Page last updated: 2024-09-05

sdz mks 492 and histamine

sdz mks 492 has been researched along with histamine in 2 studies

*Histamine: An amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscle, a vasodilator, and also a centrally acting neurotransmitter. [MeSH]

*Histamine: An amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial smooth muscle, a vasodilator, and also a centrally acting neurotransmitter. [MeSH]

Compound Research Comparison

Studies
(sdz mks 492)
Trials
(sdz mks 492)
Recent Studies (post-2010)
(sdz mks 492)
Studies
(histamine)
Trials
(histamine)
Recent Studies (post-2010) (histamine)
82037,7181,3723,457

Protein Interaction Comparison

ProteinTaxonomysdz mks 492 (IC50)histamine (IC50)
Histamine H1 receptorRattus norvegicus (Norway rat)0.1585
Histamine H1 receptorHomo sapiens (human)0.1585

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Inagaki, N; Iwama, T; Kitagaki, K; Koda, A; Nagai, H; Sakurai, T; Yamaguchi, S1
Kitagaki, K; Koda, A; Nagai, H; Tsuruoka, N; Yamaguchi, S1

Other Studies

2 other study(ies) available for sdz mks 492 and histamine

ArticleYear
Effects of MKS-492 on antigen-induced bronchoconstriction and allergic reaction in guinea pigs and rats.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:4

    Topics: Aminophylline; Animals; Antigens; Bronchial Hyperreactivity; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Female; Guinea Pigs; Histamine; Histamine Release; Hypersensitivity; Leukocyte Count; Leukotriene B4; Male; Muscle Relaxation; Muscle, Smooth; Passive Cutaneous Anaphylaxis; Phosphodiesterase Inhibitors; Platelet Activating Factor; Purinones; Rats; Rats, Wistar; Superoxides; Trachea

1993
Priming with murine recombinant interleukin-5 resulted in the augmentation of PAF-induced airway hyperresponsiveness to histamine in guinea pigs.
    Life sciences, 1993, Volume: 52, Issue:17

    Topics: Aminophylline; Animals; Bronchoconstriction; Guinea Pigs; Histamine; Interleukin-5; Leukocyte Count; Male; Naphthyridines; Phosphodiesterase Inhibitors; Platelet Activating Factor; Purinones; Recombinant Proteins

1993