Page last updated: 2024-09-05

senicapoc and tram 34

senicapoc has been researched along with tram 34 in 3 studies

Compound Research Comparison

Studies
(senicapoc)
Trials
(senicapoc)
Recent Studies (post-2010)
(senicapoc)
Studies
(tram 34)
Trials
(tram 34)
Recent Studies (post-2010) (tram 34)
423322081144

Protein Interaction Comparison

ProteinTaxonomysenicapoc (IC50)tram 34 (IC50)
Intermediate conductance calcium-activated potassium channel protein 4Homo sapiens (human)0.02
Potassium voltage-gated channel subfamily A member 3Homo sapiens (human)5

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brown, DT; Christophersen, P; Demnitz, J; Dyhring, T; Jørgensen, S; Strøbæk, D1
Dale, E; Eder, C; Möller, T; Staal, RG1
Brown, BM; Pressley, B; Wulff, H1

Reviews

1 review(s) available for senicapoc and tram 34

ArticleYear
KCa 3.1-a microglial target ready for drug repurposing?
    Glia, 2016, Volume: 64, Issue:10

    Topics: Acetamides; Animals; Drug Repositioning; Humans; Intermediate-Conductance Calcium-Activated Potassium Channels; Microglia; Pyrazoles; Trityl Compounds

2016

Other Studies

2 other study(ies) available for senicapoc and tram 34

ArticleYear
A high-throughput screening campaign for detection of ca(2+)-activated k(+) channel activators and inhibitors using a fluorometric imaging plate reader-based tl(+)-influx assay.
    Assay and drug development technologies, 2013, Volume: 11, Issue:3

    Topics: Acetamides; Algorithms; Data Interpretation, Statistical; Erythrocytes; Fluorometry; HEK293 Cells; High-Throughput Screening Assays; Humans; Inflammatory Bowel Diseases; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Pyrazoles; Small Molecule Libraries; Thallium; Thiazines; Trityl Compounds

2013
KCa3.1 Channel Modulators as Potential Therapeutic Compounds for Glioblastoma.
    Current neuropharmacology, 2018, Volume: 16, Issue:5

    Topics: Acetamides; Animals; Brain Neoplasms; Glioblastoma; Humans; Intermediate-Conductance Calcium-Activated Potassium Channels; Membrane Transport Modulators; Pyrazoles; Trityl Compounds

2018