; Guinea Pigs; Intestine, Small; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Piperidines; Purinergic P2 Receptor Antagonists; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sincalide; Spasm; Substance P; Suramin; Tetrodotoxin | 2000 |
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan | 2000 |
Potent NK1 antagonism by SR-140333 reduces rat colonic secretory response to immunocyte activation.
Topics: Animals; Benzamides; Capsaicin; Colon; Colonic Diseases, Functional; Electric Stimulation; Male; Mast Cells; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stress, Physiological; Substance P | 2001 |
NK2 tachykinin receptors mediate contraction of the pig intravesical ureter: tachykinin-induced enhancement of non-adrenergic non-cholinergic excitatory neurotransmission.
Topics: Animals; Female; In Vitro Techniques; Isometric Contraction; Male; Muscle Tonus; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-2; Substance P; Swine; Synaptic Transmission; Ureter | 2001 |
Radioligand binding and functional characterisation of tachykinin receptors in chicken small intestine.
Topics: Animals; Binding, Competitive; Chickens; Female; In Vitro Techniques; Intestine, Small; Neurokinin A; Peptide Fragments; Radioligand Assay; Radiopharmaceuticals; Receptors, Tachykinin; Substance P; Succinimides | 2001 |
Nonpeptide tachykinin receptor antagonists. III. SB 235375, a low central nervous system-penetrant, potent and selective neurokinin-3 receptor antagonist, inhibits citric acid-induced cough and airways hyper-reactivity in guinea pigs.
Topics: Acetates; Animals; Antitussive Agents; Behavior, Animal; Bronchial Hyperreactivity; Calcium; Central Nervous System; Citric Acid; Cloning, Molecular; Cough; Guinea Pigs; In Vitro Techniques; Iris; Male; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptide Fragments; Pupil; Quinolines; Rabbits; Radioligand Assay; Rats; Receptors, Neurokinin-3; Receptors, Tachykinin; Recombinant Proteins; Substance P | 2002 |
Neurokinin-receptor-mediated depolarization of cortical neurons elicits an increase in glutamate release at excitatory synapses.
Topics: Action Potentials; Animals; Entorhinal Cortex; Excitatory Postsynaptic Potentials; Glutamic Acid; Hippocampus; Interneurons; Male; Neurokinin A; Neurokinin B; Patch-Clamp Techniques; Peptide Fragments; Pyramidal Cells; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Synapses; Tetrodotoxin | 2002 |
Action of tachykinins in the rat hippocampus: modulation of inhibitory synaptic transmission.
Topics: Animals; Animals, Newborn; Bicuculline; Drug Interactions; Excitatory Amino Acid Antagonists; GABA Antagonists; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Neural Inhibition; Neurokinin A; Neurokinin-1 Receptor Antagonists; Neuropeptides; Patch-Clamp Techniques; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tachykinins; Time Factors | 2003 |
Tachykinin receptor (NK(1), NK(2), NK(3)) binding sites in the rat caudal brainstem following neonatal capsaicin administration.
Topics: Animals; Animals, Newborn; Autoradiography; Brain Stem; Capsaicin; Indicators and Reagents; Iodine Radioisotopes; Neurokinin A; Peptide Fragments; Rats; Receptors, Tachykinin; Substance P; Succinimides | 2003 |
Effects of neuropeptides on the sumatriptan-disturbed circulation in the optic nerve head of rabbits.
Topics: Animals; Arterioles; Blood-Retinal Barrier; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Female; Male; Microinjections; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neuropeptides; Optic Nerve; Peptide Fragments; Rabbits; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Retinal Vessels; Substance P; Sumatriptan; Vasodilation | 2004 |
Circular versus longitudinal myometrial contractile response to selective tachykinin receptor agonists in rat.
Topics: Animals; Female; Myometrium; Neurokinin A; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Tachykinin; Substance P; Uterine Contraction; Uterus | 2003 |
Effects of TAK-637 on NK(1) receptor-mediated mechanisms regulating colonic secretion.
Topics: Animals; Capsaicin; Colforsin; Colon; Electric Stimulation; Electrophysiology; Guinea Pigs; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Male; Naphthyridines; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Statistics, Nonparametric; Substance P; Tetrodotoxin | 2004 |
The ventral tegmental area as a putative target for tachykinins in cardiovascular regulation.
Topics: Acetates; Adrenergic beta-Antagonists; Animals; Atenolol; Behavior, Animal; Benzamides; Benzazepines; Blood Pressure; Dopamine D2 Receptor Antagonists; Glutamic Acid; Heart Rate; Indoles; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Ventral Tegmental Area | 2005 |
Senktide-induced gerbil foot tapping behaviour is blocked by selective tachykinin NK1 and NK3 receptor antagonists.
Topics: Animals; Autoradiography; Behavior, Animal; Brain; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Foot; Gerbillinae; Injections, Intraventricular; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P | 2007 |
Expression and coupling of neurokinin receptor subtypes to inositol phosphate and calcium signaling pathways in human airway smooth muscle cells.
Topics: Boron Compounds; Calcium Signaling; Humans; Imidazoles; Inositol 1,4,5-Trisphosphate; Muscle, Smooth; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; RNA, Messenger; Substance P; Trachea | 2008 |
Neurokinin receptor modulation of respiratory activity in the rabbit.
Topics: Animals; Exhalation; Inhalation; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phrenic Nerve; Piperidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Vagotomy | 2008 |
Are biological actions of neurokinin A in the adult brain mediated by a cross-talk between the NK1 and NK2 receptors?
Topics: Animals; Behavior, Animal; Benzamides; Brain; Dose-Response Relationship, Drug; Grooming; Injections, Intraventricular; Isoindoles; Male; Mice; Mice, Knockout; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Receptor Cross-Talk; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Stereoisomerism; Substance P | 2012 |
Effects of intravenous administration of neurokinin receptor subtype-selective agonists on gonadotropin-releasing hormone pulse generator activity and luteinizing hormone secretion in goats.
Topics: Animals; Estradiol; Female; Goats; Gonadotropin-Releasing Hormone; Infusions, Intravenous; Kisspeptins; Ligands; Luteinizing Hormone; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Signal Transduction; Substance P; Time Factors | 2015 |