Page last updated: 2024-08-16

sb 206553 and ketanserin

sb 206553 has been researched along with ketanserin in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (6.25)18.2507
2000's11 (68.75)29.6817
2010's4 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Bienkowski, P; Bucki, A; Jaśkowska, J; Kazek, G; Kowalski, P; Kołaczkowski, M; Marcinkowska, M; Mierzejewski, P; Mitka, K; Pawłowski, M; Siwek, A; Wasik, A; Wesołowska, A1
Caldarola-Pastuszka, M; DeLashaw, M; Uphouse, L; Wolf, A1
Fiorica-Howells, E; Gershon, MD; Maroteaux, L1
Adlersberg, M; Arango, V; Hsiung, S; Kassir, SA; Liu, K; Mann, JJ; Ruggiero, DA; Tamir, H; Underwood, MD1
Inoue, K; Ohkura, M; Sugimoto, Y; Yamada, J1
Sugimoto, Y; Yamada, J1
Bourin, M; Hascoët, M; Nic Dhonnchadha, BA1
Cunningham, KA; Filip, M; McCreary, AC1
Sinclair-Worley, L; Uphouse, L1
Arnold, JC; McGregor, IS; Morley, KC1
Bourin, M; Dailly, E; Hascoët, M; Masse, F1
Ahmad, R; Egerton, A; Grasby, PM; Hirani, E1
MacFarlane, PM; Mitchell, GS; Vinit, S1
Nagatani, H; Nakata, Y; Oshima, T; Saitoh, Y; Urano, A; Yokota, M1
Abman, SH; Delaney, C; Gien, J; Grover, TR; Roe, G1

Other Studies

16 other study(ies) available for sb 206553 and ketanserin

ArticleYear
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Novel arylsulfonamide derivatives with 5-HT₆/5-HT₇ receptor antagonism targeting behavioral and psychological symptoms of dementia.
    Journal of medicinal chemistry, 2014, Jun-12, Volume: 57, Issue:11

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Avoidance Learning; Benzoxazoles; Catalepsy; CHO Cells; Cricetulus; Dementia; Dopamine D2 Receptor Antagonists; HEK293 Cells; Humans; Male; Models, Molecular; Motor Activity; Radioligand Assay; Rats, Wistar; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Sulfonamides

2014
5-HT2C receptor involvement in female rat lordosis behavior.
    Brain research, 1999, Apr-17, Volume: 825, Issue:1-2

    Topics: Animals; Estradiol; Female; Fluorobenzenes; Indoles; Indophenol; Ketanserin; Ovariectomy; Piperidines; Posture; Pyridines; Rats; Rats, Inbred Strains; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus

1999
Serotonin and the 5-HT(2B) receptor in the development of enteric neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Jan-01, Volume: 20, Issue:1

    Topics: Age Factors; Amphetamines; Animals; Antibodies; Antigens, Differentiation; Cell Differentiation; Cells, Cultured; Female; Fetus; Fluorescent Antibody Technique; Gene Expression Regulation, Developmental; Guinea Pigs; In Situ Hybridization; Indoles; Intestines; Ketanserin; Mice; Mice, Inbred Strains; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Myenteric Plexus; Neurons; Pregnancy; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Ritanserin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Ubiquitin Thiolesterase

2000
In vitro autoradiography of serotonin 5-HT(2A/2C) receptor-activated G protein: guanosine-5'-(gamma-[(35)S]thio)triphosphate binding in rat brain.
    Journal of neuroscience research, 2000, Sep-15, Volume: 61, Issue:6

    Topics: Amphetamines; Animals; Autoradiography; Brain Chemistry; Dose-Response Relationship, Drug; Fluorobenzenes; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Image Processing, Computer-Assisted; Indoles; Ketanserin; Male; Membrane Proteins; Piperidines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Subcellular Fractions; Sulfur Radioisotopes

2000
Involvement of the 5-HT(2) receptor in hyperthermia induced by p-chloroamphetamine, a serotonin-releasing drug in mice.
    European journal of pharmacology, 2000, Sep-08, Volume: 403, Issue:3

    Topics: Animals; Body Temperature Regulation; Dose-Response Relationship, Drug; Ergolines; Fever; Indoles; Ketanserin; Male; Mice; Motor Activity; p-Chloroamphetamine; Pyridines; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists

2000
Effects of 5-HT(2) receptor antagonists on the anti-immobility effects of imipramine in the forced swimming test with mice.
    European journal of pharmacology, 2001, Sep-21, Volume: 427, Issue:3

    Topics: Animals; Antidepressive Agents, Tricyclic; Dose-Response Relationship, Drug; Ergolines; Imipramine; Indoles; Ketanserin; Male; Mice; Motor Activity; Pyridines; Receptors, Serotonin; Serotonin Antagonists; Swimming

2001
Anxiolytic-like effects of 5-HT2 ligands on three mouse models of anxiety.
    Behavioural brain research, 2003, Mar-18, Volume: 140, Issue:1-2

    Topics: Amphetamines; Animals; Anti-Anxiety Agents; Anxiety; Disease Models, Animal; Dose-Response Relationship, Drug; Ethylamines; Indoles; Ketanserin; Male; Maze Learning; Mice; Motor Activity; Naphthyridines; Piperazine; Piperazines; Psychomotor Performance; Pyridines; Reaction Time; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Thiophenes

2003
Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
    Behavioral neuroscience, 2003, Volume: 117, Issue:2

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Fenfluramine; Fluorobenzenes; Indoles; Ketanserin; Male; Piperidines; Pyrazines; Pyridines; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Thiophenes

2003
Effect of estrogen on the lordosis-inhibiting action of ketanserin and SB 206553.
    Behavioural brain research, 2004, Jun-04, Volume: 152, Issue:1

    Topics: Analysis of Variance; Animals; Dose-Response Relationship, Drug; Drug Interactions; Estradiol; Female; Hypothalamus, Middle; Indoles; Ketanserin; Posture; Progesterone; Pyridines; Rats; Rats, Inbred F344; Serotonin Antagonists; Sexual Behavior, Animal; Time Factors

2004
Serotonin (1A) receptor involvement in acute 3,4-methylenedioxymethamphetamine (MDMA) facilitation of social interaction in the rat.
    Progress in neuro-psychopharmacology & biological psychiatry, 2005, Volume: 29, Issue:5

    Topics: Animals; Hallucinogens; Indoles; Interpersonal Relations; Ketanserin; Male; N-Methyl-3,4-methylenedioxyamphetamine; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Serotonin Agents; Serotonin Antagonists; Serotonin Syndrome

2005
Anxiolytic-like effect of milnacipran in the four-plate test in mice: mechanism of action.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzylamines; Brain; Cyclopropanes; Dopamine; Dose-Response Relationship, Drug; Fenclonine; Flumazenil; Fluorobenzenes; Idazoxan; Indoles; Ketanserin; Male; Mice; Milnacipran; Motor Activity; Neurotransmitter Uptake Inhibitors; Norepinephrine; Phenols; Prazosin; Punishment; Pyridines; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2005
Modulation of striatal dopamine release by 5-HT2A and 5-HT2C receptor antagonists: [11C]raclopride PET studies in the rat.
    Psychopharmacology, 2008, Volume: 200, Issue:4

    Topics: Amphetamine; Animals; Binding, Competitive; Carbon Radioisotopes; Corpus Striatum; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Indoles; Ketanserin; Male; Positron-Emission Tomography; Protein Binding; Pyridines; Raclopride; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2008
Serotonin 2A and 2B receptor-induced phrenic motor facilitation: differential requirement for spinal NADPH oxidase activity.
    Neuroscience, 2011, Mar-31, Volume: 178

    Topics: Acetophenones; Action Potentials; Amphetamines; Animals; Indoles; Injections, Spinal; Ketanserin; Male; NADPH Oxidases; Onium Compounds; Phrenic Nerve; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Thiophenes

2011
Blockade of 5-HT(2A) and/or 5-HT(2C) receptors modulates sevoflurane-induced immobility.
    Journal of anesthesia, 2011, Volume: 25, Issue:2

    Topics: Anesthetics, Inhalation; Animals; Immobilization; Indoles; Ketanserin; Male; Methyl Ethers; Pyridines; Rats; Rats, Wistar; Serotonin 5-HT2 Receptor Antagonists; Sevoflurane

2011
Pulmonary vascular effects of serotonin and selective serotonin reuptake inhibitors in the late-gestation ovine fetus.
    American journal of physiology. Lung cellular and molecular physiology, 2011, Volume: 301, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Dose-Response Relationship, Drug; Female; Fetus; Fluoxetine; Hemodynamics; Hypertension, Pulmonary; Hysterotomy; Indoles; Ketanserin; Lung; Oxadiazoles; Piperazines; Pregnancy; Pulmonary Artery; Pyridines; Receptors, Serotonin; rho-Associated Kinases; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Sertraline; Sheep; Vascular Resistance

2011