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sdz 205-557 and tropisetron

sdz 205-557 has been researched along with tropisetron in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (81.82)18.2507
2000's2 (18.18)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ellis, ES; Gaster, LM; Jennings, AJ; Joiner, GF; King, FD; Mulholland, KR; Rahman, SK; Starr, S; Wardle, KA; Wyman, PA1
Fischmeister, R; Langlois, M1
Boulouard, M; Bureau, R; Butt-Gueulle, S; Dauphin, F; Daveu, C; Duchatelle, P; Dumuis, A; Lelong-Boulouard, V; LemaƮtre, S; Lepailleur, A; Lezoualc'h, F; Pfeiffer, B; Rault, S1
Buchheit, KH; Gamse, R; Pfannkuche, HJ1
Franks, CM; Hardcastle, J; Hardcastle, PT; Sanger, GJ1
Buchheit, KH; Buhl, T1
Cheng, CH; Costall, B; Kelly, ME; Naylor, RJ1
Bornstein, JC; Furness, JB; Yuan, SY1
Costall, B; Naylor, RJ1
Flynn, DL; Goldstin, B; Gullikson, GW; Moormann, AE; Yang, DC1
Sugimoto, Y; Yamada, J; Yoshikawa, T1

Reviews

2 review(s) available for sdz 205-557 and tropisetron

ArticleYear
5-HT4 receptor ligands: applications and new prospects.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Benzoates; Binding Sites; Cardiovascular Physiological Phenomena; Central Nervous System; Digestive System Physiological Phenomena; Humans; Indoles; Ketones; Ligands; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003
The pharmacology of the 5-HT4 receptor.
    International clinical psychopharmacology, 1993, Volume: 8 Suppl 2

    Topics: 4-Aminobenzoic Acid; 5-Hydroxytryptophan; Animals; Anxiety; Arousal; Brain; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Indoles; Mice; Neural Inhibition; Ondansetron; para-Aminobenzoates; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron

1993

Other Studies

9 other study(ies) available for sdz 205-557 and tropisetron

ArticleYear
(1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramide.
    Journal of medicinal chemistry, 1993, Dec-10, Volume: 36, Issue:25

    Topics: Animals; Dioxanes; Guinea Pigs; Metoclopramide; Muscle Contraction; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1993
Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
    Bioorganic & medicinal chemistry, 2009, Mar-15, Volume: 17, Issue:6

    Topics: Animals; Chlorocebus aethiops; COS Cells; Humans; Indoles; Models, Molecular; Molecular Structure; Pyrazines; Radioligand Assay; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides

2009
SDZ 205-557, a selective, surmountable antagonist for 5-HT4 receptors in the isolated guinea pig ileum.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:4

    Topics: 4-Aminobenzoic Acid; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Radioligand Assay; Serotonin Antagonists; Tropisetron

1992
Do 5-HT4 receptors mediate the intestinal secretory response to 5-HT in rat in-vivo?
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; 5-Methoxytryptamine; Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Colon; Dioxanes; Dose-Response Relationship, Drug; Heart Rate; Ileum; Indoles; Intestinal Mucosa; Jejunum; Male; para-Aminobenzoates; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron

1995
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron

1994
Actions of 5-hydroxytryptophan to inhibit and disinhibit mouse behaviour in the light/dark test.
    European journal of pharmacology, 1994, Apr-01, Volume: 255, Issue:1-3

    Topics: 4-Aminobenzoic Acid; 5-Hydroxytryptophan; Animals; Behavior, Animal; Brain Chemistry; Darkness; Indoles; Light; Male; Mice; Mice, Inbred Strains; Neostriatum; Neurotransmitter Agents; para-Aminobenzoates; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron

1994
Investigation of the role of 5-HT3 and 5-HT4 receptors in ascending and descending reflexes to the circular muscle of guinea-pig small intestine.
    British journal of pharmacology, 1994, Volume: 112, Issue:4

    Topics: 4-Aminobenzoic Acid; Animals; Female; Guinea Pigs; In Vitro Techniques; Indoles; Intestine, Small; Male; Muscle, Smooth; para-Aminobenzoates; Receptors, Serotonin; Reflex; Serotonin Antagonists; Tropisetron

1994
SC-53606, a potent and selective antagonist of 5-hydroxytryptamine4 receptors in isolated rat esophageal tunica muscularis mucosae.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Esophagus; Imidazoles; In Vitro Techniques; Indoles; Male; Mucous Membrane; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Pyrroles; Rats; Receptors, Cell Surface; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron; Tryptamines

1993
p-Chloroamphetamine, a serotonin-releasing drug, elicited in rats a hyperglycemia mediated by the 5-HT1A and 5-HT2B/2C receptors.
    European journal of pharmacology, 1998, Oct-23, Volume: 359, Issue:2-3

    Topics: 4-Aminobenzoic Acid; Adrenal Medulla; Adrenalectomy; Aminopyridines; Animals; Blood Glucose; Dose-Response Relationship, Drug; Ergolines; Fenclonine; Hyperglycemia; Indoles; Ketanserin; Male; Methysergide; p-Chloroamphetamine; para-Aminobenzoates; Piperazines; Propranolol; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ritanserin; Serotonin; Serotonin Agents; Serotonin Antagonists; Tropisetron

1998