Page last updated: 2024-09-02

sch 28080 and cimetidine

sch 28080 has been researched along with cimetidine in 6 studies

Compound Research Comparison

Studies
(sch 28080)
Trials
(sch 28080)
Recent Studies (post-2010)
(sch 28080)
Studies
(cimetidine)
Trials
(cimetidine)
Recent Studies (post-2010) (cimetidine)
2170209,4731,687377

Protein Interaction Comparison

ProteinTaxonomysch 28080 (IC50)cimetidine (IC50)
Solute carrier family 22 member 1Mus musculus (house mouse)0.59
Solute carrier family 22 member 2Mus musculus (house mouse)8
Potassium-transporting ATPase alpha chain 1Homo sapiens (human)0.82
Histamine H2 receptorHomo sapiens (human)1.1742
Histamine H2 receptorCavia porcellus (domestic guinea pig)1.02
Potassium-transporting ATPase subunit betaHomo sapiens (human)0.82
Multidrug and toxin extrusion protein 1Homo sapiens (human)3.0333

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19903 (50.00)18.7374
1990's3 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Conn, DJ; Domalski, MS; Elliott, AJ; Guzik, H; Hilbert, JM; Kaminski, JJ; Lovey, RG; Pramanik, BN; Rizvi, RK; Solomon, DM1
Cárdenas, P; Chacín, J; Hernández, I; Lobo, P1
Fryklund, J; Gedda, K; Sachs, G; Scott, D; Wallmark, B1
Blissard, D; Cragoe, EJ; Muallem, S; Sachs, G1
Chiu, PJ; Derelanko, MJ; Long, JF; Steinberg, M1
Carrasquer, G; Geng, Z; Rehm, WS; Schwartz, M; Zhang, JY1

Other Studies

6 other study(ies) available for sch 28080 and cimetidine

ArticleYear
Antiulcer agents. 2. Gastric antisecretory, cytoprotective, and metabolic properties of substituted imidazo[1,2-a]pyridines and analogues.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:11

    Topics: Animals; Anti-Ulcer Agents; Dogs; Gastric Acid; Gastric Mucosa; Imidazoles; Pyridines; Rats; Structure-Activity Relationship

1987
Secretory and metabolic effects of ethanol in the isolated amphibian gastric mucosa.
    Gastroenterology, 1991, Volume: 100, Issue:5 Pt 1

    Topics: Alcohol Dehydrogenase; Alcoholic Beverages; Animals; Anti-Ulcer Agents; Beer; Bufo marinus; Cimetidine; Ethanol; Gastric Acid; Gastric Mucosa; Imidazoles; In Vitro Techniques; Lactates; Lactic Acid; Oxygen Consumption; Pyruvates; Pyruvic Acid; Secretory Rate; Wine

1991
Coupling of H(+)-K(+)-ATPase activity and glucose oxidation in gastric glands.
    The American journal of physiology, 1990, Volume: 258, Issue:5 Pt 1

    Topics: Adenosine Triphosphatases; Aminopyrine; Ammonia; Animals; Anti-Ulcer Agents; Atropine; Bucladesine; Carbachol; Carbon Dioxide; Cimetidine; Gastric Mucosa; Glucose; Glycolysis; H(+)-K(+)-Exchanging ATPase; Histamine; Imidazoles; In Vitro Techniques; Kinetics; Models, Biological; Omeprazole; Oxygen Consumption; Rats

1990
Activation of the Na+/H+ and Cl-/HCO3- exchange by stimulation of acid secretion in the parietal cell.
    The Journal of biological chemistry, 1988, Oct-15, Volume: 263, Issue:29

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Aminacrine; Animals; Anti-Ulcer Agents; Bicarbonates; Cell Membrane; Chlorides; Cimetidine; Cytosol; Gastric Acid; Histamine; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Kinetics; Parietal Cells, Gastric; Rabbits; Sodium

1988
Gastric antisecretory and cytoprotective activities of SCH 28080.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Aspirin; Cimetidine; Dogs; Ethanol; Female; Gastric Acid; Gastric Mucosa; Histamine; Imidazoles; Indomethacin; Male; Membrane Potentials; Rats; Stomach Ulcer; Stress, Physiological

1983
Electrogenicity of the frog gastric mucosa proton pump based on polarization responses in the presence of H(+)-secretion inhibitors.
    Biochimica et biophysica acta, 1993, Jul-04, Volume: 1149, Issue:2

    Topics: Animals; Cimetidine; Electrophysiology; Gastric Mucosa; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Models, Biological; Proton Pumps; Rana pipiens; Thiocyanates

1993