Page last updated: 2024-08-16

sb 206553 and alpha-methylserotonin

sb 206553 has been researched along with alpha-methylserotonin in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (12.50)18.2507
2000's6 (75.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Armstrong, SR; Beattie, DT; Humphrey, PP; Mai, N; Marquess, D; McCullough, JL; Pulido-Rios, T; Richardson, C; Sandlund, C; Smith, JA; Vickery, RG1
Javid, FA; Naylor, RJ1
Fernández, MM; Martín, ML; Morán, A; San Román, L1
Calama, E; Martín, ML; Morán, A; Ortiz de Urbina, AV; San Román, L1
Hackman, JC; Holohean, AM1
Cheng, Q; Dergacheva, O; Gorini, C; Jameson, H; Kamendi, H; Mendelowitz, D; Pinol, RM; Wang, X1
Bennett, DJ; Fouad, K; Murray, KC; Rank, MM; Sanelli, L; Vavrek, R1

Other Studies

8 other study(ies) available for sb 206553 and alpha-methylserotonin

ArticleYear
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
The 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivo.
    British journal of pharmacology, 2004, Volume: 143, Issue:5

    Topics: Animals; Cell Membrane; Cells, Cultured; Colon; Cyclic AMP; Esophagus; Gastric Fundus; Gastrointestinal Transit; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Pressure; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Characterisation of 5-HT2 receptor subtypes in the Suncus murinus intestine.
    European journal of pharmacology, 1999, Sep-24, Volume: 381, Issue:2-3

    Topics: Amphetamines; Animals; Female; In Vitro Techniques; Indoles; Intestines; Male; Muscle Contraction; Pyridines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Tachyphylaxis

1999
Mesenteric vasoconstrictor response to 5-hydroxytryptamine in the in situ blood autoperfused rat mesentery: involvement of 5-HT(2B) and/or 5-HT(2C) receptor activation.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: Amphetamines; Animals; Biguanides; Dose-Response Relationship, Drug; Enalapril; Indoles; Indomethacin; Male; Mesenteric Arteries; Mesentery; Perfusion; Piperazines; Prazosin; Propranolol; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Splanchnic Circulation; Vasoconstriction

2000
Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.
    Pharmacology, 2004, Volume: 71, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Hindlimb; Indoles; Injections, Intra-Arterial; Injections, Intravenous; Male; Perfusion; Piperazines; Prazosin; Pyridines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT2; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Spiperone; Thiophenes; Vasoconstriction

2004
Mechanisms intrinsic to 5-HT2B receptor-induced potentiation of NMDA receptor responses in frog motoneurones.
    British journal of pharmacology, 2004, Volume: 143, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Ergolines; Excitatory Amino Acid Antagonists; Gallopamil; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Indoles; Magnesium; Memantine; Membrane Potentials; Motor Neurons; N-Methylaspartate; Nifedipine; Protein Kinase C; Pyridines; Rana pipiens; Receptor, Serotonin, 5-HT2B; Receptors, N-Methyl-D-Aspartate; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Staurosporine; Sulfonamides; Tetrodotoxin

2004
5HT2 receptor activation facilitates P2X receptor mediated excitatory neurotransmission to cardiac vagal neurons in the nucleus ambiguus.
    Neuropharmacology, 2008, Volume: 54, Issue:7

    Topics: Action Potentials; Animals; Animals, Newborn; Drug Interactions; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Indoles; Neurons; Nucleus Accumbens; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P2; Receptors, Purinergic P2X; Receptors, Serotonin, 5-HT2; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes; Vagus Nerve

2008
Locomotion after spinal cord injury depends on constitutive activity in serotonin receptors.
    Journal of neurophysiology, 2010, Volume: 104, Issue:6

    Topics: Aminopyridines; Animals; Cordotomy; Electromyography; Female; Gait Disorders, Neurologic; Hindlimb; Indoles; Injections, Spinal; Locomotion; Muscle Hypotonia; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT2; Recovery of Function; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Spinal Cord Injuries; Tail

2010