Compounds > sb 206553
Page last updated: 2024-08-16

sb 206553 and sb 221284

sb 206553 has been researched along with sb 221284 in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blackburn, TP; Blaney, FE; Bromidge, SM; Clarke, SE; Duckworth, M; Forbes, IT; Ham, P; Kennett, GA; King, FD; Naylor, CB; Thewlis, KM; Wood, MD1
Bailey, F; Blackburn, TP; Blaney, FE; Bromidge, SM; Dabbs, S; Davies, DT; Duckworth, DM; Forbes, IT; Ham, P; Holland, V; Jones, GE; Kennett, GA; King, FD; Naylor, CB; Riley, GJ; Saunders, DV; Starr, S; Thewlis, KM; Wood, MD; Wyman, PA1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1

Other Studies

3 other study(ies) available for sb 206553 and sb 221284

ArticleYear
6-Chloro-5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]- indoline (SB-242084): the first selective and brain penetrant 5-HT2C receptor antagonist.
    Journal of medicinal chemistry, 1997, Oct-24, Volume: 40, Issue:22

    Topics: Aminopyridines; Animals; Blood-Brain Barrier; Cell Line; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Humans; Indoles; Molecular Structure; Rats; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists

1997
Novel and selective 5-HT2C/2B receptor antagonists as potential anxiolytic agents: synthesis, quantitative structure-activity relationships, and molecular modeling of substituted 1-(3-pyridylcarbamoyl)indolines.
    Journal of medicinal chemistry, 1998, May-07, Volume: 41, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Conditioning, Operant; Conflict, Psychological; Indoles; Male; Models, Molecular; Motor Activity; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Social Behavior; Structure-Activity Relationship

1998
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004