Page last updated: 2024-09-05

sb 216763 and 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine

sb 216763 has been researched along with 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine in 1 studies

Compound Research Comparison

Studies
(sb 216763)
Trials
(sb 216763)
Recent Studies (post-2010)
(sb 216763)
Studies
(1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine)
Trials
(1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine)
Recent Studies (post-2010) (1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine)
34202251507

Protein Interaction Comparison

ProteinTaxonomysb 216763 (IC50)1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine (IC50)
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)0.13
Serine/threonine-protein kinase D3Homo sapiens (human)0.616
Tyrosine-protein kinase ABL1Homo sapiens (human)1.76
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)0.62
Proto-oncogene tyrosine-protein kinase LCK Mus musculus (house mouse)0.46
Tyrosine-protein kinase FynHomo sapiens (human)1
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)0.5
Cyclin-dependent kinase 2Homo sapiens (human)0.005
Tyrosine-protein kinase CSKHomo sapiens (human)0.51
Mitogen-activated protein kinase 8Homo sapiens (human)0.195
Serine/threonine-protein kinase D1Homo sapiens (human)0.6315
Serine/threonine-protein kinase D2Homo sapiens (human)0.786
Cyclin-dependent kinase 12Homo sapiens (human)0.1
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)0.008

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1

Other Studies

1 other study(ies) available for sb 216763 and 1-tert-butyl-3-naphthalen-1-ylmethyl-1h-pyrazolo(3,4-d)pyrimidin-4-ylemine

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007