Page last updated: 2024-09-03

sdz nvi-085 and prazosin

sdz nvi-085 has been researched along with prazosin in 6 studies

Compound Research Comparison

Studies
(sdz nvi-085)
Trials
(sdz nvi-085)
Recent Studies (post-2010)
(sdz nvi-085)
Studies
(prazosin)
Trials
(prazosin)
Recent Studies (post-2010) (prazosin)
10107,914713682

Protein Interaction Comparison

ProteinTaxonomysdz nvi-085 (IC50)prazosin (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)5.87
Interstitial collagenaseHomo sapiens (human)4.036
Alpha-2A adrenergic receptorHomo sapiens (human)2.638
Matrix metalloproteinase-9Homo sapiens (human)6.963
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0008
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)0.0078
Alpha-2B adrenergic receptorHomo sapiens (human)0.29
Alpha-2C adrenergic receptorHomo sapiens (human)0.647
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0008
Alpha-1D adrenergic receptorHomo sapiens (human)0.0007
Bromodomain-containing protein 2Homo sapiens (human)0.0009
Alpha-1A adrenergic receptorHomo sapiens (human)0.0006
Alpha-1B adrenergic receptorHomo sapiens (human)0.0006
5-hydroxytryptamine receptor 2BHomo sapiens (human)4.118
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0008
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)9.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.5849
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.6

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dement, WC; Guilleminault, C; Mignot, E; Nishino, S; Renaud, A1
Büscher, R; Insel, PA; Michel, MC1
Oriowo, MA1
Kalkman, HO; Neumann, V1
Clarke, DE; Ford, AP; Lachnit, WG1
Hasegawa, Y; Ono, H; Wada, T1

Other Studies

6 other study(ies) available for sdz nvi-085 and prazosin

ArticleYear
Effects of SDZ NVI-085, a putative subtype-selective alpha 1-agonist, on canine cataplexy, a disorder of rapid eye movement sleep.
    European journal of pharmacology, 1991, Nov-19, Volume: 205, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Body Temperature; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Cataplexy; Disease Models, Animal; Dogs; Eating; Heart Rate; Narcolepsy; Oxazines; Play and Playthings; Prazosin; Radioligand Assay; Yohimbine

1991
Is SDZ NVI-085 an alpha 1-adrenoceptor subtype-selective agonist?
    Life sciences, 1994, Volume: 54, Issue:14

    Topics: Adrenergic alpha-Agonists; Animals; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Cattle; Cell Line; Cerebral Cortex; Clonidine; In Vitro Techniques; Inositol Phosphates; Kidney; Norepinephrine; Oxazines; Prazosin; Rats; Receptors, Adrenergic, alpha; Spleen; Transfection

1994
Alpha 1-adrenoceptor subtype(s) mediating noradrenaline-induced contractions of the guinea-pig aorta.
    Fundamental & clinical pharmacology, 1994, Volume: 8, Issue:3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Clonidine; Dioxanes; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Oxazines; Prazosin; Receptors, Adrenergic, alpha-1

1994
Evidence for a 5-HT1D receptor-mediated hypothermic effect of the alpha 1-adrenoceptor agonist, SDZ NVI-085, in guinea-pigs.
    European journal of pharmacology, 1995, Oct-24, Volume: 285, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Body Temperature; Bridged-Ring Compounds; Clonidine; Guinea Pigs; In Vitro Techniques; Male; Oxadiazoles; Oxazines; Piperazines; Prazosin; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
SDZ NVI 085, an alpha 1A-adrenoceptor agonist with 5-HT2A receptor antagonist properties.
    European journal of pharmacology, 1996, Feb-15, Volume: 297, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bridged-Ring Compounds; Idazoxan; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Oxazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Regional Blood Flow; Serotonin Antagonists; Tail

1996
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
    European journal of pharmacology, 1997, Dec-04, Volume: 340, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord

1997