Page last updated: 2024-09-02

sch 28080 and linaprazan

sch 28080 has been researched along with linaprazan in 2 studies

Compound Research Comparison

Studies
(sch 28080)
Trials
(sch 28080)
Recent Studies (post-2010)
(sch 28080)
Studies
(linaprazan)
Trials
(linaprazan)
Recent Studies (post-2010) (linaprazan)
2170201849

Protein Interaction Comparison

ProteinTaxonomysch 28080 (IC50)linaprazan (IC50)
Bile salt export pumpHomo sapiens (human)10
Cytochrome P450 3A4Homo sapiens (human)8.7

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bailey, N; Bamford, M; Demont, E; Elliott, R; Farre-Gutierrez, I; Garton, N; Hayhow, T; Hutley, G; Naylor, A; Panchal, T1
Andersson, K; Geibel, JP; Kirchhoff, P; Kosiek, O; Sidani, S; Socrates, T1

Other Studies

2 other study(ies) available for sch 28080 and linaprazan

ArticleYear
Evaluation of basic, heterocyclic ring systems as templates for use as potassium competitive acid blockers (pCABs).
    Bioorganic & medicinal chemistry letters, 2009, Dec-01, Volume: 19, Issue:23

    Topics: Binding, Competitive; Drug Design; Heterocyclic Compounds; Molecular Structure; Proton Pump Inhibitors; Pyridines; Stereoisomerism; Structure-Activity Relationship

2009
Characteristics of the K+-competitive H+,K+-ATPase inhibitor AZD0865 in isolated rat gastric glands.
    American journal of physiology. Gastrointestinal and liver physiology, 2006, Volume: 291, Issue:5

    Topics: Animals; Binding, Competitive; Diagnostic Imaging; Enzyme Inhibitors; Gastric Acid; Gastric Mucosa; Histamine; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Omeprazole; Potassium; Proton Pump Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley

2006