Page last updated: 2024-09-02

sch 28080 and amiloride

sch 28080 has been researched along with amiloride in 17 studies

Compound Research Comparison

Studies
(sch 28080)
Trials
(sch 28080)
Recent Studies (post-2010)
(sch 28080)
Studies
(amiloride)
Trials
(amiloride)
Recent Studies (post-2010) (amiloride)
2170207,584339788

Protein Interaction Comparison

ProteinTaxonomysch 28080 (IC50)amiloride (IC50)
Urokinase-type plasminogen activatorHomo sapiens (human)4.7
Urokinase-type plasminogen activatorMus musculus (house mouse)2.3
Amine oxidase [flavin-containing] AHomo sapiens (human)3.909
Sodium/hydrogen exchanger 1Rattus norvegicus (Norway rat)1
Amiloride-sensitive sodium channel subunit alphaHomo sapiens (human)0.776
Sodium/hydrogen exchanger 2Oryctolagus cuniculus (rabbit)1
Acid-sensing ion channel 3Homo sapiens (human)4.4

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.88)18.7374
1990's12 (70.59)18.2507
2000's2 (11.76)29.6817
2010's2 (11.76)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abrahamse, SL; Bindels, RJ; van Os, CH1
Alpern, RJ; Hays, SR1
Blissard, D; Cragoe, EJ; Muallem, S; Sachs, G1
Abrahamse, SL; Bindels, RJ; van Os, CH; Vis, A1
Boisvert, DM; Buckman, S; Harrison, V; Iacovitti, M; Levine, DZ; Nadler, SP; Vandorpe, D1
Buckman, S; Harrison, V; Iacovitti, M; Levine, DZ; Nadler, SP; Vandorpe, D1
Cragoe Júnior, EJ; Dantas, WF; de Lira, RF; Fernandez, R; Lopes, MJ; Malnic, G1
Hayashi, M; Iyori, M; Saruta, T; Yamaji, Y1
Dagher, G; Griffiths, N; Sauterey, C; Siaume-Perez, S; Thomas, SR1
Milton, AE; Weiner, ID1
Attmane-Elakeb, A; Bichara, M; Boulanger, H; Vernimmen, C1
Wesson, DE1
Abbiati, T; Aronson, PS; Giebisch, G; Schultheis, PJ; Shull, GE; Wang, T; Yang, CL1
Fischer, H; Illek, B; Widdicombe, JH1
Bachmann, O; Heinzmann, A; Mack, A; Manns, MP; Seidler, U1
Cain, BD; Gumz, ML; Shao, J; Shull, GE; van Driel, IR; Wingo, CS; Xia, SL1
Aravena, C; Beltrán, AR; Cornejo, M; Díaz, ES; Guzmán-Gutiérrez, E; Leiva, A; Pardo, F; Ramírez, MA; Sobrevia, L; Torres, V1

Other Studies

17 other study(ies) available for sch 28080 and amiloride

ArticleYear
The colon carcinoma cell line Caco-2 contains an H+/K(+)-ATPase that contributes to intracellular pH regulation.
    Pflugers Archiv : European journal of physiology, 1992, Volume: 421, Issue:6

    Topics: Amiloride; Ammonium Chloride; Anti-Bacterial Agents; Anti-Ulcer Agents; Carcinoma; Colonic Neoplasms; Ethylmaleimide; H(+)-K(+)-Exchanging ATPase; Humans; Hydrogen-Ion Concentration; Imidazoles; Macrolides; Sodium Chloride; Tumor Cells, Cultured

1992
Apical and basolateral membrane H+ extrusion mechanisms in inner stripe of rabbit outer medullary collecting duct.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 2

    Topics: Amiloride; Animals; Cell Membrane; Ethylmaleimide; Female; Hydrochloric Acid; Hydrogen; Hydrogen-Ion Concentration; Imidazoles; Kidney Medulla; Kidney Tubules, Collecting; Protons; Rabbits; Sodium; Time Factors

1990
Activation of the Na+/H+ and Cl-/HCO3- exchange by stimulation of acid secretion in the parietal cell.
    The Journal of biological chemistry, 1988, Oct-15, Volume: 263, Issue:29

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Aminacrine; Animals; Anti-Ulcer Agents; Bicarbonates; Cell Membrane; Chlorides; Cimetidine; Cytosol; Gastric Acid; Histamine; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Kinetics; Parietal Cells, Gastric; Rabbits; Sodium

1988
Regulation of intracellular pH in crypt cells from rabbit distal colon.
    The American journal of physiology, 1994, Volume: 267, Issue:3 Pt 1

    Topics: Amiloride; Ammonia; Animals; Anti-Bacterial Agents; Buffers; Colon; Female; Fluoresceins; Fluorescent Dyes; Hydrogen-Ion Concentration; Imidazoles; Intracellular Membranes; Macrolides; Male; Quaternary Ammonium Compounds; Rabbits; Sodium

1994
In vivo adaptation of bicarbonate reabsorption by rat distal tubules during acid loading.
    The American journal of physiology, 1994, Volume: 267, Issue:5 Pt 2

    Topics: Acclimatization; Acidosis; Acute Disease; Amiloride; Ammonium Chloride; Animals; Anti-Bacterial Agents; Anti-Ulcer Agents; Antifungal Agents; Bicarbonates; Chronic Disease; Diet; Fasting; Hydrochloric Acid; Imidazoles; In Vitro Techniques; Infusions, Intravenous; Kidney Tubules, Distal; Macrolides; Male; Perfusion; Proton-Translocating ATPases; Rats; Rats, Sprague-Dawley; Reference Values

1994
Distal tubule unidirectional HCO3 reabsorption in vivo during acute and chronic metabolic alkalosis in the rat.
    The American journal of physiology, 1994, Volume: 266, Issue:6 Pt 2

    Topics: Absorption; Acute Disease; Alkalosis; Amiloride; Animals; Anti-Bacterial Agents; Bicarbonates; Chronic Disease; Imidazoles; Kidney Tubules, Distal; Macrolides; Male; Perfusion; Rats; Rats, Sprague-Dawley

1994
Mechanism of acidification along cortical distal tubule of the rat.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 2

    Topics: Amiloride; Animals; Anti-Bacterial Agents; Antifungal Agents; Bicarbonates; Epithelium; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Kidney Cortex; Kidney Tubules, Distal; Kinetics; Macrolides; Male; Membrane Potentials; Perfusion; Potassium Deficiency; Proton Pump Inhibitors; Proton-Translocating ATPases; Rats; Rats, Wistar

1994
Effects of in vivo and in vitro alkali treatment on intracellular pH regulation of OMCDis cells.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 2

    Topics: Amiloride; Ammonia; Ammonium Chloride; Animals; Carbon Dioxide; Ethylmaleimide; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Intracellular Fluid; Kidney Medulla; Kidney Tubules, Collecting; Oxygen; Partial Pressure; Rabbits

1993
Calcitonin activates an Na(+)-independent HCO3(-)-dependent pathway in the rabbit distal convoluted tubule.
    The American journal of physiology, 1997, Volume: 273, Issue:1 Pt 2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Bicarbonates; Calcitonin; Carbon Dioxide; Chlorides; Cyclic AMP; Ethylmaleimide; Glutamine; Homeostasis; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Ketoglutaric Acids; Kidney Tubules, Distal; Male; Microscopy, Fluorescence; Quaternary Ammonium Compounds; Rabbits; Sodium; Sodium-Hydrogen Exchangers

1997
Intracellular pH regulation in the rabbit cortical collecting duct A-type intercalated cell.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 2

    Topics: Amiloride; Animals; Anti-Bacterial Agents; Enzyme Inhibitors; Female; Homeostasis; Hydrogen-Ion Concentration; Imidazoles; In Vitro Techniques; Intracellular Fluid; Kidney Cortex; Kidney Tubules, Collecting; Kinetics; Macrolides; Perfusion; Proton Pump Inhibitors; Proton-Translocating ATPases; Rabbits; Sodium

1997
Apical location and inhibition by arginine vasopressin of K+/H+ antiport of the medullary thick ascending limb of rat kidney.
    The Journal of biological chemistry, 1997, Oct-10, Volume: 272, Issue:41

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Triphosphatases; Amiloride; Animals; Antiporters; Arginine Vasopressin; Barium; Calcium Channel Blockers; Cyclic AMP-Dependent Protein Kinases; Diuretics; Enzyme Inhibitors; Hydrogen; Hydrogen-Ion Concentration; Imidazoles; Loop of Henle; Male; Potassium Channels; Potassium-Hydrogen Antiporters; Rats; Rats, Sprague-Dawley; Renal Agents; Rubidium; Verapamil

1997
Na/H exchange and H-K ATPase increase distal tubule acidification in chronic alkalosis.
    Kidney international, 1998, Volume: 53, Issue:4

    Topics: Acid-Base Equilibrium; Acids; Aldosterone; Alkalosis; Amiloride; Animals; Anti-Arrhythmia Agents; Anti-Bacterial Agents; Bicarbonates; Endothelins; Enzyme Inhibitors; Female; H(+)-K(+)-Exchanging ATPase; Imidazoles; Kidney Tubules, Distal; Macrolides; Male; Rats; Rats, Wistar; Sodium-Hydrogen Exchangers

1998
Mechanism of proximal tubule bicarbonate absorption in NHE3 null mice.
    The American journal of physiology, 1999, Volume: 277, Issue:2

    Topics: Absorption; Amiloride; Animals; Anti-Bacterial Agents; Bicarbonates; Enzyme Inhibitors; H(+)-K(+)-Exchanging ATPase; Imidazoles; Kidney Tubules, Proximal; Macrolides; Mice; Mice, Knockout; Reference Values; Sodium-Hydrogen Exchanger 3; Sodium-Hydrogen Exchangers

1999
Acid secretion and proton conductance in human airway epithelium.
    American journal of physiology. Cell physiology, 2002, Volume: 282, Issue:4

    Topics: Acids; Adenosine Triphosphate; Amiloride; Biological Transport; Cells, Cultured; Chlorides; Diffusion Chambers, Culture; Diuretics; Enzyme Inhibitors; Histamine; Humans; Hydrogen-Ion Concentration; Imidazoles; Mast Cells; Membrane Potentials; Patch-Clamp Techniques; Protons; Respiratory Mucosa; Trachea; Zinc Compounds

2002
Mechanisms of secretion-associated shrinkage and volume recovery in cultured rabbit parietal cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 292, Issue:3

    Topics: Adenosine Triphosphatases; Amiloride; Animals; Carbachol; Cell Size; Cells, Cultured; Charybdotoxin; Chloride Channels; Chromans; Colforsin; Enzyme Inhibitors; Guanidines; Hydrogen-Ion Concentration; Imidazoles; Ion Channels; KCNQ1 Potassium Channel; Nitrobenzoates; Parietal Cells, Gastric; Potassium Channel Blockers; Rabbits; Sodium-Calcium Exchanger; Sodium-Hydrogen Exchangers; Sulfonamides; Sulfones

2007
Pharmacological profiles of the murine gastric and colonic H,K-ATPases.
    Biochimica et biophysica acta, 2010, Volume: 1800, Issue:9

    Topics: Amiloride; Animals; Catalytic Domain; Colon; Drug Resistance; Enzyme Inhibitors; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Imidazoles; Mice; Mice, Knockout; Organ Specificity; Ouabain; Proton Pump Inhibitors; Sodium Channel Blockers; Vanadates

2010
Potential role of sodium-proton exchangers in the low concentration arsenic trioxide-increased intracellular pH and cell proliferation.
    PloS one, 2012, Volume: 7, Issue:12

    Topics: Amiloride; Analysis of Variance; Animals; Arsenic Trioxide; Arsenicals; Blotting, Western; Carbazoles; Cell Count; Cell Fractionation; Cell Proliferation; Dogs; Flavonoids; Fluorometry; Hydrogen-Ion Concentration; Imidazoles; Macrolides; Madin Darby Canine Kidney Cells; Oxides; Sodium-Hydrogen Exchangers

2012