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selegiline and 8-(3-chlorostyryl)caffeine

selegiline has been researched along with 8-(3-chlorostyryl)caffeine in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's4 (80.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bolognesi, ML; Cavalli, A; Melchiorre, C; Minarini, A; Recanatini, M; Rosini, M; Tumiatti, V1
Bartoccini, F; Borsini, F; Cabri, W; Diamantini, G; Minetti, P; Mor, M; Pala, D; Piersanti, G; Riccioni, T; Rivara, S; Stasi, MA; Tarzia, G1
Gütschow, M; Heer, J; Hinz, S; Küppers, P; Müller, CE; Schlenk, M; Stössel, A1
Akkari, R; Borrmann, T; Brunschweiger, A; Drabczyńska, A; Hockemeyer, J; Kieć-Kononowicz, K; Koch, P; Köse, M; Küppers, P; Müller, CE; Radjainia, H; Schlenk, M1
Almos, T; Edmondson, DE; Massari, ME; Rojas, RJ; Scott, R1

Reviews

1 review(s) available for selegiline and 8-(3-chlorostyryl)caffeine

ArticleYear
Multi-target-directed ligands to combat neurodegenerative diseases.
    Journal of medicinal chemistry, 2008, Feb-14, Volume: 51, Issue:3

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Binding Sites; Calcium Channel Blockers; Chelating Agents; Cholinesterase Inhibitors; Humans; Huntington Disease; Ligands; Multiple Sclerosis; Neurodegenerative Diseases; Neurofibrillary Tangles; Neurotransmitter Agents; Parkinson Disease; Plaque, Amyloid

2008

Other Studies

4 other study(ies) available for selegiline and 8-(3-chlorostyryl)caffeine

ArticleYear
Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.
    Journal of medicinal chemistry, 2013, Feb-14, Volume: 56, Issue:3

    Topics: Caffeine; HEK293 Cells; Humans; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Docking Simulation; Monoamine Oxidase Inhibitors; Xanthines

2013
Dual targeting of adenosine A(2A) receptors and monoamine oxidase B by 4H-3,1-benzothiazin-4-ones.
    Journal of medicinal chemistry, 2013, Jun-13, Volume: 56, Issue:11

    Topics: Adenosine A2 Receptor Antagonists; Animals; Benzothiadiazines; Brain; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Humans; In Vitro Techniques; Isoenzymes; Liver; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Phenylbutyrates; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Stereoisomerism; Structure-Activity Relationship; Thiazines

2013
1,3-Dialkyl-substituted tetrahydropyrimido[1,2-f]purine-2,4-diones as multiple target drugs for the potential treatment of neurodegenerative diseases.
    Bioorganic & medicinal chemistry, 2013, Dec-01, Volume: 21, Issue:23

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Caffeine; CHO Cells; Cricetulus; Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neurodegenerative Diseases; Purinergic P1 Receptor Antagonists; Purines; Xanthines

2013
Reversible and irreversible small molecule inhibitors of monoamine oxidase B (MAO-B) investigated by biophysical techniques.
    Bioorganic & medicinal chemistry, 2015, Feb-15, Volume: 23, Issue:4

    Topics: Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Parkinson Disease; Small Molecule Libraries; Thermodynamics

2015