Page last updated: 2024-09-03

sc 53116 and mosapride

sc 53116 has been researched along with mosapride in 3 studies

Compound Research Comparison

Studies
(sc 53116)
Trials
(sc 53116)
Recent Studies (post-2010)
(sc 53116)
Studies
(mosapride)
Trials
(mosapride)
Recent Studies (post-2010) (mosapride)
200328690142

Protein Interaction Comparison

ProteinTaxonomysc 53116 (IC50)mosapride (IC50)
hepatocyte nuclear factor 4-alpha isoform 2Homo sapiens (human)4.18
perilipin-5Homo sapiens (human)1.315
perilipin-1Homo sapiens (human)1.196
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform aHomo sapiens (human)1.2753
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.3966
Cytochrome P450 1A2Homo sapiens (human)0.4
Cytochrome P450 3A4Homo sapiens (human)0.7
Alpha-2A adrenergic receptorHomo sapiens (human)3.6794
Cytochrome P450 2C9 Homo sapiens (human)1
Alpha-2B adrenergic receptorHomo sapiens (human)1.908
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.3966
Sodium-dependent serotonin transporterHomo sapiens (human)3.8117
Cytochrome P450 2C19Homo sapiens (human)1
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.2959
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)4.7932
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.3056

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fischmeister, R; Langlois, M1
Fujiwara, I; Harada, H; Hirokawa, Y; Kato, S; Suzuki, K; Yoshida, N; Yoshikawa, T1
Kamato, T; Miyata, K; Nagakura, Y; Yamano, M1

Reviews

1 review(s) available for sc 53116 and mosapride

ArticleYear
5-HT4 receptor ligands: applications and new prospects.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Benzoates; Binding Sites; Cardiovascular Physiological Phenomena; Central Nervous System; Digestive System Physiological Phenomena; Humans; Indoles; Ketones; Ligands; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

2 other study(ies) available for sc 53116 and mosapride

ArticleYear
Synthesis and structure-affinity relationships of novel N-(1-ethyl-4-methylhexahydro-1,4-diazepin-6-yl)pyridine-3-carboxamides with potent serotonin 5-HT3 and dopamine D2 receptor antagonistic activity.
    Journal of medicinal chemistry, 2003, Feb-27, Volume: 46, Issue:5

    Topics: Animals; Antiemetics; Azepines; Brain; Crystallography, X-Ray; Dogs; Dopamine Antagonists; Ferrets; In Vitro Techniques; Models, Molecular; Pyridines; Rats; Receptors, Dopamine D2; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship

2003
Effects of gastroprokinetic agents on gastroparesis in streptozotocin-induced diabetic rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: Animals; Benzamides; Benzimidazoles; Blood Glucose; Cisapride; Diabetes Mellitus, Experimental; Gastric Emptying; Gastrointestinal Motility; Gastroparesis; Granisetron; Male; Morpholines; Ondansetron; Piperidines; Pyrroles; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists; Vagotomy

1997