Page last updated: 2024-09-03

sch 39370 and phosphoramidon

sch 39370 has been researched along with phosphoramidon in 4 studies

Compound Research Comparison

Studies
(sch 39370)
Trials
(sch 39370)
Recent Studies (post-2010)
(sch 39370)
Studies
(phosphoramidon)
Trials
(phosphoramidon)
Recent Studies (post-2010) (phosphoramidon)
25107811233

Protein Interaction Comparison

ProteinTaxonomysch 39370 (IC50)phosphoramidon (IC50)
ThermolysinBacillus thermoproteolyticus0.033
NeprilysinRattus norvegicus (Norway rat)0.0578
NeprilysinOryctolagus cuniculus (rabbit)0.0028
NeprilysinHomo sapiens (human)0.0405
Angiotensin-converting enzyme Homo sapiens (human)0.615
Endothelin-converting enzyme 1Homo sapiens (human)1.0695
P2Y purinoceptor 12Homo sapiens (human)0.017

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Casley, DJ; Haslanger, MF; Johnston, CI; Kanazawa, M; Sybertz, EJ1
Fyhrquist, F; Metsärinne, K; Saijonmaa, O; Sirviö, ML1
Boublik, JH; Evans, RG; Lakat, L; Lew, RA; Pipolo, LA; Smith, AI; Tomoda, F1
Kokkonen, JO; Kovanen, PT; Kuoppala, A; Lindstedt, KA; Saarinen, J1

Other Studies

4 other study(ies) available for sch 39370 and phosphoramidon

ArticleYear
Localization and characterization of neutral metalloendopeptidase (EC 3.4.24.11), the degradative enzyme for atrial natriuretic peptide, in rat kidney using a radioiodinated neutral metalloendopeptidase inhibitor.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Animals; Atrial Natriuretic Factor; Autoradiography; Binding, Competitive; Cell Membrane; Dipeptides; Drug Interactions; Glycopeptides; Iodine Radioisotopes; Kidney; Male; Neprilysin; Phenols; Phenylalanine; Rats; Rats, Inbred Strains; Thiorphan

1992
Degradation of endothelin-1 by extracts of rat lung, kidney, and liver.
    Regulatory peptides, 1995, Feb-14, Volume: 55, Issue:3

    Topics: alpha-Amylases; Animals; Chromatography, High Pressure Liquid; Dipeptides; Edetic Acid; Endothelins; Glycopeptides; Iodine Radioisotopes; Kidney; Liver; Lung; Male; Neprilysin; Pancreatic Elastase; Plant Proteins; Rats; Rats, Wistar; Trypsin Inhibitors

1995
Synthetic inhibitors of endopeptidase EC 3.4.24.15: potency and stability in vitro and in vivo.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Analysis of Variance; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Bradykinin; Dipeptides; Dose-Response Relationship, Drug; Glycopeptides; Gonadotropin-Releasing Hormone; In Vitro Techniques; Kidney; Metalloendopeptidases; Protease Inhibitors; Rabbits; Rats; Stereoisomerism; Vasoconstrictor Agents

1996
Kallidin- and bradykinin-degrading pathways in human heart: degradation of kallidin by aminopeptidase M-like activity and bradykinin by neutral endopeptidase.
    Circulation, 1999, Apr-20, Volume: 99, Issue:15

    Topics: Angiotensin-Converting Enzyme Inhibitors; Anti-Bacterial Agents; Bradykinin; Captopril; CD13 Antigens; Dipeptides; Female; Glycopeptides; Heart Failure; Humans; Kallidin; Leucine; Male; Membrane Proteins; Middle Aged; Myocardium; Neprilysin; Peptides; Peptidyl-Dipeptidase A; Protease Inhibitors; Substrate Specificity

1999