Page last updated: 2024-09-02

sch 28080 and bafilomycin a1

sch 28080 has been researched along with bafilomycin a1 in 15 studies

Compound Research Comparison

Studies
(sch 28080)
Trials
(sch 28080)
Recent Studies (post-2010)
(sch 28080)
Studies
(bafilomycin a1)
Trials
(bafilomycin a1)
Recent Studies (post-2010) (bafilomycin a1)
2170201,1201484

Protein Interaction Comparison

ProteinTaxonomysch 28080 (IC50)bafilomycin a1 (IC50)
P2X purinoceptor 3Homo sapiens (human)0.755
V-type proton ATPase subunit S1Homo sapiens (human)0.1
Vacuolar proton pump subunit B Gallus gallus (chicken)0.03

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's13 (86.67)18.2507
2000's1 (6.67)29.6817
2010's1 (6.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abrahamse, SL; Bindels, RJ; van Os, CH; Vis, A1
Boisvert, DM; Buckman, S; Harrison, V; Iacovitti, M; Levine, DZ; Nadler, SP; Vandorpe, D1
Armitage, FE; Wingo, CS1
Cragoe Júnior, EJ; Dantas, WF; de Lira, RF; Fernandez, R; Lopes, MJ; Malnic, G1
Gillies, RJ; Lynch, RM; Martinez, GM; Martinez-Zaguilan, R1
Kohn, OF; Mitchell, PP; Steinmetz, PR1
Schwartz, GJ; Tsuruoka, S1
DuBose, TD; Truong, AV; Wall, SM1
Milton, AE; Weiner, ID1
Gekle, M; Oberleithner, H; Silbernagl, S1
Choe, H; Frindt, G; Silver, RB1
Frank, AE; Weiner, ID; Wingo, CS1
Abbiati, T; Aronson, PS; Giebisch, G; Schultheis, PJ; Shull, GE; Wang, T; Yang, CL1
Barry, CR; Youmans, SJ1
Alves-Bezerra, M; Dick, CF; Freitas-Mesquita, AL; Gondim, KC; Majerowicz, D; Meyer-Fernandes, JR; Russo-Abrahão, T1

Other Studies

15 other study(ies) available for sch 28080 and bafilomycin a1

ArticleYear
Regulation of intracellular pH in crypt cells from rabbit distal colon.
    The American journal of physiology, 1994, Volume: 267, Issue:3 Pt 1

    Topics: Amiloride; Ammonia; Animals; Anti-Bacterial Agents; Buffers; Colon; Female; Fluoresceins; Fluorescent Dyes; Hydrogen-Ion Concentration; Imidazoles; Intracellular Membranes; Macrolides; Male; Quaternary Ammonium Compounds; Rabbits; Sodium

1994
In vivo adaptation of bicarbonate reabsorption by rat distal tubules during acid loading.
    The American journal of physiology, 1994, Volume: 267, Issue:5 Pt 2

    Topics: Acclimatization; Acidosis; Acute Disease; Amiloride; Ammonium Chloride; Animals; Anti-Bacterial Agents; Anti-Ulcer Agents; Antifungal Agents; Bicarbonates; Chronic Disease; Diet; Fasting; Hydrochloric Acid; Imidazoles; In Vitro Techniques; Infusions, Intravenous; Kidney Tubules, Distal; Macrolides; Male; Perfusion; Proton-Translocating ATPases; Rats; Rats, Sprague-Dawley; Reference Values

1994
Luminal acidification in K-replete OMCDi: contributions of H-K-ATPase and bafilomycin-A1-sensitive H-ATPase.
    The American journal of physiology, 1994, Volume: 267, Issue:3 Pt 2

    Topics: Acids; Animals; Anti-Bacterial Agents; Carbon Dioxide; Electrophysiology; Female; H(+)-K(+)-Exchanging ATPase; Imidazoles; In Vitro Techniques; Kidney Medulla; Kidney Tubules, Collecting; Macrolides; Naphthoquinones; Potassium; Proton Pump Inhibitors; Proton-Translocating ATPases; Rabbits

1994
Mechanism of acidification along cortical distal tubule of the rat.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 2

    Topics: Amiloride; Animals; Anti-Bacterial Agents; Antifungal Agents; Bicarbonates; Epithelium; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Kidney Cortex; Kidney Tubules, Distal; Kinetics; Macrolides; Male; Membrane Potentials; Perfusion; Potassium Deficiency; Proton Pump Inhibitors; Proton-Translocating ATPases; Rats; Rats, Wistar

1994
Vacuolar-type H(+)-ATPases are functionally expressed in plasma membranes of human tumor cells.
    The American journal of physiology, 1993, Volume: 265, Issue:4 Pt 1

    Topics: Anti-Bacterial Agents; Cell Membrane; Humans; Hydrogen-Ion Concentration; Imidazoles; Leiomyosarcoma; Macrolides; Mesothelioma; Proton-Translocating ATPases; Rest; Tumor Cells, Cultured; Vacuoles

1993
Sch-28080 inhibits bafilomycin-sensitive H+ secretion in turtle bladder independently of luminal [K+].
    The American journal of physiology, 1993, Volume: 265, Issue:2 Pt 2

    Topics: Animals; Anti-Bacterial Agents; Hydrogen; Imidazoles; In Vitro Techniques; Macrolides; Osmolar Concentration; Potassium; Urinary Bladder

1993
Adaptation of rabbit cortical collecting duct HCO3- transport to metabolic acidosis in vitro.
    The Journal of clinical investigation, 1996, Feb-15, Volume: 97, Issue:4

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acidosis; Animals; Anti-Bacterial Agents; Bicarbonates; Biological Transport; Chlorides; Culture Techniques; Enzyme Inhibitors; Female; Imidazoles; Kidney Cortex; Kidney Tubules, Collecting; Macrolides; Membrane Potentials; Proton Pump Inhibitors; Proton-Translocating ATPases; Rabbits

1996
H(+)-K(+)-ATPase mediates net acid secretion in rat terminal inner medullary collecting duct.
    The American journal of physiology, 1996, Volume: 271, Issue:5 Pt 2

    Topics: Absorption; Acids; Animals; Anti-Bacterial Agents; Biological Transport; Carbon Dioxide; Enzyme Inhibitors; H(+)-K(+)-Exchanging ATPase; Imidazoles; Kidney Medulla; Kidney Tubules, Collecting; Macrolides; Male; Potassium; Proton Pump Inhibitors; Rats; Rats, Sprague-Dawley; Vacuoles

1996
Intracellular pH regulation in the rabbit cortical collecting duct A-type intercalated cell.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 2

    Topics: Amiloride; Animals; Anti-Bacterial Agents; Enzyme Inhibitors; Female; Homeostasis; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Intracellular Fluid; Kidney Cortex; Kidney Tubules, Collecting; Kinetics; Macrolides; Perfusion; Proton Pump Inhibitors; Proton-Translocating ATPases; Rabbits; Sodium

1997
The mineralocorticoid aldosterone activates a proton conductance in cultured kidney cells.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Aldosterone; Animals; Anti-Bacterial Agents; Cell Line; Dogs; Enzyme Inhibitors; Hydrogen-Ion Concentration; Imidazoles; Kidney; Kinetics; Macrolides; Meglumine; Membrane Potentials; Naphthalenes; Pertussis Toxin; Protein Kinase C; Protein Serine-Threonine Kinases; Proton Pump Inhibitors; Proton-Translocating ATPases; Sodium-Hydrogen Exchangers; Spironolactone; Staurosporine; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella; Zinc

1997
Low-NaCl diet increases H-K-ATPase in intercalated cells from rat cortical collecting duct.
    The American journal of physiology, 1998, Volume: 275, Issue:1

    Topics: Aldosterone; Animals; Anti-Bacterial Agents; Diet, Sodium-Restricted; Electrolytes; Enzyme Induction; Enzyme Inhibitors; Female; H(+)-K(+)-Exchanging ATPase; Hydrogen-Ion Concentration; Imidazoles; Kidney Cortex; Kidney Tubules, Collecting; Kinetics; Macrolides; Male; Ouabain; Proton Pump Inhibitors; Rats; Rats, Sprague-Dawley; Reference Values; Time Factors

1998
Apical proton secretion by the inner stripe of the outer medullary collecting duct.
    The American journal of physiology, 1999, Volume: 276, Issue:4

    Topics: Animals; Anti-Bacterial Agents; Cell Membrane; Enzyme Inhibitors; H(+)-K(+)-Exchanging ATPase; Hydrogen-Ion Concentration; Imidazoles; Kidney Medulla; Kidney Tubules, Collecting; Macrolides; Proton Pump Inhibitors; Proton Pumps; Proton-Translocating ATPases; Protons; Rabbits

1999
Mechanism of proximal tubule bicarbonate absorption in NHE3 null mice.
    The American journal of physiology, 1999, Volume: 277, Issue:2

    Topics: Absorption; Amiloride; Animals; Anti-Bacterial Agents; Bicarbonates; Enzyme Inhibitors; H(+)-K(+)-Exchanging ATPase; Imidazoles; Kidney Tubules, Proximal; Macrolides; Mice; Mice, Knockout; Reference Values; Sodium-Hydrogen Exchanger 3; Sodium-Hydrogen Exchangers

1999
Bafilomycin A1 at nanomolar concentrations saturably inhibits a portion of turtle bladder acidification current.
    The Journal of experimental biology, 2001, Volume: 204, Issue:Pt 16

    Topics: Animals; Anti-Bacterial Agents; Enzyme Inhibitors; Hydrogen-Ion Concentration; Imidazoles; Macrolides; Turtles; Urinary Bladder; Vacuolar Proton-Translocating ATPases

2001
Transport of inorganic phosphate in Leishmania infantum and compensatory regulation at low inorganic phosphate concentration.
    Biochimica et biophysica acta, 2013, Volume: 1830, Issue:3

    Topics: Amino Acid Sequence; Biological Transport; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Culture Media; Enzyme Inhibitors; Gene Expression Regulation; Imidazoles; Kinetics; Leishmania infantum; Macrolides; Molecular Sequence Data; Nigericin; Phosphates; Phosphorus Radioisotopes; Phylogeny; Proton Ionophores; Proton-Phosphate Symporters; Protozoan Proteins; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Sodium-Phosphate Cotransporter Proteins; Sodium-Potassium-Exchanging ATPase; Vacuolar Proton-Translocating ATPases

2013