Page last updated: 2024-09-02

sch 28080 and vanadates

sch 28080 has been researched along with vanadates in 17 studies

Compound Research Comparison

Studies
(sch 28080)
Trials
(sch 28080)
Recent Studies (post-2010)
(sch 28080)
Studies
(vanadates)
Trials
(vanadates)
Recent Studies (post-2010) (vanadates)
2170205,2007785

Protein Interaction Comparison

ProteinTaxonomysch 28080 (IC50)vanadates (IC50)
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)0.0254

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19905 (29.41)18.7374
1990's8 (47.06)18.2507
2000's3 (17.65)29.6817
2010's1 (5.88)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cain, BD; Curran, KA; Hebert, MJ; Wingo, CS1
Asano, S; Tabuchi, Y; Takeguchi, M; Takeguchi, N1
Anagnostopoulos, T; Cheval, L; Doucet, A; Planelles, G1
Barry, CR; Youmans, SJ1
Blostein, R; Polvani, C; Sachs, G1
Bassilian, S; Gunther, RD; Rabon, EC1
Garg, LC; Narang, N1
McBride, DE; Perrone, RD1
Kaunitz, JD; Sachs, G1
Kleinman, JG; Pscheidt, R; Tipnis, P1
Chatterjee, PK; Das, PK1
QuiƱones, L; Rodriguez, C; Specht, SC; Velazquez, S1
de Pont, JJ; Hermsen, HP; Koenderink, JB; Swarts, HG; Willems, PH1
De Pont, JJ; Koenderink, JB; Swarts, HG; Willems, PH2
De Pont, JJ; Koenderink, JB; Krieger, E; Swarts, HG; Willems, PH1
Cain, BD; Gumz, ML; Shao, J; Shull, GE; van Driel, IR; Wingo, CS; Xia, SL1

Other Studies

17 other study(ies) available for sch 28080 and vanadates

ArticleYear
Evidence for the presence of a K-dependent acidifying adenosine triphosphatase in the rabbit renal medulla.
    Kidney international, 1992, Volume: 42, Issue:5

    Topics: Adenosine Triphosphate; Animals; Female; H(+)-K(+)-Exchanging ATPase; Hydrogen-Ion Concentration; Hydrolysis; Imidazoles; Kidney Medulla; Microsomes; Proton Pump Inhibitors; Rabbits; Subcellular Fractions; Vanadates

1992
Ouabain-insensitive, vanadate-sensitive K(+)-ATPase of rat distal colon is partly similar to gastric H+,K(+)-ATPase.
    The Japanese journal of physiology, 1992, Volume: 42, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Anti-Ulcer Agents; Antibodies, Monoclonal; Binding Sites, Antibody; Cation Transport Proteins; Colon; H(+)-K(+)-Exchanging ATPase; Imidazoles; Intracellular Membranes; Male; Ouabain; Proton Pump Inhibitors; Rats; Rats, Sprague-Dawley; Sodium-Potassium-Exchanging ATPase; Stomach; Swine; Vanadates

1992
Biochemical and functional characterization of H(+)-K(+)-ATPase in distal amphibian nephron.
    The American journal of physiology, 1991, Volume: 260, Issue:6 Pt 2

    Topics: Adenosine Triphosphatases; Animals; Anti-Ulcer Agents; H(+)-K(+)-Exchanging ATPase; Hydrogen-Ion Concentration; Imidazoles; Kidney Tubules, Distal; Microinjections; Necturus maculosus; Omeprazole; Rana ridibunda; Vanadates

1991
Effects of valinomycin on vanadate-sensitive and vanadate-resistant H+ transport in vesicles from turtle bladder epithelium: evidence for a K+/H+ exchanger.
    Biochemical and biophysical research communications, 1991, May-15, Volume: 176, Issue:3

    Topics: Adenosine Triphosphate; Animals; Carrier Proteins; Epithelium; Hydrogen; Imidazoles; Kinetics; Nigericin; Potassium-Hydrogen Antiporters; Turtles; Urinary Bladder; Valinomycin; Vanadates

1991
Sodium ions as substitutes for protons in the gastric H,K-ATPase.
    The Journal of biological chemistry, 1989, Oct-25, Volume: 264, Issue:30

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Anti-Ulcer Agents; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Imidazoles; Kinetics; Protons; Sodium; Swine; Vanadates

1989
Cation transport in vesicles from secreting rabbit stomach.
    The Journal of biological chemistry, 1987, Oct-15, Volume: 262, Issue:29

    Topics: Adenosine Triphosphatases; Animals; Anti-Ulcer Agents; Cell Fractionation; Centrifugation, Density Gradient; Cytoplasmic Granules; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Imidazoles; Kinetics; Microsomes; Rabbits; Rubidium; Valinomycin; Vanadates

1987
Ouabain-insensitive K-adenosine triphosphatase in distal nephron segments of the rabbit.
    The Journal of clinical investigation, 1988, Volume: 81, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Cation Transport Proteins; H(+)-K(+)-Exchanging ATPase; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Kidney Tubules; Kidney Tubules, Distal; Omeprazole; Ouabain; Rabbits; Sodium Chloride; Sodium-Potassium-Exchanging ATPase; Vanadates

1988
Aldosterone and PCO2 enhance rubidium absorption in rat distal colon.
    The American journal of physiology, 1988, Volume: 254, Issue:6 Pt 1

    Topics: Acetazolamide; Adenosine Triphosphatases; Aldosterone; Animals; Anti-Ulcer Agents; Biological Transport, Active; Bumetanide; Carbon Dioxide; Colon; Furosemide; Hydrogen-Ion Concentration; Imidazoles; Intestinal Absorption; Male; Omeprazole; Ouabain; Potassium; Rats; Rats, Inbred Strains; Rubidium; Sodium; Vanadates

1988
Identification of a vanadate-sensitive potassium-dependent proton pump from rabbit colon.
    The Journal of biological chemistry, 1986, Oct-25, Volume: 261, Issue:30

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Chlorides; Colon; Ethylmaleimide; H(+)-K(+)-Exchanging ATPase; Hydrolysis; Imidazoles; Potassium; Rabbits; Valinomycin; Vanadates; Vanadium

1986
H(+)-K(+)-ATPase of rat inner medullary collecting duct in primary culture.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 2

    Topics: Animals; Anti-Bacterial Agents; Biological Transport; Cells, Cultured; Ethylmaleimide; H(+)-K(+)-Exchanging ATPase; Hydrogen-Ion Concentration; Imidazoles; Kidney Medulla; Kidney Tubules, Collecting; Kinetics; Macrolides; Omeprazole; Ouabain; Potassium; Proton Pump Inhibitors; Rats; Rats, Sprague-Dawley; Vanadates

1993
Characterization of Syrian hamster gastric mucosal H+,K+-ATPase.
    Molecular and cellular biochemistry, 1995, Jul-19, Volume: 148, Issue:2

    Topics: Adenosine Triphosphate; Animals; Anti-Ulcer Agents; Cricetinae; Enzyme Inhibitors; Female; Gastric Acid; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Imidazoles; Male; Mesocricetus; Nigericin; Omeprazole; Phosphorylation; Proton Pump Inhibitors; Protons; Substrate Specificity; Vanadates

1995
Effect of high ionic strength and inhibitors of H,K-ATPase on the ouabain-sensitive K-p-nitrophenylphosphatase activity in the sea anemone Stichodactyla helianthus.
    Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology, 1997, Volume: 117, Issue:2

    Topics: 4-Nitrophenylphosphatase; Animals; Choline; Enzyme Inhibitors; Hydrogen-Ion Concentration; Imidazoles; Omeprazole; Osmolar Concentration; Ouabain; Potassium; Potassium Chloride; Proton Pump Inhibitors; Rats; Sea Anemones; Sodium-Potassium-Exchanging ATPase; Vanadates

1997
Conformation-dependent inhibition of gastric H+,K+-ATPase by SCH 28080 demonstrated by mutagenesis of glutamic acid 820.
    Molecular pharmacology, 1999, Volume: 55, Issue:3

    Topics: Adenosine Triphosphate; Animals; Catalysis; Cells, Cultured; Enzyme Inhibitors; Glutamic Acid; H(+)-K(+)-Exchanging ATPase; Imidazoles; Mutagenesis; Phosphates; Phosphorylation; Potassium; Protein Conformation; Proton Pump Inhibitors; Rats; Recombinant Proteins; Stomach; Time Factors; Vanadates

1999
The E1/E2-preference of gastric H,K-ATPase mutants.
    Annals of the New York Academy of Sciences, 2003, Volume: 986

    Topics: Amino Acid Substitution; Animals; Enzyme Inhibitors; Gastric Mucosa; Imidazoles; Kinetics; Mutagenesis, Site-Directed; Potassium; Protein Conformation; Recombinant Proteins; Sodium-Potassium-Exchanging ATPase; Vanadates

2003
Asn792 participates in the hydrogen bond network around the K+-binding pocket of gastric H,K-ATPase.
    The Journal of biological chemistry, 2005, Mar-25, Volume: 280, Issue:12

    Topics: Animals; Asparagine; Binding Sites; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Hydrogen Bonding; Imidazoles; Models, Molecular; Mutation; Phosphorylation; Potassium; Rats; Vanadates

2005
The non-gastric H,K-ATPase is oligomycin-sensitive and can function as an H+,NH4(+)-ATPase.
    The Journal of biological chemistry, 2005, Sep-30, Volume: 280, Issue:39

    Topics: Adenosine Triphosphatases; Ammonia; Animals; Baculoviridae; Binding Sites; Blotting, Western; Cation Transport Proteins; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Enzyme Inhibitors; H(+)-K(+)-Exchanging ATPase; Imidazoles; Kinetics; Mutagenesis, Site-Directed; Oligomycins; Ouabain; Phosphorylation; Potassium; Protein Binding; Protein Conformation; Protein Subunits; Rats; Recombinant Proteins; Sequence Deletion; Sodium; Spodoptera; Vanadates

2005
Pharmacological profiles of the murine gastric and colonic H,K-ATPases.
    Biochimica et biophysica acta, 2010, Volume: 1800, Issue:9

    Topics: Amiloride; Animals; Catalytic Domain; Colon; Drug Resistance; Enzyme Inhibitors; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Imidazoles; Mice; Mice, Knockout; Organ Specificity; Ouabain; Proton Pump Inhibitors; Sodium Channel Blockers; Vanadates

2010