Page last updated: 2024-09-02

senktide and cp 99994

senktide has been researched along with cp 99994 in 7 studies

Compound Research Comparison

Studies
(senktide)
Trials
(senktide)
Recent Studies (post-2010)
(senktide)
Studies
(cp 99994)
Trials
(cp 99994)
Recent Studies (post-2010) (cp 99994)
292150231219

Protein Interaction Comparison

ProteinTaxonomysenktide (IC50)cp 99994 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 2Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 3Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 4Rattus norvegicus (Norway rat)0.0006
Substance-P receptorHomo sapiens (human)0.0004

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (57.14)18.2507
2000's2 (28.57)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brawner, ME; Elshourbagy, NA; Foley, JJ; Giardina, GA; Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Potts, W; Sarau, HM; Schmidt, DB; Webb, EF1
Griswold, DE; Hay, DW; Martin, LD; Medhurst, AD; Parsons, AA1
MacNaughton, W; Moore, B; Vanner, S1
Bornstein, JC; Burcher, E; Johnson, PJ1
Adolfsson, R; Ahlstedt, I; de Verdier, J; Drmota, T; Engberg, S; Johansson, A; Jussila, R; Kristensson, E; Leffler, A; Lindström, E; Novén, A; Påhlman, I; Sigfridsson, K; Sundqvist, M; von Mentzer, B1
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T1
Corboz, MR; Eckel, SP; Rivelli, MA1

Other Studies

7 other study(ies) available for senktide and cp 99994

ArticleYear
Nonpeptide tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:3

    Topics: Animals; Calcium; CHO Cells; Cricetinae; Dogs; Humans; Mice; Piperidines; Quinolines; Rabbits; Radioligand Assay; Rats; Receptors, Neurokinin-3; Receptors, Tachykinin

1997
In vitro and in vivo characterization of NK3 receptors in the rabbit eye by use of selective non-peptide NK3 receptor antagonists.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: Animals; In Vitro Techniques; Iris; Male; Miosis; Muscle Contraction; Muscle, Smooth; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Rabbits; Receptors, Neurokinin-3; Substance P

1997
Cellular pathways mediating tachykinin-evoked secretomotor responses in guinea pig ileum.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Animals; Capsaicin; Electric Stimulation; Evoked Potentials; Guinea Pigs; Ileum; In Vitro Techniques; Intestinal Mucosa; Membrane Potentials; Muscle, Smooth; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tachykinins

1997
Roles of neuronal NK1 and NK3 receptors in synaptic transmission during motility reflexes in the guinea-pig ileum.
    British journal of pharmacology, 1998, Volume: 124, Issue:7

    Topics: Animals; Female; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Neurokinin-1 Receptor Antagonists; Neurons; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Synaptic Transmission

1998
Senktide-induced gerbil foot tapping behaviour is blocked by selective tachykinin NK1 and NK3 receptor antagonists.
    European journal of pharmacology, 2007, Dec-22, Volume: 577, Issue:1-3

    Topics: Animals; Autoradiography; Behavior, Animal; Brain; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Foot; Gerbillinae; Injections, Intraventricular; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

2007
Neurokinin receptor modulation of respiratory activity in the rabbit.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Animals; Exhalation; Inhalation; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phrenic Nerve; Piperidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Vagotomy

2008
Bronchoconstrictor effect of the tachykinin NK₃-receptor agonists [MePhe⁷]-neurokinin B and senktide in the isolated guinea pig lung.
    Experimental lung research, 2010, Volume: 36, Issue:9

    Topics: Animals; Bronchoconstriction; Bronchoconstrictor Agents; CHO Cells; Cricetinae; Cricetulus; Disease Models, Animal; Guinea Pigs; In Vitro Techniques; Lung; Male; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-3; Substance P

2010