Page last updated: 2024-09-03

sc 53116 and sdz 205-557

sc 53116 has been researched along with sdz 205-557 in 4 studies

Compound Research Comparison

Studies
(sc 53116)
Trials
(sc 53116)
Recent Studies (post-2010)
(sc 53116)
Studies
(sdz 205-557)
Trials
(sdz 205-557)
Recent Studies (post-2010) (sdz 205-557)
20035609

Protein Interaction Comparison

ProteinTaxonomysc 53116 (IC50)sdz 205-557 (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.2512
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.2512

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (75.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fischmeister, R; Langlois, M1
Flynn, DL; Goldstin, B; Gullikson, GW; Moormann, AE; Yang, DC1
Lambert, HW; Lauder, JM1
Adaikan, PG; Hayes, ES; Ng, SC; Ratnam, SS1

Reviews

1 review(s) available for sc 53116 and sdz 205-557

ArticleYear
5-HT4 receptor ligands: applications and new prospects.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Benzoates; Binding Sites; Cardiovascular Physiological Phenomena; Central Nervous System; Digestive System Physiological Phenomena; Humans; Indoles; Ketones; Ligands; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

3 other study(ies) available for sc 53116 and sdz 205-557

ArticleYear
SC-53606, a potent and selective antagonist of 5-hydroxytryptamine4 receptors in isolated rat esophageal tunica muscularis mucosae.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Esophagus; Imidazoles; In Vitro Techniques; Indoles; Male; Mucous Membrane; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Pyrroles; Rats; Receptors, Cell Surface; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron; Tryptamines

1993
Serotonin receptor agonists that increase cyclic AMP positively regulate IGF-I in mouse mandibular mesenchymal cells.
    Developmental neuroscience, 1999, Volume: 21, Issue:2

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Cells, Cultured; Culture Media; Culture Media, Serum-Free; Cyclic AMP; Cysteine; Embryo, Mammalian; Insulin-Like Growth Factor I; Insulin-Like Growth Factor II; Mandible; Mesoderm; Mice; Nialamide; para-Aminobenzoates; Piperazines; Pyrroles; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
5-HT4 receptors in isolated human corpus cavernosum?
    International journal of impotence research, 1999, Volume: 11, Issue:4

    Topics: 4-Aminobenzoic Acid; Adrenergic beta-Antagonists; Benzamides; Humans; Male; Methysergide; Muscle Relaxation; Norepinephrine; para-Aminobenzoates; Penis; Pindolol; Pyrroles; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists

1999